JP2024533700A5 - - Google Patents

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Publication number
JP2024533700A5
JP2024533700A5 JP2024518606A JP2024518606A JP2024533700A5 JP 2024533700 A5 JP2024533700 A5 JP 2024533700A5 JP 2024518606 A JP2024518606 A JP 2024518606A JP 2024518606 A JP2024518606 A JP 2024518606A JP 2024533700 A5 JP2024533700 A5 JP 2024533700A5
Authority
JP
Japan
Prior art keywords
pharmaceutical composition
composition according
alopecia
compound
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024518606A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024533700A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/044346 external-priority patent/WO2023049241A1/en
Publication of JP2024533700A publication Critical patent/JP2024533700A/ja
Publication of JP2024533700A5 publication Critical patent/JP2024533700A5/ja
Pending legal-status Critical Current

Links

JP2024518606A 2021-09-23 2022-09-22 チロシンキナーゼ2(tyk2)阻害剤による脱毛症の治療方法 Pending JP2024533700A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202163247672P 2021-09-23 2021-09-23
US63/247,672 2021-09-23
PCT/US2022/044346 WO2023049241A1 (en) 2021-09-23 2022-09-22 Methods of treating hair-loss disorders with tyk2 inhibitors

Publications (2)

Publication Number Publication Date
JP2024533700A JP2024533700A (ja) 2024-09-12
JP2024533700A5 true JP2024533700A5 (https=) 2025-10-02

Family

ID=83899658

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024518606A Pending JP2024533700A (ja) 2021-09-23 2022-09-22 チロシンキナーゼ2(tyk2)阻害剤による脱毛症の治療方法

Country Status (10)

Country Link
US (1) US20240390372A1 (https=)
EP (1) EP4404930A1 (https=)
JP (1) JP2024533700A (https=)
KR (1) KR20240065283A (https=)
CN (2) CN118251222A (https=)
AU (1) AU2022350509A1 (https=)
CA (1) CA3232812A1 (https=)
IL (1) IL311624A (https=)
MX (1) MX2024003510A (https=)
WO (1) WO2023049241A1 (https=)

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LT3495358T (lt) 2012-11-08 2022-05-25 Bristol-Myers Squibb Company Amidais pakeisti heterocikliniai junginiai, naudingi kaip il-12, il-23 ir (arba) ifn alfa atsako moduliatoriai
TWI582077B (zh) * 2013-11-07 2017-05-11 必治妥美雅史谷比公司 作爲IL-12、IL-23及/或IFNα反應調節劑之經烷基-醯胺取代之吡啶化合物
TW202515876A (zh) * 2017-03-08 2025-04-16 日商武田藥品工業股份有限公司 Tyk2抑制劑及其用途
JP7113023B2 (ja) * 2017-03-30 2022-08-04 ブリストル-マイヤーズ スクイブ カンパニー 6-(シクロプロパンアミド)-4-((2-メトキシ-3-(1-メチル-1h-1,2,4-トリアゾール-3-イル)フェニル)アミノ)-n-(メチル-d3)ピリダジン-3-カルボキシアミドの製造方法
KR102848769B1 (ko) 2018-05-31 2025-08-20 브리스톨-마이어스 스큅 컴퍼니 6-(시클로프로판카르복스아미도)-4-((2-메톡시-3-(1-메틸-1h-1,2,4-트리아졸-3-일)페닐)아미노)-n-(메틸-d3) 피리다진-3-카르복스아미드의 결정질 형태
US20230093099A1 (en) * 2019-04-02 2023-03-23 Cullgen (Shanghai), Inc. Compounds and methods of treating cancers
US11357775B2 (en) * 2019-04-30 2022-06-14 Celgene Corporation Combination therapies comprising apremilast and Tyk2 inhibitors
SG11202112043PA (en) * 2019-04-30 2021-11-29 Celgene Corp Combination therapies comprising apremilast and tyk2 inhibitors
US12570637B2 (en) 2019-06-12 2026-03-10 Bristol-Myers Squibb Company Crystalline salt forms 6-(cyclopropanecarboxamido)-4-((2-methoxy-3-(1-methyl-1H-1,2,4-triazol-3-yl)phenyl)amino)-n-(methyld3) pyridazine-3-carboxamide
JP7812785B2 (ja) 2019-09-18 2026-02-10 ブリストル-マイヤーズ スクイブ カンパニー Tyk2阻害薬の剤形
AU2021205465A1 (en) * 2020-01-06 2022-07-14 Arena Pharmaceuticals, Inc. Methods of treating conditions related to the S1P1 receptor
CN111704617B (zh) * 2020-06-15 2022-08-23 嘉兴特科罗生物科技有限公司 一种小分子化合物
CN112142675B (zh) * 2020-10-09 2021-11-30 嘉兴特科罗生物科技有限公司 一种作为jak激酶抑制剂的小分子化合物及其用途

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