JP2021512893A5 - - Google Patents

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Publication number
JP2021512893A5
JP2021512893A5 JP2020542546A JP2020542546A JP2021512893A5 JP 2021512893 A5 JP2021512893 A5 JP 2021512893A5 JP 2020542546 A JP2020542546 A JP 2020542546A JP 2020542546 A JP2020542546 A JP 2020542546A JP 2021512893 A5 JP2021512893 A5 JP 2021512893A5
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JP
Japan
Prior art keywords
theta
degrees
approximately
polymorph
ray powder
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JP2020542546A
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English (en)
Japanese (ja)
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JP7550646B2 (ja
JPWO2019157225A5 (https=
JP2021512893A (ja
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Priority claimed from PCT/US2019/017117 external-priority patent/WO2019157225A2/en
Publication of JP2021512893A publication Critical patent/JP2021512893A/ja
Publication of JP2021512893A5 publication Critical patent/JP2021512893A5/ja
Publication of JPWO2019157225A5 publication Critical patent/JPWO2019157225A5/ja
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JP2020542546A 2018-02-08 2019-02-07 特定の化学物質、組成物、および方法 Active JP7550646B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862628194P 2018-02-08 2018-02-08
US62/628,194 2018-02-08
PCT/US2019/017117 WO2019157225A2 (en) 2018-02-08 2019-02-07 Certain chemical entities, compositions, and methods

Publications (4)

Publication Number Publication Date
JP2021512893A JP2021512893A (ja) 2021-05-20
JP2021512893A5 true JP2021512893A5 (https=) 2022-02-16
JPWO2019157225A5 JPWO2019157225A5 (https=) 2022-02-16
JP7550646B2 JP7550646B2 (ja) 2024-09-13

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ID=67549574

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JP2020542546A Active JP7550646B2 (ja) 2018-02-08 2019-02-07 特定の化学物質、組成物、および方法

Country Status (11)

Country Link
US (1) US11465975B2 (https=)
EP (1) EP3749310B1 (https=)
JP (1) JP7550646B2 (https=)
KR (1) KR20200143361A (https=)
CN (1) CN112105365A (https=)
AU (1) AU2019218893B2 (https=)
CA (1) CA3090528A1 (https=)
IL (1) IL276476B2 (https=)
PH (1) PH12020551193A1 (https=)
SG (1) SG11202007492XA (https=)
WO (1) WO2019157225A2 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4255434A4 (en) * 2020-12-02 2024-10-23 Neupharma, Inc. CERTAIN CHEMICALS, COMPOSITIONS AND PROCESSES

Family Cites Families (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5033252A (en) 1987-12-23 1991-07-23 Entravision, Inc. Method of packaging and sterilizing a pharmaceutical product
US5052558A (en) 1987-12-23 1991-10-01 Entravision, Inc. Packaged pharmaceutical product
US5323907A (en) 1992-06-23 1994-06-28 Multi-Comp, Inc. Child resistant package assembly for dispensing pharmaceutical medications
US6334997B1 (en) 1994-03-25 2002-01-01 Isotechnika, Inc. Method of using deuterated calcium channel blockers
CN1087725C (zh) 1994-03-25 2002-07-17 同位素技术有限公司 用氘代方法增强药物效果
GB9624482D0 (en) 1995-12-18 1997-01-15 Zeneca Phaema S A Chemical compounds
BR9707495A (pt) 1996-02-13 1999-07-27 Zeneca Ltd Derivado de quinazolina processo para a preparação do mesmo composição farmacêutica e processo para a produç o de um efeito antiangiogênico e/ou de redução de permeabilidade vascular em um animal de sangue quente
US6291455B1 (en) 1996-03-05 2001-09-18 Zeneca Limited 4-anilinoquinazoline derivatives
GB9718972D0 (en) 1996-09-25 1997-11-12 Zeneca Ltd Chemical compounds
GB9714249D0 (en) 1997-07-08 1997-09-10 Angiogene Pharm Ltd Vascular damaging agents
GB9900334D0 (en) 1999-01-07 1999-02-24 Angiogene Pharm Ltd Tricylic vascular damaging agents
GB9900752D0 (en) 1999-01-15 1999-03-03 Angiogene Pharm Ltd Benzimidazole vascular damaging agents
SK288365B6 (sk) 1999-02-10 2016-07-01 Astrazeneca Ab Medziprodukty pre chinazolínové deriváty ako inhibítory angiogenézy
NZ522074A (en) 2000-05-31 2004-06-25 Astrazeneca Ab Indole derivatives with vascular damaging activity
UA73993C2 (uk) 2000-06-06 2005-10-17 Астразенека Аб Хіназолінові похідні для лікування пухлин та фармацевтична композиція
IL153484A0 (en) 2000-07-07 2003-07-06 Angiogene Pharm Ltd Colchinol derivatives as angiogenesis inhibitors
CN1255392C (zh) 2000-07-07 2006-05-10 安吉奥金尼药品有限公司 作为血管生成抑制剂的秋水仙醇衍生物
CN103702990B (zh) * 2011-07-27 2015-09-09 阿斯利康(瑞典)有限公司 2-(2,4,5-取代苯胺)嘧啶衍生物作为egfr调谐子用于治疗癌症
CA2846574C (en) * 2011-08-26 2020-07-07 Neupharma, Inc. Quinoxaline sulfonamide derivates for use as kinase inhibitors
CN105209456B (zh) * 2013-03-06 2018-05-08 阿斯利康(瑞典)有限公司 表皮生长因子受体的活化突变形式的喹唑啉抑制剂
AU2014308616B2 (en) * 2013-08-23 2018-12-06 Neupharma, Inc. Certain chemical entities, compositions, and methods
US10689359B2 (en) * 2015-12-25 2020-06-23 Xuanzhu Pharma Co., Ltd. Crystals of quinazoline derivative and preparation method therefor

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