JP2023542548A5 - - Google Patents

Info

Publication number
JP2023542548A5
JP2023542548A5 JP2023518938A JP2023518938A JP2023542548A5 JP 2023542548 A5 JP2023542548 A5 JP 2023542548A5 JP 2023518938 A JP2023518938 A JP 2023518938A JP 2023518938 A JP2023518938 A JP 2023518938A JP 2023542548 A5 JP2023542548 A5 JP 2023542548A5
Authority
JP
Japan
Prior art keywords
nhr
alkyl
nhc
nhr2
cho
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2023518938A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023542548A (ja
JP7839786B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2021/058707 external-priority patent/WO2022064430A1/en
Publication of JP2023542548A publication Critical patent/JP2023542548A/ja
Publication of JP2023542548A5 publication Critical patent/JP2023542548A5/ja
Application granted granted Critical
Publication of JP7839786B2 publication Critical patent/JP7839786B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2023518938A 2020-09-24 2021-09-24 新規アミノピリジン及びその癌治療への使用 Active JP7839786B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
NZ768245 2020-09-24
NZ76824520 2020-09-24
PCT/IB2021/058707 WO2022064430A1 (en) 2020-09-24 2021-09-24 Novel aminopyridines and their use in treating cancer

Publications (3)

Publication Number Publication Date
JP2023542548A JP2023542548A (ja) 2023-10-10
JP2023542548A5 true JP2023542548A5 (https=) 2025-08-14
JP7839786B2 JP7839786B2 (ja) 2026-04-02

Family

ID=80844550

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023518938A Active JP7839786B2 (ja) 2020-09-24 2021-09-24 新規アミノピリジン及びその癌治療への使用

Country Status (7)

Country Link
US (1) US20230365559A1 (https=)
EP (1) EP4217357A4 (https=)
JP (1) JP7839786B2 (https=)
CN (1) CN116669725A (https=)
AU (1) AU2021346954A1 (https=)
CA (1) CA3192868A1 (https=)
WO (1) WO2022064430A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CR20230057A (es) 2020-07-02 2023-08-15 Incyte Corp Compuestos tríciclicos de urea como inhibidores de jak2 v617f
AU2023235313A1 (en) 2022-03-17 2024-10-03 Incyte Corporation Tricyclic urea compounds as jak2 v617f inhibitors
JP2026509874A (ja) * 2023-03-13 2026-03-25 インサイト・コーポレイション キナーゼ阻害剤としての二環式尿素

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2011021678A1 (ja) * 2009-08-21 2011-02-24 武田薬品工業株式会社 縮合複素環化合物
CA2902858A1 (en) * 2013-02-28 2014-09-04 Signal Pharmaceuticals, Llc Treatment of cancer with tor kinase inhibitors
ME03336B (me) * 2013-03-12 2019-10-20 Vertex Pharma Inhibitori dnk-pk
JP6883653B2 (ja) 2016-12-20 2021-06-09 アストラゼネカ・アクチエボラーグAstrazeneca Aktiebolag アミノ−トリアゾロピリジン化合物および癌の治療におけるその使用
JP7202315B2 (ja) * 2017-05-26 2023-01-11 キャンサー・リサーチ・テクノロジー・リミテッド ベンズイミダゾロン由来のbcl6阻害剤
TWI820146B (zh) * 2018-06-15 2023-11-01 瑞典商阿斯特捷利康公司 嘌呤酮化合物及其在治療癌症中之用途
GB201819126D0 (en) * 2018-11-23 2019-01-09 Cancer Research Tech Ltd Inhibitor compounds
WO2020140054A1 (en) * 2018-12-28 2020-07-02 Spv Therapeutics Inc. Cyclin-dependent kinase inhibitors

Similar Documents

Publication Publication Date Title
JP2023542548A5 (https=)
JP7778688B2 (ja) Trmp8モジュレーターとしての置換アザシル
JP2022533069A5 (https=)
JP2019034943A5 (https=)
JP2024530952A5 (https=)
ES2452868T3 (es) Nuevos inhibidores de desacetilasas de histonas basados simultáneamente en 1H-pirroles trisustituidos y en espaciadores aromáticos y heteroaromáticos
JP2021528427A5 (https=)
JP2019535672A5 (https=)
JP2019524702A5 (https=)
JP2010515756A5 (https=)
JP2009544602A5 (https=)
CO6310968A2 (es) Derivados de 3,5-diamino sustituido-n-tetrahidropirimidin/imidazolin/diazepam-2-ilidenpirazin-2-carboxamida, utiles como bloqueadores de la actividad del canal de sodio epitelial (enac)
JP2016515096A5 (https=)
JP2017536395A5 (https=)
CN110023292B (zh) 细胞凋亡抑制剂
JP2019531279A5 (https=)
CN108778288A (zh) 可用于治疗疾病的FimH的甘露糖衍生的拮抗剂
JP2019505502A5 (https=)
JP2018535930A5 (https=)
JP2022505257A5 (https=)
JP2024507139A5 (https=)
JP2010505865A5 (https=)
JP2017538697A5 (https=)
JP2004525183A5 (https=)
GT200600457A (es) Sal de fosfato dihidrogeno como antagonistas del receptor de prostaglandina d2