JP2025512957A5 - - Google Patents

Info

Publication number
JP2025512957A5
JP2025512957A5 JP2024559157A JP2024559157A JP2025512957A5 JP 2025512957 A5 JP2025512957 A5 JP 2025512957A5 JP 2024559157 A JP2024559157 A JP 2024559157A JP 2024559157 A JP2024559157 A JP 2024559157A JP 2025512957 A5 JP2025512957 A5 JP 2025512957A5
Authority
JP
Japan
Prior art keywords
alkyl
independently selected
appropriately substituted
membered
halo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024559157A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025512957A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2023/017384 external-priority patent/WO2023196283A1/en
Publication of JP2025512957A publication Critical patent/JP2025512957A/ja
Publication of JP2025512957A5 publication Critical patent/JP2025512957A5/ja
Pending legal-status Critical Current

Links

JP2024559157A 2022-04-05 2023-04-04 Egfr阻害剤 Pending JP2025512957A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202263327631P 2022-04-05 2022-04-05
US63/327,631 2022-04-05
PCT/US2023/017384 WO2023196283A1 (en) 2022-04-05 2023-04-04 Egfr inhibitors

Publications (2)

Publication Number Publication Date
JP2025512957A JP2025512957A (ja) 2025-04-22
JP2025512957A5 true JP2025512957A5 (enExample) 2026-04-13

Family

ID=86286433

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024559157A Pending JP2025512957A (ja) 2022-04-05 2023-04-04 Egfr阻害剤

Country Status (14)

Country Link
US (1) US20250236608A1 (enExample)
EP (1) EP4504719A1 (enExample)
JP (1) JP2025512957A (enExample)
KR (1) KR20250012554A (enExample)
CN (1) CN119325471A (enExample)
AR (1) AR129002A1 (enExample)
AU (1) AU2023250382A1 (enExample)
CA (1) CA3247645A1 (enExample)
IL (1) IL315980A (enExample)
MX (1) MX2024012267A (enExample)
PY (1) PY2325218A (enExample)
TW (1) TW202404590A (enExample)
UY (1) UY40220A (enExample)
WO (1) WO2023196283A1 (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2025080786A1 (en) * 2023-10-11 2025-04-17 Blueprint Medicines Corporation Salt and solid forms of an egfr inhibitor
WO2025080784A1 (en) * 2023-10-11 2025-04-17 Blueprint Medicines Corporation Egfr inhibitors

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2012066122A1 (en) * 2010-11-18 2012-05-24 Syngenta Participations Ag 2 - (pyridin- 2 -yl) -quinazoline derivatives and their use as microbicides
CN110498804A (zh) * 2018-05-18 2019-11-26 山东轩竹医药科技有限公司 喹唑啉衍生物类酪氨酸激酶抑制剂的新用途
TW202012391A (zh) * 2018-07-04 2020-04-01 日商第一三共股份有限公司 二芳基醚型喹唑啉衍生物
JP7752617B2 (ja) 2019-12-23 2025-10-10 ブループリント メディシンズ コーポレイション Egfrの変異型の阻害剤

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