JP2025504028A - セラグノスティクス葉酸コンジュゲート - Google Patents
セラグノスティクス葉酸コンジュゲート Download PDFInfo
- Publication number
- JP2025504028A JP2025504028A JP2024544934A JP2024544934A JP2025504028A JP 2025504028 A JP2025504028 A JP 2025504028A JP 2024544934 A JP2024544934 A JP 2024544934A JP 2024544934 A JP2024544934 A JP 2024544934A JP 2025504028 A JP2025504028 A JP 2025504028A
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- JP
- Japan
- Prior art keywords
- compound
- compound according
- radiometal
- dota
- effective amount
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
- A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
- A61K51/04—Organic compounds
- A61K51/0497—Organic compounds conjugates with a carrier being an organic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
- A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
- A61K51/04—Organic compounds
- A61K51/0402—Organic compounds carboxylic acid carriers, fatty acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
- A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
- A61K51/04—Organic compounds
- A61K51/041—Heterocyclic compounds
- A61K51/044—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
- A61K51/0459—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
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- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Optics & Photonics (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Physics & Mathematics (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP22154653 | 2022-02-01 | ||
| EP22154653.4 | 2022-02-01 | ||
| PCT/EP2023/052116 WO2023148115A1 (en) | 2022-02-01 | 2023-01-30 | Theragnostic folate conjugates |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2025504028A true JP2025504028A (ja) | 2025-02-06 |
| JP2025504028A5 JP2025504028A5 (enExample) | 2026-02-12 |
Family
ID=80119142
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024544934A Pending JP2025504028A (ja) | 2022-02-01 | 2023-01-30 | セラグノスティクス葉酸コンジュゲート |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US20250108138A1 (enExample) |
| EP (1) | EP4472676A1 (enExample) |
| JP (1) | JP2025504028A (enExample) |
| KR (1) | KR20240142514A (enExample) |
| CN (1) | CN118660723A (enExample) |
| AU (1) | AU2023214599A1 (enExample) |
| CA (1) | CA3243526A1 (enExample) |
| IL (1) | IL314507A (enExample) |
| WO (1) | WO2023148115A1 (enExample) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2025220711A1 (ja) * | 2024-04-17 | 2025-10-23 | 日本メジフィジックス株式会社 | 化合物、放射性標識化合物及びその製造方法、並びに放射性医薬組成物 |
| WO2026014283A1 (ja) * | 2024-07-09 | 2026-01-15 | 日本メジフィジックス株式会社 | 化合物、放射性標識化合物およびその製造方法、並びに放射性医薬組成物 |
-
2023
- 2023-01-30 CA CA3243526A patent/CA3243526A1/en active Pending
- 2023-01-30 JP JP2024544934A patent/JP2025504028A/ja active Pending
- 2023-01-30 WO PCT/EP2023/052116 patent/WO2023148115A1/en not_active Ceased
- 2023-01-30 KR KR1020247028953A patent/KR20240142514A/ko active Pending
- 2023-01-30 AU AU2023214599A patent/AU2023214599A1/en active Pending
- 2023-01-30 IL IL314507A patent/IL314507A/en unknown
- 2023-01-30 CN CN202380019559.6A patent/CN118660723A/zh active Pending
- 2023-01-30 US US18/834,637 patent/US20250108138A1/en active Pending
- 2023-01-30 EP EP23702011.0A patent/EP4472676A1/en active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| AU2023214599A1 (en) | 2024-09-19 |
| IL314507A (en) | 2024-09-01 |
| CN118660723A (zh) | 2024-09-17 |
| US20250108138A1 (en) | 2025-04-03 |
| EP4472676A1 (en) | 2024-12-11 |
| KR20240142514A (ko) | 2024-09-30 |
| CA3243526A1 (en) | 2023-08-10 |
| WO2023148115A1 (en) | 2023-08-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| A521 | Request for written amendment filed |
Free format text: JAPANESE INTERMEDIATE CODE: A523 Effective date: 20260113 |
|
| A621 | Written request for application examination |
Free format text: JAPANESE INTERMEDIATE CODE: A621 Effective date: 20260113 |
|
| A521 | Request for written amendment filed |
Free format text: JAPANESE INTERMEDIATE CODE: A523 Effective date: 20260203 |