JP2021510680A5 - - Google Patents

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Publication number
JP2021510680A5
JP2021510680A5 JP2020535980A JP2020535980A JP2021510680A5 JP 2021510680 A5 JP2021510680 A5 JP 2021510680A5 JP 2020535980 A JP2020535980 A JP 2020535980A JP 2020535980 A JP2020535980 A JP 2020535980A JP 2021510680 A5 JP2021510680 A5 JP 2021510680A5
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JP
Japan
Prior art keywords
cancer
compound
pharmaceutically acceptable
antibody
pharmaceutical composition
Prior art date
Application number
JP2020535980A
Other languages
English (en)
Japanese (ja)
Other versions
JP2021510680A (ja
JP7539151B2 (ja
JPWO2019140324A5 (https=
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Priority claimed from PCT/US2019/013377 external-priority patent/WO2019140324A1/en
Publication of JP2021510680A publication Critical patent/JP2021510680A/ja
Publication of JPWO2019140324A5 publication Critical patent/JPWO2019140324A5/ja
Publication of JP2021510680A5 publication Critical patent/JP2021510680A5/ja
Application granted granted Critical
Publication of JP7539151B2 publication Critical patent/JP7539151B2/ja
Active legal-status Critical Current
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JP2020535980A 2018-01-12 2019-01-11 Etbr活性化に関連する癌を処置するための重水素化化合物、組成物、および方法 Active JP7539151B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862616729P 2018-01-12 2018-01-12
US62/616,729 2018-01-12
PCT/US2019/013377 WO2019140324A1 (en) 2018-01-12 2019-01-11 Deuterated compounds, compositions, and methods for treating cancers associated with etbr activation

Publications (4)

Publication Number Publication Date
JP2021510680A JP2021510680A (ja) 2021-04-30
JPWO2019140324A5 JPWO2019140324A5 (https=) 2022-02-07
JP2021510680A5 true JP2021510680A5 (https=) 2022-02-07
JP7539151B2 JP7539151B2 (ja) 2024-08-23

Family

ID=67212721

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020535980A Active JP7539151B2 (ja) 2018-01-12 2019-01-11 Etbr活性化に関連する癌を処置するための重水素化化合物、組成物、および方法

Country Status (10)

Country Link
US (4) US10435434B2 (https=)
EP (1) EP3713571A4 (https=)
JP (1) JP7539151B2 (https=)
KR (1) KR102846292B1 (https=)
CN (1) CN111886010A (https=)
AU (1) AU2019206652B2 (https=)
CA (1) CA3087009A1 (https=)
EA (1) EA202091630A1 (https=)
MX (1) MX2020007293A (https=)
WO (1) WO2019140324A1 (https=)

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Publication number Priority date Publication date Assignee Title
US10695400B2 (en) 2015-08-03 2020-06-30 Enb Therapeutics, Inc. Compositions and methods for treating cancers associated with ETBR activation
AU2019206652B2 (en) * 2018-01-12 2024-11-14 Enb Therapeutics, Inc. Deuterated compounds, compositions, and methods for treating cancers associated with ETBR activation
CN114423425A (zh) * 2019-07-17 2022-04-29 Enb治疗公司 通过使用内皮素b受体拮抗剂治疗尿路上皮癌和肾癌
TW202120486A (zh) * 2019-08-09 2021-06-01 英商阿帝歐斯製藥有限公司 新穎化合物
EP4608447A1 (en) * 2022-10-28 2025-09-03 ENB Therapeutics, Inc. Methods for treating cancers associated with etbr activation

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