JP2016510787A5 - - Google Patents
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- Publication number
- JP2016510787A5 JP2016510787A5 JP2015562144A JP2015562144A JP2016510787A5 JP 2016510787 A5 JP2016510787 A5 JP 2016510787A5 JP 2015562144 A JP2015562144 A JP 2015562144A JP 2015562144 A JP2015562144 A JP 2015562144A JP 2016510787 A5 JP2016510787 A5 JP 2016510787A5
- Authority
- JP
- Japan
- Prior art keywords
- crizotinib
- lubricant
- tablet
- optionally
- tablets
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 238000000034 method Methods 0.000 claims 13
- 239000002146 L01XE16 - Crizotinib Substances 0.000 claims 8
- KTEIFNKAUNYNJU-GFCCVEGCSA-N crizotinib Chemical compound O([C@H](C)C=1C(=C(F)C=CC=1Cl)Cl)C(C(=NC=1)N)=CC=1C(=C1)C=NN1C1CCNCC1 KTEIFNKAUNYNJU-GFCCVEGCSA-N 0.000 claims 8
- 229960005061 crizotinib Drugs 0.000 claims 8
- 239000000314 lubricant Substances 0.000 claims 8
- 239000012458 free base Substances 0.000 claims 3
- 239000000546 pharmaceutical excipient Substances 0.000 claims 3
- 229940124531 pharmaceutical excipient Drugs 0.000 claims 3
- 239000011230 binding agent Substances 0.000 claims 2
- 239000007884 disintegrant Substances 0.000 claims 2
- 239000002552 dosage form Substances 0.000 claims 2
- 239000000945 filler Substances 0.000 claims 2
- 239000000203 mixture Substances 0.000 claims 2
- 125000004432 carbon atom Chemical group C* 0.000 claims 1
- 230000006835 compression Effects 0.000 claims 1
- 238000007906 compression Methods 0.000 claims 1
- 239000007888 film coating Substances 0.000 claims 1
- 238000009501 film coating Methods 0.000 claims 1
- 238000002156 mixing Methods 0.000 claims 1
- 239000002245 particle Substances 0.000 claims 1
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201361780015P | 2013-03-13 | 2013-03-13 | |
| EP13001257 | 2013-03-13 | ||
| US61/780,015 | 2013-03-13 | ||
| EP13001257.8 | 2013-03-13 | ||
| PCT/EP2014/054933 WO2014140159A1 (en) | 2013-03-13 | 2014-03-13 | Dosage form comprising crizotinib |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2016510787A JP2016510787A (ja) | 2016-04-11 |
| JP2016510787A5 true JP2016510787A5 (https=) | 2017-04-13 |
Family
ID=47900469
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015562144A Pending JP2016510787A (ja) | 2013-03-13 | 2014-03-13 | クリゾチニブを含む剤形 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US20160022661A1 (https=) |
| EP (1) | EP2968167A1 (https=) |
| JP (1) | JP2016510787A (https=) |
| EA (1) | EA201591644A1 (https=) |
| WO (1) | WO2014140159A1 (https=) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN108721243B (zh) * | 2017-04-25 | 2022-07-08 | 正大天晴药业集团股份有限公司 | 克唑替尼药物组合物及其制备方法 |
| CA3166050C (en) * | 2019-12-31 | 2024-02-20 | Pfizer R&D Uk Limited | Stable immediate release tablet and capsule formulations of 1-((2s,5r)-5-((7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino)-2-methylpiperidin-1-yl)prop-2-en-1-one |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9518953D0 (en) * | 1995-09-15 | 1995-11-15 | Pfizer Ltd | Pharmaceutical formulations |
| PL1959955T3 (pl) * | 2005-12-05 | 2011-04-29 | Pfizer Prod Inc | Sposób traktowania nieprawidłowego wzrostu komórek |
| DE102009015702A1 (de) * | 2009-03-31 | 2010-10-07 | Ratiopharm Gmbh | Tabletten enthaltend Dapoxetin und Trockenverarbeitungsverfahren zu deren Herstellung |
-
2014
- 2014-03-13 JP JP2015562144A patent/JP2016510787A/ja active Pending
- 2014-03-13 EA EA201591644A patent/EA201591644A1/ru unknown
- 2014-03-13 EP EP14709950.1A patent/EP2968167A1/en not_active Withdrawn
- 2014-03-13 US US14/774,072 patent/US20160022661A1/en not_active Abandoned
- 2014-03-13 WO PCT/EP2014/054933 patent/WO2014140159A1/en not_active Ceased
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