JP5250029B2 - ２ｈ−インダゾールの遷移金属触媒合成 - Google Patents

２ｈ−インダゾールの遷移金属触媒合成 Download PDF

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Publication number
JP5250029B2
JP5250029B2 JP2010513708A JP2010513708A JP5250029B2 JP 5250029 B2 JP5250029 B2 JP 5250029B2 JP 2010513708 A JP2010513708 A JP 2010513708A JP 2010513708 A JP2010513708 A JP 2010513708A JP 5250029 B2 JP5250029 B2 JP 5250029B2
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JP
Japan
Prior art keywords
unsubstituted
indazole
phenyl
independently
substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
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JP2010513708A
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English (en)
Japanese (ja)
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JP2010531311A (ja
JP2010531311A5 (enExample
Inventor
ニス・ハールラント
マルク・ナツァーレ
アンドレーアス・リンデンシュミット
ホルヘ・アロンソ
オマール・ルカイク
マティーアス・ウルマン
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Sanofi SA
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Sanofi SA
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Publication of JP2010531311A5 publication Critical patent/JP2010531311A5/ja
Application granted granted Critical
Publication of JP5250029B2 publication Critical patent/JP5250029B2/ja
Expired - Fee Related legal-status Critical Current
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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Catalysts (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
JP2010513708A 2007-06-26 2008-06-11 ２ｈ−インダゾールの遷移金属触媒合成 Expired - Fee Related JP5250029B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP07290799.1 2007-06-26
EP07290799 2007-06-26
PCT/EP2008/004637 WO2009000411A1 (en) 2007-06-26 2008-06-11 A transition metal catalyzed synthesis of 2h-indazoles

Publications (3)

Publication Number Publication Date
JP2010531311A JP2010531311A (ja) 2010-09-24
JP2010531311A5 JP2010531311A5 (enExample) 2011-07-07
JP5250029B2 true JP5250029B2 (ja) 2013-07-31

Family

ID=38577414

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010513708A Expired - Fee Related JP5250029B2 (ja) 2007-06-26 2008-06-11 ２ｈ−インダゾールの遷移金属触媒合成

Country Status (12)

Country Link
US (1) US8283476B2 (enExample)
EP (1) EP2170833B1 (enExample)
JP (1) JP5250029B2 (enExample)
KR (1) KR20100024963A (enExample)
CN (1) CN101687809A (enExample)
AT (1) ATE511501T1 (enExample)
AU (1) AU2008267442A1 (enExample)
BR (1) BRPI0813870A2 (enExample)
CA (1) CA2693024A1 (enExample)
IL (1) IL202825A0 (enExample)
MX (1) MX2009014203A (enExample)
WO (1) WO2009000411A1 (enExample)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9487506B2 (en) 2011-04-13 2016-11-08 Merck Sharp & Dohme Corp. Mineralocorticoid receptor antagonists
BR112015009738A8 (pt) * 2012-10-31 2019-09-17 Raqualia Pharma Inc composto , uso do referido composto no tratamento de uma condição ou distúrbio em que bloqueadores de canal ttx-s, composição farmacêutica contendo o referido composto e processo para preparar a referida composição
CN103232462B (zh) * 2013-05-13 2016-03-02 湖北科技学院 香豆素-吡咯类化合物的合成方法
MX2017011579A (es) * 2015-03-12 2018-03-15 Du Pont Pesticidas de tipo azol bicíclicos sustituidos con un heterociclo.
WO2017138783A1 (ko) * 2016-02-12 2017-08-17 주식회사 엘지화학 신규한 리간드 화합물 및 전이금속 화합물
KR101931234B1 (ko) 2016-02-12 2018-12-21 주식회사 엘지화학 신규한 리간드 화합물 및 전이금속 화합물
KR102095007B1 (ko) * 2016-02-12 2020-03-30 주식회사 엘지화학 신규한 리간드 화합물 및 전이금속 화합물의 제조방법
KR102038977B1 (ko) * 2016-12-30 2019-11-01 사빅 에스케이 넥슬렌 컴퍼니 피티이 엘티디 신규한 시클로펜타[ｂ]티오펜일 전이금속 화합물, 이를 포함하는 전이금속 촉매 조성물, 및 이를 이용한 에틸렌 단독중합체 또는 에틸렌과 α-올레핀의 공중합체의 제조방법
US11786528B2 (en) 2018-06-04 2023-10-17 Exscientia Ltd. Pyrazolopyrimidine compounds as adenosine receptor antagonists
CN110317204B (zh) * 2019-08-02 2022-02-08 安徽农业大学 吡唑并嘧啶酮类衍生物及其制备方法和应用
CN113698349B (zh) * 2021-09-02 2023-08-01 河南师范大学 一种2-(2-苯基-2h-吲唑-3-基)乙酸酯类化合物的水相光催化制备方法
CN114920699B (zh) * 2022-05-31 2024-03-19 甘肃皓天科技股份有限公司 一种制备6-氯-2-甲基-2h-吲唑-5-胺的方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2322194C (en) * 1998-02-26 2011-04-26 Massachusetts Institute Of Technology Metal-catalyzed arylations and vinylations of hydrazines, hydrazones, hydroxylamines and oximes

Also Published As

Publication number Publication date
JP2010531311A (ja) 2010-09-24
CA2693024A1 (en) 2008-12-31
BRPI0813870A2 (pt) 2015-01-06
US20100234601A1 (en) 2010-09-16
EP2170833A1 (en) 2010-04-07
EP2170833B1 (en) 2011-06-01
US8283476B2 (en) 2012-10-09
CN101687809A (zh) 2010-03-31
MX2009014203A (es) 2010-01-28
ATE511501T1 (de) 2011-06-15
WO2009000411A1 (en) 2008-12-31
IL202825A0 (en) 2010-06-30
KR20100024963A (ko) 2010-03-08
AU2008267442A1 (en) 2008-12-31

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