JP2018524337A5 - - Google Patents
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- JP2018524337A5 JP2018524337A5 JP2017567379A JP2017567379A JP2018524337A5 JP 2018524337 A5 JP2018524337 A5 JP 2018524337A5 JP 2017567379 A JP2017567379 A JP 2017567379A JP 2017567379 A JP2017567379 A JP 2017567379A JP 2018524337 A5 JP2018524337 A5 JP 2018524337A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- cycloalkyl
- cyano
- formula
- halogen
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 125000004093 cyano group Chemical group *C#N 0.000 claims description 36
- 125000000217 alkyl group Chemical group 0.000 claims description 35
- 229910052736 halogen Inorganic materials 0.000 claims description 34
- 150000002367 halogens Chemical class 0.000 claims description 34
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims description 30
- 150000001875 compounds Chemical class 0.000 claims description 30
- 125000001424 substituent group Chemical group 0.000 claims description 23
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 claims description 16
- -1 C 2 -C 6 haloalkynyl Chemical group 0.000 claims description 16
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 claims description 14
- 125000004770 (C1-C4) haloalkylsulfanyl group Chemical group 0.000 claims description 14
- 125000004771 (C1-C4) haloalkylsulfinyl group Chemical group 0.000 claims description 12
- 229910052717 sulfur Inorganic materials 0.000 claims description 12
- 125000003545 alkoxy group Chemical group 0.000 claims description 10
- 229910052739 hydrogen Inorganic materials 0.000 claims description 10
- 239000001257 hydrogen Substances 0.000 claims description 10
- 125000004435 hydrogen atom Chemical class [H]* 0.000 claims description 10
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 claims description 8
- 229910052760 oxygen Inorganic materials 0.000 claims description 8
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims description 7
- 241000607479 Yersinia pestis Species 0.000 claims description 7
- 238000000034 method Methods 0.000 claims description 7
- 125000004769 (C1-C4) alkylsulfonyl group Chemical group 0.000 claims description 6
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 claims description 6
- 125000006643 (C2-C6) haloalkenyl group Chemical group 0.000 claims description 6
- 125000001188 haloalkyl group Chemical group 0.000 claims description 6
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims description 6
- 125000000753 cycloalkyl group Chemical group 0.000 claims description 5
- 125000004768 (C1-C4) alkylsulfinyl group Chemical group 0.000 claims description 4
- 125000002915 carbonyl group Chemical group [*:2]C([*:1])=O 0.000 claims description 4
- 125000001559 cyclopropyl group Chemical group [H]C1([H])C([H])([H])C1([H])* 0.000 claims description 4
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 claims description 4
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims description 4
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 claims description 4
- 150000003839 salts Chemical class 0.000 claims description 4
- 125000004749 (C1-C6) haloalkylsulfinyl group Chemical group 0.000 claims description 3
- 125000004738 (C1-C6) alkyl sulfinyl group Chemical group 0.000 claims description 2
- 125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 claims description 2
- 125000004740 (C1-C6) haloalkylsulfanyl group Chemical group 0.000 claims description 2
- 125000004741 (C1-C6) haloalkylsulfonyl group Chemical group 0.000 claims description 2
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 claims description 2
- 150000001204 N-oxides Chemical class 0.000 claims description 2
- 239000004480 active ingredient Substances 0.000 claims description 2
- 125000004644 alkyl sulfinyl group Chemical group 0.000 claims description 2
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 claims description 2
- SNOOUWRIMMFWNE-UHFFFAOYSA-M sodium;6-[(3,4,5-trimethoxybenzoyl)amino]hexanoate Chemical compound [Na+].COC1=CC(C(=O)NCCCCCC([O-])=O)=CC(OC)=C1OC SNOOUWRIMMFWNE-UHFFFAOYSA-M 0.000 claims description 2
- 239000012752 auxiliary agent Substances 0.000 claims 1
- 125000004441 haloalkylsulfonyl group Chemical group 0.000 description 7
- 125000004414 alkyl thio group Chemical group 0.000 description 3
- 241001465754 Metazoa Species 0.000 description 2
- 125000000232 haloalkynyl group Chemical group 0.000 description 2
- 0 *C(CC1)=CC(*2)=C1N=C2C(*1)=C(CI)C([P+])=C1N=P Chemical compound *C(CC1)=CC(*2)=C1N=C2C(*1)=C(CI)C([P+])=C1N=P 0.000 description 1
- 241000256118 Aedes aegypti Species 0.000 description 1
- 125000004448 alkyl carbonyl group Chemical group 0.000 description 1
- 238000002405 diagnostic procedure Methods 0.000 description 1
- 125000004692 haloalkylcarbonyl group Chemical group 0.000 description 1
- 125000004440 haloalkylsulfinyl group Chemical group 0.000 description 1
- 238000003359 percent control normalization Methods 0.000 description 1
- 230000000361 pesticidal effect Effects 0.000 description 1
- 238000001356 surgical procedure Methods 0.000 description 1
- 238000002560 therapeutic procedure Methods 0.000 description 1
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP15174759.9 | 2015-07-01 | ||
| EP15174759 | 2015-07-01 | ||
| EP15184066 | 2015-09-07 | ||
| EP15184066.7 | 2015-09-07 | ||
| PCT/EP2016/064778 WO2017001311A1 (en) | 2015-07-01 | 2016-06-27 | Pesticidally active tetracyclic derivatives with sulfur containing substituents |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2018524337A JP2018524337A (ja) | 2018-08-30 |
| JP2018524337A5 true JP2018524337A5 (https=) | 2019-08-08 |
Family
ID=56203411
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017567379A Pending JP2018524337A (ja) | 2015-07-01 | 2016-06-27 | 硫黄含有置換基を有する有害生物防除に活性な四環式誘導体 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US10202380B2 (https=) |
| EP (1) | EP3317275B1 (https=) |
| JP (1) | JP2018524337A (https=) |
| CN (1) | CN107810186B (https=) |
| BR (1) | BR112018000052A2 (https=) |
| ES (1) | ES2762958T3 (https=) |
| WO (1) | WO2017001311A1 (https=) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2017144341A1 (de) * | 2016-02-23 | 2017-08-31 | Bayer Cropscience Aktiengesellschaft | Kondensierte bicyclische heterocyclen-derivate als schädlingsbekämpfungsmittel |
| EP3428166A4 (en) | 2016-03-10 | 2019-11-13 | Nissan Chemical Corporation | CONDENSED HETEROCYCLIC COMPOUND AND PESTICIDES |
| WO2018197257A1 (de) * | 2017-04-24 | 2018-11-01 | Bayer Aktiengesellschaft | Kondensierte bicyclische heterocyclen-derivate als schädlingsbekämpfungsmittel |
| WO2019038195A1 (de) | 2017-08-22 | 2019-02-28 | Bayer Aktiengesellschaft | Heterocyclen-derivate als schädlingsbekämpfungsmittel |
| CN111741958A (zh) | 2018-02-21 | 2020-10-02 | 拜耳公司 | 作为害虫防治剂的稠合双环杂环衍生物 |
| KR20200131268A (ko) * | 2018-03-12 | 2020-11-23 | 바이엘 악티엔게젤샤프트 | 해충 방제제로서의 융합된 비시클릭 헤테로시클릭 유도체 |
| WO2019219689A1 (en) | 2018-05-18 | 2019-11-21 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulfoximine containing substituents |
| BR112021003665A2 (pt) | 2018-09-13 | 2021-05-18 | Bayer Aktiengesellschaft | derivados de heterocicleno como agentes de controle de pragas |
| ES2974634T3 (es) | 2018-12-21 | 2024-06-28 | Celgene Corp | Inhibidores de tienopiridinas de RIPK2 |
| AR119140A1 (es) | 2019-06-13 | 2021-11-24 | Pi Industries Ltd | Compuestos heterocíclicos fusionados y su uso como agentes de control de plagas |
| TW202132300A (zh) | 2020-01-06 | 2021-09-01 | 瑞士商先正達農作物保護公司 | 具有含硫取代基的殺有害生物活性雜環衍生物 |
| EP4680028A1 (en) | 2023-03-14 | 2026-01-21 | Syngenta Crop Protection AG | Control of pests resistant to insecticides |
Family Cites Families (46)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BR8600161A (pt) | 1985-01-18 | 1986-09-23 | Plant Genetic Systems Nv | Gene quimerico,vetores de plasmidio hibrido,intermediario,processo para controlar insetos em agricultura ou horticultura,composicao inseticida,processo para transformar celulas de plantas para expressar uma toxina de polipeptideo produzida por bacillus thuringiensis,planta,semente de planta,cultura de celulas e plasmidio |
| CA1340685C (en) | 1988-07-29 | 1999-07-27 | Frederick Meins | Dna sequences encoding polypeptides having beta-1,3-glucanase activity |
| US5169629A (en) | 1988-11-01 | 1992-12-08 | Mycogen Corporation | Process of controlling lepidopteran pests, using bacillus thuringiensis isolate denoted b.t ps81gg |
| EP0374753A3 (de) | 1988-12-19 | 1991-05-29 | American Cyanamid Company | Insektizide Toxine, Gene, die diese Toxine kodieren, Antikörper, die sie binden, sowie transgene Pflanzenzellen und transgene Pflanzen, die diese Toxine exprimieren |
| DK0392225T3 (da) | 1989-03-24 | 2003-09-22 | Syngenta Participations Ag | Sygdomsresistente transgene planter |
| GB8910624D0 (en) | 1989-05-09 | 1989-06-21 | Ici Plc | Bacterial strains |
| CA2015951A1 (en) | 1989-05-18 | 1990-11-18 | Mycogen Corporation | Novel bacillus thuringiensis isolates active against lepidopteran pests, and genes encoding novel lepidopteran-active toxins |
| EP0427529B1 (en) | 1989-11-07 | 1995-04-19 | Pioneer Hi-Bred International, Inc. | Larvicidal lectins and plant insect resistance based thereon |
| US5639949A (en) | 1990-08-20 | 1997-06-17 | Ciba-Geigy Corporation | Genes for the synthesis of antipathogenic substances |
| UA48104C2 (uk) | 1991-10-04 | 2002-08-15 | Новартіс Аг | Фрагмент днк, який містить послідовність,що кодує інсектицидний протеїн, оптимізовану для кукурудзи,фрагмент днк, який забезпечує направлену бажану для серцевини стебла експресію зв'язаного з нею структурного гена в рослині, фрагмент днк, який забезпечує специфічну для пилку експресію зв`язаного з нею структурного гена в рослині, рекомбінантна молекула днк, спосіб одержання оптимізованої для кукурудзи кодуючої послідовності інсектицидного протеїну, спосіб захисту рослин кукурудзи щонайменше від однієї комахи-шкідника |
| US5530195A (en) | 1994-06-10 | 1996-06-25 | Ciba-Geigy Corporation | Bacillus thuringiensis gene encoding a toxin active against insects |
| US5631072A (en) | 1995-03-10 | 1997-05-20 | Avondale Incorporated | Method and means for increasing efficacy and wash durability of insecticide treated fabric |
| BR9913745B1 (pt) | 1998-09-15 | 2011-05-31 | cetonas de piridina, composição herbicida e inibidora do crescimento de plantas, seu uso, método para controle de crescimento de plantas indesejáveis, bem como método para inibir o crescimento de plantas. | |
| AU8590001A (en) | 2000-08-25 | 2002-03-04 | Syngenta Participations Ag | Novel insecticidal toxins derived from bacillus thuringiensis insecticidal crystal proteins |
| JP3789749B2 (ja) | 2000-12-19 | 2006-06-28 | エア・ウォーター・ケミカル株式会社 | チオサリチル酸の製造方法 |
| US7777097B2 (en) | 2001-06-22 | 2010-08-17 | Syngenta Participations Ag | Plant disease resistance genes |
| US7230167B2 (en) | 2001-08-31 | 2007-06-12 | Syngenta Participations Ag | Modified Cry3A toxins and nucleic acid sequences coding therefor |
| WO2003034823A1 (en) | 2001-10-25 | 2003-05-01 | Siamdutch Mosquito Netting Company Limited | Treatment of fabric materials with an insecticide |
| WO2003052073A2 (en) | 2001-12-17 | 2003-06-26 | Syngenta Participations Ag | Novel corn event |
| US20050132500A1 (en) | 2003-12-22 | 2005-06-23 | Basf Aktiengesellschaft | Composition for impregnation of fibers, fabrics and nettings imparting a protective activity against pests |
| DE102004023894A1 (de) | 2004-05-12 | 2005-12-08 | Basf Ag | Verfahren zur Behandlung von flexiblen Substraten |
| JP2008505167A (ja) | 2004-07-05 | 2008-02-21 | アステックス、セラピューティックス、リミテッド | 医薬組成物 |
| DE102005007160A1 (de) | 2005-02-16 | 2006-08-24 | Basf Ag | Pyrazolcarbonsäureanilide, Verfahren zu ihrer Herstellung und sie enthaltende Mittel zur Bekämpfung von Schadpilzen |
| DE102005020889A1 (de) | 2005-05-04 | 2006-11-09 | Fritz Blanke Gmbh & Co.Kg | Verfahren zur antimikrobiellen Ausrüstung von textilen Flächengebilden |
| AP2007004257A0 (en) | 2005-06-03 | 2007-12-31 | Basf Ag | Composition for impregnation of fibres fabrics andnettings imparting a protective activity against pests |
| BRPI0617076B1 (pt) | 2005-09-02 | 2021-07-06 | Nissan Chemical Corporation | Composto benzamida substituída por isoxazolina da fórmula (1) ou sal do mesmo; composto benzamida substituido por 4-hidroxiiminametila da fórmula (2) ou sal do mesmo; pesticida; agente agroquímico; parasiticida interno ou externo para mamíferos ou aves; inseticida ou acaricida |
| US7732469B2 (en) | 2005-10-25 | 2010-06-08 | Syngenta Crop Protection, Inc. | Heterocyclic amide derivatives useful as microbiocides |
| ES2586569T3 (es) | 2006-02-03 | 2016-10-17 | Basf Se | Procedimiento para el tratamiento de sustratos textiles |
| MX2009011208A (es) | 2007-04-19 | 2009-10-30 | Novartis Ag | Derivados de acido nicotinico como moduladores del receptor de glutamato metabotropico-5. |
| JP5230731B2 (ja) | 2007-06-12 | 2013-07-10 | ビーエーエスエフ ソシエタス・ヨーロピア | 害虫からの保護活性を付与するための非生物材料への含浸用水性製剤及び含浸方法 |
| JP5369854B2 (ja) | 2008-04-21 | 2013-12-18 | 住友化学株式会社 | 有害節足動物防除組成物および縮合複素環化合物 |
| US8273764B2 (en) | 2009-04-28 | 2012-09-25 | Sumitomo Chemical Company, Limited | Fused heterocyclic compounds and use thereof |
| CN102573488A (zh) | 2009-09-30 | 2012-07-11 | 住友化学株式会社 | 用于防治节肢动物害虫的组合物和方法 |
| JP5540640B2 (ja) | 2009-10-07 | 2014-07-02 | 住友化学株式会社 | 複素環化合物及びその有害節足動物防除用途 |
| WO2012086848A1 (en) | 2010-12-24 | 2012-06-28 | Sumitomo Chemical Company, Limited | Fused heterocyclic compound and use for pest control thereof |
| TWI528899B (zh) | 2010-12-29 | 2016-04-11 | 杜邦股份有限公司 | 中離子性殺蟲劑 |
| US20120309796A1 (en) | 2011-06-06 | 2012-12-06 | Fariborz Firooznia | Benzocycloheptene acetic acids |
| TWI545119B (zh) | 2011-08-04 | 2016-08-11 | 住友化學股份有限公司 | 稠合雜環化合物及其在病蟲害防制上之用途 |
| JP2013170151A (ja) * | 2012-02-22 | 2013-09-02 | Nagoya Institute Of Technology | インドール‐３−トリフロン類の直接的製造法及びインドールトリフロン誘導体 |
| EP2857397B1 (en) * | 2012-05-30 | 2020-04-08 | Sumitomo Chemical Company Limited | Fused heterocyclic compound |
| WO2013180193A1 (ja) * | 2012-05-31 | 2013-12-05 | 住友化学株式会社 | 縮合複素環化合物 |
| EP2862853B1 (en) | 2012-06-18 | 2020-01-22 | Sumitomo Chemical Co., Ltd | Fused heterocyclic compound |
| WO2015000715A1 (en) * | 2013-07-02 | 2015-01-08 | Syngenta Participations Ag | Pesticidally active bi- or tricyclic heterocycles with sulfur containing substituents |
| JP6779225B2 (ja) * | 2015-03-12 | 2020-11-04 | シンジェンタ パーティシペーションズ アーゲー | 硫黄含有置換基を有する有害生物防除に活性な四環式誘導体 |
| CN107428751B (zh) * | 2015-03-12 | 2020-06-30 | 先正达参股股份有限公司 | 具有含硫取代基的杀有害生物活性四环衍生物 |
| WO2016169882A1 (en) * | 2015-04-24 | 2016-10-27 | Syngenta Participations Ag | Pesticidally active polycyclic derivatives with sulfur substituted five membered ring heterocyles |
-
2016
- 2016-06-27 JP JP2017567379A patent/JP2018524337A/ja active Pending
- 2016-06-27 EP EP16731935.9A patent/EP3317275B1/en active Active
- 2016-06-27 WO PCT/EP2016/064778 patent/WO2017001311A1/en not_active Ceased
- 2016-06-27 CN CN201680038616.5A patent/CN107810186B/zh not_active Expired - Fee Related
- 2016-06-27 BR BR112018000052-3A patent/BR112018000052A2/pt not_active Application Discontinuation
- 2016-06-27 ES ES16731935T patent/ES2762958T3/es active Active
- 2016-06-27 US US15/732,804 patent/US10202380B2/en not_active Expired - Fee Related
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