JP2025512583A5 - - Google Patents

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Publication number
JP2025512583A5
JP2025512583A5 JP2024562812A JP2024562812A JP2025512583A5 JP 2025512583 A5 JP2025512583 A5 JP 2025512583A5 JP 2024562812 A JP2024562812 A JP 2024562812A JP 2024562812 A JP2024562812 A JP 2024562812A JP 2025512583 A5 JP2025512583 A5 JP 2025512583A5
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JP
Japan
Prior art keywords
solution
pharmaceutical composition
organic solvent
filler
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024562812A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025512583A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2023/061060 external-priority patent/WO2023209062A1/en
Publication of JP2025512583A publication Critical patent/JP2025512583A/ja
Publication of JP2025512583A5 publication Critical patent/JP2025512583A5/ja
Pending legal-status Critical Current

Links

JP2024562812A 2022-04-28 2023-04-27 3-((1R,3R)-1-(2,6-ジフルオロ-4-((1-(3-フルオロプロピル)アゼチジン-3-イル)アミノ)フェニル)-3-メチル-1,3,4,9-テトラヒドロ-2H-ピリド[3,4-b]インドール-2-イル)-2,2-ジフルオロプロパン-1-オール酒石酸塩の固体形態 Pending JP2025512583A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP22170407.5 2022-04-28
EP22170407 2022-04-28
PCT/EP2023/061060 WO2023209062A1 (en) 2022-04-28 2023-04-27 Solid form of 3-((1r,3r)-1-(2,6-difluoro-4-((1-(3- fluoropropyl)azetidin-3-yl)amino)phenyl)-3-methyl-1,3,4,9- tetrahydro-2h-pyrido[3,4-b]indol-2-yl)-2,2-difluoropropan-1-ol tartrate

Publications (2)

Publication Number Publication Date
JP2025512583A JP2025512583A (ja) 2025-04-17
JP2025512583A5 true JP2025512583A5 (https=) 2026-05-07

Family

ID=81392840

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024562812A Pending JP2025512583A (ja) 2022-04-28 2023-04-27 3-((1R,3R)-1-(2,6-ジフルオロ-4-((1-(3-フルオロプロピル)アゼチジン-3-イル)アミノ)フェニル)-3-メチル-1,3,4,9-テトラヒドロ-2H-ピリド[3,4-b]インドール-2-イル)-2,2-ジフルオロプロパン-1-オール酒石酸塩の固体形態

Country Status (11)

Country Link
US (1) US20250282775A1 (https=)
EP (1) EP4514792A1 (https=)
JP (1) JP2025512583A (https=)
KR (1) KR20250006222A (https=)
CN (1) CN119156386A (https=)
AU (1) AU2023262166A1 (https=)
CA (1) CA3255956A1 (https=)
IL (1) IL316096A (https=)
MX (1) MX2024013116A (https=)
TW (1) TW202400141A (https=)
WO (1) WO2023209062A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW202602868A (zh) * 2024-04-15 2026-01-16 瑞士商諾華公司 瑞波西利的藥物組成物

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI874834B (zh) 2014-12-18 2025-03-01 瑞士商赫孚孟拉羅股份公司 四氫-吡啶并[3,4-b]吲哚雌激素受體調節劑及其用途
CR20200621A (es) 2018-06-21 2021-02-03 Hoffmann La Roche Formas sólidas de 3-((1r,3r)-1-(2,6-difluoro-4-((1-(3 fluoropropil)azetidin-3-il)amino)fenil)-3-(metil-1,3,4,9-tetrahidro-2h-pirido[3,4-b]indol-2-il)-2,2-difluoropropan-1-ol y procesos para preparar compuestos tricíclicos fusionados que comprenden un resto fenilo o piridinilo sustituido, incluidos métodos para su uso

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