JP4847275B2 - ピラゾロ［１，５−ａ］ピリミジン化合物 - Google Patents

ピラゾロ［１，５−ａ］ピリミジン化合物 Download PDF

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Publication number
JP4847275B2
JP4847275B2 JP2006285609A JP2006285609A JP4847275B2 JP 4847275 B2 JP4847275 B2 JP 4847275B2 JP 2006285609 A JP2006285609 A JP 2006285609A JP 2006285609 A JP2006285609 A JP 2006285609A JP 4847275 B2 JP4847275 B2 JP 4847275B2
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Japan
Prior art keywords
group
chlorophenyl
pyrimidine
alkyl
pyrazolo
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JP2006285609A
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English (en)
Japanese (ja)
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JP2008007493A5 (https=
JP2008007493A (ja
Inventor
恭典 盛谷
公博 白井
真利子 大井
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Tanabe Pharma Corp
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Mitsubishi Tanabe Pharma Corp
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  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2006285609A 2005-10-21 2006-10-20 ピラゾロ［１，５−ａ］ピリミジン化合物 Expired - Fee Related JP4847275B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2006285609A JP4847275B2 (ja) 2005-10-21 2006-10-20 ピラゾロ［１，５−ａ］ピリミジン化合物

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
JP2005306816 2005-10-21
JP2005306816 2005-10-21
JP2006151470 2006-05-31
JP2006151470 2006-05-31
JP2006285609A JP4847275B2 (ja) 2005-10-21 2006-10-20 ピラゾロ［１，５−ａ］ピリミジン化合物

Publications (3)

Publication Number Publication Date
JP2008007493A JP2008007493A (ja) 2008-01-17
JP2008007493A5 JP2008007493A5 (https=) 2008-11-13
JP4847275B2 true JP4847275B2 (ja) 2011-12-28

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ID=39066005

Family Applications (1)

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JP2006285609A Expired - Fee Related JP4847275B2 (ja) 2005-10-21 2006-10-20 ピラゾロ［１，５−ａ］ピリミジン化合物

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JP (1) JP4847275B2 (https=)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW201345908A (zh) * 2006-07-05 2013-11-16 Mitsubishi Tanabe Pharma Corp 吡唑并〔１，５-ａ〕嘧啶化合物
RU2369600C1 (ru) * 2008-01-24 2009-10-10 Андрей Александрович Иващенко ЗАМЕЩЕННЫЕ 4-СУЛЬФОНИЛ-ПИРАЗОЛЫ И 3-СУЛЬФОНИЛ-ПИРАЗОЛО[1,5-a]ПИРИМИДИНЫ - АНТАГОНИСТЫ СЕРОТОНИНОВЫХ5-HT6 РЕЦЕПТОРОВ, АКТИВНЫЙ КОМПОНЕНТ, ФАРМАЦЕВТИЧЕСКАЯ КОМПОЗИЦИЯ, ЛЕКАРСТВЕННОЕ СРЕДСТВО И СПОСОБЫ ИХ ПОЛУЧЕНИЯ
CN102223798A (zh) * 2008-09-24 2011-10-19 巴斯夫欧洲公司 用于防治无脊椎动物害虫的吡唑化合物
EA024353B1 (ru) * 2010-07-29 2016-09-30 Астеллас Фарма Инк. Конденсированные циклические соединения пиридина
EP2834243B1 (en) * 2012-03-09 2018-04-25 Lexicon Pharmaceuticals, Inc. PYRAZOLO[1,5-a]PYRIMIDINE-BASED COMPOUNDS, COMPOSITIONS COMPRISING THEM, AND METHODS OF THEIR USE
TW201542550A (zh) * 2013-09-06 2015-11-16 Lexicon Pharmaceuticals Inc 吡唑并［１，５－ａ］嘧啶基化合物、包含彼之組合物以及使用彼之方法
EP3156405A1 (en) 2015-10-13 2017-04-19 Boehringer Ingelheim International GmbH Spirocyclic ether derivatives of pyrazolo[1,5-a]pyrimidine-3-carboxamide
WO2018093698A1 (en) * 2016-11-18 2018-05-24 Merck Sharp & Dohme Corp. Indole derivatives useful as inhibitors of diacylglyceride o-acyltransferase 2

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7196111B2 (en) * 2002-06-04 2007-03-27 Schering Corporation Pyrazolo[1,5a]pyrimidine compounds as antiviral agents
US7329658B2 (en) * 2003-02-06 2008-02-12 Pfizer Inc Cannabinoid receptor ligands and uses thereof
US7176210B2 (en) * 2003-02-10 2007-02-13 Pfizer Inc. Cannabinoid receptor ligands and uses thereof
DE102004008807A1 (de) * 2004-02-20 2005-09-08 Bayer Cropscience Ag Pyrazolopyrimidine
WO2005103052A1 (en) * 2004-04-21 2005-11-03 Pfizer Products Inc. Pyrazolo [1,5-a] pyrimidin-7-one compounds and uses thereof

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Publication number Publication date
JP2008007493A (ja) 2008-01-17

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