JP2017531616A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2017531616A5 JP2017531616A5 JP2017510336A JP2017510336A JP2017531616A5 JP 2017531616 A5 JP2017531616 A5 JP 2017531616A5 JP 2017510336 A JP2017510336 A JP 2017510336A JP 2017510336 A JP2017510336 A JP 2017510336A JP 2017531616 A5 JP2017531616 A5 JP 2017531616A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- haloalkyl
- cycloalkyl
- group
- halogen
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims description 37
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 claims description 36
- 229910052736 halogen Inorganic materials 0.000 claims description 36
- 150000002367 halogens Chemical group 0.000 claims description 36
- 125000001424 substituent group Chemical group 0.000 claims description 35
- 125000000217 alkyl group Chemical group 0.000 claims description 32
- 125000004093 cyano group Chemical group *C#N 0.000 claims description 32
- 150000001875 compounds Chemical class 0.000 claims description 29
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims description 25
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 claims description 23
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims description 19
- -1 C 1 -C 4 alkyl Chemical group 0.000 claims description 12
- 125000001181 organosilyl group Chemical group [SiH3]* 0.000 claims description 10
- 125000004770 (C1-C4) haloalkylsulfanyl group Chemical group 0.000 claims description 8
- 125000004771 (C1-C4) haloalkylsulfinyl group Chemical group 0.000 claims description 8
- 238000000034 method Methods 0.000 claims description 7
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 claims description 6
- 241000607479 Yersinia pestis Species 0.000 claims description 6
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims description 6
- 239000000463 material Substances 0.000 claims description 6
- 239000000203 mixture Substances 0.000 claims description 6
- 125000000753 cycloalkyl group Chemical group 0.000 claims description 5
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 claims description 4
- IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 claims description 4
- 125000004186 cyclopropylmethyl group Chemical group [H]C([H])(*)C1([H])C([H])([H])C1([H])[H] 0.000 claims description 4
- 125000001188 haloalkyl group Chemical group 0.000 claims description 4
- 229910052739 hydrogen Inorganic materials 0.000 claims description 4
- 239000001257 hydrogen Substances 0.000 claims description 4
- 125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 claims description 4
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims description 4
- 125000004123 n-propyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])* 0.000 claims description 4
- 150000003839 salts Chemical class 0.000 claims description 4
- SNOOUWRIMMFWNE-UHFFFAOYSA-M sodium;6-[(3,4,5-trimethoxybenzoyl)amino]hexanoate Chemical compound [Na+].COC1=CC(C(=O)NCCCCCC([O-])=O)=CC(OC)=C1OC SNOOUWRIMMFWNE-UHFFFAOYSA-M 0.000 claims description 3
- 125000006643 (C2-C6) haloalkenyl group Chemical group 0.000 claims description 2
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 claims description 2
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 claims description 2
- 150000001204 N-oxides Chemical class 0.000 claims description 2
- 239000004480 active ingredient Substances 0.000 claims description 2
- 238000002405 diagnostic procedure Methods 0.000 claims description 2
- 150000002431 hydrogen Chemical class 0.000 claims description 2
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims description 2
- 125000001434 methanylylidene group Chemical group [H]C#[*] 0.000 claims description 2
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 claims description 2
- 229910052757 nitrogen Inorganic materials 0.000 claims description 2
- 229910052760 oxygen Inorganic materials 0.000 claims description 2
- 229910052717 sulfur Inorganic materials 0.000 claims description 2
- 238000001356 surgical procedure Methods 0.000 claims description 2
- 239000002671 adjuvant Substances 0.000 claims 1
- 230000000361 pesticidal effect Effects 0.000 claims 1
- 238000002560 therapeutic procedure Methods 0.000 claims 1
- 125000003545 alkoxy group Chemical group 0.000 description 4
- 125000004441 haloalkylsulfonyl group Chemical group 0.000 description 4
- IAZDPXIOMUYVGZ-UHFFFAOYSA-N Dimethylsulphoxide Chemical compound CS(C)=O IAZDPXIOMUYVGZ-UHFFFAOYSA-N 0.000 description 3
- 0 **c1c(C(*2)=Nc3c2cnc(*)c3)ncc(*)c1 Chemical compound **c1c(C(*2)=Nc3c2cnc(*)c3)ncc(*)c1 0.000 description 2
- 241001465754 Metazoa Species 0.000 description 2
- 125000003342 alkenyl group Chemical group 0.000 description 2
- 125000000392 cycloalkenyl group Chemical group 0.000 description 2
- 125000006727 (C1-C6) alkenyl group Chemical group 0.000 description 1
- 229920001817 Agar Polymers 0.000 description 1
- 241000196324 Embryophyta Species 0.000 description 1
- 241000927584 Frankliniella occidentalis Species 0.000 description 1
- 241000208818 Helianthus Species 0.000 description 1
- 235000003222 Helianthus annuus Nutrition 0.000 description 1
- 206010061217 Infestation Diseases 0.000 description 1
- 241001414989 Thysanoptera Species 0.000 description 1
- 239000008272 agar Substances 0.000 description 1
- 239000007864 aqueous solution Substances 0.000 description 1
- 239000012752 auxiliary agent Substances 0.000 description 1
- 238000001035 drying Methods 0.000 description 1
- 239000000575 pesticide Substances 0.000 description 1
- 239000011550 stock solution Substances 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP14181715 | 2014-08-21 | ||
| EP14181715.5 | 2014-08-21 | ||
| PCT/EP2015/068928 WO2016026848A1 (en) | 2014-08-21 | 2015-08-18 | Pesticidally active heterocyclic derivatives with sulphur containing substituents |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2017531616A JP2017531616A (ja) | 2017-10-26 |
| JP2017531616A5 true JP2017531616A5 (cg-RX-API-DMAC7.html) | 2018-09-27 |
| JP6695326B2 JP6695326B2 (ja) | 2020-05-20 |
Family
ID=51383620
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017510336A Active JP6695326B2 (ja) | 2014-08-21 | 2015-08-18 | 硫黄含有置換基を有する殺有害生物的に活性な複素環式誘導体 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US10081641B2 (cg-RX-API-DMAC7.html) |
| EP (1) | EP3183245B1 (cg-RX-API-DMAC7.html) |
| JP (1) | JP6695326B2 (cg-RX-API-DMAC7.html) |
| CN (1) | CN106573891B (cg-RX-API-DMAC7.html) |
| AR (1) | AR101586A1 (cg-RX-API-DMAC7.html) |
| BR (1) | BR112017003168B1 (cg-RX-API-DMAC7.html) |
| ES (1) | ES2701859T3 (cg-RX-API-DMAC7.html) |
| WO (1) | WO2016026848A1 (cg-RX-API-DMAC7.html) |
Families Citing this family (50)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US11229208B2 (en) | 2013-07-02 | 2022-01-25 | Syngenta Participations Ag | Pesticidally active bi- or tricyclic heterocycles with sulfur containing substituents |
| MX2015017821A (es) * | 2013-07-02 | 2016-04-15 | Syngenta Participations Ag | Heterociclos bi-o triciclicos activos como plaguicidas con sustituyentes que contienen azufre. |
| BR112017003366B1 (pt) * | 2014-08-25 | 2020-12-08 | Syngenta Participations Ag | derivados de heterocíclicos ativos do ponto de vista pesticida com substituintes contendo enxofre, composição pesticida, método para controle de pragas e método para a proteção de material de propagação de plantas do ataque por pragas |
| CN107074865B (zh) * | 2014-11-07 | 2020-06-30 | 先正达参股股份有限公司 | 具有含硫取代基的杀有害生物活性多环衍生物 |
| US10494366B2 (en) * | 2014-12-01 | 2019-12-03 | Syngenta Participations Ag | Pesticidally active amide heterocyclic derivatives with sulphur containing substituents |
| US10071997B2 (en) * | 2014-12-01 | 2018-09-11 | Syngenta Participations Ag | Pesticidally active amide heterocyclic derivatives with sulphur containing substituents |
| TWI696612B (zh) * | 2015-01-29 | 2020-06-21 | 日商日本農藥股份有限公司 | 具有環烷基吡啶基的稠合雜環化合物或其鹽類及含有該化合物的農園藝用殺蟲劑以及其使用方法 |
| UY36547A (es) * | 2015-02-05 | 2016-06-01 | Bayer Cropscience Ag | Derivados heterocíclicos condensados bicíclicos sustituidos por 2-(het)arilo como pesticidas |
| MX2018001417A (es) | 2015-08-07 | 2018-03-15 | Bayer Cropscience Ag | Derivados heterociclicos condensados sustituidos por 2-(het)-arilo como pesticidas. |
| WO2017055185A1 (de) | 2015-09-28 | 2017-04-06 | Bayer Cropscience Aktiengesellschaft | 2-(het)aryl-substituierte kondensierte heterocyclen-derivate als schädlingsbekämpfungsmittel |
| CA3002888A1 (en) | 2015-10-26 | 2017-05-04 | Bayer Cropscience Aktiengesellschaft | Condensed bicyclic heterocycle derivatives as pest control agents |
| JP2019502713A (ja) | 2016-01-11 | 2019-01-31 | バイエル・クロップサイエンス・アクチェンゲゼルシャフト | 有害生物防除剤としてのヘテロサイクレン誘導体 |
| ES2877814T3 (es) | 2016-10-06 | 2021-11-17 | Bayer Cropscience Ag | Derivados de heterociclos bicíclicos condensados sustituidos con 2-(het)arilo como pesticidas |
| WO2018065288A1 (de) | 2016-10-07 | 2018-04-12 | Bayer Cropscience Aktiengesellschaft | 2-[2-phenyl-1-(sulfonylmethyl)vinyl]-imidazo[4,5-b]pyridin-derivate und verwandte verbindungen als schädlingsbekämpfungsmittel im pflanzenschutz |
| CN117624038A (zh) | 2016-12-01 | 2024-03-01 | 先正达参股股份有限公司 | 具有含硫取代基的杀有害生物活性杂环衍生物 |
| KR102515694B1 (ko) | 2017-01-10 | 2023-03-29 | 바이엘 악티엔게젤샤프트 | 해충 방제제로서의 헤테로사이클 유도체 |
| WO2018130443A1 (de) | 2017-01-10 | 2018-07-19 | Bayer Aktiengesellschaft | Heterocyclen-derivate als schädlingsbekämpfungsmittel |
| TWI793104B (zh) * | 2017-02-21 | 2023-02-21 | 瑞士商先正達合夥公司 | 具有含硫取代基的殺有害生物活性雜環衍生物 |
| EP3615531A1 (en) | 2017-04-25 | 2020-03-04 | Syngenta Participations AG | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| JP2020128341A (ja) * | 2017-04-27 | 2020-08-27 | 日本農薬株式会社 | 共役したオキシムエーテル基を有する複素環化合物又はその塩類及び該化合物を含有する農園芸用殺虫剤並びにその使用方法 |
| JP7309615B2 (ja) | 2017-05-02 | 2023-07-18 | シンジェンタ パーティシペーションズ アーゲー | 硫黄含有置換基を有する有害生物防除に活性な複素環式誘導体 |
| CN110891949B (zh) | 2017-07-05 | 2023-05-23 | 先正达参股股份有限公司 | 具有含硫取代基的杀有害生物活性杂环衍生物 |
| EP3649128A1 (en) | 2017-07-07 | 2020-05-13 | Syngenta Participations AG | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| ES2975315T3 (es) | 2017-09-18 | 2024-07-04 | Syngenta Participations Ag | Derivados heterocíclicos plaguicidamente activos con sustituyentes que contienen azufre |
| US11252962B2 (en) | 2017-09-21 | 2022-02-22 | Nihon Nohyaku Co., Ltd. | Cyclopropylpyridyl group-containing benzimidazole compound or salt thereof, agricultural and horticultural insecticide comprising the compound or the salt, and method for using the insecticide |
| WO2019076778A1 (en) | 2017-10-16 | 2019-04-25 | Syngenta Participations Ag | HETEROCYCLIC DERIVATIVES HAVING PESTICIDAL ACTIVITY HAVING SUBSTITUENTS CONTAINING SULFUR AND SULFONIMIDAMIDES |
| CN111836810B (zh) | 2018-01-15 | 2024-06-25 | 先正达参股股份有限公司 | 具有含硫取代基的杀有害生物活性的杂环衍生物 |
| WO2019229089A1 (en) | 2018-05-31 | 2019-12-05 | Syngenta Participations Ag | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| AR115495A1 (es) | 2018-06-06 | 2021-01-27 | Syngenta Crop Protection Ag | Derivados heterocíclicos con sustituyentes que contienen azufre activos como plaguicidas |
| MA52751A (fr) | 2018-06-06 | 2021-04-14 | Syngenta Crop Protection Ag | Dérivés hétérocycliques à action pesticide comportant des substituants contenant de la sulfoximine |
| AU2019296166B2 (en) | 2018-06-26 | 2024-01-18 | Bayer Aktiengesellschaft | Heterocyclene derivatives as pest control agents |
| EP3835301B1 (en) | 2018-07-10 | 2024-10-09 | Nihon Nohyaku Co., Ltd. | Benzimidazole compound having alkylenedioxy group which may be halogenated or salt thereof, agricultural and horticultural pesticide containing said compound, and method of using same |
| TW202035404A (zh) | 2018-10-24 | 2020-10-01 | 瑞士商先正達農作物保護公司 | 具有含亞碸亞胺的取代基之殺有害生物活性雜環衍生物 |
| CN113348169A (zh) | 2018-12-31 | 2021-09-03 | 先正达农作物保护股份公司 | 具有含硫取代基的杀有害生物活性的杂环衍生物 |
| US12439920B2 (en) | 2019-02-26 | 2025-10-14 | Nippon Soda Co., Ltd. | Pyridine n-oxide compound and pest control agent |
| JP7664166B2 (ja) * | 2019-02-26 | 2025-04-17 | バイエル・アクチエンゲゼルシヤフト | 有害生物防除剤としての縮合二環式複素環式誘導体 |
| BR112021010400A2 (pt) | 2019-02-26 | 2021-08-24 | Bayer Aktiengesellschaft | Derivados heterocíclicos bicíclicos condensados como agentes de controle de praga |
| TW202045011A (zh) | 2019-02-28 | 2020-12-16 | 瑞士商先正達農作物保護公司 | 具有含硫取代基之殺有害生物活性雜環衍生物 |
| AR118243A1 (es) | 2019-03-07 | 2021-09-22 | Pi Industries Ltd | Compuestos heterocíclicos fusionados y su uso como agentes de control de plagas |
| KR102335886B1 (ko) * | 2020-03-11 | 2021-12-07 | 서울대학교병원 | 엘리오카퍼스 페티오라투스를 포함하는 심혈관 대사 질환의 예방 또는 치료용 조성물 |
| EP4132927A1 (en) | 2020-04-06 | 2023-02-15 | Basf Se | Imidazo-pyrimidone compounds as pesticides |
| TW202200570A (zh) | 2020-04-21 | 2022-01-01 | 德商拜耳廠股份有限公司 | 作為殺蟲劑之經２—（雜）芳基取代的稠合雜環衍生物 |
| EP4143177A1 (en) | 2020-04-30 | 2023-03-08 | Syngenta Crop Protection AG | Pesticidally active heterocyclic derivatives with sulfur containing substituents |
| CN116033828B (zh) | 2020-07-02 | 2025-05-16 | 拜耳公司 | 作为害虫防治剂的杂环衍生物 |
| EP4204422A1 (en) | 2020-08-26 | 2023-07-05 | Syngenta Crop Protection AG | Process for the preparation of 2,2-difluoro-1,3-benzodioxole derivatives with sulfur containing substituents |
| AU2021403544A1 (en) | 2020-12-14 | 2023-06-29 | Basf Se | Sulfoximine pesticides |
| KR20240007207A (ko) | 2021-05-12 | 2024-01-16 | 바이엘 악티엔게젤샤프트 | 살충제로서의 2-(헤트)아릴-치환된 융합된 헤테로사이클 유도체 |
| KR20240016326A (ko) | 2021-06-02 | 2024-02-06 | 신젠타 크롭 프로텍션 아게 | 설폭시민 함유 치환체를 갖는 살충 활성 헤테로사이클릭 유도체 |
| AU2024235487A1 (en) | 2023-03-14 | 2025-09-25 | Syngenta Crop Protection Ag | Control of pests resistant to insecticides |
| WO2025026738A1 (en) | 2023-07-31 | 2025-02-06 | Bayer Aktiengesellschaft | 6-[5-(ethylsulfonyl)-1-methyl-1h-imidazol-4-yl]-7-methyl-3-(pentafluoroethyl)-7h-imidazo[4,5-c]pyridazine derivatives as pesticides |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES517193A0 (es) * | 1981-11-10 | 1983-12-01 | Wellcome Found | Un procedimiento para la preparacion de nuevos derivados de imidazo (4,5-c)piridina. |
| ZA828213B (en) * | 1981-11-10 | 1984-06-27 | Wellcome Found | New bicyclic compounds,processes for their preparation and pharmaceutical formulations containing such compounds |
| BR112013016022B1 (pt) * | 2010-12-24 | 2019-05-07 | Sumitomo Chemical Company, Limited | Composto heterocíclico fundido e uso do mesmo para controle de peste. |
| TWI545119B (zh) * | 2011-08-04 | 2016-08-11 | 住友化學股份有限公司 | 稠合雜環化合物及其在病蟲害防制上之用途 |
| ITMI20120225A1 (it) * | 2012-02-16 | 2013-08-17 | Ecoct Tecnologie Ambientali S P A | Macchina di lavaggio a tamburo rotante |
| MX2015017821A (es) * | 2013-07-02 | 2016-04-15 | Syngenta Participations Ag | Heterociclos bi-o triciclicos activos como plaguicidas con sustituyentes que contienen azufre. |
| KR101545215B1 (ko) * | 2013-10-30 | 2015-08-18 | 삼성에스디에스 주식회사 | 데이터 센터 장애 이벤트 관리 자동화 시스템 및 방법 |
| ES2987367T3 (es) * | 2014-02-17 | 2024-11-14 | Bayer Cropscience Ag | Derivados de heterociclos bicíclicos condensados sustituidos con 2-(het)arilo como agentes para combatir parásitos |
| MX2017000305A (es) * | 2014-07-08 | 2017-04-27 | Syngenta Participations Ag | Derivados heterociclicos activos con sustituyentes que contienen azufre como plaguicidas. |
| CN107074846B (zh) * | 2014-08-12 | 2020-05-19 | 先正达参股股份有限公司 | 具有含硫取代基的杀有害生物活性杂环衍生物 |
| BR112017003366B1 (pt) * | 2014-08-25 | 2020-12-08 | Syngenta Participations Ag | derivados de heterocíclicos ativos do ponto de vista pesticida com substituintes contendo enxofre, composição pesticida, método para controle de pragas e método para a proteção de material de propagação de plantas do ataque por pragas |
-
2015
- 2015-08-18 JP JP2017510336A patent/JP6695326B2/ja active Active
- 2015-08-18 EP EP15753672.3A patent/EP3183245B1/en active Active
- 2015-08-18 ES ES15753672T patent/ES2701859T3/es active Active
- 2015-08-18 CN CN201580044808.2A patent/CN106573891B/zh active Active
- 2015-08-18 US US15/504,688 patent/US10081641B2/en active Active
- 2015-08-18 WO PCT/EP2015/068928 patent/WO2016026848A1/en not_active Ceased
- 2015-08-18 BR BR112017003168-0A patent/BR112017003168B1/pt active IP Right Grant
- 2015-08-19 AR ARP150102661A patent/AR101586A1/es unknown