JP2023543299A5 - - Google Patents

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Publication number
JP2023543299A5
JP2023543299A5 JP2023519522A JP2023519522A JP2023543299A5 JP 2023543299 A5 JP2023543299 A5 JP 2023543299A5 JP 2023519522 A JP2023519522 A JP 2023519522A JP 2023519522 A JP2023519522 A JP 2023519522A JP 2023543299 A5 JP2023543299 A5 JP 2023543299A5
Authority
JP
Japan
Application number
JP2023519522A
Other languages
Japanese (ja)
Other versions
JP2023543299A (ja
JPWO2022069520A5 (https=
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2021/076752 external-priority patent/WO2022069520A1/en
Publication of JP2023543299A publication Critical patent/JP2023543299A/ja
Publication of JPWO2022069520A5 publication Critical patent/JPWO2022069520A5/ja
Publication of JP2023543299A5 publication Critical patent/JP2023543299A5/ja
Pending legal-status Critical Current

Links

JP2023519522A 2020-09-30 2021-09-29 化合物及び癌の治療におけるそれらの使用 Pending JP2023543299A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063085384P 2020-09-30 2020-09-30
US63/085,384 2020-09-30
PCT/EP2021/076752 WO2022069520A1 (en) 2020-09-30 2021-09-29 Compounds and their use in treating cancer

Publications (3)

Publication Number Publication Date
JP2023543299A JP2023543299A (ja) 2023-10-13
JPWO2022069520A5 JPWO2022069520A5 (https=) 2024-10-07
JP2023543299A5 true JP2023543299A5 (https=) 2024-10-07

Family

ID=78085628

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023519522A Pending JP2023543299A (ja) 2020-09-30 2021-09-29 化合物及び癌の治療におけるそれらの使用

Country Status (17)

Country Link
US (1) US20230374007A1 (https=)
EP (1) EP4221756A1 (https=)
JP (1) JP2023543299A (https=)
KR (1) KR20230079408A (https=)
CN (1) CN116249554A (https=)
AU (2) AU2021353968B2 (https=)
BR (1) BR112023005708A2 (https=)
CA (1) CA3195695A1 (https=)
CL (1) CL2023000881A1 (https=)
CO (1) CO2023005188A2 (https=)
CR (1) CR20230185A (https=)
DO (1) DOP2023000062A (https=)
EC (1) ECSP23030959A (https=)
IL (1) IL301626A (https=)
MX (1) MX2023003564A (https=)
PE (1) PE20230782A1 (https=)
WO (1) WO2022069520A1 (https=)

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Publication number Priority date Publication date Assignee Title
CN115141179B (zh) * 2021-03-31 2024-09-13 江苏恒瑞医药股份有限公司 一种新型苯并杂环基类衍生物、其制备方法及其在医药上的应用
CN119301111A (zh) 2022-03-24 2025-01-10 葛兰素史密斯克莱知识产权发展有限公司 作为protac中的降解决定子的2,4-二氧代四氢嘧啶基衍生物
USD1018676S1 (en) * 2022-04-15 2024-03-19 Puttshack LTD Miniature golf hole
USD1018746S1 (en) * 2022-04-15 2024-03-19 Puttshack LTD Miniature golf hole
USD1020957S1 (en) * 2022-04-15 2024-04-02 Puttshack LTD Miniature golf hole
USD1018747S1 (en) * 2022-04-15 2024-03-19 Puttshack LTD Miniature golf hole
CN119855812A (zh) * 2022-09-14 2025-04-18 海南先声再明医药股份有限公司 多并环类化合物及其用途
US20240374588A1 (en) 2023-04-07 2024-11-14 Astrazeneca Ab Irak4 protacs
TW202515566A (zh) 2023-06-14 2025-04-16 瑞典商阿斯特捷利康公司 Smarca2降解劑及其用途
MX2025015084A (es) * 2023-06-14 2026-02-03 Astrazeneca Ab Degradadores de smarca2 y usos de estos
WO2025036489A1 (zh) * 2023-08-17 2025-02-20 海思科医药集团股份有限公司 一种氰基芳香环衍生物及其在医药上的应用
IL326555A (en) 2023-09-22 2026-04-01 Glaxosmithkline Ip Dev Ltd Androgen receptor protax
CN117430605A (zh) * 2023-10-26 2024-01-23 广西天铭药业有限公司 一种kras g12c抑制剂amg-510中间体的合成方法
US20250177539A1 (en) * 2023-12-01 2025-06-05 Astrazeneca Ab Er degraders and uses thereof
WO2025125575A1 (en) 2023-12-14 2025-06-19 Astrazeneca Ab Irak4 protacs

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0422263D0 (en) 2004-10-07 2004-11-10 Glaxo Group Ltd Novel compounds
PH12012502079A1 (en) 2010-04-16 2013-02-11 Ac Immune Sa Novel compounds for the treatment of diseases associated with amyloid or amyloid-like proteins
JP6509838B2 (ja) 2013-06-26 2019-05-08 アッヴィ・インコーポレイテッド Btk阻害薬としての一級カルボキサミド類
ES2826443T3 (es) 2014-09-25 2021-05-18 Araxes Pharma Llc Inhibidores de proteínas mutantes KRAS G12C
JP6815318B2 (ja) * 2014-12-23 2021-01-20 ダナ−ファーバー キャンサー インスティテュート,インコーポレイテッド 二官能性分子によって標的化タンパク質分解を誘導する方法
BR112019015484A2 (pt) * 2017-01-31 2020-04-28 Arvinas Operations Inc ligantes de cereblon e compostos bifuncionais compreendendo os mesmos
WO2019057757A1 (en) * 2017-09-20 2019-03-28 Astrazeneca Ab 1,3-DIHYDROIMIDAZO [4,5-C] CINNOLIN-2-ONE COMPOUNDS AND THEIR USE IN THE TREATMENT OF CANCER
WO2019140387A1 (en) * 2018-01-12 2019-07-18 Kymera Therapeutics, Inc. Crbn ligands and uses thereof
CN120698983A (zh) * 2018-12-20 2025-09-26 C4医药公司 靶向蛋白降解

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