JP2021515749A5 - - Google Patents

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Publication number
JP2021515749A5
JP2021515749A5 JP2020544266A JP2020544266A JP2021515749A5 JP 2021515749 A5 JP2021515749 A5 JP 2021515749A5 JP 2020544266 A JP2020544266 A JP 2020544266A JP 2020544266 A JP2020544266 A JP 2020544266A JP 2021515749 A5 JP2021515749 A5 JP 2021515749A5
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JP
Japan
Prior art keywords
compound according
pharmaceutically acceptable
acceptable salt
treatment
alkyl
Prior art date
Application number
JP2020544266A
Other languages
English (en)
Japanese (ja)
Other versions
JP2021515749A (ja
JP7225255B2 (ja
JPWO2019166822A5 (https=
Filing date
Publication date
Priority claimed from GBGB1803340.7A external-priority patent/GB201803340D0/en
Application filed filed Critical
Publication of JP2021515749A publication Critical patent/JP2021515749A/ja
Publication of JP2021515749A5 publication Critical patent/JP2021515749A5/ja
Publication of JPWO2019166822A5 publication Critical patent/JPWO2019166822A5/ja
Application granted granted Critical
Publication of JP7225255B2 publication Critical patent/JP7225255B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2020544266A 2018-03-01 2019-03-01 Ampa受容体機能を調節する化合物 Active JP7225255B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB1803340.7A GB201803340D0 (en) 2018-03-01 2018-03-01 Compounds
GB1803340.7 2018-03-01
PCT/GB2019/050578 WO2019166822A1 (en) 2018-03-01 2019-03-01 Compounds that modulates ampa receptor function

Publications (4)

Publication Number Publication Date
JP2021515749A JP2021515749A (ja) 2021-06-24
JP2021515749A5 true JP2021515749A5 (https=) 2022-02-25
JPWO2019166822A5 JPWO2019166822A5 (https=) 2022-02-25
JP7225255B2 JP7225255B2 (ja) 2023-02-20

Family

ID=61903711

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020544266A Active JP7225255B2 (ja) 2018-03-01 2019-03-01 Ampa受容体機能を調節する化合物

Country Status (16)

Country Link
US (3) US11298345B2 (https=)
EP (1) EP3759092B1 (https=)
JP (1) JP7225255B2 (https=)
KR (2) KR20250093578A (https=)
CN (1) CN112004811B (https=)
AU (1) AU2019226718C1 (https=)
BR (1) BR112020017739A2 (https=)
CA (1) CA3091783A1 (https=)
DK (1) DK3759092T3 (https=)
ES (1) ES2970784T3 (https=)
FI (1) FI3759092T3 (https=)
GB (1) GB201803340D0 (https=)
MX (1) MX2020009097A (https=)
PL (1) PL3759092T3 (https=)
RU (1) RU2020127537A (https=)
WO (1) WO2019166822A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB201702221D0 (en) 2017-02-10 2017-03-29 Univ Of Sussex Compounds
GB201803340D0 (en) 2018-03-01 2018-04-18 Univ Of Sussex Compounds

Family Cites Families (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW575561B (en) 1999-03-25 2004-02-11 Hoffmann La Roche 1-arenesulfonyl-2-aryl-pyrrolidine and piperidine derivatives
IL152848A0 (en) 2000-06-12 2003-06-24 Eisai Co Ltd 1,2-dihydropyridine derivatives, pharmaceutical compositions containing the same and methods for the production thereof
RU2279428C2 (ru) 2000-09-18 2006-07-10 Эйсай Ко., Лтд. Производные пиридазинона и триазинона и их применение в качестве фармацевтических препаратов
AU2003302027A1 (en) 2002-11-21 2004-06-15 Vicore Pharma Ab New tricyclic angiotensin ii agonists
JP5289043B2 (ja) 2005-04-12 2013-09-11 ヴィコール・ファルマ・アーベー 新規な三環系アンジオテンシンiiアゴニスト
CA2646585A1 (en) 2006-03-20 2007-09-27 Glaxo Group Limited Compounds which potentiate ampa receptor and uses thereof in medicine
EP2049475B1 (en) 2006-04-24 2012-02-01 Eli Lilly & Company Cyclohexyl substituted pyrrolidinones as inhibitors of 11-beta-hydroxysteroid dehydrogenase 1
TW200817385A (en) 2006-07-04 2008-04-16 Organon Nv Heterocyclic derivatives
DE602007013450D1 (de) 2006-11-03 2011-05-05 Glaxo Group Ltd Verbindungen, die den ampa-rezeptor verstärken, und deren anwendung in der medizin
GB0711088D0 (en) 2007-06-08 2007-07-18 Glaxo Group Ltd Compounds
GB0711089D0 (en) 2007-06-08 2007-07-18 Glaxo Group Ltd Compounds
EP2183228B1 (en) 2007-07-26 2014-08-20 Vitae Pharmaceuticals, Inc. CYCLIC INHIBITORS OF 11ß -HYDROXYSTERIOD DEHYDROGENASE 1
KR20100063087A (ko) 2007-09-20 2010-06-10 코텍스 파마슈티칼스, 인크. 글루타메이트 시냅스 반응 향상을 위한 3-치환된 1,2,3-트리아진-4-온 및 3-치환된 1,3-피리미디논
GB0721094D0 (en) 2007-10-26 2007-12-05 Glaxo Group Ltd Compounds
TW200934497A (en) 2007-11-13 2009-08-16 Organon Nv Heterocyclic derivatives
AR071236A1 (es) 2008-05-01 2010-06-02 Vitae Pharmaceuticals Inc Inhibidores ciclicos de la 11beta-hidroxiesteroide deshidrogenasa 1
TW201012803A (en) 2008-06-06 2010-04-01 Organon Nv Heterocyclic derivatives
TW201031649A (en) 2008-12-02 2010-09-01 Organon Nv 1-(4-(pyridin-2-yl)benzyl)imidazolidine-2,4-dione derivatives
AP3066A (en) 2009-06-26 2014-12-31 Pfizer Heterocyclic sulfonamides, uses and pharmaceuticalcompositions thereof
WO2011132051A2 (en) * 2010-04-19 2011-10-27 Glenmark Pharmaceuticals S.A. Tricycle compounds as phosphodiesterase-10 inhibitors
UY33930A (es) 2011-03-04 2012-10-31 Novartis Ag Inhibidores novedosos de quinasas
GB201702221D0 (en) 2017-02-10 2017-03-29 Univ Of Sussex Compounds
GB201803340D0 (en) 2018-03-01 2018-04-18 Univ Of Sussex Compounds

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