JP2024542199A5 - - Google Patents

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Publication number
JP2024542199A5
JP2024542199A5 JP2024529504A JP2024529504A JP2024542199A5 JP 2024542199 A5 JP2024542199 A5 JP 2024542199A5 JP 2024529504 A JP2024529504 A JP 2024529504A JP 2024529504 A JP2024529504 A JP 2024529504A JP 2024542199 A5 JP2024542199 A5 JP 2024542199A5
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JP
Japan
Application number
JP2024529504A
Other languages
Japanese (ja)
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JPWO2023088441A5 (https=
JP2024542199A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/CN2022/132954 external-priority patent/WO2023088441A1/zh
Publication of JP2024542199A publication Critical patent/JP2024542199A/ja
Publication of JPWO2023088441A5 publication Critical patent/JPWO2023088441A5/ja
Publication of JP2024542199A5 publication Critical patent/JP2024542199A5/ja
Pending legal-status Critical Current

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JP2024529504A 2021-11-19 2022-11-18 Kif18a阻害剤 Pending JP2024542199A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
CN202111399876.4 2021-11-19
CN202111399876 2021-11-19
CN202210225663.8 2022-03-09
CN202210225663 2022-03-09
CN202210667619.2 2022-06-13
CN202210667619 2022-06-13
PCT/CN2022/132954 WO2023088441A1 (zh) 2021-11-19 2022-11-18 Kif18a抑制剂

Publications (3)

Publication Number Publication Date
JP2024542199A JP2024542199A (ja) 2024-11-13
JPWO2023088441A5 JPWO2023088441A5 (https=) 2025-11-25
JP2024542199A5 true JP2024542199A5 (https=) 2025-11-25

Family

ID=86396297

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024529504A Pending JP2024542199A (ja) 2021-11-19 2022-11-18 Kif18a阻害剤

Country Status (8)

Country Link
EP (1) EP4434979A4 (https=)
JP (1) JP2024542199A (https=)
KR (1) KR20240108489A (https=)
CN (1) CN118215657A (https=)
AU (1) AU2022389558A1 (https=)
CA (1) CA3237625A1 (https=)
MX (1) MX2024005996A (https=)
WO (1) WO2023088441A1 (https=)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI844602B (zh) 2018-12-20 2024-06-11 美商安進公司 Kif18a抑制劑
CN119241504A (zh) 2021-08-26 2025-01-03 沃拉斯查疗法公司 Kif18a的螺吲哚啉抑制剂
WO2024022508A1 (zh) * 2022-07-29 2024-02-01 武汉人福创新药物研发中心有限公司 Kif18a抑制剂及用途
TW202416973A (zh) 2022-08-18 2024-05-01 美商雅客森醫療公司 Kif18a抑制劑及其用途
CN117917405A (zh) * 2022-10-21 2024-04-23 杭州邦顺制药有限公司 Kif18a蛋白抑制剂
CN120202002A (zh) * 2022-11-30 2025-06-24 微境生物医药科技(上海)有限公司 一种用于癌症治疗的药物组合物
EP4628486A1 (en) * 2022-12-02 2025-10-08 Shenzhen Zhongge Biological Technology Co., Ltd. Amide or urea compound
WO2024146593A1 (zh) * 2023-01-05 2024-07-11 浙江海正药业股份有限公司 芳香酰胺类衍生物及其制备方法和医药上的用途
WO2024244972A1 (zh) * 2023-05-30 2024-12-05 浙江海正药业股份有限公司 芳香酰胺类衍生物及其制备方法和用途
CN121532380A (zh) * 2023-07-21 2026-02-13 浙江海正药业股份有限公司 芳香酰胺类衍生物及其制备方法和用途
WO2025026392A1 (zh) * 2023-08-02 2025-02-06 上海湃隆生物科技有限公司 驱动蛋白kif18a抑制剂及其应用
WO2025036479A1 (zh) * 2023-08-16 2025-02-20 上海湃隆生物科技有限公司 驱动蛋白kif18a抑制剂及其应用
WO2025190888A1 (en) * 2024-03-12 2025-09-18 F. Hoffmann-La Roche Ag Macrocyclic kif18a inhibitors and their use thereof
TW202547479A (zh) * 2024-03-27 2025-12-16 大陸商上海齊魯製藥研究中心有限公司 驅動蛋白kif18a抑制劑及其使用方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AUPO395396A0 (en) * 1996-12-02 1997-01-02 Fujisawa Pharmaceutical Co., Ltd. Benzamide derivatives
WO2020132651A1 (en) * 2018-12-20 2020-06-25 Amgen Inc. Kif18a inhibitors
EP3898616B1 (en) * 2018-12-20 2024-10-02 Amgen Inc. Heteroaryl amides useful as kif18a inhibitors
TWI844602B (zh) 2018-12-20 2024-06-11 美商安進公司 Kif18a抑制劑
JP7676308B2 (ja) * 2018-12-20 2025-05-14 アムジエン・インコーポレーテツド Kif18a阻害剤として有用なヘテロアリールアミド
US12540129B2 (en) * 2019-08-02 2026-02-03 Amgen Inc. KIF18A inhibitors
AU2020326627B2 (en) * 2019-08-02 2026-01-29 Amgen Inc. KIF18A inhibitors
WO2021026099A1 (en) * 2019-08-02 2021-02-11 Amgen Inc. Kif18a inhibitors
JP2023521802A (ja) * 2020-04-14 2023-05-25 アムジエン・インコーポレーテツド 新生物疾患の処置のためのkif18a阻害剤
JP2024534572A (ja) * 2021-09-24 2024-09-20 ゼノン・ファーマシューティカルズ・インコーポレイテッド ナトリウムチャンネル活性化剤としてのピリジニルアセトアミド誘導体

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