JP2024534510A5 - - Google Patents

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Publication number
JP2024534510A5
JP2024534510A5 JP2024517459A JP2024517459A JP2024534510A5 JP 2024534510 A5 JP2024534510 A5 JP 2024534510A5 JP 2024517459 A JP2024517459 A JP 2024517459A JP 2024517459 A JP2024517459 A JP 2024517459A JP 2024534510 A5 JP2024534510 A5 JP 2024534510A5
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JP
Japan
Application number
JP2024517459A
Other languages
Japanese (ja)
Other versions
JP2024534510A (ja
JPWO2023046698A5 (https=
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2022/076130 external-priority patent/WO2023046698A1/en
Publication of JP2024534510A publication Critical patent/JP2024534510A/ja
Publication of JP2024534510A5 publication Critical patent/JP2024534510A5/ja
Publication of JPWO2023046698A5 publication Critical patent/JPWO2023046698A5/ja
Withdrawn legal-status Critical Current

Links

JP2024517459A 2021-09-21 2022-09-20 Alk5阻害剤としてのピリダジニルアミノ誘導体 Withdrawn JP2024534510A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
EP21198025.5 2021-09-21
EP21198025 2021-09-21
EP21216519 2021-12-21
EP21216519.5 2021-12-21
PK598/2022 2022-09-13
PK5982022 2022-09-13
PCT/EP2022/076130 WO2023046698A1 (en) 2021-09-21 2022-09-20 Pyridazinyl amino derivatives as alk5 inhibitors

Publications (3)

Publication Number Publication Date
JP2024534510A JP2024534510A (ja) 2024-09-20
JP2024534510A5 true JP2024534510A5 (https=) 2025-09-30
JPWO2023046698A5 JPWO2023046698A5 (https=) 2025-09-30

Family

ID=83978901

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024517459A Withdrawn JP2024534510A (ja) 2021-09-21 2022-09-20 Alk5阻害剤としてのピリダジニルアミノ誘導体

Country Status (11)

Country Link
US (1) US20250011299A1 (https=)
EP (1) EP4405343A1 (https=)
JP (1) JP2024534510A (https=)
KR (1) KR20240069773A (https=)
CN (1) CN118201915A (https=)
AR (1) AR127108A1 (https=)
AU (1) AU2022351219A1 (https=)
CA (1) CA3232178A1 (https=)
MX (1) MX2024003399A (https=)
TW (1) TW202328102A (https=)
WO (1) WO2023046698A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2024180206A1 (en) * 2023-03-02 2024-09-06 Chiesi Farmaceutici S.P.A. Pyridazinyl amino derivatives as alk5 inhibitors
WO2024180207A1 (en) 2023-03-02 2024-09-06 Chiesi Farmaceutici S.P.A. Pyridazinyl amino derivatives as alk5 inhibitors
WO2025132458A1 (en) 2023-12-18 2025-06-26 Chiesi Farmaceutici S.P.A. Pyridazinyl amino derivatives as alk5 inhibitors
WO2025132460A1 (en) 2023-12-18 2025-06-26 Chiesi Farmaceutici S.P.A. Pyridazinyl amino derivatives as alk5 inhibitors

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR029803A1 (es) 2000-02-21 2003-07-16 Smithkline Beecham Plc Imidazoles sustituidos con piridilo y composiciones farmaceuticas que las comprenden
GB0007405D0 (en) 2000-03-27 2000-05-17 Smithkline Beecham Corp Compounds
EP1317450B1 (en) 2000-09-15 2006-11-22 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
CA2423050A1 (en) 2000-09-20 2002-03-28 Ortho-Mcneil Pharmaceutical, Inc. Pyrazine derivatives as modulators of tyrosine kinases
AR039241A1 (es) 2002-04-04 2005-02-16 Biogen Inc Heteroarilos trisustituidos y metodos para su produccion y uso de los mismos
AU2004278382B2 (en) 2003-09-30 2008-09-18 Amgen Inc. Vanilloid receptor ligands and their use in treatments
WO2005080377A1 (ja) * 2004-02-20 2005-09-01 Kirin Beer Kabushiki Kaisha TGFβ阻害活性を有する化合物およびそれを含んでなる医薬組成物
BRPI0714409A2 (pt) 2006-07-14 2013-03-12 Novartis Ag derivados de pirimidina como inibidores de alk-5
ES2375425T3 (es) 2007-07-26 2012-02-29 Novartis Ag Compuestos org�?nicos.
BRPI0817434A2 (pt) 2007-10-17 2015-06-16 Novartis Ag Composto orgânicos
AR070127A1 (es) 2008-01-11 2010-03-17 Novartis Ag Pirrolo - pirimidinas y pirrolo -piridinas
MX2010007604A (es) 2008-01-11 2010-08-02 Novartis Ag Pirimidinas como inhibidores de cinasa.
US8343966B2 (en) 2008-01-11 2013-01-01 Novartis Ag Organic compounds
EA201001687A1 (ru) 2008-04-29 2011-06-30 Новартис Аг Производные имидазопиридина в качестве ингибиторов активиноподобной рецепторной киназы ( alk-4 или alk-5 )
US9073918B2 (en) * 2010-05-20 2015-07-07 Takeda Pharmaceutical Company Limited Pyrazolo[4,3-b]pyridine-7-amine inhibitors of ALK5
US20200247812A1 (en) * 2018-07-10 2020-08-06 Integral Biosciences Private Limited Heterocyclic compounds and methods of use

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