JP2017516777A5 - - Google Patents

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Publication number
JP2017516777A5
JP2017516777A5 JP2016568934A JP2016568934A JP2017516777A5 JP 2017516777 A5 JP2017516777 A5 JP 2017516777A5 JP 2016568934 A JP2016568934 A JP 2016568934A JP 2016568934 A JP2016568934 A JP 2016568934A JP 2017516777 A5 JP2017516777 A5 JP 2017516777A5
Authority
JP
Japan
Prior art keywords
pharmaceutical composition
subject
infection
oxazino
oxazolo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2016568934A
Other languages
English (en)
Japanese (ja)
Other versions
JP2017516777A (ja
JP6502387B2 (ja
JP6502387B6 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2015/001585 external-priority patent/WO2015181637A1/en
Publication of JP2017516777A publication Critical patent/JP2017516777A/ja
Publication of JP2017516777A5 publication Critical patent/JP2017516777A5/ja
Publication of JP6502387B2 publication Critical patent/JP6502387B2/ja
Application granted granted Critical
Publication of JP6502387B6 publication Critical patent/JP6502387B6/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2016568934A 2014-05-29 2015-05-27 細菌感染の治療のための融合スピロ環ヘテロ芳香族化合物 Expired - Fee Related JP6502387B6 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201462004246P 2014-05-29 2014-05-29
US62/004,246 2014-05-29
PCT/IB2015/001585 WO2015181637A1 (en) 2014-05-29 2015-05-27 Fused, spirocyclic heteroaromatic compounds for the treatment of bacterial infections

Publications (4)

Publication Number Publication Date
JP2017516777A JP2017516777A (ja) 2017-06-22
JP2017516777A5 true JP2017516777A5 (enExample) 2018-06-07
JP6502387B2 JP6502387B2 (ja) 2019-04-17
JP6502387B6 JP6502387B6 (ja) 2019-05-29

Family

ID=54329851

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2016568934A Expired - Fee Related JP6502387B6 (ja) 2014-05-29 2015-05-27 細菌感染の治療のための融合スピロ環ヘテロ芳香族化合物

Country Status (14)

Country Link
US (1) US10238661B2 (enExample)
EP (1) EP3148546A1 (enExample)
JP (1) JP6502387B6 (enExample)
KR (1) KR20170007818A (enExample)
CN (1) CN106659725A (enExample)
AU (1) AU2015265620B2 (enExample)
CA (1) CA2948438A1 (enExample)
EA (1) EA033459B1 (enExample)
IL (1) IL248838B (enExample)
MX (1) MX365261B (enExample)
PH (1) PH12016502271A1 (enExample)
SG (2) SG10201906842WA (enExample)
TW (1) TWI657818B (enExample)
WO (1) WO2015181637A1 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN109111465B (zh) * 2017-06-22 2021-01-12 中国科学院上海药物研究所 噻唑烷酮螺嘧啶三酮类化合物及制备方法和用途
US11905286B2 (en) 2018-08-09 2024-02-20 Antabio Sas Diazabicyclooctanones as inhibitors of serine beta-lactamases
SG11202101255UA (en) 2018-08-09 2021-03-30 Antabio Sas Diazabicyclooctanones as inhibitors of serine beta-lactamases

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7208490B2 (en) * 2002-10-07 2007-04-24 Pharmacia & Upjohn Company Llc Tricyclic tetrahydroquinoline antibacterial agents
ATE423122T1 (de) 2003-08-15 2009-03-15 Astrazeneca Ab Kondensierte heterocyclen als inhibitoren von glutamatracemase (muri)
WO2006120563A2 (en) 2005-05-09 2006-11-16 Warner-Lambert Company Llc Antibacterial agents
DOP2006000268A (es) 2005-12-22 2007-07-31 Pfizer Prod Inc Agentes antibacterianos
CL2007003332A1 (es) 2006-11-24 2008-06-20 Actelion Pharmaceuticals Ltd Compuestos derivados de heterociclos condensados; compuestos intermediarios; composicion farmaceutica; y uso en la prevencion o tratamiento de infecciones bacterianas.
CN101784553A (zh) 2007-07-02 2010-07-21 阿斯利康(瑞典)有限公司 3-螺嘧啶三酮-喹啉衍生物及其作为抗菌药物的应用
UY32174A (es) * 2008-10-14 2010-05-31 Astrazeneca Ab Nuevos heterociclos sustituidos, composiciones farmaceuticas conteniendolos, procedimientos de preparacion y aplicaciones
US9040528B2 (en) 2008-10-14 2015-05-26 Astrazeneca Ab Chemical compounds 542
AR084070A1 (es) 2010-12-02 2013-04-17 Constellation Pharmaceuticals Inc Inhibidores del bromodominio y usos de los mismos
US8952149B2 (en) 2012-09-26 2015-02-10 Zoetis Llc Tricyclic tetrahydroquinoline antibacterial agents
US8889671B2 (en) 2013-01-23 2014-11-18 Astrazeneca Ab Compounds and methods for treating bacterial infections

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