JP2016204377A

JP2016204377A - Acylhydrazone derivative and pest control agent

Info

Publication number: JP2016204377A
Application number: JP2016085760A
Authority: JP
Inventors: 基浩梶; Motohiro Kaji; 伊藤　幸子; Sachiko Ito; 幸子伊藤; 西尾　晃一; Koichi Nishio; 晃一西尾; 優樹植村; Yuki Uemura
Original assignee: Nissan Chemical Corp
Current assignee: Nissan Chemical Corp
Priority date: 2015-04-24
Filing date: 2016-04-22
Publication date: 2016-12-08

Abstract

PROBLEM TO BE SOLVED: To provide a novel bactericidal agent, particularly a bactericide for agricultural and horticultural use.SOLUTION: The present invention provides an acylhydrazone derivative represented by formula (I) or salt thereof, or N-oxide thereof, and a bactericide for agricultural and horticultural use comprising the same [W is O or S; A is O or S; Ris alkyl or cycloalkyl; and Ris phenyl substituted by (Z)and the like].SELECTED DRAWING: None

Description

本発明は、新規なアシルヒドラゾン誘導体及びその塩、並びに該化合物を有効成分として含有する有害生物防除剤に関するものである。 The present invention relates to a novel acyl hydrazone derivative and a salt thereof, and a pest control agent containing the compound as an active ingredient.

ある種のアシルヒドラゾン誘導体が殺菌活性を有することが知られている（例えば、特許文献１参照。）。 It is known that certain acyl hydrazone derivatives have bactericidal activity (see, for example, Patent Document 1).

また、ある種のヘテロ環、例えばテトラゾリノン環を有する化合物が殺菌活性を有することが知られている（例えば、特許文献２〜特許文献３参照。）。 Moreover, it is known that the compound which has a certain kind of heterocyclic ring, for example, a tetrazolinone ring, has bactericidal activity (for example, refer patent document 2-patent document 3).

しかしながら、本発明に係るアシルヒドラゾン誘導体に関しては何ら開示されてなく、また、それらの有害生物防除剤としての有用性は知られていない。 However, no acyl hydrazone derivatives according to the present invention are disclosed, and their usefulness as pest control agents is not known.

特開平７−１７９３０号公報JP-A-7-17930 国際公開第１９９６／０３６２２９号International Publication No. 1996/036229 国際公開第２０１３／１６２０７２号International Publication No. 2013/162072

農園芸作物の病害に対する防除剤の開発が進み、多種多様な薬剤が今日まで実用に供されてきた。しかしながら、こうした薬剤の長年にわたる使用により、近年、病原菌が薬剤抵抗性を獲得し、従来用いられてきた既存の殺菌剤による防除が困難となる場面が増えてきている。また、既存の薬剤の一部のものは毒性が高く、或いはあるものは環境中に長期間残留することにより、生態系を攪乱するという問題も顕在化しつつある。このような状況下、高度な防除活性ならびに対象となる作物に対する高い安全性を有するのみならず、低毒性且つ低残留性の新規な薬剤の開発が常に期待されている。 The development of control agents for diseases of agricultural and horticultural crops has progressed, and a wide variety of drugs have been put to practical use until now. However, due to the long-term use of such drugs, in recent years, pathogens have acquired drug resistance, and the number of scenes where it is difficult to control with existing bactericides that have been used in the past has increased. In addition, some existing drugs are highly toxic, or some remain in the environment for a long time, causing problems that disturb the ecosystem. Under such circumstances, development of a new drug having not only high control activity and high safety for target crops but also low toxicity and low persistence is always expected.

本発明者らは、上記の課題解決を目標に鋭意研究を重ねた結果、本発明に係る下記式（Ｉ）で表される新規なアシルヒドラゾン誘導体が殺菌剤、特に農園芸用殺菌剤として優れた防除活性ならびに対象となる作物に対する高い安全性を有し、且つ、ホ乳動物、魚類及び益虫等の非標的生物に対してほとんど悪影響の無い、極めて有用な化合物であることを見い出し、本発明を完成した。 As a result of intensive studies aimed at solving the above problems, the present inventors have found that the novel acylhydrazone derivative represented by the following formula (I) according to the present invention is excellent as a bactericidal agent, particularly an agricultural and horticultural fungicide. The present invention has been found to be a very useful compound that has a high control activity and a high safety against the target crop and has almost no adverse effect on non-target organisms such as mammals, fish and beneficial insects. Was completed.

すなわち、本発明は下記〔１〕〜〔８〕に関するものである。 That is, the present invention relates to the following [1] to [8].

〔１〕
式（Ｉ）： [1]
Formula (I):

［式中、Ｗは、酸素原子又は硫黄原子を表し、
Ａは、酸素原子又は硫黄原子を表し、
Ｒ^１は、Ｃ_１〜Ｃ_６アルキル、ハロ（Ｃ_１〜Ｃ_６）アルキル、Ｒ^ａ１によって任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_３〜Ｃ_６シクロアルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^ｂによって任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_１〜Ｃ_６アルコキシ、フェニル、（Ｚ）_ｍによって置換されたフェニル、ピリジン−２−イル、（Ｚ）_ｎによって置換されたピリジン−２−イル、ピリジン−３−イル、（Ｚ）_ｎによって置換されたピリジン−３−イル、ピリジン−４−イル、（Ｚ）_ｎによって置換されたピリジン−４−イル、チオフェン−２−イル、（Ｚ）_ｐによって置換されたチオフェン−２−イル、チオフェン−３−イル、（Ｚ）_ｐによって置換されたチオフェン−３−イル、チアゾール−２−イル、（Ｚ）_ｒによって置換されたチアゾール−２−イル、チアゾール−４−イル、（Ｚ）_ｒによって置換されたチアゾール−４−イル、チアゾール−５−イル、（Ｚ）_ｒによって置換されたチアゾール−５−イル、ナフタレン−１−イル、（Ｚ）_ｑによって置換されたナフタレン−１−イル、ナフタレン−２−イル又は（Ｚ）_ｑによって置換されたナフタレン−２−イルを表し、
Ｒ^２は、水素原子、ハロゲン原子、ニトロ、シアノ、Ｃ_１〜Ｃ_６アルキル、ハロ（Ｃ_１〜Ｃ_６）アルキル、Ｒ^ｂ１によって任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_３〜Ｃ_６シクロアルキル、Ｃ_２〜Ｃ_６アルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｃ_１〜Ｃ_６アルコキシ、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_１〜Ｃ_６アルキルカルボニル、Ｃ_１〜Ｃ_６アルコキシカルボニル、フェニル又は（Ｙ^１）_ｔ１によって置換されたフェニルを表し、
ｔ１が２、３、４又は５の整数を表すとき、各々のＹ^１は互いに同一であっても又は互いに異なっていてもよく、
Ｒ^３は、水素原子、ハロゲン原子、ニトロ、シアノ、Ｃ_１〜Ｃ_６アルキル、Ｃ_３〜Ｃ_６シクロアルキル、ハロ（Ｃ_１〜Ｃ_６）アルキル、Ｒ^ａよって任意に置換された（Ｃ_１〜Ｃ_６）アルキル、ハロ（Ｃ_３〜Ｃ_６）シクロアルキル、Ｒ^ｂによって任意に置換された（Ｃ_３〜Ｃ_６）シクロアルキル、Ｃ_２〜Ｃ_６アルケニル、ハロ（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_２〜Ｃ_６アルキニル、ハロ（Ｃ_２〜Ｃ_６）アルキニル、Ｃ_１〜Ｃ_６アルコキシ、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_１〜Ｃ_６アルキルカルボニル、Ｃ_１〜Ｃ_６アルコキシカルボニル、−Ｃ（＝ＮＯＲ^ｃ）Ｃ（＝ＮＯＲ^ｃ１）Ｒ^ｄ、フェニル、（Ｙ^２）_ｔ２によって置換されたフェニル、ピリジン−２−イル、ピリジン−３−イル、ピリジン−４−イル、オキセタン−２−イル又はテトラヒドロフラン−２−イルを表し、
ｔ２が２、３、４又は５の整数を表すとき、各々のＹ^２は互いに同一であっても又は互いに異なっていてもよく、
Ｒ^４及びＲ^５は、互いに独立して、水素原子、ハロゲン原子、Ｃ_１〜Ｃ_６アルキル、ハロ（Ｃ_１〜Ｃ_６）アルキル、Ｃ_１〜Ｃ_６アルコキシ又はＣ_１〜Ｃ_６アルキルチオを表すか、或いは、Ｒ^４とＲ^５とが一緒になってＣ_２〜Ｃ_５アルキレン鎖を形成することにより、Ｒ^４及びＲ^５が結合する炭素原子と共に３〜６員環を形成することを表し、
Ｒ^６、Ｒ^７、Ｒ^８及びＲ^９は、互いに独立して、水素原子、ハロゲン原子、ニトロ、シアノ、Ｃ_１〜Ｃ_６アルキル、ハロ（Ｃ_１〜Ｃ_６）アルキル、Ｒ^ｂ２によって任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_３〜Ｃ_６シクロアルキル、ハロ（Ｃ_３〜Ｃ_６）シクロアルキル、Ｃ_２〜Ｃ_６アルケニル、ハロ（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_２〜Ｃ_６アルキニル、ハロ（Ｃ_２〜Ｃ_６）アルキニル、Ｃ_１〜Ｃ_６アルコキシ、ハロ（Ｃ_１〜Ｃ_６）アルコキシ、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_１〜Ｃ_６アルキルスルフィニル又はＣ_１〜Ｃ_６アルキルスルホニルを表し、
Ｒ^１０は、水素原子、Ｃ_１〜Ｃ_６アルキル、ハロ（Ｃ_１〜Ｃ_６）アルキル、Ｒ^ｂ３によって任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_２〜Ｃ_６アルケニル又はＣ_２〜Ｃ_６アルキニルを表し、
Ｚは、ハロゲン原子、ニトロ、シアノ、ホルミル、ヒドロキシ、カルボキシ、メルカプト、アミノ、Ｃ_１〜Ｃ_６アルキル、ハロ（Ｃ_１〜Ｃ_６）アルキル、Ｒ^ｂ４によって任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_３〜Ｃ_６シクロアルキル、ハロ（Ｃ_３〜Ｃ_６）シクロアルキル、Ｃ_２〜Ｃ_６アルケニル、ハロ（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_１〜Ｃ_６アルコキシ、ハロ（Ｃ_１〜Ｃ_６）アルコキシ、Ｒ^ｂ４によって任意に置換された（Ｃ_１〜Ｃ_６）アルコキシ、Ｃ_３〜Ｃ_６シクロアルコキシ、Ｃ_２〜Ｃ_６アルケニルオキシ、ハロ（Ｃ_２〜Ｃ_６）アルケニルオキシ、Ｃ_２〜Ｃ_６アルキニルオキシ、ハロ（Ｃ_２〜Ｃ_６）アルキニルオキシ、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_２〜Ｃ_６アルケニルチオ、Ｃ_２〜Ｃ_６アルキニルチオ、ハロ（Ｃ_１〜Ｃ_６）アルキルチオ、Ｃ_１〜Ｃ_６アルキルスルフィニル、Ｃ_２〜Ｃ_６アルケニルスルフィニル、Ｃ_２〜Ｃ_６アルキニルスルフィニル、ハロ（Ｃ_１〜Ｃ_６）アルキルスルフィニル、Ｃ_１〜Ｃ_６アルキルスルホニル、Ｃ_２〜Ｃ_６アルケニルスルホニル、Ｃ_２〜Ｃ_６アルキニルスルホニル、ハロ（Ｃ_１〜Ｃ_６）アルキルスルホニル、Ｃ_１〜Ｃ_６アルキルアミノ、ジ（Ｃ_１〜Ｃ_６）アルキルアミノ、Ｃ_１〜Ｃ_６アルキルカルボニル、ハロ（Ｃ_１〜Ｃ_６）アルキルカルボニル、Ｃ_１〜Ｃ_６アルコキシカルボニル、Ｃ_１〜Ｃ_６アルキルアミノカルボニル、ジ（Ｃ_１〜Ｃ_６）アルキルアミノカルボニル、Ｃ_１〜Ｃ_６アルコキシ（Ｃ_１〜Ｃ_６）アルキル、Ｃ_１〜Ｃ_６アルコキシ（Ｃ_１〜Ｃ_６）アルコキシ、−Ｃ（＝ＮＯＲ^ｃ）Ｒ^ｄ、−Ｃ≡ＣＲ^ｅ、フェニル、（Ｚ^１）_ｍ１によって置換されたフェニル、フェノキシ又は（Ｚ^１）_ｍ１によって置換されたフェノキシを表し、
ｍが２、３、４若しくは５の整数を表すか、ｎが２、３若しくは４の整数を表すか、ｐが２若しくは３の整数を表すか、ｑが２、３、４、５、６若しくは７の整数を表すか、又はｒが２の整数を表すとき、各々のＺは互いに同一であっても又は互いに異なっていてもよく、
ｍ１が２、３、４又は５の整数を表すとき、各々のＺ^１は互いに同一であっても又は互いに異なっていてもよく、
Ｚ^１、Ｚ^２、Ｚ^３、Ｚ^４、Ｚ^５、Ｙ^１及びＹ^２は、互いに独立して、ハロゲン原子、Ｃ_１〜Ｃ_６アルキル又はＣ_１〜Ｃ_６アルコキシを表し、
Ｒ^ａは、ニトロ、シアノ、ヒドロキシ、Ｃ_３〜Ｃ_６シクロアルキル、Ｃ_１〜Ｃ_６アルコキシ、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_１〜Ｃ_６アルキルスルフィニル、Ｃ_１〜Ｃ_６アルキルスルホニル、Ｃ_１〜Ｃ_６アルキルカルボニルオキシ、フェニル又は（Ｚ）_ｍによって置換されたフェニルを表し、
Ｒ^ａ１は、フェニル、（Ｚ）_ｍによって置換されたフェニル、フェノキシ又は（Ｚ）_ｍによって置換されたフェノキシを表し、
Ｒ^ｂは、フェニル、（Ｚ）_ｍによって置換されたフェニル、ピリジン−２−イル、（Ｚ）_ｎによって置換されたピリジン−２−イル、ピリジン−３−イル、（Ｚ）_ｎによって置換されたピリジン−３−イル、ピリジン−４−イル又は（Ｚ）_ｎによって置換されたピリジン−４−イルを表し、
Ｒ^ｂ１は、ヒドロキシ、Ｃ_３〜Ｃ_６シクロアルキル、ハロ（Ｃ_１〜Ｃ_６）アルキル、Ｃ_１〜Ｃ_６アルコキシ、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_１〜Ｃ_６アルキルスルフィニル、Ｃ_１〜Ｃ_６アルキルスルホニル、Ｃ_１〜Ｃ_６アルキルカルボニルオキシ、フェニル又は（Ｚ^２）_ｍ２によって置換されたフェニルを表し、
ｍ２が２、３、４又は５の整数を表すとき、各々のＺ^２は互いに同一であっても又は互いに異なっていてもよく、
Ｒ^ｂ２は、ヒドロキシ、Ｃ_３〜Ｃ_６シクロアルキル、ハロ（Ｃ_１〜Ｃ_６）アルキル、Ｃ_１〜Ｃ_６アルコキシ、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_１〜Ｃ_６アルキルスルフィニル、Ｃ_１〜Ｃ_６アルキルスルホニル、Ｃ_１〜Ｃ_６アルキルカルボニルオキシ、フェニル又は（Ｚ^３）_ｍ３によって置換されたフェニルを表し、
ｍ３が２、３、４又は５の整数を表すとき、各々のＺ^３は互いに同一であっても又は互いに異なっていてもよく、
Ｒ^ｂ３は、ヒドロキシ、Ｃ_３〜Ｃ_６シクロアルキル、ハロ（Ｃ_１〜Ｃ_６）アルキル、Ｃ_１〜Ｃ_６アルコキシ、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_１〜Ｃ_６アルキルスルフィニル、Ｃ_１〜Ｃ_６アルキルスルホニル、Ｃ_１〜Ｃ_６アルキルカルボニルオキシ、フェニル又は（Ｚ^４）_ｍ４によって置換されたフェニルを表し、
ｍ４が２、３、４又は５の整数を表すとき、各々のＺ^４は互いに同一であっても又は互いに異なっていてもよく、
Ｒ^ｂ４は、ヒドロキシ、Ｃ_３〜Ｃ_６シクロアルキル、ハロ（Ｃ_１〜Ｃ_６）アルキル、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_１〜Ｃ_６アルキルスルフィニル、Ｃ_１〜Ｃ_６アルキルスルホニル、Ｃ_１〜Ｃ_６アルキルカルボニルオキシ、フェニル又は（Ｚ^５）_ｍ５によって置換されたフェニルを表し、
ｍ５が２、３、４又は５の整数を表すとき、各々のＺ^５は互いに同一であっても又は互いに異なっていてもよく、
Ｒ^ｃ、Ｒ^ｃ１及びＲ^ｄは、互いに独立して、水素原子又はＣ_１〜Ｃ_６アルキルを表し、
Ｒ^ｅは、水素原子、ハロゲン原子、Ｃ_１〜Ｃ_６アルキル、Ｃ_３〜Ｃ_６シクロアルキル又はトリ（Ｃ_１〜Ｃ_６）アルキルシリルを表し、
ｐは、１、２又は３の整数を表し、
ｑは、１、２、３、４、５、６又は７の整数を表し、
ｒは、１又は２の整数を表し、
ｍ、ｍ１、ｍ２、ｍ３、ｍ４、ｍ５、ｔ１及びｔ２は、互いに独立して、１、２、３、４又は５の整数を表し、
ｎは、１、２、３又は４の整数を表す。］で表されるアシルヒドラゾン誘導体若しくはその塩又はそれらのＮ−オキシド。 [Wherein W represents an oxygen atom or a sulfur atom,
A represents an oxygen atom or a sulfur atom,
R ¹ _is, C 1 -C ₆ alkyl, halo _(C 1 ~C ₆₎ ^alkyl, optionally substituted by ^{R a1} _(C 1 ~C ₆₎ _alkyl, C 3 -C ₆ _cycloalkyl, C 2 -C ₆ alkenyl, (C ₂ -C ₆ ) alkenyl optionally substituted by R ^b , C ₁ -C ₆ alkoxy, phenyl, phenyl substituted by (Z) _m , pyridin-2-yl, (Z) _n Substituted pyridin-2-yl, pyridin-3-yl, pyridin-3-yl substituted by (Z) _n , pyridin-4-yl, pyridin-4-yl substituted by (Z) _n , thiophene 2-yl, _(Z) is replaced by _p thiophene-2-yl, thiophen-3-yl, _(Z) thiophene was replaced by _p-3-yl, thiazol-2-yl, (Z replaced by _r thiazol-2-yl, thiazol-4-yl, _(Z) is replaced by _r thiazol-4-yl, thiazol-5-yl, _(Z) thiazol-5-yl which is substituted by _r , Naphthalen-1-yl, naphthalen-1-yl substituted by (Z) _q , naphthalen-2-yl or naphthalen-2-yl substituted by (Z) _q ,
R ² represents a hydrogen atom, a halogen atom, nitro, _cyano, C 1 -C ₆ alkyl, halo _(C 1 ~C ₆₎ ^alkyl, optionally substituted by ^{R b1} _(C 1 ~C ₆₎ alkyl, _{C 3} -C ₆ _cycloalkyl, C 2 -C ₆ _alkenyl, C 2 -C ₆ _alkynyl, C 1 -C ₆ _alkoxy, C 1 -C ₆ _alkylthio, C 1 -C ₆ _{alkylcarbonyl,} C 1 -C ₆ alkoxycarbonyl, Represents phenyl or phenyl substituted by (Y ¹ ) _t1 ;
when t1 represents an integer of 2, 3, 4 or 5, each Y ¹ may be the same as or different from each other;
R ³ is hydrogen atom, halogen atom, nitro, cyano, C ₁ -C ₆ alkyl, C ₃ -C ₆ cycloalkyl, halo (C ₁ -C ₆ ) alkyl, R ^a optionally substituted (C ₁ -C ₆₎ alkyl, halo _(C 3 ~C ₆₎ cycloalkyl, optionally substituted by ^{R b} _(C 3 ~C ₆₎ _cycloalkyl, C 2 -C ₆ alkenyl, halo _{_(C} 2 _~C 6) _alkenyl, C 2 -C ₆ alkynyl, halo _(C 2 ~C ₆₎ _alkynyl, C 1 -C ₆ _alkoxy, C 1 -C ₆ _alkylthio, C 1 -C ₆ _{alkylcarbonyl,} C 1 -C ₆ alkoxycarbonyl, - ^{C (= NOR c) C (} = NOR c1) R d, ^phenyl, (Y ₂₎ phenyl substituted by _t2, pyridin-2-yl, pyridin-3-yl, pyridin-4-yl Represent oxetane-2-yl or tetrahydrofuran-2-yl,
when t2 represents an integer of 2, 3, 4 or 5, each Y ² may be the same as or different from each other;
R ⁴ and R ⁵ each independently represent a hydrogen atom, a halogen atom, C ₁ -C ₆ alkyl, halo (C ₁ -C ₆ ) alkyl, C ₁ -C ₆ alkoxy or C ₁ -C ₆ alkylthio. Or R ⁴ and R ⁵ together form a C _{2 to} C ₅ alkylene chain to form a 3 to 6 membered ring with the carbon atom to which R ⁴ and R ⁵ are bonded. ,
R ⁶ , R ⁷ , R ⁸ and R ⁹ are independently of one another optionally selected from a hydrogen atom, halogen atom, nitro, cyano, C ₁ -C ₆ alkyl, halo (C ₁ -C ₆ ) alkyl, R ^b2 Substituted (C ₁ -C ₆ ) alkyl, C ₃ -C ₆ cycloalkyl, halo (C ₃ -C ₆ ) cycloalkyl, C ₂ -C ₆ alkenyl, halo (C ₂ -C ₆ ) alkenyl, C ₂ -C ₆ alkynyl, halo _(C 2 ~C ₆₎ _alkynyl, C 1 -C ₆ alkoxy, halo _(C 1 ~C ₆₎ _alkoxy, C 1 -C ₆ _alkylthio, C 1 -C ₆ alkylsulfinyl or _C 1 ~ It represents C ₆ alkylsulfonyl,
R ¹⁰ is a hydrogen atom, C ₁ -C ₆ alkyl, halo (C ₁ -C ₆ ) alkyl, (C ₁ -C ₆ ) alkyl, C ₂ -C ₆ alkenyl, or C ₂ optionally substituted with R ^b3 . ~C ₆ alkynyl,
Z is a halogen atom, nitro, cyano, formyl, hydroxy, carboxy, mercapto, _amino, C 1 -C ₆ alkyl, halo _(C 1 ~C ₆₎ ^alkyl, optionally substituted by ^{R b4} _(C 1 ~C ₆₎ _alkyl, C 3 -C ₆ cycloalkyl, halo _(C 3 -C ₆₎ _cycloalkyl, C 2 -C ₆ alkenyl, halo _(C 2 -C ₆₎ _alkenyl, C 1 -C ₆ alkoxy, halo (C ₁ -C ₆₎ ^alkoxy, optionally substituted by ^{R b4} _(C 1 ~C ₆₎ _alkoxy, C 3 -C ₆ _cycloalkoxy, C 2 -C ₆ alkenyloxy, halo _(C 2 ~C ₆₎ alkenyloxy , _C 2 -C ₆ alkynyloxy, halo _(C 2 ~C ₆₎ _alkynyloxy, C 1 -C ₆ _alkylthio, C 2 -C ₆ _{alkenylthio, C} 2 ~ ₆ alkynylthio, halo _(C 1 -C ₆₎ _alkylthio, C 1 -C ₆ _{alkylsulfinyl,} C 2 -C ₆ _{alkenylsulfinyl,} C 2 -C ₆ alkynylsulfinyl, halo _(C 1 -C ₆₎ alkylsulfinyl, C ₁ -C ₆ _{alkylsulfonyl,} C 2 -C ₆ _{alkenylsulfonyl,} C 2 -C ₆ alkynylsulfonyl, halo _(C 1 ~C ₆₎ _{alkylsulfonyl,} C 1 -C ₆ alkylamino, di _{_(C} 1 ~C 6) _alkylamino, C 1 -C ₆ alkylcarbonyl, halo _(C 1 ~C ₆₎ _{alkylcarbonyl,} C 1 -C ₆ _{alkoxycarbonyl,} C 1 -C ₆ alkylaminocarbonyl, di _(C 1 ~C ₆₎ alkylaminocarbonyl , _C 1 -C ₆ alkoxy _(C 1 ~C ₆₎ _alkyl, C 1 -C ₆ alkoxy _(C 1 ~C ₆₎ ^{^{alkoxy, -C (= NOR c) R}} d, -C≡CR e, ^phenyl, phenoxy which is substituted by the (Z ₁₎ phenyl substituted by _m1, phenoxy or ^(Z _{1) m1} Represents
m represents an integer of 2, 3, 4 or 5, n represents an integer of 2, 3 or 4, p represents an integer of 2 or 3, q is 2, 3, 4, 5, 6 Or when R represents an integer of 7, or when r represents an integer of 2, each Z may be the same as or different from each other;
when m1 represents an integer of 2, 3, 4 or 5, each Z ¹ may be the same as or different from each other;
Z ¹ , Z ² , Z ³ , Z ⁴ , Z ⁵ , Y ¹ and Y ² each independently represent a halogen atom, C ₁ -C ₆ alkyl or C ₁ -C ₆ alkoxy,
R ^a is nitro, cyano, hydroxy, C ₃ -C ₆ cycloalkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ alkylsulfonyl, C ₁ -C ₆ alkylcarbonyloxy, phenyl substituted by phenyl or _{(Z) m,}
R ^a1 represents phenyl, phenoxy which is substituted by phenyl which is substituted, phenoxy or _{(Z) m} by _{(Z) m,}
^Rb was substituted by phenyl, phenyl substituted by (Z) _m , pyridin-2-yl, pyridin-2-yl substituted by (Z) _n , pyridin-3-yl, (Z) _n Represents pyridin-4-yl substituted by pyridin-3-yl, pyridin-4-yl or (Z) _n ;
R ^b1 is hydroxy, C ₃ -C ₆ cycloalkyl, halo (C ₁ -C ₆ ) alkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ _{alkylsulfonyl,} C 1 -C ₆ alkylcarbonyloxy, phenyl substituted by phenyl or ^(Z _{2) m @ 2,}
when m2 represents an integer of 2, 3, 4 or 5, each Z ² may be the same as or different from each other;
R ^b2 is hydroxy, C ₃ -C ₆ cycloalkyl, halo (C ₁ -C ₆ ) alkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ alkylsulfonyl, C ₁ -C ₆ alkylcarbonyloxy, phenyl or phenyl substituted by (Z ³ ) _m3
when m3 represents an integer of 2, 3, 4 or 5, each Z ³ may be the same as or different from each other;
R ^b3 is hydroxy, C ₃ -C ₆ cycloalkyl, halo (C ₁ -C ₆ ) alkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ _{alkylsulfonyl,} C 1 -C ₆ alkylcarbonyloxy, phenyl substituted by phenyl or ^(Z _{4) m4,}
when m4 represents an integer of 2, 3, 4 or 5, each Z ⁴ may be the same as or different from each other;
R ^b4 is hydroxy, C ₃ -C ₆ cycloalkyl, halo (C ₁ -C ₆ ) alkyl, C ₁ -C ₆ alkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ alkylsulfonyl, C _1- C ₆ alkylcarbonyloxy, phenyl or phenyl substituted by (Z ⁵ ) _m5
when m5 represents an integer of 2, 3, 4 or 5, each Z ⁵ may be the same as or different from each other;
R ^c , R ^c1 and R ^d each independently represent a hydrogen atom or C ₁ -C ₆ alkyl;
R ^e represents a hydrogen atom, a halogen atom, C ₁ -C ₆ alkyl, C ₃ -C ₆ cycloalkyl or tri (C ₁ -C ₆ ) alkylsilyl;
p represents an integer of 1, 2 or 3,
q represents an integer of 1, 2, 3, 4, 5, 6 or 7,
r represents an integer of 1 or 2,
m, m1, m2, m3, m4, m5, t1 and t2 each independently represent an integer of 1, 2, 3, 4 or 5;
n represents an integer of 1, 2, 3 or 4. ] The acyl hydrazone derivative represented by these, its salt, or those N-oxides.

〔２〕
Ｗは、酸素原子を表し、
Ａは、酸素原子を表し、
Ｒ^１は、Ｃ_１〜Ｃ_６アルキル、Ｒ^ａ１によって任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_３〜Ｃ_６シクロアルキル、Ｒ^bによって任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、フェニル、（Ｚ）_ｍによって置換されたフェニル、ピリジン−２−イル、（Ｚ）_ｎによって置換されたピリジン−２−イル、ピリジン−３−イル、（Ｚ）_ｎによって置換されたピリジン−３−イル、ピリジン−４−イル、（Ｚ）_ｎによって置換されたピリジン−４−イル、チオフェン−２−イル、（Ｚ）_ｐによって置換されたチオフェン−２−イル、チオフェン−３−イル、（Ｚ）_ｐによって置換されたチオフェン−３−イル、チアゾール−２−イル、（Ｚ）_ｒによって置換されたチアゾール−２−イル、（Ｚ）_ｒによって置換されたチアゾール−４−イル、チアゾール−５−イル、ナフタレン−１−イル又はナフタレン−２−イルを表し、
Ｒ^２は、水素原子、Ｃ_１〜Ｃ_６アルキル、ハロ（Ｃ_１〜Ｃ_６）アルキル、Ｒ^ｂ１によって任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_３〜Ｃ_６シクロアルキル、Ｃ_１〜Ｃ_６アルコキシ又はフェニルを表し、
Ｒ^３は、水素原子、Ｃ_１〜Ｃ_６アルキル、Ｃ_３〜Ｃ_６シクロアルキル、ハロ（Ｃ_１〜Ｃ_６）アルキル、Ｒ^aによって任意に置換された（Ｃ_１〜Ｃ_６）アルキル、ハロ（Ｃ_３〜Ｃ_６）シクロアルキル、Ｃ_２〜Ｃ_６アルケニル、Ｃ_１〜Ｃ_６アルコキシ、Ｃ_１〜Ｃ_６アルコキシカルボニル、−Ｃ（＝ＮＯＲ^ｃ）Ｃ（＝ＮＯＲ^ｃ１）Ｒ^ｄ、フェニル、ピリジン−２−イル、ピリジン−３−イル又はピリジン−４−イルを表し、
Ｒ^４及びＲ^５は、水素原子を表し、
Ｒ^６は、水素原子、ハロゲン原子、シアノ、Ｃ_１〜Ｃ_６アルキル、ハロ（Ｃ_１〜Ｃ_６）アルキル、Ｃ_２〜Ｃ_６アルケニル、Ｃ_１〜Ｃ_６アルコキシ、Ｃ_１〜Ｃ_６アルキルチオ又はＣ_１〜Ｃ_６アルキルスルフィニルを表し、
Ｒ^１０は、Ｃ_１〜Ｃ_６アルキルを表し、
Ｚは、ハロゲン原子、ニトロ、シアノ、ヒドロキシ、カルボキシ、Ｃ_１〜Ｃ_６アルキル、ハロ（Ｃ_１〜Ｃ_６）アルキル、Ｃ_３〜Ｃ_６シクロアルキル、Ｃ_２〜Ｃ_６アルケニル、Ｃ_１〜Ｃ_６アルコキシ、ハロ（Ｃ_１〜Ｃ_６）アルコキシ、Ｒ^ｂ４によって任意に置換された（Ｃ_１〜Ｃ_６）アルコキシ、Ｃ_２〜Ｃ_６アルケニルオキシ、Ｃ_２〜Ｃ_６アルキニルオキシ、Ｃ_１〜Ｃ_６アルキルチオ、ハロ（Ｃ_１〜Ｃ_６）アルキルチオ、Ｃ_１〜Ｃ_６アルキルスルフィニル、Ｃ_１〜Ｃ_６アルキルスルホニル、ジ（Ｃ_１〜Ｃ_６）アルキルアミノ、Ｃ_１〜Ｃ_６アルキルカルボニル、Ｃ_１〜Ｃ_６アルコキシカルボニル、Ｃ_１〜Ｃ_６アルキルアミノカルボニル、Ｃ_１〜Ｃ_６アルコキシ（Ｃ_１〜Ｃ_６）アルコキシ、−Ｃ（＝ＮＯＲ^ｃ）Ｒ^ｄ、−Ｃ≡ＣＲ^ｅ、フェニル、（Ｚ^１）_ｍ１によって置換されたフェニル又は（Ｚ^１）_ｍ１によって置換されたフェノキシを表し、
Ｒ^ａは、ヒドロキシ、Ｃ_３〜Ｃ_６シクロアルキル、Ｃ_１〜Ｃ_６アルコキシ、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_１〜Ｃ_６アルキルスルフィニル、Ｃ_１〜Ｃ_６アルキルカルボニルオキシ又は（Ｚ）_ｍによって置換されたフェニルを表し、
Ｒ^ａ１は、（Ｚ）_ｍによって置換されたフェニル又はフェノキシを表し、
Ｒ^ｂは、（Ｚ）_ｍによって置換されたフェニル又は（Ｚ）_ｎによって置換されたピリジン−２−イルを表し、
Ｒ^ｂ１は、Ｃ_１〜Ｃ_６アルコキシを表し、
Ｒ^ｂ４は、フェニルを表し、
Ｒ^ｃ、Ｒ^ｃ１及びＲ^ｄは、互いに独立して、Ｃ_１〜Ｃ_６アルキルを表す、上記〔１〕記載のアシルヒドラゾン誘導体若しくはその塩又はそれらのＮ−オキシド。 [2]
W represents an oxygen atom,
A represents an oxygen atom,
R ¹ is C ₁ -C ₆ alkyl, (C ₁ -C ₆ ) alkyl optionally substituted by R ^a1 , C ₃ -C ₆ cycloalkyl, optionally substituted by R ^b (C ₂ -C ₆ ) Alkenyl, phenyl, phenyl substituted by (Z) _m , pyridin-2-yl, pyridin-2-yl substituted by (Z) _n , pyridin-3-yl, pyridine substituted by (Z) _n -3-yl, pyridin-4-yl, (Z) _n- substituted pyridin-4-yl, thiophen-2-yl, (Z) _p- substituted thiophen-2-yl, thiophen-3-yl , _(Z) thiophene was replaced by _p-3-yl, thiazol-2-yl, _(Z) is replaced by _r thiazol-2-yl, Chiazo substituted by _{(Z) r} It represents 4-yl, thiazol-5-yl, naphthalene-1-yl or naphthalen-2-yl,
R ² is a hydrogen _atom, C 1 -C ₆ alkyl, halo _(C 1 ~C ₆₎ ^alkyl, optionally substituted by ^{R b1} _(C 1 ~C ₆₎ _alkyl, C 3 -C ₆ cycloalkyl alkyl, C ₁ -C ₆ alkoxy or phenyl,
R ³ represents a hydrogen _atom, C 1 -C ₆ _alkyl, C 3 -C ₆ cycloalkyl, halo _(C 1 ~C ₆₎ alkyl, optionally substituted by R ^a _(C 1 ~C ₆₎ alkyl, halo (C ₃ -C ₆ ) cycloalkyl, C ₂ -C ₆ alkenyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ alkoxycarbonyl, -C (= NOR ^c ) C (= NOR ^{c 1} ) R ^d , phenyl, Represents pyridin-2-yl, pyridin-3-yl or pyridin-4-yl,
R ⁴ and R ⁵ represent a hydrogen atom,
R ⁶ is a hydrogen atom, halogen atom, cyano, C ₁ -C ₆ alkyl, halo (C ₁ -C ₆ ) alkyl, C ₂ -C ₆ alkenyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ alkylthio or C ₁ -C ₆ alkyl sulfinyl,
R ¹⁰ represents C ₁ -C ₆ alkyl,
Z is a halogen atom, nitro, cyano, hydroxy, _carboxy, C 1 -C ₆ alkyl, halo _(C 1 ~C ₆₎ _alkyl, C 3 -C ₆ _cycloalkyl, C 2 -C ₆ _alkenyl, C 1 -C ₆ alkoxy, halo _(C 1 -C ₆₎ ^alkoxy, optionally substituted by ^{R b4} _(C 1 ~C ₆₎ _alkoxy, C 2 -C ₆ _alkenyloxy, C 2 -C ₆ _alkynyloxy, C 1 -C ₆ alkylthio, halo (C ₁ -C ₆ ) alkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ alkylsulfonyl, di (C ₁ -C ₆ ) alkylamino, C ₁ -C ₆ alkylcarbonyl, C ₁ -C ₆ _{alkoxycarbonyl,} C 1 -C ₆ _{alkylaminocarbonyl,} C 1 -C ₆ alkoxy _(C 1 ~C ₆₎ alkoxy, -C (= N Represents ^{^{^{OR c) R d, -C≡CR e}}} , ^phenyl, phenoxy which is substituted by the (Z ₁₎ phenyl or substituted by _{_m1} ^(Z ₁₎ _m1,
R ^a is hydroxy, C ₃ -C ₆ cycloalkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ alkylcarbonyloxy or (Z) _m Represents substituted phenyl,
R ^a1 represents phenyl or phenoxy substituted by (Z) _m ,
R ^b represents phenyl substituted by (Z) _m or pyridin-2-yl substituted by (Z) _n ;
R ^b1 represents C ₁ -C ₆ alkoxy;
R ^b4 represents phenyl,
R ^c , R ^c1 and R ^d each independently represent C ₁ -C ₆ alkyl, the acyl hydrazone derivative of the above-mentioned [1] or a salt thereof, or an N-oxide thereof.

〔３〕
Ｒ^１は、Ｃ_１〜Ｃ_６アルキル、Ｒ^ｂによって任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、フェニル、（Ｚ）_ｍによって置換されたフェニル、（Ｚ）_ｎによって置換されたピリジン−２−イル、（Ｚ）_ｐによって置換されたチオフェン−２−イル又は（Ｚ）_ｐによって置換されたチオフェン−３−イルを表し、
Ｒ^２は、Ｃ_１〜Ｃ_６アルキル又はフェニルを表し、
Ｒ^３は、水素原子、Ｃ_１〜Ｃ_６アルキル、Ｃ_３〜Ｃ_６シクロアルキル、ハロ（Ｃ_１〜Ｃ_６）アルキル、Ｒ^ａによって任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_１〜Ｃ_６アルコキシ又はＣ_１〜Ｃ_６アルコキシカルボニルを表し、
Ｒ^６は、水素原子、ハロゲン原子、Ｃ_１〜Ｃ_６アルキル、Ｃ_１〜Ｃ_６アルコキシを表し、
Ｒ^７及びＲ^８は、水素原子を表し、
Ｒ^９は、水素原子又はハロゲン原子を表し、
Ｚは、ハロゲン原子、シアノ、Ｃ_１〜Ｃ_６アルキル、ハロ（Ｃ_１〜Ｃ_６）アルキル、Ｃ_１〜Ｃ_６アルコキシ、ハロ（Ｃ_１〜Ｃ_６）アルコキシ、Ｒ^ｂ４によって任意に置換された（Ｃ_１〜Ｃ_６）アルコキシ、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_１〜Ｃ_６アルキルカルボニル、Ｃ_１〜Ｃ_６アルコキシカルボニル、−Ｃ（＝ＮＯＲ^ｃ）Ｒ^ｄ又はフェニルを表し、
Ｒ^ｂは、（Ｚ）_ｍによって置換されたフェニルを表し、
Ｒ^ａは、Ｃ_１〜Ｃ_６アルコキシ、Ｃ_１〜Ｃ_６アルキルチオ又はＣ_１〜Ｃ_６アルキルカルボニルオキシを表す、上記〔２〕に記載のアシルヒドラゾン誘導体若しくはその塩又はそれらのＮ−オキシド。 [3]
R ¹ is C ₁ -C ₆ alkyl, (C ₂ -C ₆ ) alkenyl optionally substituted by R ^b , phenyl, phenyl substituted by (Z) _m , pyridine- substituted by (Z) _n 2-yl, represents a thiophene-3-yl substituted by the _(Z) thiophene was replaced by _p-2-yl or _{(Z) p,}
R ² represents C ₁ -C ₆ alkyl or phenyl,
R ³ represents a hydrogen _atom, C 1 -C ₆ _alkyl, C 3 -C ₆ cycloalkyl, halo _(C 1 ~C ₆₎ alkyl, optionally substituted by ^{R a} _(C 1 ~C ₆₎ alkyl, C Represents ₁ -C ₆ alkoxy or C ₁ -C ₆ alkoxycarbonyl,
R ⁶ represents a hydrogen atom, a halogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ alkoxy,
R ⁷ and R ⁸ represent a hydrogen atom,
R ⁹ represents a hydrogen atom or a halogen atom,
Z is optionally substituted with a halogen atom, cyano, C ₁ -C ₆ alkyl, halo (C ₁ -C ₆ ) alkyl, C ₁ -C ₆ alkoxy, halo (C ₁ -C ₆ ) alkoxy, R ^b4 _(C 1 _~C ₆₎ _-alkoxy, C 1 -C ₆ _alkylthio, C 1 -C ₆ _{alkylcarbonyl,} C 1 -C ₆ alkoxycarbonyl, -C a (= ^NOR c) ^{R d} or phenyl,
R ^b represents (Z) phenyl substituted by _m ;
R ^a _is, C 1 -C ₆ _alkoxy, C 1 -C ₆ alkylthio or _C 1 -C ₆ alkyl carbonyloxy acylhydrazone derivative or a salt thereof, or their N- oxide according to [2].

〔４〕
上記〔１〕〜〔３〕記載のアシルヒドラゾン誘導体若しくはその塩又はそれらのＮ−オキシドから選ばれる１種又は２種以上を有効成分として含有する農薬。 [4]
An agrochemical containing one or more selected from the acylhydrazone derivatives or salts thereof according to the above [1] to [3] or their N-oxides as an active ingredient.

〔５〕
上記〔１〕〜〔３〕記載のアシルヒドラゾン誘導体若しくはその塩又はそれらのＮ−オキシドから選ばれる１種又は２種以上を有効成分として含有する殺菌剤。 [5]
A fungicide containing, as an active ingredient, one or more selected from the acylhydrazone derivatives or salts thereof according to the above [1] to [3] or their N-oxides.

〔６〕
上記〔１〕〜〔３〕記載のアシルヒドラゾン誘導体若しくはその塩又はそれらのＮ−オキシドから選ばれる１種又は２種以上を有効成分として含有する農園芸用殺菌剤。 [6]
An agricultural and horticultural fungicide containing, as an active ingredient, one or more selected from the acylhydrazone derivatives according to the above [1] to [3], salts thereof, or N-oxides thereof.

〔７〕
上記〔１〕〜〔３〕のいずれかに記載のアシルヒドラゾン誘導体若しくはその塩又はそれらのＮ−オキシドから選ばれる１種又は２種以上を有効成分として含有する抗真菌剤。 [7]
The antifungal agent which contains as an active ingredient 1 type, or 2 or more types chosen from the acyl hydrazone derivative in any one of said [1]-[3], its salt, or those N-oxides.

〔８〕
上記〔１〕〜〔３〕のいずれかに記載のアシルヒドラゾン誘導体若しくはその塩又はそれらのＮ−オキシドから選ばれる１種又は２種以上を有効成分として含有する内部寄生虫防除剤。 [8]
An endoparasite control agent comprising, as an active ingredient, one or more selected from the acylhydrazone derivatives or salts thereof according to any one of the above [1] to [3] or their N-oxides.

本発明化合物は多くの病原菌に対して優れた防除活性を有し、既存の殺菌剤に対して抵抗性を獲得した病原菌に対しても十分な防除効果を発揮する。さらに、対象となる作物に薬害を生じることがなく、ホ乳類、魚類及び益虫に対してほとんど悪影響を及ぼさず、低残留性で環境に対する負荷も軽い。 The compound of the present invention has an excellent control activity against many pathogenic bacteria, and also exhibits a sufficient control effect against pathogenic bacteria that have acquired resistance to existing fungicides. Furthermore, it does not cause phytotoxicity on the target crop, has almost no adverse effect on mammals, fish and beneficial insects, has low persistence, and has a low environmental impact.

従って、本発明は有用な殺菌剤、特に農園芸用殺菌剤を提供することができる。 Therefore, the present invention can provide useful fungicides, particularly agricultural and horticultural fungicides.

本発明に包含される化合物には、置換基の種類によってはＥ−体及びＺ−体の幾何異性体が存在する場合があるが、本発明はこれらＥ−体、Ｚ−体又はＥ−体及びＺ−体を任意の割合で含む混合物を包含するものである。また、本発明に包含される化合物は、置換基同士の立体障害を原因とする制限された結合回転により、１種又は２種以上の回転異性体として存在する場合があるが、本発明は全ての回転異性体又は任意の割合で含むジアステレオマーの混合物を包含するものである。また、本発明に包含される化合物は、１個又は２個以上の不斉炭素原子の存在に起因する光学活性体が存在するが、本発明は全ての光学活性体又はラセミ体を包含する。 The compounds included in the present invention may have geometrical isomers of E-form and Z-form depending on the type of substituent, and the present invention is not limited to these E-form, Z-form or E-form. And a mixture containing the Z-form in an arbitrary ratio. In addition, the compounds included in the present invention may exist as one or more rotational isomers due to limited bond rotation caused by steric hindrance between substituents, but all of the present invention Or a mixture of diastereomers including any proportions. In addition, the compounds included in the present invention include optically active substances resulting from the presence of one or more asymmetric carbon atoms, but the present invention includes all optically active substances or racemates.

本発明に包含される化合物のうちで、常法に従って酸付加塩にすることができるものは、例えば、フッ化水素酸、塩酸、臭化水素酸、沃化水素酸等のハロゲン化水素酸の塩、硝酸、硫酸、燐酸、塩素酸、過塩素酸等の無機酸の塩、メタンスルホン酸、エタンスルホン酸、トリフルオロメタンスルホン酸、ベンゼンスルホン酸、ｐ−トルエンスルホン酸等のスルホン酸の塩、ギ酸、酢酸、プロピオン酸、トリフルオロ酢酸、フマル酸、酒石酸、蓚酸、マレイン酸、リンゴ酸、コハク酸、安息香酸、マンデル酸、アスコルビン酸、乳酸、グルコン酸、クエン酸等のカルボン酸の塩又はグルタミン酸、アスパラギン酸等のアミノ酸の塩とすることができる。 Among the compounds included in the present invention, those that can be converted into acid addition salts according to a conventional method include, for example, hydrohalic acids such as hydrofluoric acid, hydrochloric acid, hydrobromic acid, hydroiodic acid, and the like. Salts of inorganic acids such as salts, nitric acid, sulfuric acid, phosphoric acid, chloric acid, perchloric acid, salts of sulfonic acids such as methanesulfonic acid, ethanesulfonic acid, trifluoromethanesulfonic acid, benzenesulfonic acid, p-toluenesulfonic acid, Salts of carboxylic acids such as formic acid, acetic acid, propionic acid, trifluoroacetic acid, fumaric acid, tartaric acid, succinic acid, maleic acid, malic acid, succinic acid, benzoic acid, mandelic acid, ascorbic acid, lactic acid, gluconic acid, citric acid or the like A salt of an amino acid such as glutamic acid or aspartic acid can be used.

或いは、本発明に包含される化合物のうちで、常法に従って金属塩にすることができるものは、例えば、リチウム、ナトリウム、カリウムといったアルカリ金属の塩、カルシウム、バリウム、マグネシウムといったアルカリ土類金属の塩又はアルミニウムの塩とすることができる。 Alternatively, among the compounds included in the present invention, those that can be converted into a metal salt according to a conventional method include, for example, alkali metal salts such as lithium, sodium, and potassium, and alkaline earth metals such as calcium, barium, and magnesium. It can be a salt or a salt of aluminum.

本発明化合物において、Ｎ−オキシドとは、複素環基上の環を構成する窒素原子が酸化された化合物である。Ｎ−オキシドを形成しうる複素環基としては、例えば、ピリジン環又はチアゾール環が挙げられる。 In the compound of the present invention, N-oxide is a compound in which a nitrogen atom constituting a ring on a heterocyclic group is oxidized. Examples of the heterocyclic group that can form an N-oxide include a pyridine ring or a thiazole ring.

次に本明細書において示した各置換基の具体例を以下に示す。ここで、ｎ−はノルマル、ｉ−はイソ、ｓ−はセカンダリー及びｔｅｒｔ−はターシャリーを各々意味し、Ｐｈはフェニルを意味する。 Next, specific examples of each substituent shown in the present specification are shown below. Here, n- represents normal, i- represents iso, s- represents secondary, and tert- represents tertiary, and Ph represents phenyl.

本発明化合物におけるハロゲン原子としては、フッ素原子、塩素原子、臭素原子及びヨウ素原子が挙げられる。尚、本明細書中「ハロ」の表記もこれらのハロゲン原子を表す。 As a halogen atom in this invention compound, a fluorine atom, a chlorine atom, a bromine atom, and an iodine atom are mentioned. In the present specification, the notation “halo” also represents these halogen atoms.

本明細書におけるＣ_ａ〜Ｃ_ｂアルキルの表記は、炭素原子数がａ〜ｂ個よりなる直鎖状又は分岐鎖状の炭化水素基を表し、例えばメチル基、エチル基、ｎ−プロピル基、ｉ−プロピル基、ｎ−ブチル基、ｉ−ブチル基、ｓ−ブチル基、ｔｅｒｔ−ブチル基、ｎ−ペンチル基、１，１−ジメチルプロピル基、ｎ−ヘキシル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkyl in the present specification represents a linear or branched hydrocarbon group having a carbon number of _a to _b , for example, methyl group, ethyl group, n-propyl group, Specific examples include i-propyl group, n-butyl group, i-butyl group, s-butyl group, tert-butyl group, n-pentyl group, 1,1-dimethylpropyl group, n-hexyl group, and the like. Each selected range of carbon atoms is selected.

ハロ（Ｃ_ａ〜Ｃ_ｂ）アルキルの表記は、炭素原子に結合した水素原子が、ハロゲン原子によって任意に置換された、炭素原子数がａ〜ｂ個よりなる直鎖状又は分岐鎖状の炭化水素基を表し、このとき、２個以上のハロゲン原子によって置換されている場合、それらのハロゲン原子は互いに同一でも、又は互いに相異なっていてもよい。例えばフルオロメチル基、クロロメチル基、ブロモメチル基、ヨードメチル基、ジフルオロメチル基、ジクロロメチル基、トリフルオロメチル基、クロロジフルオロメチル基、トリクロロメチル基、ブロモジフルオロメチル基、２−フルオロエチル基、２−クロロエチル基、２−ブロモエチル基、２，２−ジフルオロエチル基、２，２，２−トリフルオロエチル基、２−クロロ−２，２−ジフルオロエチル基、２，２，２−トリクロロエチル基、１，１，２，２−テトラフルオロエチル基、２−クロロ−１，１，２−トリフルオロエチル基、ペンタフルオロエチル基、３，３，３−トリフルオロプロピル基、２，２，３，３，３−ペンタフルオロプロピル基、１，１，２，３，３，３−ヘキサフルオロプロピル基、ヘプタフルオロプロピル基、２，２，２−トリフルオロ−１−（トリフルオロメチル）エチル基、１，２，２，２−テトラフルオロ−１−（トリフルオロメチル）エチル基、２，２，３，３，４，４，４−ヘプタフルオロブチル基、ノナフルオロブチル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of halo (C _a -C _b ) alkyl is a linear or branched carbon atom having a carbon number of _a to _b in which a hydrogen atom bonded to a carbon atom is optionally substituted with a halogen atom Represents a hydrogen group, and when substituted by two or more halogen atoms, these halogen atoms may be the same as or different from each other; For example, fluoromethyl group, chloromethyl group, bromomethyl group, iodomethyl group, difluoromethyl group, dichloromethyl group, trifluoromethyl group, chlorodifluoromethyl group, trichloromethyl group, bromodifluoromethyl group, 2-fluoroethyl group, 2- Chloroethyl group, 2-bromoethyl group, 2,2-difluoroethyl group, 2,2,2-trifluoroethyl group, 2-chloro-2,2-difluoroethyl group, 2,2,2-trichloroethyl group, 1 , 1,2,2-tetrafluoroethyl group, 2-chloro-1,1,2-trifluoroethyl group, pentafluoroethyl group, 3,3,3-trifluoropropyl group, 2,2,3,3 , 3-pentafluoropropyl group, 1,1,2,3,3,3-hexafluoropropyl group, heptafluoropropyl group 2,2,2-trifluoro-1- (trifluoromethyl) ethyl group, 1,2,2,2-tetrafluoro-1- (trifluoromethyl) ethyl group, 2,2,3,3,4, Specific examples include 4,4-heptafluorobutyl group, nonafluorobutyl group and the like, and each is selected within the range of the number of carbon atoms designated.

Ｃ_ａ〜Ｃ_ｂシクロアルキルの表記は、炭素原子数がａ〜ｂ個よりなる環状の炭化水素基を表し、３員環から１０員環までの単環又は複合環構造を形成することが出来る。また、各々の環は指定の炭素原子数の範囲でアルキル基によって任意に置換されていてもよい。例えばシクロプロピル基、１−メチルシクロプロピル基、２−メチルシクロプロピル基、２，２−ジメチルシクロプロピル基、シクロブチル基、シクロペンチル基、シクロヘキシル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _{a to} C _b cycloalkyl represents a cyclic hydrocarbon group having _a to _b carbon atoms, and can form a monocyclic or complex ring structure having 3 to 10 members. . Each ring may be optionally substituted with an alkyl group within the range of the specified number of carbon atoms. Specific examples include cyclopropyl group, 1-methylcyclopropyl group, 2-methylcyclopropyl group, 2,2-dimethylcyclopropyl group, cyclobutyl group, cyclopentyl group, cyclohexyl group, etc. Selected in a range of numbers.

ハロ（Ｃ_ａ〜Ｃ_ｂ）シクロアルキルの表記は、炭素原子に結合した水素原子がハロゲン原子によって任意に置換された、炭素原子数がａ〜ｂ個よりなる環状の炭化水素基を表し、３員環から６員環までの単環又は複合環構造を形成することが出来る。また、各々の環は指定の炭素原子数の範囲でアルキル基によって任意に置換されていてもよく、ハロゲン原子による置換は環構造部分であっても、側鎖部分であっても、或いはそれらの両方であってもよく、さらに、２個以上のハロゲン原子によって置換されている場合、それらのハロゲン原子は互いに同一でも、または互いに相異なっていてもよい。具体例として、２，２−ジフルオロシクロプロピル基、２，２−ジクロロシクロプロピル基、２，２−ジブロモシクロプロピル基、２，２−ジフルオロ−１−メチルシクロプロピル基、２，２−ジクロロ−１−メチルシクロプロピル基、２，２−ジブロモ−１−メチルシクロプロピル基、１−トリフルオロメチルシクロプロピル基、２−トリフルオロメチルシクロプロピル基、１−トリクロロメチルシクロプロピル基、２−トリクロロメチルシクロプロピル基、２，２，３，３−テトラフルオロシクロブチル基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of halo (C _a -C _b ) cycloalkyl represents a cyclic hydrocarbon group consisting of _a to _b carbon atoms in which a hydrogen atom bonded to a carbon atom is optionally substituted with a halogen atom, 3 A monocyclic or complex ring structure from a member ring to a 6-member ring can be formed. Each ring may be optionally substituted with an alkyl group within the range of the specified number of carbon atoms, and the substitution with a halogen atom may be a ring structure part, a side chain part, They may be both, and when they are substituted by two or more halogen atoms, the halogen atoms may be the same as or different from each other. Specific examples include 2,2-difluorocyclopropyl group, 2,2-dichlorocyclopropyl group, 2,2-dibromocyclopropyl group, 2,2-difluoro-1-methylcyclopropyl group, 2,2-dichloro- 1-methylcyclopropyl group, 2,2-dibromo-1-methylcyclopropyl group, 1-trifluoromethylcyclopropyl group, 2-trifluoromethylcyclopropyl group, 1-trichloromethylcyclopropyl group, 2-trichloromethyl A cyclopropyl group, a 2,2,3,3-tetrafluorocyclobutyl group and the like can be mentioned, and each is selected within the range of the designated number of carbon atoms.

Ｃ_ａ〜Ｃ_ｂアルケニルの表記は、炭素原子数がａ〜ｂ個よりなる直鎖状又は分岐鎖状で、且つ、分子内に１個又は２個以上の二重結合を有する不飽和炭化水素基を表す。具体例として、ビニル基、１−プロペニル基、２−プロペニル基、１−メチルエテニル基、２−ブテニル基、２−メチル−２−プロペニル基、３−メチル−２−ブテニル基、１，１−ジメチル−２−プロペニル基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkenyl is an unsaturated hydrocarbon having a linear or branched chain composed of _a to _b carbon atoms and having one or more double bonds in the molecule. Represents a group. Specific examples include vinyl group, 1-propenyl group, 2-propenyl group, 1-methylethenyl group, 2-butenyl group, 2-methyl-2-propenyl group, 3-methyl-2-butenyl group, 1,1-dimethyl. -2-propenyl group and the like, and each selected within the range of the specified number of carbon atoms.

ハロ（Ｃ_ａ〜Ｃ_ｂ）アルケニルの表記は、炭素原子に結合した水素原子がハロゲン原子によって任意に置換された、炭素原子数がａ〜ｂ個よりなる直鎖状又は分岐鎖状で、且つ、分子内に１個又は２個以上の二重結合を有する不飽和炭化水素基を表す。２個以上のハロゲン原子によって置換されている場合、それらのハロゲン原子は互いに同一でも、又は互いに相異なっていてもよい。具体例として、２−フルオロビニル基、２−クロロビニル基、１，２−ジクロロビニル基、２，２−ジクロロビニル基、２，２−ジブロモビニル基、２−フルオロ−２−プロペニル基、２−クロロ−２−プロペニル基、３−クロロ−２−プロペニル基、３，３−ジフルオロ−２−プロペニル基、２，３−ジクロロ−２−プロペニル基、３，３−ジクロロ−２−プロペニル基、２，３，３−トリフルオロ−２−プロペニル基、２，３，３−トリクロロ−２−プロペニル基、１−（トリフルオロメチル）エテニル基、４，４−ジフルオロ−３−ブテニル基、３，４，４−トリフルオロ−３−ブテニル基、２，４，４，４−テトラフルオロ−２−ブテニル基、３−クロロ−４，４，４−トリフルオロ−２−ブテニル基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of halo (C _a -C _b ) alkenyl is linear or branched consisting of _a to _b carbon atoms, in which a hydrogen atom bonded to a carbon atom is optionally substituted with a halogen atom, and Represents an unsaturated hydrocarbon group having one or more double bonds in the molecule. When substituted by two or more halogen atoms, the halogen atoms may be the same as or different from each other. Specific examples include 2-fluorovinyl group, 2-chlorovinyl group, 1,2-dichlorovinyl group, 2,2-dichlorovinyl group, 2,2-dibromovinyl group, 2-fluoro-2-propenyl group, 2 -Chloro-2-propenyl group, 3-chloro-2-propenyl group, 3,3-difluoro-2-propenyl group, 2,3-dichloro-2-propenyl group, 3,3-dichloro-2-propenyl group, 2,3,3-trifluoro-2-propenyl group, 2,3,3-trichloro-2-propenyl group, 1- (trifluoromethyl) ethenyl group, 4,4-difluoro-3-butenyl group, 3, 4,4-trifluoro-3-butenyl group, 2,4,4,4-tetrafluoro-2-butenyl group, 3-chloro-4,4,4-trifluoro-2-butenyl group, etc. Each specified charcoal It may be selected from the range number of atoms.

Ｃ_ａ〜Ｃ_ｂアルキニルの表記は、炭素原子数がａ〜ｂ個よりなる直鎖状又は分岐鎖状で、且つ分子内に１個又は２個以上の三重結合を有する不飽和炭化水素基を表す。具体例として、エチニル基、１−プロピニル基、２−プロピニル基、１−ブチニル基、２−ブチニル基、３−ブチニル基、１，１−ジメチル−２−プロピニル基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkynyl refers to an unsaturated hydrocarbon group having a linear or branched chain consisting of _a to _b carbon atoms and having one or more triple bonds in the molecule. Represent. Specific examples include ethynyl group, 1-propynyl group, 2-propynyl group, 1-butynyl group, 2-butynyl group, 3-butynyl group, 1,1-dimethyl-2-propynyl group and the like. In the range of the number of carbon atoms.

ハロ（Ｃ_ａ〜Ｃ_ｂ）アルキニルの表記は、炭素原子に結合した水素原子がハロゲン原子によって任意に置換された、炭素原子数がａ〜ｂ個よりなる直鎖状又は分岐鎖状で、且つ、分子内に１個又は２個以上の三重結合を有する不飽和炭化水素基を表す。２個以上のハロゲン原子によって置換されている場合、それらのハロゲン原子は互いに同一でも、又は互いに相異なっていても良い。具体例として、２−クロロエチニル基、２−ブロモエチニル基、２−ヨードエチニル基、３−フルオロ−１−プロピニル基、３−クロロ−１−プロピニル基、３−クロロ−２−プロピニル基、３−ブロモ−１−プロピニル基、３−ブロモ−２−プロピニル基、３−ヨード−２−プロピニル基、３，３−ジフルオロ−１−プロピニル基、３，３，３−トリフルオロ−１−プロピニル基、３−ブロモ−１−ブチニル基、３−フルオロ−３−メチル−１−ブチニル基、３−クロロ−３−メチル−１−ブチニル基、３−ブロモ−３−メチル−１−ブチニル基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of halo (C _a -C _b ) alkynyl is linear or branched consisting of _a to _b carbon atoms, in which a hydrogen atom bonded to a carbon atom is optionally substituted with a halogen atom, and Represents an unsaturated hydrocarbon group having one or more triple bonds in the molecule. When substituted with two or more halogen atoms, the halogen atoms may be the same as or different from each other. Specific examples include 2-chloroethynyl group, 2-bromoethynyl group, 2-iodoethynyl group, 3-fluoro-1-propynyl group, 3-chloro-1-propynyl group, 3-chloro-2-propynyl group, 3 -Bromo-1-propynyl group, 3-bromo-2-propynyl group, 3-iodo-2-propynyl group, 3,3-difluoro-1-propynyl group, 3,3,3-trifluoro-1-propynyl group 3-bromo-1-butynyl group, 3-fluoro-3-methyl-1-butynyl group, 3-chloro-3-methyl-1-butynyl group, 3-bromo-3-methyl-1-butynyl group, etc. Each of which is selected for each specified number of carbon atoms.

Ｃ_ａ〜Ｃ_ｂアルコキシの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル−Ｏ−基を表す。具体例として、メトキシ基、エトキシ基、ｎ−プロピルオキシ基、ｉ−プロピルオキシ基、ｎ−ブチルオキシ基、ｉ−ブチルオキシ基、ｓ−ブチルオキシ基、ｔｅｒｔ−ブチルオキシ基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation C _a -C _b alkoxy represents an alkyl-O— group with the above meaning consisting of _a to _b carbon atoms. Specific examples include methoxy group, ethoxy group, n-propyloxy group, i-propyloxy group, n-butyloxy group, i-butyloxy group, s-butyloxy group, tert-butyloxy group and the like. Selected in the range of the number of carbon atoms.

ハロ（Ｃ_ａ〜Ｃ_ｂ）アルコキシの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるハロアルキル−Ｏ−基を表し、例えばジフルオロメトキシ基、トリフルオロメトキシ基、クロロジフルオロメトキシ基、ブロモジフルオロメトキシ基、２−フルオロエトキシ基、２−クロロエトキシ基、２，２，２−トリフルオロエトキシ基、１，１，２，２−テトラフルオロエトキシ基、２−クロロ−１，１，２−トリフルオロエトキシ基、１，１，２，３，３，３−ヘキサフルオロプロピルオキシ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of halo (C _a -C _b ) alkoxy represents a haloalkyl-O— group having the above-mentioned meaning consisting of _a to _b carbon atoms, such as a difluoromethoxy group, a trifluoromethoxy group, a chlorodifluoromethoxy group. Bromodifluoromethoxy group, 2-fluoroethoxy group, 2-chloroethoxy group, 2,2,2-trifluoroethoxy group, 1,1,2,2-tetrafluoroethoxy group, 2-chloro-1,1, Specific examples include 2-trifluoroethoxy group, 1,1,2,3,3,3-hexafluoropropyloxy group, and the like are selected in the range of the respective designated number of carbon atoms.

Ｃ_ａ〜Ｃ_ｂシクロアルコキシの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるシクロアルキル−Ｏ−基を表す。具体例として、シクロプロピルオキシ基、シクロブチルオキシ基、シクロペンチルオキシ基、シクロヘキシルオキシ基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b cycloalkoxy represents a cycloalkyl-O— group having the above meaning consisting of _a to _b carbon atoms. Specific examples include a cyclopropyloxy group, a cyclobutyloxy group, a cyclopentyloxy group, a cyclohexyloxy group, and the like, and each is selected within the range of the designated number of carbon atoms.

Ｃ_ａ〜Ｃ_ｂアルケニルオキシの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルケニル−Ｏ−基を表す。具体例として、２−プロペニルオキシ基、２−ブテニルオキシ基、１−メチル−２−プロペニルオキシ基、２−メチル−２−プロペニルオキシ基、３−メチル−２−ブテニルオキシ基、１，１−ジメチル−２−プロペニルオキシ基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkenyloxy represents an alkenyl-O— group having the above meaning consisting of _a to _b carbon atoms. Specific examples include 2-propenyloxy group, 2-butenyloxy group, 1-methyl-2-propenyloxy group, 2-methyl-2-propenyloxy group, 3-methyl-2-butenyloxy group, 1,1-dimethyl- 2-propenyloxy group and the like can be mentioned, and each is selected within the range of the designated number of carbon atoms.

ハロ（Ｃ_ａ〜Ｃ_ｂ）アルケニルオキシの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるハロアルケニル−Ｏ−基を表す。具体例として、２−フルオロ−２−プロペニルオキシ基、２−クロロ−２−プロペニルオキシ基、３−クロロ−２−プロペニルオキシ基、３，３−ジフルオロ−２−プロペニルオキシ基、２，３−ジクロロ−２−プロペニルオキシ基、３，３−ジクロロ−２−プロペニルオキシ基、２，３，３−トリフルオロ−２−プロペニルオキシ基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation halo (C _a -C _b ) alkenyloxy represents a haloalkenyl-O— group with the above meaning consisting of _a to _b carbon atoms. Specific examples include 2-fluoro-2-propenyloxy group, 2-chloro-2-propenyloxy group, 3-chloro-2-propenyloxy group, 3,3-difluoro-2-propenyloxy group, 2,3- Examples include dichloro-2-propenyloxy group, 3,3-dichloro-2-propenyloxy group, 2,3,3-trifluoro-2-propenyloxy group, etc. Is done.

Ｃ_ａ〜Ｃ_ｂアルキニルオキシの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキニル−Ｏ−基を表す。具体例として、２−プロピニルオキシ基、２−ブチニルオキシ基、１−メチル−２−プロピニルオキシ基、１，１−ジメチル−２−プロピニルオキシ基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation C _a -C _b alkynyloxy represents an alkynyl-O— group with the above meaning consisting of _a to _b carbon atoms. Specific examples include a 2-propynyloxy group, a 2-butynyloxy group, a 1-methyl-2-propynyloxy group, a 1,1-dimethyl-2-propynyloxy group, and the like. Selected.

ハロ（Ｃ_ａ〜Ｃ_ｂ）アルキニルオキシの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるハロアルキニル−Ｏ−基を表す。具体例として、３−クロロ−２−プロピニルオキシ基、３−ブロモ−２−プロピニルオキシ基、３−ヨード−２−プロピニルオキシ基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation halo (C _a -C _b ) alkynyloxy represents a haloalkynyl-O— group with the above meaning consisting of _a to _b carbon atoms. Specific examples include a 3-chloro-2-propynyloxy group, a 3-bromo-2-propynyloxy group, a 3-iodo-2-propynyloxy group, and the like, which are selected within the range of each designated number of carbon atoms. The

Ｃ_ａ〜Ｃ_ｂアルキルチオの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル−Ｓ−基を表し、例えばメチルチオ基、エチルチオ基、ｎ−プロピルチオ基、ｉ−プロピルチオ基、ｎ−ブチルチオ基、ｉ−ブチルチオ基、ｓ−ブチルチオ基、ｔｅｒｔ−ブチルチオ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkylthio represents an alkyl-S-group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, methylthio group, ethylthio group, n-propylthio group, i-propylthio group, Specific examples include an n-butylthio group, an i-butylthio group, an s-butylthio group, a tert-butylthio group, and the like, and each is selected within the range of the designated number of carbon atoms.

ハロ（Ｃ_ａ〜Ｃ_ｂ）アルキルチオの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるハロアルキル−Ｓ−基を表す。具体例として、ジフルオロメチルチオ基、トリフルオロメチルチオ基、クロロジフルオロメチルチオ基、トリクロロメチルチオ基、ブロモジフルオロメチルチオ基、２，２，２−トリフルオロエチルチオ基、１，１，２，２−テトラフルオロエチルチオ基、２−クロロ−１，１，２−トリフルオロエチルチオ基、ペンタフルオロエチルチオ基、１，１，２，３，３，３−ヘキサフルオロプロピルチオ基、ヘプタフルオロプロピルチオ基、１，２，２，２−テトラフルオロ−１−（トリフルオロメチル）エチルチオ基、ノナフルオロブチルチオ基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation halo (C _a -C _b ) alkylthio represents a haloalkyl-S— group with the above meaning consisting of _a to _b carbon atoms. Specific examples include difluoromethylthio group, trifluoromethylthio group, chlorodifluoromethylthio group, trichloromethylthio group, bromodifluoromethylthio group, 2,2,2-trifluoroethylthio group, 1,1,2,2-tetrafluoroethyl. Thio group, 2-chloro-1,1,2-trifluoroethylthio group, pentafluoroethylthio group, 1,1,2,3,3,3-hexafluoropropylthio group, heptafluoropropylthio group, 1 , 2,2,2-tetrafluoro-1- (trifluoromethyl) ethylthio group, nonafluorobutylthio group, and the like, and each is selected in the range of the designated number of carbon atoms.

Ｃ_ａ〜Ｃ_ｂアルケニルチオの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルケニル−Ｓ−基を表す。具体例として、２−プロペニルチオ基、２−ブテニルチオ基、１−メチル−２−プロペニルチオ基、２−メチル−２−プロペニルチオ基、３−メチル−２−ブテニルチオ基、１，１−ジメチル−２−プロペニルチオ基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation C _a -C _b alkenylthio represents an alkenyl-S— group with the above meaning consisting of _a to _b carbon atoms. Specific examples include 2-propenylthio group, 2-butenylthio group, 1-methyl-2-propenylthio group, 2-methyl-2-propenylthio group, 3-methyl-2-butenylthio group, 1,1-dimethyl- 2-propenylthio group etc. are mentioned, It selects in the range of each designated carbon atom number.

Ｃ_ａ〜Ｃ_ｂアルキニルチオの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキニル−Ｓ−基を表す。具体例として、２−プロピニルチオ基、２−ブチニルチオ基、１−メチル−２−プロピニルチオ基、１，１−ジメチル−２−プロピニルチオ基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation C _a -C _b alkynylthio represents an alkynyl-S— group with the above meaning consisting of _a to _b carbon atoms. Specific examples include 2-propynylthio group, 2-butynylthio group, 1-methyl-2-propynylthio group, 1,1-dimethyl-2-propynylthio group, etc. Selected.

Ｃ_ａ〜Ｃ_ｂアルキルスルフィニルの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル−Ｓ（Ｏ）−基を表す。具体例として、メチルスルフィニル基、エチルスルフィニル基、ｎ−プロピルスルフィニル基、ｉ−プロピルスルフィニル基、ｎ−ブチルスルフィニル基、ｉ−ブチルスルフィニル基、ｓ−ブチルスルフィニル基、ｔｅｒｔ−ブチルスルフィニル基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation C _a -C _b alkylsulfinyl represents an alkyl-S (O) — group with the above meaning consisting of _a to _b carbon atoms. Specific examples include methylsulfinyl group, ethylsulfinyl group, n-propylsulfinyl group, i-propylsulfinyl group, n-butylsulfinyl group, i-butylsulfinyl group, s-butylsulfinyl group, tert-butylsulfinyl group and the like. Selected within a range of each specified number of carbon atoms.

ハロ（Ｃ_ａ〜Ｃ_ｂ）アルキルスルフィニルの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるハロアルキル−Ｓ（Ｏ）−基を表す。具体例として、ジフルオロメチルスルフィニル基、トリフルオロメチルスルフィニル基、クロロジフルオロメチルスルフィニル基、トリクロロメチルスルフィニル基、ブロモジフルオロメチルスルフィニル基、２，２，２−トリフルオロエチルスルフィニル基、１，１，２，２−テトラフルオロエチルスルフィニル基、２−クロロ−１，１，２−トリフルオロエチルスルフィニル基、ペンタフルオロエチルスルフィニル基、１，１，２，３，３，３−ヘキサフルオロプロピルスルフィニル基、ヘプタフルオロプロピルスルフィニル基、１，２，２，２−テトラフルオロ−１−（トリフルオロメチル）エチルスルフィニル基、ノナフルオロブチルスルフィニル基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation halo (C _a -C _b ) alkylsulfinyl represents a haloalkyl-S (O) — group with the above meaning consisting of _a to _b carbon atoms. Specific examples include difluoromethylsulfinyl group, trifluoromethylsulfinyl group, chlorodifluoromethylsulfinyl group, trichloromethylsulfinyl group, bromodifluoromethylsulfinyl group, 2,2,2-trifluoroethylsulfinyl group, 1,1,2, 2-tetrafluoroethylsulfinyl group, 2-chloro-1,1,2-trifluoroethylsulfinyl group, pentafluoroethylsulfinyl group, 1,1,2,3,3,3-hexafluoropropylsulfinyl group, heptafluoro Examples thereof include a propylsulfinyl group, 1,2,2,2-tetrafluoro-1- (trifluoromethyl) ethylsulfinyl group, nonafluorobutylsulfinyl group, and the like, and each is selected within the range of the designated number of carbon atoms.

Ｃ_ａ〜Ｃ_ｂアルケニルスルフィニルの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルケニル−Ｓ（Ｏ）−基を表す。具体例として、２−プロペニルスルフィニル基、２−ブテニルスルフィニル基、１−メチル−２−プロペニルスルフィニル基、２−メチル−２−プロペニルスルフィニル基、３−メチル−２−ブテニルスルフィニル基、１，１−ジメチル−２−プロペニルスルフィニル基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation C _a -C _b alkenylsulfinyl represents an alkenyl-S (O) — group with the above meaning consisting of _a to _b carbon atoms. Specific examples include 2-propenylsulfinyl group, 2-butenylsulfinyl group, 1-methyl-2-propenylsulfinyl group, 2-methyl-2-propenylsulfinyl group, 3-methyl-2-butenylsulfinyl group, 1, Examples include 1-dimethyl-2-propenylsulfinyl group and the like, and each is selected within the range of the designated number of carbon atoms.

Ｃ_ａ〜Ｃ_ｂアルキニルスルフィニルの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキニル−Ｓ（Ｏ）−基を表す。具体例として、２−プロピニルスルフィニル基、２−ブチニルスルフィニル基、１−メチル−２−プロピニルスルフィニル基、１，１−ジメチル−２−プロピニルスルフィニル基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation C _a -C _b alkynylsulfinyl represents an alkynyl-S (O) — group with the above meaning consisting of _a to _b carbon atoms. Specific examples include 2-propynylsulfinyl group, 2-butynylsulfinyl group, 1-methyl-2-propynylsulfinyl group, 1,1-dimethyl-2-propynylsulfinyl group, etc. The range is selected.

Ｃ_ａ〜Ｃ_ｂアルキルスルホニルの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル−Ｓ（Ｏ）_２−基を表す。具体例として、メチルスルホニル基、エチルスルホニル基、ｎ−プロピルスルホニル基、ｉ−プロピルスルホニル基、ｎ−ブチルスルホニル基、ｉ−ブチルスルホニル基、ｓ−ブチルスルホニル基、ｔｅｒｔ−ブチルスルホニル基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation C _a -C _b alkylsulfonyl represents an alkyl-S (O) ₂ -group having the above-mentioned meaning consisting of _a to _b carbon atoms. Specific examples include methylsulfonyl group, ethylsulfonyl group, n-propylsulfonyl group, i-propylsulfonyl group, n-butylsulfonyl group, i-butylsulfonyl group, s-butylsulfonyl group, tert-butylsulfonyl group and the like. Selected within a range of each specified number of carbon atoms.

ハロ（Ｃ_ａ〜Ｃ_ｂ）アルキルスルホニルの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるハロアルキル−Ｓ（Ｏ）_２−基を表す。具体例として、ジフルオロメチルスルホニル基、トリフルオロメチルスルホニル基、クロロジフルオロメチルスルホニル基、トリクロロメチルスルホニル基、ブロモジフルオロメチルスルホニル基、２，２，２−トリフルオロエチルスルホニル基、１，１，２，２−テトラフルオロエチルスルホニル基、２−クロロ−１，１，２−トリフルオロエチルスルホニル基、ペンタフルオロエチルスルホニル基、１，１，２，３，３，３−ヘキサフルオロプロピルスルホニル基、ヘプタフルオロプロピルスルホニル基、１，２，２，２−テトラフルオロ−１−（トリフルオロメチル）エチルスルホニル基、ノナフルオロブチルスルホニル基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of halo (C _a -C _b ) alkylsulfonyl represents a haloalkyl-S (O) ₂ — group with the above meaning consisting of _a to _b carbon atoms. Specific examples include difluoromethylsulfonyl group, trifluoromethylsulfonyl group, chlorodifluoromethylsulfonyl group, trichloromethylsulfonyl group, bromodifluoromethylsulfonyl group, 2,2,2-trifluoroethylsulfonyl group, 1,1,2, 2-tetrafluoroethylsulfonyl group, 2-chloro-1,1,2-trifluoroethylsulfonyl group, pentafluoroethylsulfonyl group, 1,1,2,3,3,3-hexafluoropropylsulfonyl group, heptafluoro Examples thereof include a propylsulfonyl group, 1,2,2,2-tetrafluoro-1- (trifluoromethyl) ethylsulfonyl group, nonafluorobutylsulfonyl group and the like, and each is selected within the range of the designated number of carbon atoms.

Ｃ_ａ〜Ｃ_ｂアルケニルスルホニルの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルケニル−Ｓ（Ｏ）_２−基を表す。具体例として、２−プロペニルスルホニル基、２−ブテニルスルホニル基、１−メチル−２−プロペニルスルホニル基、２−メチル−２−プロペニルスルホニル基、３−メチル−２−ブテニルスルホニル基、１，１−ジメチル−２−プロペニルスルホニル基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation C _a -C _b alkenylsulfonyl represents an alkenyl-S (O) ₂ -group having the above-mentioned meaning consisting of _a to _b carbon atoms. Specific examples include 2-propenylsulfonyl group, 2-butenylsulfonyl group, 1-methyl-2-propenylsulfonyl group, 2-methyl-2-propenylsulfonyl group, 3-methyl-2-butenylsulfonyl group, 1, Examples include 1-dimethyl-2-propenylsulfonyl group and the like, and each is selected within the range of the designated number of carbon atoms.

Ｃ_ａ〜Ｃ_ｂアルキニルスルホニルの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキニル−Ｓ（Ｏ）_２−基を表す。具体例として、２−プロピニルスルホニル基、２−ブチニルスルホニル基、１−メチル−２−プロピニルスルホニル基、１，１−ジメチル−２−プロピニルスルホニル基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation C _a -C _b alkynylsulfonyl represents an alkynyl-S (O) ₂ -group having the above meaning consisting of _a to _b carbon atoms. Specific examples include 2-propynylsulfonyl group, 2-butynylsulfonyl group, 1-methyl-2-propynylsulfonyl group, 1,1-dimethyl-2-propynylsulfonyl group, etc. The range is selected.

Ｃ_ａ〜Ｃ_ｂアルキルアミノの表記は、それぞれ同一でも又は互いに相異なっていてもよい炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル基によって置換されたアミノ基を表す。具体例として、メチルアミノ基、エチルアミノ基、ｎ−プロピルアミノ基、ｉ−プロピルアミノ基、ｎ−ブチルアミノ基、ｉ−ブチルアミノ基、ｓ−ブチルアミノ基、ｔｅｒｔ−ブチルアミノ基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkylamino represents an amino group substituted by an alkyl group having the above-mentioned meanings consisting of _a to _b carbon atoms, which may be the same or different from each other. Specific examples include methylamino group, ethylamino group, n-propylamino group, i-propylamino group, n-butylamino group, i-butylamino group, s-butylamino group, tert-butylamino group and the like. Selected within a range of each specified number of carbon atoms.

ジ（Ｃ_ａ〜Ｃ_ｂ）アルキルアミノの表記は、それぞれ同一でも又は互いに相異なっていてもよい炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル基によって置換されたアミノ基を表す。具体例として、ジメチルアミノ基、エチルメチルアミノ基、ジエチルアミノ基、ジ（ｎ−プロピル）アミノ基、ジ（ｎ−ブチル）アミノ基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of di (C _a -C _b ) alkylamino represents an amino group substituted with an alkyl group having the above-mentioned meaning consisting of _a to _b carbon atoms, which may be the same or different from each other. . Specific examples include a dimethylamino group, an ethylmethylamino group, a diethylamino group, a di (n-propyl) amino group, a di (n-butyl) amino group, and the like. The

トリ（Ｃ_ａ〜Ｃ_ｂ）アルキルシリルの表記は、それぞれ同一でも又は互いに相異なっていてもよい炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル基によって置換されたシリル基を表す。具体例として、トリメチルシリル基、トリエチルシリル基、トリ（ｎ−プロピル）シリル基、エチルジメチルシリル基、ｎ−プロピルジメチルシリル基、ｎ−ブチルジメチルシリル基、ｉ−ブチルジメチルシリル基、ｔｅｒｔ−ブチルジメチルシリル基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of tri (C _a -C _b ) alkylsilyl represents a silyl group substituted by an alkyl group having the above-mentioned meanings consisting of _a to _b carbon atoms which may be the same or different from each other. . Specific examples include trimethylsilyl group, triethylsilyl group, tri (n-propyl) silyl group, ethyldimethylsilyl group, n-propyldimethylsilyl group, n-butyldimethylsilyl group, i-butyldimethylsilyl group, tert-butyldimethyl. A silyl group etc. are mentioned, It selects in the range of each designated carbon atom number.

Ｃ_ａ〜Ｃ_ｂアルキルカルボニルの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル−Ｃ（Ｏ）−基を表す。具体例として、アセチル基、プロピオニル基、ブチリル基、イソブチリル基、バレリル基、イソバレリル基、２−メチルブタノイル基、ピバロイル基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation C _a -C _b alkylcarbonyl represents an alkyl-C (O) — group with the above meaning consisting of _a to _b carbon atoms. Specific examples include an acetyl group, a propionyl group, a butyryl group, an isobutyryl group, a valeryl group, an isovaleryl group, a 2-methylbutanoyl group, a pivaloyl group, and the like, and each is selected within the range of the designated number of carbon atoms.

ハロ（Ｃ_ａ〜Ｃ_ｂ）アルキルカルボニルの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるハロアルキル−Ｃ（Ｏ）−基を表す。具体例として、ジフルオロアセチル基、トリフルオロアセチル基、クロロジフルオロアセチル基、ブロモジフルオロアセチル基、２−フルオロプロピオニル基、２−クロロプロピオニル基、２，２，２−フルオロプロピオニル基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of halo (C _a -C _b ) alkylcarbonyl represents a haloalkyl-C (O) — group with the above meaning consisting of _a to _b carbon atoms. Specific examples include difluoroacetyl group, trifluoroacetyl group, chlorodifluoroacetyl group, bromodifluoroacetyl group, 2-fluoropropionyl group, 2-chloropropionyl group, 2,2,2-fluoropropionyl group, etc. Is selected within the range of the specified number of carbon atoms.

Ｃ_ａ〜Ｃ_ｂアルコキシカルボニルの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル−Ｏ−Ｃ（Ｏ）−基を表す。具体例として、メトキシカルボニル基、エトキシカルボニル基、ｎ−プロピルオキシカルボニル基、ｉ−プロピルオキシカルボニル基、ｎ−ブトキシカルボニル基、ｉ−ブトキシカルボニル基、ｔｅｒｔ−ブトキシカルボニル基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation C _a -C _b alkoxycarbonyl represents an alkyl-O—C (O) — group with the above meaning consisting of _a to _b carbon atoms. Specific examples include methoxycarbonyl group, ethoxycarbonyl group, n-propyloxycarbonyl group, i-propyloxycarbonyl group, n-butoxycarbonyl group, i-butoxycarbonyl group, tert-butoxycarbonyl group and the like. Selected within the specified number of carbon atoms.

Ｃ_ａ〜Ｃ_ｂアルキルカルボニルオキシの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル−Ｃ（Ｏ）−Ｏ−基を表す。具体例として、アセチルオキシ基、プロピオニルオキシ基、ブチリルオキシ基、イソブチリルオキシ基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation C _a -C _b alkylcarbonyloxy represents an alkyl-C (O) —O— group with the above meaning consisting of _a to _b carbon atoms. Specific examples include an acetyloxy group, a propionyloxy group, a butyryloxy group, an isobutyryloxy group, and the like, and each is selected within the range of the designated number of carbon atoms.

Ｃ_ａ〜Ｃ_ｂアルキルアミノカルボニルの表記は、水素原子の一方が、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル基によって置換されたカルバモイル基を表す。具体例として、メチルカルバモイル基、エチルカルバモイル基、ｎ−プロピルカルバモイル基、ｉ−プロピルカルバモイル基、ｎ−ブチルカルバモイル基、ｉ−ブチルカルバモイル基、ｓ−ブチルカルバモイル基、ｔｅｒｔ−ブチルカルバモイル基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkylaminocarbonyl represents a carbamoyl group in which one of the hydrogen atoms is substituted with an alkyl group having the above meaning consisting of _a to _b carbon atoms. Specific examples include methylcarbamoyl group, ethylcarbamoyl group, n-propylcarbamoyl group, i-propylcarbamoyl group, n-butylcarbamoyl group, i-butylcarbamoyl group, s-butylcarbamoyl group, tert-butylcarbamoyl group and the like. Selected within a range of each specified number of carbon atoms.

ジ（Ｃ_ａ〜Ｃ_ｂ）アルキルアミノカルボニルの表記は、水素原子が両方とも、それぞれ同一でも又は互いに相異なっていてもよい炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル基によって置換されたカルバモイル基を表す。具体例として、Ｎ，Ｎ−ジメチルカルバモイル基、Ｎ−エチル−Ｎ−メチルカルバモイル基、Ｎ，Ｎ−ジエチルカルバモイル基、Ｎ，Ｎ−ジ（ｎ−プロピル）カルバモイル基、Ｎ，Ｎ−ジ（ｎ−ブチル）カルバモイル基等が挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of di (C _a -C _b ) alkylaminocarbonyl refers to an alkyl group as defined above comprising a to b carbon atoms in which both hydrogen atoms may be the same or different from each other. Represents a substituted carbamoyl group. Specific examples include N, N-dimethylcarbamoyl group, N-ethyl-N-methylcarbamoyl group, N, N-diethylcarbamoyl group, N, N-di (n-propyl) carbamoyl group, N, N-di (n -Butyl) carbamoyl group and the like, and each is selected within the range of the designated number of carbon atoms.

Ｃ_ａ〜Ｃ_ｂアルコキシ（Ｃ_ｄ〜Ｃ_ｅ）アルキルの表記は、それぞれ前記の意味である任意のＣ_ａ〜Ｃ_ｂアルコキシ基によって、炭素原子に結合した水素原子が任意に置換された、炭素原子数がｄ〜ｅ個よりなる前記の意味であるアルキル基を表す。具体例として、メトキシメチル基等があげられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkoxy (C _d -C _e ) alkyl is a carbon in which a hydrogen atom bonded to a carbon atom is optionally substituted by any C _a -C _b alkoxy group having the aforementioned meaning, respectively. It represents an alkyl group having the above-mentioned meaning consisting of de to e atoms. Specific examples include a methoxymethyl group and the like, which are selected in the range of each designated number of carbon atoms.

Ｃ_ａ〜Ｃ_ｂアルコキシ（Ｃ_ｄ〜Ｃ_ｅ）アルコキシの表記は、それぞれ前記の意味である任意のＣ_ａ〜Ｃ_ｂアルコキシ基によって、炭素原子に結合した水素原子が任意に置換された、炭素原子数がｄ〜ｅ個よりなる前記の意味であるアルコキシ基を表す。具体例として、メトキシメトキシ基等があげられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkoxy (C _d -C _e ) alkoxy is a carbon in which a hydrogen atom bonded to a carbon atom is optionally substituted by any C _a -C _b alkoxy group having the aforementioned meaning, respectively. An alkoxy group having the above-mentioned meaning consisting of d to e atoms is represented. Specific examples include a methoxymethoxy group and the like, which are selected within the range of each designated number of carbon atoms.

「Ｒ^ａによって任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルキル」の表記は、任意のＲ^ａによって、炭素原子に結合した水素原子が任意に置換された、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル基を表し、各々の指定の炭素原子数の範囲で選択される。それぞれの（Ｃ_ａ〜Ｃ_ｂ）アルキル基上の置換基Ｒ^ａが２個以上存在するとき、それぞれのＲ^ａは互いに同一でも、または互いに相異なっていてもよい。 Designation "optionally substituted by R ^a _(C ^a ~C _b) alkyl", by any R ^a, hydrogen atoms bonded to carbon atoms are optionally substituted, to b number carbon atoms Each of which is selected within the range of the designated number of carbon atoms. When two or more substituents R ^a on each (C _a -C _b ) alkyl group are present, each R ^a may be the same as or different from each other.

「Ｒ^ａ１によって任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルキル」の表記は、任意のＲ^ａ１によって、炭素原子に結合した水素原子が任意に置換された、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル基を表し、各々の指定の炭素原子数の範囲で選択される。それぞれの（Ｃ_ａ〜Ｃ_ｂ）アルキル基上の置換基Ｒ^ａ１が２個以上存在するとき、それぞれのＲ^ａ１は互いに同一でも、または互いに相異なっていてもよい。 The notation “(C _a -C _b ) alkyl optionally substituted with R ^a1 ” indicates that a hydrogen atom bonded to a carbon atom is optionally substituted with any R ^a1 and the number of carbon atoms is a to b Each of which is selected within the range of the designated number of carbon atoms. When two or more substituents R ^a1 on each (C _a -C _b ) alkyl group are present, each R ^a1 may be the same as or different from each other.

「Ｒ^ｂによって任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルケニル」の表記は、任意のＲ^ｂによって、炭素原子に結合した水素原子が任意に置換された、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルケニル基を表し、各々の指定の炭素原子数の範囲で選択される。それぞれの（Ｃ_ａ〜Ｃ_ｂ）アルケニル基上の置換基Ｒ^ｂが２個以上存在するとき、それぞれのＲ^ｂは互いに同一でも、または互いに相異なっていてもよい。 The notation “(C _a -C _b ) alkenyl optionally substituted with R ^b ” refers to the number of carbon atoms a to ^b in which a hydrogen atom bonded to a carbon atom is optionally substituted with any R ^b Each of which is selected within the range of the designated number of carbon atoms. When there are two or more substituents R ^b on each (C _a -C _b ) alkenyl group, each R ^b may be the same as or different from each other.

「Ｒ^ｂ１によって任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルキル」の表記は、任意のＲ^ｂ１によって、炭素原子に結合した水素原子が任意に置換された炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル基を表し、各々の指定の炭素原子数の範囲で選択される。それぞれの（Ｃ_ａ〜Ｃ_ｂ）アルキル基上の置換基Ｒ^ｂ１が２個以上存在するとき、それぞれのＲ^ｂ１は互いに同一でも、または互いに相異なっていてもよい。 Designation "optionally substituted by R ^b1 _(C a ~C _b) alkyl", by any R ^b1, number of carbon atoms in which the hydrogen atoms bonded to carbon atom is optionally substituted from a~b pieces The above-mentioned meaning is an alkyl group, and each is selected within the range of the designated number of carbon atoms. When two or more substituents R ^b1 are present on each (C _a -C _b ) alkyl group, each R ^b1 may be the same as or different from each other.

「Ｒ^ｂ２によって任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルキル」の表記は、任意のＲ^ｂ２によって、炭素原子に結合した水素原子が任意に置換された、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル基を表し、各々の指定の炭素原子数の範囲で選択される。それぞれの（Ｃ_ａ〜Ｃ_ｂ）アルキル基上の置換基Ｒ^ｂ２が２個以上存在するとき、それぞれのＲ^ｂ２は互いに同一でも、または互いに相異なっていてもよい。 Designation "optionally substituted by R ^b2 _(C a ~C _b) alkyl", by any R ^b2, hydrogen atoms bonded to carbon atoms are optionally substituted, to b number carbon atoms Each of which is selected within the range of the designated number of carbon atoms. When two or more substituents R ^b2 on each (C _a -C _b ) alkyl group are present, each R ^b2 may be the same as or different from each other.

「Ｒ^ｂ３によって任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルキル」の表記は、任意のＲ^ｂ３によって、炭素原子に結合した水素原子が任意に置換された、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル基を表し、各々の指定の炭素原子数の範囲で選択される。それぞれの（Ｃ_ａ〜Ｃ_ｂ）アルキル基上の置換基Ｒ^ｂ３が２個以上存在するとき、それぞれのＲ^ｂ３は互いに同一でも、または互いに相異なっていてもよい。 The notation “(C _a -C _b ) alkyl optionally substituted with R ^b3 ” refers to any number of carbon atoms a to ^b in which a hydrogen atom bonded to a carbon atom is optionally substituted with any R ^b3 . Each of which is selected within the range of the designated number of carbon atoms. When there are two or more substituents R ^b3 on each (C _a -C _b ) alkyl group, each R ^b3 may be the same as or different from each other.

「Ｒ^ｂ４によって任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルキル」の表記は、任意のＲ^ｂ４によって、炭素原子に結合した水素原子が任意に置換された、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル基を表し、各々の指定の炭素原子数の範囲で選択される。それぞれの（Ｃ_ａ〜Ｃ_ｂ）アルキル基上の置換基Ｒ^ｂ４が２個以上存在するとき、それぞれのＲ^ｂ４は互いに同一でも、または互いに相異なっていてもよい。 The notation “(C _a -C _b ) alkyl optionally substituted with R ^b4 ” refers to any number of carbon atoms a to ^b in which a hydrogen atom bonded to a carbon atom is optionally substituted with any R ^b4 . Each of which is selected within the range of the designated number of carbon atoms. When two or more substituents R ^b4 on each (C _a -C _b ) alkyl group are present, each R ^b4 may be the same as or different from each other.

「Ｒ^ｂによって任意に置換された（Ｃ_ａ〜Ｃ_ｂ）シクロアルキル」の表記は、任意のＲ^ａによって、炭素原子に結合した水素原子が任意に置換された、炭素原子数がａ〜ｂ個よりなる前記の意味であるシクロアルキル基を表し、各々の指定の炭素原子数の範囲で選択される。それぞれの（Ｃ_ａ〜Ｃ_ｂ）シクロアルキル基上の置換基Ｒ^ａが２個以上存在するとき、それぞれのＲ^ａは互いに同一でも、または互いに相異なっていてもよい。 The notation “(C _a -C _b ) cycloalkyl optionally substituted with R ^b ” refers to the case where the hydrogen atom bonded to the carbon atom is optionally substituted with any R ^a , and the number of carbon atoms is ab Represents a cycloalkyl group having the above-mentioned meaning, and is selected in the range of the respective designated number of carbon atoms. When two or more substituents R ^a are present on each (C _a -C _b ) cycloalkyl group, each R ^a may be the same as or different from each other.

「Ｒ^ｂ４によって任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルコキシ」の表記は、任意のＲ^ｂ４によって、炭素原子に結合した水素原子が任意に置換された、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルコキシ基を表し、各々の指定の炭素原子数の範囲で選択される。それぞれの（Ｃ_ａ〜Ｃ_ｂ）アルコキシ基上の置換基Ｒ^ｂ４が２個以上存在するとき、それぞれのＲ^ｂ４は互いに同一でも、または互いに相異なっていてもよい。 The notation “(C _a -C _b ) alkoxy optionally substituted with R ^b4 ” refers to any number of carbon atoms a to ^b in which a hydrogen atom bonded to a carbon atom is optionally substituted with any R ^b4 . Each of which is selected within the range of the designated number of carbon atoms. When there are two or more substituents R ^b4 on each (C _a -C _b ) alkoxy group, each R ^b4 may be the same as or different from each other.

「Ｒ^４とＲ^５とが一緒になってＣ_２〜Ｃ_５アルキレン鎖を形成することにより、Ｒ^４及びＲ^５が結合する炭素原子と共に３〜６員環を形成すること」の表記の具体例として、例えば、シクロプロパン、シクロブタン、シクロペンタン、シクロヘキサン等の環が挙げられ、各々の指定の原子数の範囲で選択される。 "By forming the ^{R 4} and ^{R 5} and together _C 2 -C ₅ alkylene chain, to form a 3-6 membered ring together with the carbon atom ^{to which R 4} and ^{R 5} are bonded" specific notation Examples include, for example, rings such as cyclopropane, cyclobutane, cyclopentane, cyclohexane, etc., each selected within the specified number of atoms.

本発明のアシルヒドラゾン誘導体の農薬として許容される塩としては、例えば塩酸塩、臭化水素酸塩、ヨウ化水素酸塩、ギ酸塩、酢酸塩又はシュウ酸塩等が挙げられる。 Examples of the pesticidally acceptable salt of the acyl hydrazone derivative of the present invention include hydrochloride, hydrobromide, hydroiodide, formate, acetate, oxalate and the like.

本発明の化合物は、一般的には農園芸用の殺菌・殺かび剤として、ネコブカビ類、卵菌類、接合菌類、子嚢菌類、担子菌類、不完全菌類、細菌類又はウイルスによる種々の病害に対し使用することができる。 The compounds of the present invention are generally used as fungicides and fungicides for agricultural and horticultural use in various diseases caused by root-knot fungi, oomycetes, zygomycetes, ascomycetes, basidiomycetes, imperfect fungi, bacteria or viruses. Can be used against.

本発明化合物の防除対象となる植物病害としては、
イネのいもち病（Ｐｙｒｉｃｕｌａｒｉａｏｒｙｚａｅ）、ごま葉枯病（Ｃｏｃｈｌｉｏｂｏｌｕｓｍｉｙａｂｅａｎｕｓ）、紋枯病（Ｒｈｉｚｏｃｔｏｎｉａｓｏｌａｎｉ）、イネこうじ病（Ｃｌａｖｉｃｅｐｓｖｉｒｅｎｓ）、ばか苗病（Ｇｉｂｂｅｒｅｌｌａｆｕｊｉｋｕｒｏｉ）、苗立枯病（Ｐｙｔｈｉｕｍｇｒａｍｉｎｉｃｏｌａ，Ｐ．ｓｐｉｎｏｓｕｍ，Ｆｕｓａｒｉｕｍａｖｅｎａｃｅｕｍ，Ｆｕｓａｒｉｕｍｓｏｌａｎｉ，Ｆｕｓａｒｉｕｍｓｐｐ．，Ｒｈｉｚｏｐｕｓｃｈｉｎｅｎｓｉｓ，Ｒ．ｏｒｙｚａｅ，Ｒｈｉｚｏｐｕｓｓｐｐ．，Ｔｒｉｃｈｏｄｅｒｍａｖｉｒｉｄｅ）、もみ枯細菌病（Ｂｕｒｋｈｏｌｄｅｒｉａｇｌｕｍａｅ）、苗立枯細菌病（Ｂｕｒｋｈｏｌｄｅｒｉａｐｌａｎｔａｒｉｉ）、褐条病（Ａｃｉｄｏｖｏｒａｘａｖｅｎａｅ）、白葉枯病（Ｘａｎｔｈｏｍｏｎａｓｏｒｙｚａｅ）、内頴褐変病（Ｅｒｗｉｎｉａａｎａｎａｓ）、
コムギ縞萎縮病（Ｗｈｅａｔｙｅｌｌｏｗｍｏｓａｉｃｖｉｒｕｓ）、オオムギ縞萎縮病（Ｂａｒｌｅｙｙｅｌｌｏｗｍｏｓａｉｃｖｉｒｕｓ）、ムギ類のうどんこ病（Ｅｒｙｓｉｐｈｅｇｒａｍｉｎｉｓｆ．ｓｐ．ｈｏｒｄｅｉ，Ｅ．ｇｒａｍｉｎｉｓｆ．ｓｐ．ｔｒｉｔｉｃｉ）、斑葉病（Ｐｙｒｅｎｏｐｈｏｒａｇｒａｍｉｎｅａ）、網斑病（Ｐｙｒｅｎｏｐｈｏｒａｔｅｒｅｓ）、赤かび病（Ｇｉｂｂｅｒｅｌｌａｚｅａｅ）、さび病（Ｐｕｃｃｉｎｉａｓｔｒｉｉｆｏｒｍｉｓ，Ｐ．ｇｒａｍｉｎｉｓ，Ｐ．ｒｅｃｏｎｄｉｔａ，Ｐ．ｈｏｒｄｅｉ）、褐色雪腐病（Ｐｙｔｈｉｕｍｉｗａｙａｍａｉ）、雪腐病（Ｔｉｐｕｌａｓｐ．，Ｍｉｃｒｏｎｅｃｔｒｉｅｌｌａｎｉｖａｉｓ）、裸黒穂病（Ｕｓｔｉｌａｇｏｔｒｉｔｉｃｉ，Ｕ．ｎｕｄａ）、雲形病（Ｒｈｙｎｃｈｏｓｐｏｒｉｕｍｓｅｃａｌｉｓ）、葉枯病（Ｓｅｐｔｏｒｉａｔｒｉｔｉｃｉ）、ふ枯病（Ｌｅｐｔｏｓｐｈａｅｒｉａｎｏｄｏｒｕｍ）、眼紋病（Ｐｓｅｕｄｏｃｅｒｃｏｓｐｏｒｅｌｌａｈｅｒｐｏｔｒｉｃｈｏｉｄｅｓ）、雪腐小粒菌核病（Ｔｙｐｈｕｌａｉｎｃａｒｎａｔａ）、雪腐大粒菌核病（Ｍｙｒｉｏｓｃｌｅｒｏｔｉｎｉａｂｏｒｅａｌｉｓ）、コムギの紅色雪腐病（Ｍｏｎｏｇｒａｐｈｅｌｌａｎｉｖａｌｉｓ）、立枯病（Ｇａｅｕｍａｎｏｍｙｃｅｓｇｒａｍｉｎｉｓ）、
カンキツの黒点病（Ｄｉａｐｏｒｔｈｅｃｉｔｒｉ）、そうか病（Ｅｌｓｉｎｏｅｆａｗｃｅｔｔｉｉ）、果実腐敗病（Ｐｅｎｉｃｉｌｌｉｕｍｄｉｇｉｔａｔｕｍ，Ｐ．ｉｔａｌｉｃｕｍ）、かいよう病（Ｘａｎｔｈｏｍｏｎａｓｃａｍｐｅｓｔｒｉｓ）、灰色かび病（Ｂｏｔｒｙｔｉｓｃｉｎｅｒｅａ）、
リンコ゛のモニリア病（Ｍｏｎｉｌｉｎｉａｍａｌｉ）、腐らん病（Ｖａｌｓａｍａｌｉ）、うどんこ病（Ｐｏｄｏｓｐｈａｅｒａｌｅｕｃｏｔｒｉｃｈａ）、斑点落葉病（Ａｌｔｅｒｎａｒｉａｍａｌｉ）、黒星病（Ｖｅｎｔｕｒｉａｉｎａｅｑｕａｌｉｓ）、
ナシの黒星病（Ｖｅｎｔｕｒｉａｎａｓｈｉｃｏｌａ）、黒斑病（Ａｌｔｅｒｎａｒｉａｋｉｋｕｃｈｉａｎａ）、赤星病（Ｇｙｍｎｏｓｐｏｒａｎｇｉｕｍａｓｉａｔｉｃｕｍ）、疫病（Ｐｈｙｔｏｐｈｔｈｏｒａｃａｃｔｏｒｕｎ，Ｐ．ｓｙｒｉｎｇａｅ）、葉炭そ病（Ｃｏｌｌｅｔｏｔｒｉｃｈｕｍｇｌｏｅｏｓｐｒｉｏｉｄｅｓ）、輪紋病（Ｂｏｔｒｙｏｓｐｈａｅｒｉａｂｅｒｅｎｇｅｒｉａｎａ）、うどんこ病（Ｐｈｙｌｌａｃｔｉｎｉａｍａｌｉ）、
モモの灰星病（Ｍｏｎｉｌｉｎｉａｆｒｕｃｔｉｃｏｌａ）、黒星病（Ｃｌａｄｏｓｐｏｒｉｕｍｃａｒｐｏｐｈｉｌｕｍ）、フォモプシス腐敗病（Ｐｈｏｍｏｐｓｉｓｓｐ．）、せん孔病（Ｐｓｅｕｄｏｃｅｒｃｏｓｐｏｒａｃｉｒｃｕｍｓｃｉｓｓａ，Ｐｈｙｌｌｏｓｔｉｃｔａｐｅｒｓｉｃａｅ）、白紋羽病（Ｒｏｓｅｌｌｉｎｉａｎｅｃａｔｒｉｘ）、縮葉病（Ｔａｐｈｒｉｎａｄｅｆｏｒｍａｎｓ）、スモモのかいよう病（Ｐｓｅｕｄｏｍｏｎａｓｓｙｒｉｎｇａｅｐｖ．ｍｏｒｓｐｒｕｎｏｒｕｍ）、灰星病（Ｍｏｎｉｌｉｎｉａｆｒｕｃｔｉｃｏｌａ）、黒斑病（Ｘａｎｔｈｏｍｏｎａｓｃａｍｐｅｓｔｒｉｓｐｖ．ｐｒｕｎｉ）、アンズの灰星病（Ｍｏｎｉｌｉｎｉａｆｒｕｃｔｉｃｏｌａ）、
ウメのかいよう病（Ｐｓｅｕｄｏｍｏｎａｓｓｙｒｉｎｇａｅｐｖ．ｍｏｒｓｐｒｕｎｏｒｕｍ）、黒星病（Ｃｌａｄｏｓｐｏｒｉｕｍｃａｒｐｏｐｈｉｌｕｍ）、
ブドウのべと病（Ｐｌａｓｍｏｐａｒａｖｉｔｉｃｏｌａ）、黒とう病（Ｅｌｓｉｎｏｅａｍｐｅｌｉｎａ）、晩腐病（Ｇｌｏｍｅｒｅｌｌａｃｉｎｇｕｌａｔａ）、うどんこ病（Ｕｎｃｉｎｕｌａｎｅｃａｔｏｒ）、さび病（Ｐｈｙｓｐｐｅｌｌａａｍｐｅｌｏｐｓｉｄｉｓ）、芽枯病（Ｄｉａｐｏｒｔｈｅｍｅｄｕｓａ）、灰色かび病（Ｂｏｔｒｙｔｉｓｃｉｎｅｒｅａ）、
カキの炭そ病（Ｇｌｏｍｅｒｅｌｌａｏｒｂｉｃｕｌａ）、落葉病（Ｍｙｃｏｓｐｈａｅｒｅｌｌａｎａｗａｉ）、灰色かび病（Ｂｏｔｒｙｔｉｓｃｉｎｅｒｅａ）、うどんこ病（Ｐｈｙｌｌａｃｔｉｎｉａｋａｋｉｃｏｌａ）、
ウリ類のべと病（Ｐｓｅｕｄｏｐｅｒｅｎｏｓｐｏｒａｃｕｂｅｎｓｉｓ）、炭そ病（Ｃｏｌｌｅｔｏｔｒｉｃｈｕｍｏｒｂｉｃｕｌａ）、うどんこ病（Ｓｐｈａｅｒｏｔｈｅｃａｆｕｌｉｇｉｎｅａ）、つる枯病（Ｄｉｄｌｙｍｅｌｌａｂｒｙｏｎｉａｅ）、つる割病（Ｆｕｓａｒｉｕｍｏｘｙｓｐｏｒｕｍ）、灰色かび病（Ｂｏｔｒｙｔｉｓｃｉｎｅｒｅａ）、菌核病（Ｓｃｌｅｒｏｔｉｎｉａｓｃｌｅｒｏｔｉｏｒｕｍ）、立枯病（Ｆｕｓａｒｉｕｍｓｏｌａｎｉ）、白絹病（Ｓｃｌｅｒｏｔｉｕｍｒｏｌｆｓｉｉ）、ホモプシス根腐病（Ｐｈｏｍｏｐｓｉｓｓｃｌｅｒｏｔｉｏｉｄｅｓ）、
キュウリの褐斑病（Ｃｏｒｙｎｅｓｐｏｒａｃａｓｓｉｉｃｏｌａ）、苗立枯病（Ｐｙｔｈｉｕｍｃｕｃｕｒｂｉｔａｃｅａｒｕｍ，Ｐ．ｄｅｂａｒｙａｎｕｍ，Ｒｈｉｚｏｃｔｏｎｉａｓｏｌａｎｉ）、根腐病（Ｐｙｔｈｉｕｍｍｙｒｉｏｔｙｌｕｍ，Ｐ．ｖｏｌｕｔｕｍ）、疫病（Ｐｈｙｔｏｐｈｔｈｏｒａｍｅｒｏｎｉｓ，Ｐ．ｎｉｃｏｔｉａｎａｅ）、斑点細菌病（Ｐｓｅｕｄｏｍｏｎａｓｓｙｒｉｎｇａｅｐｖ．ｌａｃｈｒｙｍａｎｓ）、紫紋羽病（Ｈｅｌｉｃｏｂａｓｉｄｉｕｍｍｏｍｐａ）、
スイカの褐色腐敗病（Ｐｈｙｔｏｐｈｔｈｏｒａｃａｐｓｉｃｉ）、疫病（Ｐｈｙｔｏｐｈｔｈｏｒａｃｒｙｐｔｏｇｅａ）、
メロンの立枯病（Ｐｙｔｈｉｕｍｄｅｂａｒｙａｎｕｍ）、疫病（Ｐｈｙｔｏｐｈｔｈｏｒａｎｉｃｏｔｉａｎａｅ）、
カボチャの疫病（Ｐｈｙｔｏｐｈｔｈｏｒａｃａｐｓｉｃｉ）、
ナス科の青枯病（Ｒａｌｓｔｏｎｉａｓｏｌａｎａｃｅａｒｕｍ）、萎凋病（Ｆｕｓａｒｉｕｍｏｘｙｓｐｏｒｕｍ）、灰色かび病（Ｂｏｔｒｙｔｉｓｃｉｎｅｒｅａ）、菌核病（Ｓｃｌｅｒｏｔｉｎｉａｓｃｌｅｒｏｔｉｏｒｕｍ）、白絹病（Ｓｃｌｅｒｏｔｉｕｍｒｏｌｆｓｉｉ）、
ジャガイモの疫病（Ｐｈｙｔｏｐｈｔｈｏｒａｉｎｆｅｓｔａｎｓ）、夏疫病（Ａｌｔｅｒｎａｒｉａｓｏｌａｎｉ）、黒あざ病（Ｔｈａｎａｔｅｐｈｏｒｕｓｃｕｃｕｍｅｒｉｓ）、黒あし病（Ｅｒｗｉｎｉａｃａｒｏｔｏｖｏｒａ）、そうか病（Ｓｔｒｅｐｔｏｍｙｃｅｓｓｐｐ．）、軟腐病（Ｅｒｗｉｎｉａｃａｒｏｔｏｖｏｒａ）、粉状そうか病（Ｓｐｏｎｇｏｓｐｏｒａｓｕｂｔｅｒｒａｎｅａ）、
トマトの疫病（Ｐｈｙｔｏｐｈｔｈｏｒａｉｎｆｅｓｔａｎｓ）、根腐疫病（Ｐｈｙｔｏｐｈｔｈｏｒａｃｒｙｐｔｏｇｅａ）、灰色疫病（Ｐｈｙｔｏｐｈｔｈｏｒａｃａｐｓｉｃｉ）、輪紋病（Ａｌｔｅｒｎａｒｉａｓｏｌａｎｉ）、葉かび病（Ｆｕｌｖｉａｆｕｌｖａ）、うどんこ病（Ｏｉｄｉｕｍｓｐ．，Ｏｉｄｉｏｐｓｉｓｉｓｉｃｕｌａ）、褐色腐敗病（Ｐｈｙｔｏｐｈｔｈｏｒａｎｉｃｏｔｉａｎａｅ）、かいよう病（Ｃｌａｖｉｂａｃｔｅｒｍｉｃｈｉｇａｎｅｎｓｉｓ）、褐色根腐病（Ｐｙｒｅｎｏｃｈａｅｔａｌｙｃｏｐｅｒｓｉｃｉ）、炭そ病（Ｃｏｌｌｅｔｏｔｒｉｃｈｕｍｇｌｏｅｏｓｐｏｒｉｏｉｄｅｓ）、苗立枯病（Ｐｙｔｈｉｕｍｖｅｘａｎｓ、Ｒｈｉｚｏｃｔｏｎｉａｓｏｌａｎｉ）、半身萎凋病（Ｖｅｒｔｉｃｉｌｌｉｕｍｄａｈｌｉａｅ）、斑点病（Ｓｔｅｍｐｈｙｌｉｕｍｌｙｃｏｐｅｒｓｉｃｉ）、
ピーマンの疫病（Ｐｈｙｔｏｐｈｔｈｏｒａｃａｐｓｉｃｉ）、うどんこ病（Ｏｉｄｉｏｐｓｉｓｓｉｃｕｌａ）、苗立枯病（Ｒｈｉｚｏｃｔｏｎｉａｓｏｌａｎｉ）、斑点病（Ｃｅｒｃｏｓｐｏｒａｃａｐｓｉｃｉ）、
ナスの疫病（Ｐｈｙｔｏｐｈｔｈｏｒａｉｎｆｅｓｔａｎｓ）、褐色腐敗病（Ｐｈｙｔｏｐｈｔｈｏｒａｃａｐｓｉｃｉ）、褐紋病（Ｐｈｏｍｏｐｓｉｓｖｅｘａｎｓ）、うどんこ病（Ｅｒｙｓｉｐｈｅｃｉｃｈｏｒａｃｅｒｕｍ，Ｏｉｄｉｏｐｓｉｓｓｉｃｕｌａ）、
ホウレンソウの疫病（Ｐｈｙｔｏｐｈｔｈｏｒａｓｐ．）、べと病（Ｐｅｒｏｎｏｓｐｏｒａｅｆｆｕｓａ）、立枯病（Ｐｙｔｈｉｕｍａｐｈａｎｉｄｅｒｍａｔｕｍ，Ｐ．ｍｙｒｉｏｔｙｌｕｍ、Ｐ．ｐａｒｏｅｃａｎｄｒｕｍ，Ｐ．ｕｌｔｉｍｕｍ）、萎凋病（Ｆｕｓａｒｉｕｍｏｘｙｓｐｏｒｕｍ）、株腐病（Ｒｈｉｚｏｃｔｏｎｉａｓｏｌａｎｉ）、根腐病（Ａｐｈａｎｏｍｙｃｅｓｃｏｃｈｌｉｏｉｄｅｓ）、斑点病（Ｈｅｔｅｒｏｓｐｏｒｉｕｍｖａｒｉａｂｉｌｅ）、
ネギ類の白色疫病（Ｐｈｙｔｏｐｈｔｈｏｒａｐｏｒｒｉ）、疫病（Ｐｈｙｔｏｐｈｔｈｏｒａｎｉｃｏｔｉａｎａｅ）、白絹病（Ｓｃｌｅｒｏｔｉｕｍｒｏｌｆｓｉｉ）、苗立枯病（Ｒｈｉｚｏｃｔｏｎｉａｓｏｌａｎｉ）、黒斑病（Ａｌｔｅｒｎａｒｉａｐｏｒｒｉ）、軟腐病（Ｅｒｗｉｎｉａｃａｒｏｔｏｖｏｒａ，Ｅ．ｃｈｒｙｓａｎｔｈｍｉ）、べと病（Ｐｅｒｏｎｏｓｐｏｒａｄｅｓｔｒｕｃｔｏｒ）、さび病（Ｐｕｃｃｉｎｉａａｌｌｉｉ）、
ネギの萎凋病（Ｆｕｓａｒｉｕｍｏｘｙｓｐｏｒｕｍ）、黄斑病（Ｈｅｔｅｒｏｓｐｏｒｉｕｍａｌｉｉ）、紅色根腐病（Ｐｙｒｅｎｏｃｈａｅｔａｔｅｒｒｅｓｔｒｉｓ）、小菌核腐敗病（Ｂｏｔｒｙｔｉｓｓｑｕａｍｏｓａ）、
タマネギの乾腐病（Ｆｕｓａｒｉｕｍｏｘｙｓｐｏｒｕｍ）、黒穂病（Ｕｒｏｃｙｓｔｉｓｃｅｐｕｌａｅ）、小菌核病（Ｃｉｂｏｒｉｎｉａａｌｌｉ）、灰色かび病（Ｂｏｔｒｙｔｉｓｃｉｎｅｒｅａ）、灰色腐敗病（Ｂｏｔｒｙｔｉｓａｌｌｉｉ）、腐敗病（Ｅｒｗｉｎｉａｒｈａｐｏｎｔｉｃｉ）、りん片腐敗病（Ｂｕｒｋｈｏｌｄｅｒｉａｇｌａｄｉｏｌｉ）、
アブラナ科野菜のべと病（Ｐｅｒｏｎｏｓｐｏｒａｐａｒａｓｉｔｉｃａ）、根こぶ病（Ｐｌａｓｍｏｄｉｏｐｈｏｒａｂｒａｓｓｉｃａｅ）、白さび病（Ａｌｂｕｇｏｍａｃｒｏｓｐｏｒａ）、黒斑病（Ａｌｔｅｒｎａｒｉａｊａｐｏｎｉｃａ，Ａ．ｂｒａｓｓｉｃａｅ）、白斑病（Ｃｅｒｃｏｓｐｏｒｅｌｌａｂｒａｓｓｉｃａｅ）、軟腐病（Ｅｒｗｉｎｉａｃａｒｏｔｏｖｏｒａ）、菌核病（Ｓｃｌｅｒｏｔｉｎｉａｓｃｌｅｒｏｔｉｏｒｕｍ）、
キャベツの株腐病（Ｔｈａｎａｔｅｐｈｏｒｕｓｃｕｃｕｍｅｒｉｓ）、バーティシリウム萎凋病（Ｖｅｒｔｉｃｉｌｌｉｕｍｄａｈｌｉａｅ）、ハクサイの黄化病（Ｖｅｒｔｉｃｉｌｌｉｕｍｄａｈｌｉａｅ）、尻腐病（Ｒｈｉｚｏｃｔｏｎｉａｓｏｌａｎｉ）、根くびれ病（Ａｐｈａｎｏｍｙｃｅｓｒａｐｈａｎｉ）、灰色かび病（Ｂｏｔｒｙｔｉｓｃｉｎｅｒｅａ）、ピシウム腐敗病（Ｐｙｔｈｉｕｍｕｌｔｉｍｕｍ）、
ダイコンの炭そ病（Ｃｏｌｌｅｔｏｔｒｉｃｈｕｍｈｉｇｇｉｎｓｉａｎｕｍ）、バーティシリウム黒点病（Ｖｅｒｔｉｃｉｌｌｉｕａｌｂｏ−ａｔｒｕｍ）、
マメ類の青枯病（Ｒａｌｓｔｏｎｉａｓｏｌａｎａｃｅａｒｕｍ）、萎凋病（Ｖｅｒｔｉｃｉｌｌｉｕｍｄａｈｌｉａｅ）、菌核病（Ｓｃｌｅｒｏｔｉｎｉａｓｃｌｅｒｏｔｉｏｒｕｍ）、黒根病（Ｔｈｉｅｌａｖｉｏｐｓｉｓｓｐ．）、さび病（Ｐｈａｋｏｐｓｏｒａｐａｃｈｙｒｈｉｚｉ）、白絹病（Ｓｃｌｅｒｏｔｉｕｍｒｏｌｆｓｉｉ）、立枯病（Ｆｕｓａｒｉｕｍｏｘｙｓｐｏｒｕｍ）、炭そ病（Ｃｏｌｌｅｔｏｔｒｉｃｈｕｍｔｒｕｎｃａｔｕｍ，Ｃ．ｔｒｉｆｏｌｉｉ，Ｇｌｏｍｅｒｅｌｌａｇｌｙｃｉｎｅｓ，Ｇｌｏｅｏｓｐｏｒｉｕｍｓｐ．）、灰色かび病（Ｂｏｔｒｙｔｉｓｃｉｎｅｒｅａ）、
ダイズのべと病（Ｐｅｒｏｎｏｓｐｏｒａｍａｎｓｈｕｒｉｃａ）、茎疫病（Ｐｈｙｔｏｐｈｔｈｏｒａｓｏｊａｅ）、葉焼病（Ｘａｎｔｈｏｍｏｎａｓｃａｍｐｅｓｔｒｉｓｐｖ．ｇｌｙｃｉｎｅｓ）、紫斑病（Ｃｅｒｃｏｓｐｏｒａｋｉｋｕｃｈｉｉ）、黒とう病（Ｅｌｓｉｎｏｅｇｌｙｃｉｎｅｓ）、黒点病（Ｄｉａｐｏｒｔｈｅｐｈａｓｅｏｌｏｒｕｍ）、
ラッカセイの黒渋病（Ｍｙｃｏｓｐｈａｅｒｅｌｌａｐｅｒｓｏｎａｔａ）、褐斑病（Ｍｙｃｏｓｐｈａｅｒｅｌｌａａｒａｃｈｉｄｉｓ）、エンドウのうどんこ病（Ｅｒｙｓｉｐｈｅｐｉｓｉ）、
イチゴのうどんこ病（Ｓｐｈａｅｒｏｔｈｅｃａａｐｈａｎｉｓ）、萎黄病（Ｆｕｓａｒｉｕｍｏｘｙｓｐｏｒｕｍ）、萎凋病（Ｖｅｒｔｉｃｉｌｌｉｕｍｄａｈｌｉａｅ）、疫病（Ｐｈｙｔｏｐｈｔｈｏｒａｃａｃｔｏｒｕｍ）、角斑細菌病（Ｘａｎｔｈｏｍｏｎａｓｃａｍｐｅｓｔｒｉｓ，Ｘ．ｆｒａｇａｒｉａｅ）、黒斑病（Ａｌｔｅｒｎａｒｉａａｌｔｅｒｎａｔｅ）、じゃのめ病（Ｍｙｃｏｓｐｈａｅｒｅｌｌａｆｒａｇａｒｉａｅ）、炭そ病（Ｃｏｌｌｅｔｏｔｒｉｃｈｕｍａｃｕｔａｔｕｍ，Ｃ．ｆｒａｇａｒｉａｅ，Ｇｌｏｍｅｒｅｌｌａｃｉｎｇｕｌａｔａ）、根腐病（Ｐｈｙｔｏｐｈｔｈｏｒａｆｒａｇａｒｉａｅ）、灰色かび病（Ｂｏｔｒｙｔｉｓｃｉｎｅｒｅａ）、芽枯病（Ｒｈｉｚｏｃｔｏｎｉａｓｏｌａｎｉ）、輪斑病（Ｄｒｅｎｅｒｏｐｈｏｍａｏｂｓｃｕｒａｎｓ）、
レタスの菌核病（Ｓｃｌｅｒｏｔｉｎｉａｓｃｌｅｒｏｔｉｏｒｕｍ）、すそ枯病（Ｒｈｉｚｏｂａｃｔｅｒｓｏｌａｎｉ）、軟腐病（Ｅｒｗｉｎｉａｃａｒｏｔｏｖｏｒａ）、立枯病（Ｐｙｔｈｉｕｍｓｐ．）、根腐病（Ｆｕｓａｒｉｕｍｏｘｙｓｐｏｒｕｍ）、灰色かび病（Ｂｏｔｒｙｔｉｓｃｉｎｅｒｅａ）、斑点細菌病（Ｘａｎｔｈｏｍｏｎａｓｃａｍｐｅｓｔｒｉｓｐｖ．ｖｉｔｉａｎｓ）、ビッグベイン病（Ｌｅｔｔｕｃｅｂｉｇ−ｖｅｉｎｖｉｒｕｓ）、腐敗病（Ｐｓｅｕｄｏｍｏｎａｓｃｉｃｈｏｒｉｉ，Ｐ．ｍａｒｇｉｎａｌｉｓｐｖ．ｍａｒｇｉｎａｌｉｓ，Ｐ．ｖｉｒｉｄｉｆｌａｖａ）、べと病（Ｂｒｅｍｉａｌａｃｔｕｃａｅ）、
ゴボウの萎凋病（Ｆｕｓａｒｉｕｍｏｘｙｓｐｏｒｕｍ）、黒あざ病（Ｒｈｉｚｏｃｔｏｎｉａｓｏｌａｎｉ）、黒条病（Ｉｔｅｒｓｏｎｉｌｉａｐｅｒｐｌｅｘａｎｓ）、黒斑細菌病（Ｘａｎｔｈｏｍｏｎａｓｃａｍｐｅｓｔｒｉｓｐｖ．ｎｉｇｒｏｍａｃｕｌａｎｓ）、黒斑病（Ａｓｃｏｃｈｙｔａｐｈａｓｅｏｌｏｒｕｍ）、根腐病（Ｐｙｔｈｉｕｍｉｒｒｅｇｕｌａｒｅ）、紫紋羽病（Ｈｅｌｉｃｏｂａｓｉｄｉｕｍｍｏｍｐａ）、
ニンジンの萎凋病（Ｆｕｓａｒｉｕｍｏｘｙｓｐｏｒｕｍ）、うどんこ病（Ｅｒｙｓｉｐｈｅｈｅｒａｃｌｅｉ）、黒葉枯病（Ａｌｔｅｒｎａｒｉａｄａｕｃｉ）、こぶ病（Ｒｈｉｚｏｃｔｏｎｉａｄａｕｃｉ）、しみ腐病（Ｐｙｔｈｉｕｍｓｕｌｃａｔｕｍ）、白絹病（Ｓｃｌｅｒｏｔｉｕｍｒｏｌｆｓｉｉ）、軟腐病（Ｅｒｗｉｎｉａｃａｒｏｔｏｖｏｒａ）、根腐病（Ｒｈｉｚｏｃｔｏｎｉａｓｏｌａｎｉ）、斑点病（Ｃｅｒｃｏｓｐｏｒａｃａｒｏｔａｅ）、紫紋羽病（Ｈｅｌｉｃｏｂａｓｉｄｉｕｍｍｏｍｐａ）、
チャの網もち病（Ｅｘｏｂａｓｉｄｉｕｍｒｅｔｉｃｕｌａｔｕｍ）、白星病（Ｅｌｓｉｎｏｅｌｅｕｃｏｓｐｉｌａ）、褐色円星病（Ｐｓｅｕｄｏｃｅｒｃｏｓｐｏｒａｏｃｅｌｌａｔａ，Ｃｅｒｏｓｐｏｒａｃｈａａｅ）、もち病（Ｅｘｏｂａｓｉｄｉｕｍｖｅｘａｎｓ）、輪紋病（Ｐｅｓｔａｌｔｉｏｐｓｉｓｌｏｎｇｉｓｅｔａ，Ｐ．ｔｈｅａｅ）、炭そ病（Ｃｏｌｌｅｔｏｔｒｉｃｈｕｍｔｈｅａ−ｓｉｎｅｎｓｉｓ）、
タバコの赤星病（Ａｌｔｅｒｎａｒｉａａｌｔｅｒｎａｔａ）、うどんこ病（Ｅｒｙｓｉｐｈｅｃｉｃｈｏｒａｃｅａｒｕｍ）、炭そ病（Ｃｏｌｌｅｔｏｔｒｉｃｈｕｍｃｉｃｈｏｒａｃｅａｒｕｍ）、
テンサイの褐斑病（Ｃｅｒｃｏｓｐｏｒａｂｅｔｉｃｏｌａ）、黒根病（Ａｐｈａｎｏｍｙｃｅｓｃｏｃｈｌｉｏｉｄｅｓ）そう根病（Ｂｅｅｔｎｅｃｒｏｔｉｃｙｅｌｌｏｗｖｅｉｎｖｉｒｕｓ）、苗立枯病（Ｐｙｔｈｉｕｍｄｅｂａｒｙａｎｕｍ、Ｐｈｏｍａｂｅｔａｅ，Ｒｈｉｚｏｃｔｏｎｉａｓｏｌａｎｉ，Ａｐｈａｎｏｍｙｃｅｓｃｏｃｈｌｉｏｉｄｅｓ，Ｆｕｓａｒｉｕｍｓｐ．）
バラの黒星病（Ｄｉｐｌｏｃａｒｐｏｎｒｏｓａｅ）、うどんこ病（Ｓｐｈａｅｒｏｔｈｅｃａｐａｎｎｏｓａ）、
キクの褐斑病（Ｓｅｐｔｏｒｉａｃｈｒｙｓａｎｔｈｅｍｉｉｎｄｉｃｉ）、白さび病（Ｐｕｃｃｉｎｉａｈｏｒｉａｎａ）、
シバ類のファリーリング病（Ｌｙｃｏｐｅｒｄｏｎｐｅｒｌａｔｕｍ，Ｌｅｐｉｓｔａｓｕｂｎｕｄｏ，Ｍａｒａｓｍｉｕｓｏｒｅａｄｅｓ）、擬似葉腐病（Ｃｅｒａｔｏｂａｓｉｄｉｕｍｓｐｐ．）、立枯病（Ｇａｅｍａｎｎｏｍｙｃｅｓｇｒａｍｉｎｉｓ）、カーブラリア葉枯病（Ｃｕｒｖｕｌａｒｉａｇｅｎｉｃｕｌａｔａ）、葉腐病（Ｒｈｉｚｏｃｔｏｎｉａｓｏｌａｎｉ）、ピシウム病（Ｐｙｔｈｉｕｍｐｅｒｉｐｌｏｃｕｍ、Ｐ．ｇｒａｍｉｎｉｃｏｌａ，Ｐ．ｖａｎｔｅｒｐｏｏｌｉｉ）、さび病（Ｐｕｃｃｉｎｉａｓｐｐ．）、うどんこ病（ＥｒｙｓｉｐｈｅｇｒａｍｉｎｉｓＤＣ）、ダラースポット病（Ｓｃｌｅｒｏｔｉｎｉａｈｏｍｏｅｏｃａｒｐａ）、雪腐病（Ｐｙｔｈｉｕｍｉｗａｙａｍａｉ，Ｐ．ｓｐｐ．，Ｔｙｐｈｕｌａｉｎｃａｒｎａｔａ，Ｔ．ｉｓｉｋａｒｉｅｎｓｉｓ，Ｆｕｓａｒｉｕｍｎｉｖａｌｅ，Ｓｃｌｅｒｏｔｉｎｉａｂｏｒｅａｌｉｓ）、
ベントグラスの赤焼病（Ｐｙｔｈｉｕｍａｐｈａｎｉｄｅｒｍａｔｕｍ）、炭そ病（Ｃｏｌｌｅｔｏｔｒｉｃｈｕｍｓｐ．）等が挙げられるが、本発明はこれらのみに限定されるものではない。 As plant diseases to be controlled by the compounds of the present invention,
Rice blast (Piculararia oryzae), sesame leaf blight (Cochliobolus miyabeanus), blight (Rhizoctonia solani), rice mildew (Claviceps virenk), leaf seedling (Gibberk) P. spinosum, Fusarium avenaceum, Fusarium solani, Fusarium spp., Rhizopus chinensis, R. oryzae, Rhizopus spp., Trichoderma virulence ), 褐条 disease (Acidovorax avenae), bacterial leaf blight (Xanthomonas oryzae), the inner 頴褐 Henbyo (Erwinia ananas),
Wheat stripe atrophy, Barley yellow mosaic virus, wheat powdery mildew (Erysiphe graminis f. Sp. Hordei, E. f. (Pyrenophora graminea), reticular rot (Pyrenophora teres), red mold (Gibberella zeae), rust (Puccinia striformis, P. graminis, P. recondita, P. yhorde) Rot (Tipula sp., Micronelliella nipivais), Bare Scab (Ustil) go tritici, U. nuda), cloud disease (Rhynchosporium secalis), leaf blight (Septoria trihortici), leaf blight (Leptospharia nodorum), small spot disease (Pseudocercosporella pallet) Snow rot large grain sclerotia (Myrioclerotinia borealis), wheat red snow rot (Monographella nivalis), withering disease (Gaeumanomyces graminis),
Citrus spot disease (Diaporthe citri), scab (Elsinoe fawcetii), fruit rot (Penicillium digitatum, P. italicum), scab (Xanthomonas campestris), gray mold (B)
Mongolia disease of Mongolia (Monilinia mali), rot (Valsa mali), powdery mildew (Podosphaera leukotricha), spotted leaf disease (Alternaria maria), scab (Venturia inaequalis)
Pear black spot disease (Venturia nashikocola), black spot disease (Alternaria kikuchiana), red star disease (Gymnosporium erbiotic asiaticum), plague (Phytophthora cergocterun, P. syringae), leaf syringae , Powdery mildew (Phyllactinia mary),
Peach ash streak (Monilinia fracticola), black streak (Cladosporium carpophilum), pomopsis rot (Phomophsis disease), pneumotrophic disease (Pseudocercospora circumscis, saury) deformans), plum scab (Pseudomonas syringae pv. morsprunorum), ash scab (Monilinia fracticola), black spot (Xanthomonas campestri pv. punil disease).
Pseudomonas syringae pv. Morsprunorum, black scab (Cladosporium carpophilum),
Grape downy mildew (Plasmopara viticola), black scab (Elsinoe ampelina), late rot (Glomerella gingulata), powdery mildew (Uncinula necatoris), rust (Amphidiaploid bud) Mold disease (Botrytis cinerea),
Oyster anthracnose (Glomerella orbicula), defoliation (Mycosphaerella nawai), gray mold (Botrytis cinerea), powdery mildew (Phyllactinia kakicola),
Downy mildew (Pseudoperenospora cubensis), anthracnose (Colletotrichumum orbicula), powdery mildew (Sphaerotheca fuliginea), vine blight (Didlymella brionum) , Sclerotia sclerotiorum, Fusarium solani, white silkworm (Sclerotium rolfsii), homopsis root rot (Phomopsis sclerotioides),
Cucumber brown spot (Corynespora casicicola), seedling blight (Pythium cucurbitaceacerum, P. debaryanum, Rhizoctonia solani), root rot (Pytium myriotrum, P.) Disease (Pseudomonas syringae pv. Lacrymans), purple coat rot (Helicobasidium mompa),
Brown rot of watermelon (Phytophthora capsici), plague (Phytophthora cryptogea),
Melon blight (Phythium debaryanum), plague (Phytophthora nicotianae),
Pumpkin plague (Phytophthora capsici),
Eggplant blight (Ralstonia solanacerum), wilt disease (Fusarium oxysporum), gray mold disease (Botrytis cinereaa), mycorrhizal disease (Sclerotinia sclerotiorum), white silkworm (Sclerotium olfactory)
Potato plague (Phytophthora infestans), summer plague (Alternaria solani), black scab (Thanatephorus cucumeris), black scab (Erwinia carotovora), common scab (Streptomyc spp.) Spongespora subterranea,
Phytophthora infestans, Phytophthora criptogea, Phytophathora capsici, Alternaria sulani, leaf mold disease (Fulvia uldus). , Brown rot, Phytophthora nicotianae, scab (Clavibacter michiganensis), brown root rot (Pyrenochaeta lycopersii), anthracnose (Colletotrichum gloesporis), (Verticillium dahliae), leaf spot (Stemphylium lycopersici),
Pepper plague (Phytophthora capsici), powdery mildew (Oidiopsis sicula), seedling blight (Rhizotonia solani), spot disease (Cercospora capsici),
Eggplant plague (Phytophthora infestans), brown rot (Phytophthora capsici), brown rot (Phomopsis vexans), powdery mildew (Erysiphe cichoracerum, Oidiopsis sicula)
Phytophthora sp., Downy mildew (Peronospora effusa), withering disease (Pythium aphanidermatum, P. myriotylum, P. paraecandrum, P. ultimum, sprout disease) ), Root rot (Aphanomyces cochlioides), spot disease (Heterosporia variabile),
White leaf blight of leeks (Phytophthora porori), blight (Phytophthora nicotianae), white silkworm (Sclerotium rolfsiii), seedling blight (Rhizoctonia solanii), black spot disease (Alternaria poultry disease) ), Downy mildew (Peronospora destructor), rust (Puccinia allii),
Leek wilt (Fusarium oxysporum), macular disease (Heterosporia aliii), red root rot (Pyrenochaeta terrestris), bacterium rot (Botrytis squamosa),
Onion dry rot (Fusarium oxysporum), smut (Urocystis cepulae), sclerotia nuclei (Cibolinia alli), gray mold (Botrytis cinerea), gray rot (Botrytis allirp), rot Burkholderia gladioli,
Brassicaceae vegetable downy mildew (Peronospora parasitica), root-knot disease (Plasmodiophora brassicae), white rust (Albuguoma macrospora), black spot (Alternaria japonica), A. brasco disease, A. brasic disease Erwinia carotovora), mycorrhizal disease (Sclerotinia sclerotiorum),
Strains of cabbage (Thanatephorus cucumeris), Verticillium dahliae, yellow cabbage (Verticillium dahliae), rot rot (Rhizotonia solani), gray scab Botrytis cinerea), Pythium ultimum,
Japanese radish anthracnose (Colletotrichum higginsianum), Verticillium albo-atrum,
Legume blight (Ralstonia solanacearum), wilt disease (Verticillium dahlliae), mycorrhizal disease (Sclerotinisia sclerotiorum), black root disease (Thielaviopsis sp.), Rust disease (Phakopsorapirosis) Fusarium oxysporum, Anthracnose (Colletotrichum truncatum, C. trifolii, Glomerella glycines, Gloeosporium sp.), Gray mold (Botrytis cinerea)
Soybean downy mildew (Peronospora manshurica), stem rot (Phytophthora sojae), leaf burning (Xanthomonas campestris pv. Glycines), purpura (Cercospora kikuchii), black spot (Cercospora kikuchii), black spot (Cercospora kikuchii)
Peanut black astringency (Mycosphaerella personata), brown spot (Mycosphaerella arachidis), pea powdery mildew (Erysiphe pisi),
Strawberry powdery mildew (Sphaerotheca aphanis), yellowing (Fusarium oxysporum), wilt (Verticillium dahliae), plague (Phytophthora cactrum, black spot bacterial disease (Xanthomonasca). , Potato disease (Mycosphaerella fragaliae), anthracnose (Colletotrichum acutatum, C. fragariae, Glomerella singularata), root rot (Phytophthora fragriae), gray mold disease lani), Wamadarabyo (Drenerophoma obscurans),
Lettuce sclerotia (Sclerotinia sclerotiorum), Blight blight (Rhizobacter solani), Soft rot (Erwinia carotovora), Blight (Pythium sp.), Root rot (Fusarium oxysporum), Gray rot, and gray rot Bacterial disease (Xanthomonas campestris pv. Vitians), Big vein disease (Lettuce big-vein virus), rot disease (Pseudomonas cichoris, P. marginalis pv. Virgin disease, P. marginalis pv. Virgin disease).
Burdock wilt disease (Fusarium oxysporum), black bruise (Rhizoctonia solani), black stripe disease (Itersonilia perplexans), black spot bacterial disease (Xanthomomonas camphorsis disease pv. irregulare), purple coat feather (Helicobasidium mompa),
Carrot wilt (Fusarium oxysporum), powdery mildew (Erysiphe heraclei), black leaf blight (Alternaria dauci), mildew (Rhizoctonia dauci), leaf rot (Pythium sulcium rot) Disease (Erwinia carotovora), root rot (Rhizoctonia solani), spot disease (Cercospora carrotae), purple coat (Helicobasidium mompa),
Chamochi rice blast (Exobasidium reticulatum), white scab (Elsinoe leucospila), brown scab (Pseudocercospora ocellata, Cerospora chas), rice blast (Exobasidium pex. Disease (Colletotrichum thea-sinensis),
Tobacco Red Star Disease (Alternaria alternata), Powdery Mildew (Erysiphe cichoacearum), Anthracnose (Colletotrichum cichoacearum),
Brown beet disease of sugar beet (Cercospora beticola), black root disease (Aphanomyces cochlioides), root beetle (Beet necrous yellow sp.), Phythium bebarium, Phomae horzole physic rape,
Rose scab (Diplocarpon rosae), powdery mildew (Sphaerotheca pannosa),
Chrysanthemum brown spot (Septoria chrysanthemiindicii), white rust (Puccinia horiana),
Fevering disease (Lycoperdon perlatum, Lepista subnudo, Marasmius oradees), pseudoleaf rot (Ceratobasidium spp.), Leaf disease (Gaemnomyces graminis) ), Pythium periplocum, P. graminicola, P. vanterpoulii, Rust (Puccinia spp.), Powdery mildew (Erysiphegramyis DC), Dollar spot disease (Sclerotinoposis) . pp., Typhula incarnata, T. isikariensis, Fusarium nivale, Sclerotinia borealis),
Bentgrass red blight (Pythium aphanidermatum), anthracnose (Colletotrichum sp.) And the like can be mentioned, but the present invention is not limited thereto.

本発明の化合物は、農園芸用殺菌剤としての使用以外に、医療用抗菌剤、動物用抗菌剤、木材、紙・パルプ、接着剤・塗料、繊維、皮革などの防菌・防かび剤、製造工場の冷却水路などの工業用殺菌剤としても使用できる。 In addition to use as agricultural and horticultural fungicides, the compounds of the present invention are antibacterial and antifungal agents such as medical antibacterial agents, animal antibacterial agents, wood, paper / pulp, adhesives / paints, fibers, leather, etc. It can also be used as an industrial disinfectant such as a cooling water channel in a manufacturing plant.

本発明化合物の、医療用抗菌剤、動物用抗菌剤として対象となる病原菌は、
Ｔｒｉｃｈｏｐｈｙｔｏｎｒｕｂｒｕｍ、Ｔｒｉｃｈｏｐｈｙｔｏｎｍｅｎｔａｇｒｏｐｈｙｔｅｓなどの白癬菌類、Ｃａｎｄｉｄａａｌｂｉｃａｎｓなどのカンジダ菌類、Ａｓｐｅｒｇｉｌｌｕｓｆｕｍｉｇａｔｕｓなどのアスペルギルス菌類Ｃｒｙｐｔｏｃｏｃｃｕｓｎｅｏｆｏｒｍａｓなどのクリプトコックス菌類などの真菌類、大腸菌（Ｅｓｃｈｅｒｉｃｈｉａｃｏｌｉ）、緑膿菌（Ｐｓｅｕｄｏｍｏｎａｓａｅｒｕｇｉｎｏｓａ）、インフルエンザ菌（Ｈａｅｍｏｐｈｉｌｕｓｉｎｆｌｕｅｎｚａｅ）などのグラム陰性細菌類、黄色ブドウ球菌（Ｓｔａｐｈｙｌｏｃｏｃｃｕｓａｕｒｅｕｓ）、化膿レンサ球菌（Ｓｔｒｅｐｔｏｃｏｃｃｕｓｐｙｏｇｅｎｅｓ）などのグラム陽性細菌類等が挙げられるが、本発明はこれらのみに限定されるものではない。 The antimicrobial agent for medical use of the compound of the present invention, the pathogenic bacteria that are targeted as animal antimicrobial agents,
Trichophyton rubrum, Trichophyton mentagrophytes, etc. Ringworm fungi, Candida albicans, Candida fungi, Aspergillus fumigatus fungi, E. coli, etc. Gram-negative bacteria such as Haemophilus influenzae, Gram-positive bacteria such as Staphylococcus aureus, Streptococcus pyogenes, and the like. It is not limited to only.

また、木材、紙・パルプ、接着剤・塗料、繊維、皮革などの防菌・防かび剤として対象となる菌株としては、
Ｔｙｒｏｍｙｃｅｓｐａｌｕｓｔｒｉｓ、Ｃｏｒｉｏｌｕｓｖｅｒｓｉｃｏｌｏｒなどの木材腐朽菌類、Ａｓｐｅｒｇｉｌｌｕｓｎｉｇｅｒ、Ａｓｐｅｒｇｉｌｌｕｓｔｅｒｒｅｕｓ、Ｅｕｒｏｔｉｕｍｔｏｎｏｐｈｉｌｕｍ、Ｐｅｎｉｃｉｌｌｉｕｍｃｉｔｒｉｎｕｍ、Ｐｅｎｉｃｉｌｌｉｕｍｆｕｎｉｃｕｌｏｓｕｍ、Ｒｈｉｚｏｐｕｓｏｒｙｚａｅ、Ｃｌａｄｏｓｐｏｒｉｕｍｃｌａｄｏｓｐｏｒｉｏｉｄｅｓ、Ａｕｒｅｏｂａｓｉｄｉｕｍｐｕｌｌｕｌａｎｓ、Ｇｌｉｏｃｌａｄｉｕｍｖｉｒｅｎｓ、Ｃｈａｅｔｏｍｉｕｍｇｌｏｂｏｓｕｍ、Ｆｕｓａｒｉｕｍｍｏｎｉｌｉｆｏｒｍｅ、Ｍｙｒｏｔｈｅｃｉｕｍｖｅｒｒｕｃａｒｉａなどの資材の劣化微生物類が挙げられる。 In addition, as strains targeted as antibacterial and antifungal agents for wood, paper / pulp, adhesives / paints, fibers, leather, etc.
Tyromyces palustris, wood-rotting fungi such as Coriolus versicolor, Aspergillus niger, Aspergillus terreus, Eurotium tonophilum, Penicillium citrinum, Penicillium funiculosum, Rhizopus oryzae, Cladosporium cladosporioides, Aureobasidium pullulans, Gliocladium virens, Chaetomium globosum, Fusarium moniliforme, of materials such as Myrothecium verrucaria Examples include degraded microorganisms.

工業用殺菌剤として対象となる菌株としては
Ｓｐｈａｅｒｏｔｉｌｉｓｎａｔａｎｓ、Ｚｏｏｇｌｏｅａｒａｍｉｇｅｒａなどのスライム菌類が挙げられるが、本発明はこれらのみに限定されるものではない。 Examples of strains that are targeted as industrial fungicides include slime fungi such as Sphaerotilis natans and Zoogloea ramigera, but the present invention is not limited thereto.

本発明の化合物は、農園芸用殺菌剤としての使用以外に、家畜、家禽、愛玩動物等の内部寄生虫防除剤としても使用できる。 The compound of the present invention can be used not only as an agricultural and horticultural fungicide but also as an endoparasite control agent for livestock, poultry, pets and the like.

本発明化合物の、内部寄生虫防除剤として対象となる内部寄生虫は、
ヘモンクス属（Ｈａｅｍｏｎｃｈｕｓ）、トリコストロンギルス属（Ｔｒｉｃｈｏｓｔｒｏｎｇｙｌｕｓ）、オステルターギヤ属（Ｏｓｔｅｒｔａｇｉａ）、ネマトディルス属（Ｎｅｍａｔｏｄｉｒｕｓ）、クーペリア属（Ｃｏｏｐｅｒｉａ）、アスカリス属（Ａｓｃａｒｉｓ）、ブノストムーム属（Ｂｕｎｏｓｔｏｍｕｍ）、エスファゴストムーム属（Ｏｅｓｏｐｈａｇｏｓｔｏｍｕｍ）、チャベルチア属（Ｃｈａｂｅｒｔｉａ）、トリキュリス属（Ｔｒｉｃｈｕｒｉｓ）、ストロンギルス属（Ｓｔｏｒｏｎｇｙｌｕｓ）、トリコネマ属（Ｔｒｉｃｈｏｎｅｍａ）、ディクチオカウルス属（Ｄｉｃｔｙｏｃａｕｌｕｓ）、キャピラリア属（Ｃａｐｉｌｌａｒｉａ）、ヘテラキス属（Ｈｅｔｅｒａｋｉｓ）、トキソカラ属（Ｔｏｘｏｃａｒａ）、アスカリディア属（Ａｓｃａｒｉｄｉａ）、オキシウリス属（Ｏｘｙｕｒｉｓ）、アンキロストーマ属（Ａｎｃｙｌｏｓｔｏｍａ）、ウンシナリア属（Ｕｎｃｉｎａｒｉａ）、トキサスカリス属（Ｔｏｘａｓｃａｒｉｓ）、パラスカリス属（Ｐａｒａｓｃａｒｉｓ）などの線虫類、
ブツヘレリア属（Ｗｕｃｈｅｒｅｒｉａ）、ブルージア属（Ｂｒｕｇｉａ）、オンコセルカ属（Ｏｎｃｈｏｃｅｃａ）、ディロフィラリア属（Ｄｉｒｏｆｉｌａｒｉａ）、ロア糸状虫属（Ｌｏａ）などのフィラリア科（Ｆｉｌａｒｉｉｄａｅ）線虫類、
ドラクンクルス属（Ｄｅａｃｕｎｃｕｌｕｓ）などの蛇状線虫科（Ｄｒａｃｕｎｃｕｌｉｄａｅ）線虫類、
犬条虫（Ｄｉｐｙｌｉｄｉｕｍｃａｎｉｎｕｍ）、猫条虫（Ｔａｅｎｉａｔａｅｎｉａｅｆｏｒｍｉｓ）、有鉤条虫（Ｔａｅｎｉａｓｏｌｉｕｍ）、無鉤条虫（Ｔａｅｎｉａｓａｇｉｎａｔａ）、縮小条虫（Ｈｙｍｅｎｏｌｅｐｉｓｄｉｍｉｎｕｔａ）、ベネデン条虫（Ｍｏｎｉｅｚｉａｂｅｎｅｄｅｎｉ）、広節裂頭条虫（Ｄｉｐｈｙｌｌｏｂｏｔｈｒｉｕｍｌａｔｕｍ）、マンソン裂頭条虫（Ｄｉｐｈｙｌｌｏｂｏｔｈｒｉｕｍｅｒｉｎａｃｅｉ）、単包条虫（Ｅｃｈｉｎｏｃｏｃｃｕｓｇｒａｎｕｌｏｓｕｓ）、多包条虫（Ｅｃｈｉｎｏｃｏｃｃｕｓｍｕｌｔｉｌｏｃｕｌａｒｉｓ）などの条虫類、
肝蛭（Ｆａｓｃｉｏｌａｈｅｐａｔｉｃａ，Ｆ．ｇｉｇａｎｔｉｃａ）、ウエステルマン肺吸虫（Ｐａｒａｇｏｎｉｍｕｓｗｅｓｔｅｒｍａｎｉｉ）、肥大吸虫（Ｆａｓｃｉｏｌｏｐｓｉｃｂｒｕｓｋｉ）、膵吸虫（Ｅｕｒｙｔｒｅｍａｐａｎｃｒｅａｔｉｃｕｍ，Ｅ．ｃｏｅｌｏｍａｔｉｃｕｍ）、肝吸虫（Ｃｌｏｎｏｒｃｈｉｓｓｉｎｅｎｓｉｓ）、日本住血吸虫（Ｓｃｈｉｓｔｏｓｏｍａｊａｐｏｎｉｃｕｍ）、ビルハルツ住血吸虫（Ｓｃｈｉｓｔｏｓｏｍａｈａｅｍａｔｏｂｉｕｍ）、マンソン住血吸虫（Ｓｃｈｉｓｔｏｓｏｍａｍａｎｓｏｎｉ）などの吸虫類、
エイメリア・テネラ（Ｅｉｍｅｒｉａｔｅｎｅｌｌａ）、エイメリア・アセルブリナ（Ｅｉｍｅｒｉａａｃｅｒｖｕｌｉｎａ）、エイメリア・ブルネッチ（Ｅｉｍｅｒｉａｂｒｕｎｅｔｔｉ）、エイメリア・マクシマ（Ｅｉｍｅｒｉａｍａｘｉｍａ）、エイメリア・ネカトリクス（Ｅｉｍｅｒｉａｎｅｃａｔｒｉｘ）、エイメリア・ボビス（Ｅｉｍｅｒｉａｂｏｖｉｓ）、エイメリア・オビノイダリス（Ｅｉｍｅｒｉａｏｖｉｎｏｉｄａｌｉｓ）のようなエイメリア類（Ｅｉｍｅｒｉａｓｐｐ．）、
クルーズトリパノソーマ（Ｔｒｙｐａｎｏｓｏｍｓａｃｒｕｚｉ）、リーシュマニア類（Ｌｅｉｓｈｍａｎｉａｓｐｐ．）、マラリア原虫（Ｐｌａｓｍｏｄｉｕｍｓｐｐ．）、バベシア類（Ｂａｂｅｓｉｓｓｐｐ．）、トリコモナス類（Ｔｒｉｃｈｏｍｏｎａｄｉｄａｅｓｐｐ．）、ヒストモナス類（Ｈｉｓｔｏｍａｎａｓｓｐｐ．）、ジアルディア類（Ｇｉａｒｄｉａｓｐｐ．）、トキソプラズマ類（Ｔｏｘｏｐｌａｓｍａｓｐｐ．）、赤痢アメーバ（Ｅｎｔａｍｏｅｂａｈｉｓｔｏｌｙｔｉｃａ）、タイレリア類（Ｔｈｅｉｌｅｒｉａｓｐｐ．）等が挙げられるが、本発明はこれらのみに限定されるものではない。
（製造法）
式（Ｉ）で表される化合物は、例えば、式（ＩＩ）で表される化合物と、式（ＩＩＩ）で表される化合物とを反応させることにより製造することができる。 The endoparasite which is a target of the present invention compound as an endoparasite control agent,
Haemonchus, Trichostrongillus, Ostertagia, Nematodirus, Cooperia, Ascarisum, Bnost Genus (Oesophagostoumum), Chabertia (Chabertia), Trichuris (Trichuris), Strongylus (Storongylus), Trichonema (Trichonema), Dictiocaurus (Dictyocaurus), Capriella i ), Toxocara , Asuka Lydia genus (Ascaridia), Okishiurisu genus (Oxyuris), Anne kilometers stoma genus (Ancylostoma), Unshinaria genus (Uncinaria), Tokisasukarisu genus (Toxascaris), nematodes such as Parasukarisu genus (Parascaris),
Filariidae nematodes such as Wuchereria, Brugia, Onchocerca, Dirofilaria, Loa, and the like,
Dracunculus nematodes such as the genus Deacunculus,
Dogpyridium (Dipyridium caninum), caterpillar (Taenia taeniaeformis), potato tapeworm (Taenia solium), scabies tapeworm (Taenia saginata), tapeworm (Hymenolepis diminta), Beneden edenedia C. elegans (Diphyllobothrium latum), C. elegans (Diphyllobothrium erinacei), Echinococcus granulosus, Echinococcus multiloculus, etc.
Fasciola hepatica (F. gigantica), Westermann pulmonary fluke (Paragonimus westermanii), hypertrophic fluke (Fasciolopsic brilliant), C. pulmonary fluke (E.) japonicum), Schistosoma haematobium, Schistosoma mansoni, etc.,
Eimeria tenella, Eimeria acervulina, Eimeria brunetti, Eimeria bimetti, Eimeria maxima, Eimeria maxima Eimerias such as Eimeria ovinoidalis (Eimeria spp.),
Trypanosoma cruzi, Leishmania spp., Plasmodium spp., Babesis spp., Trichomonida spp., Trichomonadida spp. (Giadia spp.), Toxoplasma spp., Shigella amoeba (Entamoeba histolytica), Theylerias (Theileria spp.) And the like, but the present invention is not limited thereto.
(Production method)
The compound represented by the formula (I) can be produced, for example, by reacting the compound represented by the formula (II) with the compound represented by the formula (III).

［式中、Ｘは塩素原子、臭素原子、ヨウ素原子、Ｃ_１〜Ｃ_４アルキルスルホニルオキシ（例えば、メタンスルホニルオキシ）、ハロスルホニルオキシ（例えば、フルオロスルホニルオキシ）、ハロ（Ｃ_１〜Ｃ_４）アルキルスルホニルオキシ（例えば、トリフルオロメタンスルホニルオキシ）又はアリールスルホニルオキシ（例えば、ベンゼンスルホニルオキシ）等の脱離基を表し、Ｒ^１、Ｒ^２、Ｒ^３、Ｒ^４、Ｒ^５、Ｒ^６、Ｒ^７、Ｒ^８、Ｒ^９、Ｒ^１０、Ａ及びＷは前記と同じ意味を表す。］
式（Ｉ）で表される本発明化合物は、式（ＩＩ）で表される化合物と式（ＩＩＩ）で表される化合物とを溶媒中又は無溶媒で、場合によっては塩基存在下反応させることにより得ることができる。溶媒を用いる場合、用いられる溶媒としては反応に不活性であればよく、例えばジエチルエーテル、テトラヒドロフラン、１，４−ジオキサン、１，２−ジメトキシエタン等のエーテル溶媒、ベンゼン、キシレン、トルエン等の芳香族炭化水素溶媒、ペンタン、ヘキサン、シクロヘキサン等の脂肪族炭化水素溶媒、ジクロロメタン、クロロホルム、１，２−ジクロロエタン等のハロゲン化炭化水素溶媒、アセトニトリル、プロピオニトリル等のニトリル溶媒、Ｎ，Ｎ−ジメチルホルムアミド、Ｎ，Ｎ−ジメチルアセトアミド、Ｎ−メチルピロリドン、Ｎ，Ｎ’−ジメチルイミダゾリジノン等のアミド溶媒、ジメチルスルホキシド或いはこれらの混合溶媒等が挙げられる。好ましくは、アセトニトリル、テトラヒドロフラン、Ｎ，Ｎ−ジメチルホルムアミド、Ｎ−メチルピロリドン、ジメチルスルホキシド及びこれらの混合物等が挙げられる。 [Wherein, X is a chlorine atom, a bromine atom, an iodine atom, a C ₁ -C ₄ alkylsulfonyloxy (eg, methanesulfonyloxy), a halosulfonyloxy (eg, fluorosulfonyloxy), a halo (C ₁ -C ₄ ) It represents a leaving group such as alkylsulfonyloxy (for example, trifluoromethanesulfonyloxy) or arylsulfonyloxy (for example, benzenesulfonyloxy), and R ¹ , R ² , R ³ , R ⁴ , R ⁵ , R ⁶ , R ⁷ , R ⁸ , R ⁹ , R ¹⁰ , A and W represent the same meaning as described above. ]
The compound of the present invention represented by the formula (I) is obtained by reacting the compound represented by the formula (II) and the compound represented by the formula (III) in a solvent or without a solvent, and optionally in the presence of a base. Can be obtained. When a solvent is used, the solvent used may be inert to the reaction. For example, an ether solvent such as diethyl ether, tetrahydrofuran, 1,4-dioxane, 1,2-dimethoxyethane, an aromatic such as benzene, xylene, and toluene. Hydrocarbon solvents, aliphatic hydrocarbon solvents such as pentane, hexane and cyclohexane, halogenated hydrocarbon solvents such as dichloromethane, chloroform and 1,2-dichloroethane, nitrile solvents such as acetonitrile and propionitrile, N, N-dimethyl Examples include amide solvents such as formamide, N, N-dimethylacetamide, N-methylpyrrolidone, N, N′-dimethylimidazolidinone, dimethyl sulfoxide, or a mixed solvent thereof. Preferably, acetonitrile, tetrahydrofuran, N, N-dimethylformamide, N-methylpyrrolidone, dimethyl sulfoxide, and a mixture thereof can be used.

該反応は塩基の存在下に行うことができる。用いることのできる塩基としては、例えばピリジン、２，６−ルチジン、４−ジメチルアミノピリジン、トリエチルアミン、ジイソプロピルエチルアミン、トリブチルアミン、Ｎ，Ｎ−ジメチルアニリン、１，４−ジアザビシクロ［２．２．２］オクタン（ＤＡＢＣＯ）、１，８−ジアザビシクロ［５．４．０］−７−ウンデセン（ＤＢＵ）又は１，５−ジアザビシクロ［４．３．０］−５−ノネン（ＤＢＮ）等の有機塩基、水酸化ナトリウム、水酸化カリウム、水素化ナトリウム、炭酸水素ナトリウム、炭酸カリウム、炭酸セシウム等の無機塩基が挙げられる。塩基の当量としては、式（ＩＩ）で表される化合物に対して０．１から１００当量の範囲で用いることができ、１から４０当量の範囲が好ましい。 The reaction can be performed in the presence of a base. Examples of the base that can be used include pyridine, 2,6-lutidine, 4-dimethylaminopyridine, triethylamine, diisopropylethylamine, tributylamine, N, N-dimethylaniline, and 1,4-diazabicyclo [2.2.2]. Organic base such as octane (DABCO), 1,8-diazabicyclo [5.4.0] -7-undecene (DBU) or 1,5-diazabicyclo [4.3.0] -5-nonene (DBN), water Inorganic bases such as sodium oxide, potassium hydroxide, sodium hydride, sodium hydrogen carbonate, potassium carbonate, cesium carbonate and the like can be mentioned. As an equivalent of a base, it can be used in the range of 0.1 to 100 equivalents with respect to the compound represented by the formula (II), and a range of 1 to 40 equivalents is preferable.

反応温度は−８０℃から反応混合物の還流温度まで任意の温度を設定することができ、０℃から反応混合物の還流温度の範囲が好ましい。 The reaction temperature can be set at an arbitrary temperature from −80 ° C. to the reflux temperature of the reaction mixture, and the range of 0 ° C. to the reflux temperature of the reaction mixture is preferable.

反応時間は、反応基質の濃度、反応温度によって変化するが、通常５分から１００時間の範囲で任意に設定でき、１時間から４８時間の範囲が好ましい。 The reaction time varies depending on the concentration of the reaction substrate and the reaction temperature, but can usually be arbitrarily set in the range of 5 minutes to 100 hours, and preferably in the range of 1 hour to 48 hours.

基質の当量としては、化合物（ＩＩ）は化合物（ＩＩＩ）に対して、０．５から５０当量の範囲で用いることができ、１から２０当量の範囲が好ましい。 As the equivalent of the substrate, compound (II) can be used in the range of 0.5 to 50 equivalents relative to compound (III), and preferably in the range of 1 to 20 equivalents.

反応終了後は、反応溶液中から通常の後処理により式（Ｉ）で表される化合物を得ることができる。例えば、反応混合物に水及びトルエン、酢酸エチル、ジエチルエーテル又はクロロホルム等の抽出溶媒を加えて抽出後、有機層を乾燥、濃縮することにより化合物（Ｉ）が得られる。化合物を精製する必要が生じた場合には、再結晶、カラムクロマトグラフィー等の任意の精製法によって分離、精製することができる。 After completion of the reaction, the compound represented by the formula (I) can be obtained from the reaction solution by ordinary post-treatment. For example, water and an extraction solvent such as toluene, ethyl acetate, diethyl ether or chloroform are added to the reaction mixture for extraction, and then the organic layer is dried and concentrated to obtain compound (I). When it becomes necessary to purify the compound, it can be separated and purified by any purification method such as recrystallization or column chromatography.

式（ＩＩ）で表される化合物の或るものは公知化合物であり、文献記載の公知の方法、例えばシンセシス［Ｓｙｎｔｈｅｓｉｓ］１９９５年、４巻、４３５頁等に記載の合成方法に準じて製造することができる。 Some of the compounds represented by formula (II) are known compounds, and are prepared according to known methods described in the literature, for example, synthesis methods described in Synthesis, 1995, Vol. 4, page 435, etc. be able to.

式（ＩＩＩ）で表される化合物の或るものは公知化合物であり、文献記載の公知の方法、例えば国際公開第２０１３／１６２９７２号等に記載の合成方法に準じて製造することができる。 Some of the compounds represented by the formula (III) are known compounds and can be produced according to known methods described in the literature, for example, synthetic methods described in International Publication No. 2013/162972.

本発明に包含される活性化合物としては、具体的には、第１表乃至第４表に示す化合物が挙げられる。但し、第１表乃至第４表の化合物は例示のためのものであって、本発明はこれらのみに限定されるものではない。 Specific examples of the active compound included in the present invention include compounds shown in Tables 1 to 4. However, the compounds in Tables 1 to 4 are for illustrative purposes, and the present invention is not limited thereto.

尚、表中、Ｍｅはメチル基を、Ｅｔはエチル基を、ｎＰｒはｎ−プロピル基を、ｉＰｒはｉ−プロピル基を、ｃＰｒはシクロプロピル基を、ｎＢｕはｎ−ブチル基を、ｃＢｕはシクロブチル基を、ｃＰｅｎはシクロペンチル基を、ｃＨｅｘはシクロヘキシル基を、Ｐｈはフェニル基を、Ａｃはアセチル基を、＝は２重結合を、≡は３重結合をそれぞれ表す。 In the table, Me represents a methyl group, Et represents an ethyl group, nPr represents an n-propyl group, iPr represents an i-propyl group, cPr represents a cyclopropyl group, nBu represents an n-butyl group, and cBu represents A cyclobutyl group, cPen represents a cyclopentyl group, cHex represents a cyclohexyl group, Ph represents a phenyl group, Ac represents an acetyl group, = represents a double bond, and ≡ represents a triple bond.

また、表中、Ｕ−１ａ、Ｕ−１ｂ、Ｕ−１ｅ、Ｕ−３ｂ、Ｕ−４ａ、Ｕ−４ｂ、Ｕ−４ｃ、Ｕ−４ｄ、Ｕ−４ｅ、Ｕ−４ｆ、及びＵ−４ｇで表される置換基は、それぞれ下記の構造を表す。 In the table, U-1a, U-1b, U-1e, U-3b, U-4a, U-4b, U-4c, U-4d, U-4e, U-4f, and U-4g The substituents represented represent the following structures, respectively.

［第１表］［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
Me 2-F U-4a 3-Cl-5-OMe U-4f 2-F-5-OCF₃
Me 2-Cl U-4a 3-Cl-5-OCF₃ U-4f 2-Cl-5-F
Me 2-Br U-4a 3-Br-5-F U-4f 2,5-di-Cl
Me 2-Me U-4a 3-Br-5-Cl U-4f 2-Cl-5-Br
Me 2-CF₃ U-4a 3,5-di-Br U-4f 2-Cl-5-Me
Me 2-OMe U-4a 3-Br-5-Me U-4f 2-Cl-5-CF₃
Me 2-OCF₃ U-4a 3-Br-5-CF₃ U-4f 2-Cl-5-OMe
Me 3-F U-4a 3-Br-5-OMe U-4f 2-Cl-5-OCF₃
Me 3-Cl U-4a 3-Br-5-OCF₃ U-4f 2-Br-5-F
Me 3-Br U-4a 3-Me-5-F U-4f 2-Br-5-Cl
Me 3-Me U-4a 3-Me-5-Cl U-4f 2,5-di-Br
Me 3-CF₃ U-4a 3-Me-5-Br U-4f 2-Br-5-Me
Me 3-OMe U-4a 3,5-di-Me U-4f 2-Br-5-CF₃
Me 3-OCF₃ U-4a 3-Me-5-CF₃ U-4f 2-Br-5-OMe
Me 4-F U-4a 3-Me-5-OMe U-4f 2-Br-5-OCF₃
Me 4-Cl U-4a 3-Me-5-OCF₃ U-4f 2-Me-5-F
Me 4-Br U-4a 3-CF₃-5-F U-4f 2-Me-5-Cl
Me 4-Me U-4a 3-CF₃-5-Cl U-4f 2-Me-5-Br
Me 4-CF₃ U-4a 3-CF₃-5-Br U-4f 2,5-di-Me
Me 4-OMe U-4a 3-CF₃-5-Me U-4f 2-Me-5-CF₃
Me 4-OCF₃ U-4a 3,5-di-CF₃ U-4f 2-Me-5-OMe
Me 5-F U-4a 3-CF₃-5-OMe U-4f 2-Me-5-OCF₃
Me 5-Cl U-4a 3-CF₃-5-OCF₃ U-4f 2-CF₃-5-F
Me 5-Br U-4a 3-OMe-5-F U-4f 2-CF₃-5-Cl
Me 5-Me U-4a 3-OMe-5-Cl U-4f 2-CF₃-5-Br
Me 5-CF₃ U-4a 3-OMe-5-Br U-4f 2-CF₃-5-Me
Me 5-OMe U-4a 3-OMe-5-Me U-4f 2,5-di-CF₃
Me 5-OCF₃ U-4a 3-OMe-5-CF₃ U-4f 2-CF₃-5-OMe
Et 2-F U-4a 3,5-di-OMe U-4f 2-CF₃-5-OCF₃
Et 2-Cl U-4a 3-OMe-5-OCF₃ U-4f 2-OMe-5-F
Et 2-Br U-4a 3-OCF₃-5-F U-4f 2-OMe-5-Cl
Et 2-Me U-4a 3-OCF₃-5-Cl U-4f 2-OMe-5-Br
Et 2-CF₃ U-4a 3-OCF₃-5-Br U-4f 2-OMe-5-Me
Et 2-OMe U-4a 3-OCF₃-5-Me U-4f 2-OMe-5-CF₃
Et 2-OCF₃ U-4a 3-OCF₃-5-CF₃ U-4f 2,5-di-OMe
Et 3-F U-4a 3-OCF₃-5-OMe U-4f 2-OMe-5-OCF₃
Et 3-Cl U-4a 3,5-di-OCF₃ U-4f 2-OCF₃-5-F
Et 3-Br CF₃ 2,3-di-F U-4f 2-OCF₃-5-Cl
Et 3-Me CF₃ 2-F-3-Cl U-4f 2-OCF₃-5-Br
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
Et 3-CF₃ CF₃ 2-F-3-Br U-4f 2-OCF₃-5-Me
Et 3-OMe CF₃ 2-F-3-Me U-4f 2-OCF₃-5-CF₃
Et 3-OCF₃ CF₃ 2-F-3-CF₃ U-4f 2-OCF₃-5-OMe
Et 4-F CF₃ 2-F-3-OMe U-4f 2,5-di-OCF₃
Et 4-Cl CF₃ 2-F-3-OCF₃ U-4f 3,4-di-F
Et 4-Br CF₃ 2-Cl-3-F U-4f 3-F-4-Cl
Et 4-Me CF₃ 2,3-di-Cl U-4f 3-F-4-Br
Et 4-CF₃ CF₃ 2-Cl-3-Br U-4f 3-F-4-Me
Et 4-OMe CF₃ 2-Cl-3-Me U-4f 3-F-4-CF₃
Et 4-OCF₃ CF₃ 2-Cl-3-CF₃ U-4f 3-F-4-OMe
Et 5-F CF₃ 2-Cl-3-OMe U-4f 3-F-4-OCF₃
Et 5-Cl CF₃ 2-Cl-3-OCF₃ U-4f 3-Cl-4-F
Et 5-Br CF₃ 2-Br-3-F U-4f 3,4-di-Cl
Et 5-Me CF₃ 2-Br-3-Cl U-4f 3-Cl-4-Br
Et 5-CF₃ CF₃ 2,3-di-Br U-4f 3-Cl-4-Me
Et 5-OMe CF₃ 2-Br-3-Me U-4f 3-Cl-4-CF₃
Et 5-OCF₃ CF₃ 2-Br-3-CF₃ U-4f 3-Cl-4-OMe
iPr 2-F CF₃ 2-Br-3-OMe U-4f 3-Cl-4-OCF₃
iPr 2-Cl CF₃ 2-Br-3-OCF₃ U-4f 3-Br-4-F
iPr 2-Br CF₃ 2-Me-3-F U-4f 3-Br-4-Cl
iPr 2-Me CF₃ 2-Me-3-Cl U-4f 3,4-di-Br
iPr 2-CF₃ CF₃ 2-Me-3-Br U-4f 3-Br-4-Me
iPr 2-OMe CF₃ 2,3-di-Me U-4f 3-Br-4-CF₃
iPr 2-OCF₃ CF₃ 2-Me-3-CF₃ U-4f 3-Br-4-OMe
iPr 3-F CF₃ 2-Me-3-OMe U-4f 3-Br-4-OCF₃
iPr 3-Cl CF₃ 2-Me-3-OCF₃ U-4f 3-Me-4-F
iPr 3-Br CF₃ 2-CF₃-3-F U-4f 3-Me-4-Cl
iPr 3-Me CF₃ 2-CF₃-3-Cl U-4f 3-Me-4-Br
iPr 3-CF₃ CF₃ 2-CF₃-3-Br U-4f 3,4-di-Me
iPr 3-OMe CF₃ 2-CF₃-3-Me U-4f 3-Me-4-CF₃
iPr 3-OCF₃ CF₃ 2,3-di-CF₃ U-4f 3-Me-4-OMe
iPr 4-F CF₃ 2-CF₃-3-OMe U-4f 3-Me-4-OCF₃
iPr 4-Cl CF₃ 2-CF₃-3-OCF₃ U-4f 3-CF₃-4-F
iPr 4-Br CF₃ 2-OMe-3-F U-4f 3-CF₃-4-Cl
iPr 4-Me CF₃ 2-OMe-3-Cl U-4f 3-CF₃-4-Br
iPr 4-CF₃ CF₃ 2-OMe-3-Br U-4f 3-CF₃-4-Me
iPr 4-OMe CF₃ 2-OMe-3-Me U-4f 3,4-di-CF₃
iPr 4-OCF₃ CF₃ 2-OMe-3-CF₃ U-4f 3-CF₃-4-OMe
iPr 5-F CF₃ 2,3-di-OMe U-4f 3-CF₃-4-OCF₃
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
iPr 5-Cl CF₃ 2-OMe-3-OCF₃ U-4f 3-OMe-4-F
iPr 5-Br CF₃ 2-OCF₃-3-F U-4f 3-OMe-4-Cl
iPr 5-Me CF₃ 2-OCF₃-3-Cl U-4f 3-OMe-4-Br
iPr 5-CF₃ CF₃ 2-OCF₃-3-Br U-4f 3-OMe-4-Me
iPr 5-OMe CF₃ 2-OCF₃-3-Me U-4f 3-OMe-4-CF₃
iPr 5-OCF₃ CF₃ 2-OCF₃-3-CF₃ U-4f 3,4-di-OMe
U-4a 2-F CF₃ 2-OCF₃-3-OMe U-4f 3-OMe-4-OCF₃
U-4a 2-Cl CF₃ 2,3-di-OCF₃ U-4f 3-OCF₃-4-F
U-4a 2-Br CF₃ 2,4-di-F U-4f 3-OCF₃-4-Cl
U-4a 2-Me CF₃ 2-F-4-Cl U-4f 3-OCF₃-4-Br
U-4a 2-CF₃ CF₃ 2-F-4-Br U-4f 3-OCF₃-4-Me
U-4a 2-OMe CF₃ 2-F-4-Me U-4f 3-OCF₃-4-CF₃
U-4a 2-OCF₃ CF₃ 2-F-4-CF₃ U-4f 3-OCF₃-4-OMe
U-4a 3-F CF₃ 2-F-4-OMe U-4f 3,4-di-OCF₃
U-4a 3-Cl CF₃ 2-F-4-OCF₃ U-4f 3,5-di-F
U-4a 3-Br CF₃ 2-Cl-4-F U-4f 3-F-5-Cl
U-4a 3-Me CF₃ 2,4-di-Cl U-4f 3-F-5-Br
U-4a 3-CF₃ CF₃ 2-Cl-4-Br U-4f 3-F-5-Me
U-4a 3-OMe CF₃ 2-Cl-4-Me U-4f 3-F-5-CF₃
U-4a 3-OCF₃ CF₃ 2-Cl-4-CF₃ U-4f 3-F-5-OMe
U-4a 4-F CF₃ 2-Cl-4-OMe U-4f 3-F-5-OCF₃
U-4a 4-Cl CF₃ 2-Cl-4-OCF₃ U-4f 3-Cl-5-F
U-4a 4-Br CF₃ 2-Br-4-F U-4f 3,5-di-Cl
U-4a 4-Me CF₃ 2-Br-4-Cl U-4f 3-Cl-5-Br
U-4a 4-CF₃ CF₃ 2,4-di-Br U-4f 3-Cl-5-Me
U-4a 4-OMe CF₃ 2-Br-4-Me U-4f 3-Cl-5-CF₃
U-4a 4-OCF₃ CF₃ 2-Br-4-CF₃ U-4f 3-Cl-5-OMe
U-4a 5-F CF₃ 2-Br-4-OMe U-4f 3-Cl-5-OCF₃
U-4a 5-Cl CF₃ 2-Br-4-OCF₃ U-4f 3-Br-5-F
U-4a 5-Br CF₃ 2-Me-4-F U-4f 3-Br-5-Cl
U-4a 5-Me CF₃ 2-Me-4-Cl U-4f 3,5-di-Br
U-4a 5-CF₃ CF₃ 2-Me-4-Br U-4f 3-Br-5-Me
U-4a 5-OMe CF₃ 2,4-di-Me U-4f 3-Br-5-CF₃
U-4a 5-OCF₃ CF₃ 2-Me-4-CF₃ U-4f 3-Br-5-OMe
CF₃ 2-F CF₃ 2-Me-4-OMe U-4f 3-Br-5-OCF₃
CF₃ 2-Cl CF₃ 2-Me-4-OCF₃ U-4f 3-Me-5-F
CF₃ 2-Br CF₃ 2-CF₃-4-F U-4f 3-Me-5-Cl
CF₃ 2-Me CF₃ 2-CF₃-4-Cl U-4f 3-Me-5-Br
CF₃ 2-CF₃ CF₃ 2-CF₃-4-Br U-4f 3,5-di-Me
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
CF₃ 2-OMe CF₃ 2-CF₃-4-Me U-4f 3-Me-5-CF₃
CF₃ 2-OCF₃ CF₃ 2,4-di-CF₃ U-4f 3-Me-5-OMe
CF₃ 3-F CF₃ 2-CF₃-4-OMe U-4f 3-Me-5-OCF₃
CF₃ 3-Cl CF₃ 2-CF₃-4-OCF₃ U-4f 3-CF₃-5-F
CF₃ 3-Br CF₃ 2-OMe-4-F U-4f 3-CF₃-5-Cl
CF₃ 3-Me CF₃ 2-OMe-4-Cl U-4f 3-CF₃-5-Br
CF₃ 3-CF₃ CF₃ 2-OMe-4-Br U-4f 3-CF₃-5-Me
CF₃ 3-OMe CF₃ 2-OMe-4-Me U-4f 3,5-di-CF₃
CF₃ 3-OCF₃ CF₃ 2-OMe-4-CF₃ U-4f 3-CF₃-5-OMe
CF₃ 4-F CF₃ 2,4-di-OMe U-4f 3-CF₃-5-OCF₃
CF₃ 4-Cl CF₃ 2-OMe-4-OCF₃ U-4f 3-OMe-5-F
CF₃ 4-Br CF₃ 2-OCF₃-4-F U-4f 3-OMe-5-Cl
CF₃ 4-Me CF₃ 2-OCF₃-4-Cl U-4f 3-OMe-5-Br
CF₃ 4-CF₃ CF₃ 2-OCF₃-4-Br U-4f 3-OMe-5-Me
CF₃ 4-OMe CF₃ 2-OCF₃-4-Me U-4f 3-OMe-5-CF₃
CF₃ 4-OCF₃ CF₃ 2-OCF₃-4-CF₃ U-4f 3,5-di-OMe
CF₃ 5-F CF₃ 2-OCF₃-4-OMe U-4f 3-OMe-5-OCF₃
CF₃ 5-Cl CF₃ 2,4-di-OCF₃ U-4f 3-OCF₃-5-F
CF₃ 5-Br CF₃ 2,5-di-F U-4f 3-OCF₃-5-Cl
CF₃ 5-Me CF₃ 2-F-5-Cl U-4f 3-OCF₃-5-Br
CF₃ 5-CF₃ CF₃ 2-F-5-Br U-4f 3-OCF₃-5-Me
CF₃ 5-OMe CF₃ 2-F-5-Me U-4f 3-OCF₃-5-CF₃
CF₃ 5-OCF₃ CF₃ 2-F-5-CF₃ U-4f 3-OCF₃-5-OMe
cPr 2-F CF₃ 2-F-5-OMe U-4f 3,5-di-OCF₃
cPr 2-Cl CF₃ 2-F-5-OCF₃ U-4g 2,3-di-F
cPr 2-Br CF₃ 2-Cl-5-F U-4g 2-F-3-Cl
cPr 2-Me CF₃ 2,5-di-Cl U-4g 2-F-3-Br
cPr 2-CF₃ CF₃ 2-Cl-5-Br U-4g 2-F-3-Me
cPr 2-OMe CF₃ 2-Cl-5-Me U-4g 2-F-3-CF₃
cPr 2-OCF₃ CF₃ 2-Cl-5-CF₃ U-4g 2-F-3-OMe
cPr 3-F CF₃ 2-Cl-5-OMe U-4g 2-F-3-OCF₃
cPr 3-Cl CF₃ 2-Cl-5-OCF₃ U-4g 2-Cl-3-F
cPr 3-Br CF₃ 2-Br-5-F U-4g 2,3-di-Cl
cPr 3-Me CF₃ 2-Br-5-Cl U-4g 2-Cl-3-Br
cPr 3-CF₃ CF₃ 2,5-di-Br U-4g 2-Cl-3-Me
cPr 3-OMe CF₃ 2-Br-5-Me U-4g 2-Cl-3-CF₃
cPr 3-OCF₃ CF₃ 2-Br-5-CF₃ U-4g 2-Cl-3-OMe
cPr 4-F CF₃ 2-Br-5-OMe U-4g 2-Cl-3-OCF₃
cPr 4-Cl CF₃ 2-Br-5-OCF₃ U-4g 2-Br-3-F
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
cPr 4-Br CF₃ 2-Me-5-F U-4g 2-Br-3-Cl
cPr 4-Me CF₃ 2-Me-5-Cl U-4g 2,3-di-Br
cPr 4-CF₃ CF₃ 2-Me-5-Br U-4g 2-Br-3-Me
cPr 4-OMe CF₃ 2,5-di-Me U-4g 2-Br-3-CF₃
cPr 4-OCF₃ CF₃ 2-Me-5-CF₃ U-4g 2-Br-3-OMe
cPr 5-F CF₃ 2-Me-5-OMe U-4g 2-Br-3-OCF₃
cPr 5-Cl CF₃ 2-Me-5-OCF₃ U-4g 2-Me-3-F
cPr 5-Br CF₃ 2-CF₃-5-F U-4g 2-Me-3-Cl
cPr 5-Me CF₃ 2-CF₃-5-Cl U-4g 2-Me-3-Br
cPr 5-CF₃ CF₃ 2-CF₃-5-Br U-4g 2,3-di-Me
cPr 5-OMe CF₃ 2-CF₃-5-Me U-4g 2-Me-3-CF₃
cPr 5-OCF₃ CF₃ 2,5-di-CF₃ U-4g 2-Me-3-OMe
U-4b 2-F CF₃ 2-CF₃-5-OMe U-4g 2-Me-3-OCF₃
U-4b 2-Cl CF₃ 2-CF₃-5-OCF₃ U-4g 2-CF₃-3-F
U-4b 2-Br CF₃ 2-OMe-5-F U-4g 2-CF₃-3-Cl
U-4b 2-Me CF₃ 2-OMe-5-Cl U-4g 2-CF₃-3-Br
U-4b 2-CF₃ CF₃ 2-OMe-5-Br U-4g 2-CF₃-3-Me
U-4b 2-OMe CF₃ 2-OMe-5-Me U-4g 2,3-di-CF₃
U-4b 2-OCF₃ CF₃ 2-OMe-5-CF₃ U-4g 2-CF₃-3-OMe
U-4b 3-F CF₃ 2,5-di-OMe U-4g 2-CF₃-3-OCF₃
U-4b 3-Cl CF₃ 2-OMe-5-OCF₃ U-4g 2-OMe-3-F
U-4b 3-Br CF₃ 2-OCF₃-5-F U-4g 2-OMe-3-Cl
U-4b 3-Me CF₃ 2-OCF₃-5-Cl U-4g 2-OMe-3-Br
U-4b 3-CF₃ CF₃ 2-OCF₃-5-Br U-4g 2-OMe-3-Me
U-4b 3-OMe CF₃ 2-OCF₃-5-Me U-4g 2-OMe-3-CF₃
U-4b 3-OCF₃ CF₃ 2-OCF₃-5-CF₃ U-4g 2,3-di-OMe
U-4b 4-F CF₃ 2-OCF₃-5-OMe U-4g 2-OMe-3-OCF₃
U-4b 4-Cl CF₃ 2,5-di-OCF₃ U-4g 2-OCF₃-3-F
U-4b 4-Br CF₃ 3,4-di-F U-4g 2-OCF₃-3-Cl
U-4b 4-Me CF₃ 3-F-4-Cl U-4g 2-OCF₃-3-Br
U-4b 4-CF₃ CF₃ 3-F-4-Br U-4g 2-OCF₃-3-Me
U-4b 4-OMe CF₃ 3-F-4-Me U-4g 2-OCF₃-3-CF₃
U-4b 4-OCF₃ CF₃ 3-F-4-CF₃ U-4g 2-OCF₃-3-OMe
U-4b 5-F CF₃ 3-F-4-OMe U-4g 2,3-di-OCF₃
U-4b 5-Cl CF₃ 3-F-4-OCF₃ U-4g 2,4-di-F
U-4b 5-Br CF₃ 3-Cl-4-F U-4g 2-F-4-Cl
U-4b 5-Me CF₃ 3,4-di-Cl U-4g 2-F-4-Br
U-4b 5-CF₃ CF₃ 3-Cl-4-Br U-4g 2-F-4-Me
U-4b 5-OMe CF₃ 3-Cl-4-Me U-4g 2-F-4-CF₃
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
U-4b 5-OCF₃ CF₃ 3-Cl-4-CF₃ U-4g 2-F-4-OMe
U-4c 2-F CF₃ 3-Cl-4-OMe U-4g 2-F-4-OCF₃
U-4c 2-Cl CF₃ 3-Cl-4-OCF₃ U-4g 2-Cl-4-F
U-4c 2-Br CF₃ 3-Br-4-F U-4g 2,4-di-Cl
U-4c 2-Me CF₃ 3-Br-4-Cl U-4g 2-Cl-4-Br
U-4c 2-CF₃ CF₃ 3,4-di-Br U-4g 2-Cl-4-Me
U-4c 2-OMe CF₃ 3-Br-4-Me U-4g 2-Cl-4-CF₃
U-4c 2-OCF₃ CF₃ 3-Br-4-CF₃ U-4g 2-Cl-4-OMe
U-4c 3-F CF₃ 3-Br-4-OMe U-4g 2-Cl-4-OCF₃
U-4c 3-Cl CF₃ 3-Br-4-OCF₃ U-4g 2-Br-4-F
U-4c 3-Br CF₃ 3-Me-4-F U-4g 2-Br-4-Cl
U-4c 3-Me CF₃ 3-Me-4-Cl U-4g 2,4-di-Br
U-4c 3-CF₃ CF₃ 3-Me-4-Br U-4g 2-Br-4-Me
U-4c 3-OMe CF₃ 3,4-di-Me U-4g 2-Br-4-CF₃
U-4c 3-OCF₃ CF₃ 3-Me-4-CF₃ U-4g 2-Br-4-OMe
U-4c 4-F CF₃ 3-Me-4-OMe U-4g 2-Br-4-OCF₃
U-4c 4-Cl CF₃ 3-Me-4-OCF₃ U-4g 2-Me-4-F
U-4c 4-Br CF₃ 3-CF₃-4-F U-4g 2-Me-4-Cl
U-4c 4-Me CF₃ 3-CF₃-4-Cl U-4g 2-Me-4-Br
U-4c 4-CF₃ CF₃ 3-CF₃-4-Br U-4g 2,4-di-Me
U-4c 4-OMe CF₃ 3-CF₃-4-Me U-4g 2-Me-4-CF₃
U-4c 4-OCF₃ CF₃ 3,4-di-CF₃ U-4g 2-Me-4-OMe
U-4c 5-F CF₃ 3-CF₃-4-OMe U-4g 2-Me-4-OCF₃
U-4c 5-Cl CF₃ 3-CF₃-4-OCF₃ U-4g 2-CF₃-4-F
U-4c 5-Br CF₃ 3-OMe-4-F U-4g 2-CF₃-4-Cl
U-4c 5-Me CF₃ 3-OMe-4-Cl U-4g 2-CF₃-4-Br
U-4c 5-CF₃ CF₃ 3-OMe-4-Br U-4g 2-CF₃-4-Me
U-4c 5-OMe CF₃ 3-OMe-4-Me U-4g 2,4-di-CF₃
U-4c 5-OCF₃ CF₃ 3-OMe-4-CF₃ U-4g 2-CF₃-4-OMe
U-4d 2-F CF₃ 3,4-di-OMe U-4g 2-CF₃-4-OCF₃
U-4d 2-Cl CF₃ 3-OMe-4-OCF₃ U-4g 2-OMe-4-F
U-4d 2-Br CF₃ 3-OCF₃-4-F U-4g 2-OMe-4-Cl
U-4d 2-Me CF₃ 3-OCF₃-4-Cl U-4g 2-OMe-4-Br
U-4d 2-CF₃ CF₃ 3-OCF₃-4-Br U-4g 2-OMe-4-Me
U-4d 2-OMe CF₃ 3-OCF₃-4-Me U-4g 2-OMe-4-CF₃
U-4d 2-OCF₃ CF₃ 3-OCF₃-4-CF₃ U-4g 2,4-di-OMe
U-4d 3-F CF₃ 3-OCF₃-4-OMe U-4g 2-OMe-4-OCF₃
U-4d 3-Cl CF₃ 3,4-di-OCF₃ U-4g 2-OCF₃-4-F
U-4d 3-Br CF₃ 3,5-di-F U-4g 2-OCF₃-4-Cl
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
U-4d 3-Me CF₃ 3-F-5-Cl U-4g 2-OCF₃-4-Br
U-4d 3-CF₃ CF₃ 3-F-5-Br U-4g 2-OCF₃-4-Me
U-4d 3-OMe CF₃ 3-F-5-Me U-4g 2-OCF₃-4-CF₃
U-4d 3-OCF₃ CF₃ 3-F-5-CF₃ U-4g 2-OCF₃-4-OMe
U-4d 4-F CF₃ 3-F-5-OMe U-4g 2,4-di-OCF₃
U-4d 4-Cl CF₃ 3-F-5-OCF₃ U-4g 2,5-di-F
U-4d 4-Br CF₃ 3-Cl-5-F U-4g 2-F-5-Cl
U-4d 4-Me CF₃ 3,5-di-Cl U-4g 2-F-5-Br
U-4d 4-CF₃ CF₃ 3-Cl-5-Br U-4g 2-F-5-Me
U-4d 4-OMe CF₃ 3-Cl-5-Me U-4g 2-F-5-CF₃
U-4d 4-OCF₃ CF₃ 3-Cl-5-CF₃ U-4g 2-F-5-OMe
U-4d 5-F CF₃ 3-Cl-5-OMe U-4g 2-F-5-OCF₃
U-4d 5-Cl CF₃ 3-Cl-5-OCF₃ U-4g 2-Cl-5-F
U-4d 5-Br CF₃ 3-Br-5-F U-4g 2,5-di-Cl
U-4d 5-Me CF₃ 3-Br-5-Cl U-4g 2-Cl-5-Br
U-4d 5-CF₃ CF₃ 3,5-di-Br U-4g 2-Cl-5-Me
U-4d 5-OMe CF₃ 3-Br-5-Me U-4g 2-Cl-5-CF₃
U-4d 5-OCF₃ CF₃ 3-Br-5-CF₃ U-4g 2-Cl-5-OMe
U-4e 2-F CF₃ 3-Br-5-OMe U-4g 2-Cl-5-OCF₃
U-4e 2-Cl CF₃ 3-Br-5-OCF₃ U-4g 2-Br-5-F
U-4e 2-Br CF₃ 3-Me-5-F U-4g 2-Br-5-Cl
U-4e 2-Me CF₃ 3-Me-5-Cl U-4g 2,5-di-Br
U-4e 2-CF₃ CF₃ 3-Me-5-Br U-4g 2-Br-5-Me
U-4e 2-OMe CF₃ 3,5-di-Me U-4g 2-Br-5-CF₃
U-4e 2-OCF₃ CF₃ 3-Me-5-CF₃ U-4g 2-Br-5-OMe
U-4e 3-F CF₃ 3-Me-5-OMe U-4g 2-Br-5-OCF₃
U-4e 3-Cl CF₃ 3-Me-5-OCF₃ U-4g 2-Me-5-F
U-4e 3-Br CF₃ 3-CF₃-5-F U-4g 2-Me-5-Cl
U-4e 3-Me CF₃ 3-CF₃-5-Cl U-4g 2-Me-5-Br
U-4e 3-CF₃ CF₃ 3-CF₃-5-Br U-4g 2,5-di-Me
U-4e 3-OMe CF₃ 3-CF₃-5-Me U-4g 2-Me-5-CF₃
U-4e 3-OCF₃ CF₃ 3,5-di-CF₃ U-4g 2-Me-5-OMe
U-4e 4-F CF₃ 3-CF₃-5-OMe U-4g 2-Me-5-OCF₃
U-4e 4-Cl CF₃ 3-CF₃-5-OCF₃ U-4g 2-CF₃-5-F
U-4e 4-Br CF₃ 3-OMe-5-F U-4g 2-CF₃-5-Cl
U-4e 4-Me CF₃ 3-OMe-5-Cl U-4g 2-CF₃-5-Br
U-4e 4-CF₃ CF₃ 3-OMe-5-Br U-4g 2-CF₃-5-Me
U-4e 4-OMe CF₃ 3-OMe-5-Me U-4g 2,5-di-CF₃
U-4e 4-OCF₃ CF₃ 3-OMe-5-CF₃ U-4g 2-CF₃-5-OMe
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
U-4e 5-F CF₃ 3,5-di-OMe U-4g 2-CF₃-5-OCF₃
U-4e 5-Cl CF₃ 3-OMe-5-OCF₃ U-4g 2-OMe-5-F
U-4e 5-Br CF₃ 3-OCF₃-5-F U-4g 2-OMe-5-Cl
U-4e 5-Me CF₃ 3-OCF₃-5-Cl U-4g 2-OMe-5-Br
U-4e 5-CF₃ CF₃ 3-OCF₃-5-Br U-4g 2-OMe-5-Me
U-4e 5-OMe CF₃ 3-OCF₃-5-Me U-4g 2-OMe-5-CF₃
U-4e 5-OCF₃ CF₃ 3-OCF₃-5-CF₃ U-4g 2,5-di-OMe
U-4f 2-F CF₃ 3-OCF₃-5-OMe U-4g 2-OMe-5-OCF₃
U-4f 2-Cl CF₃ 3,5-di-OCF₃ U-4g 2-OCF₃-5-F
U-4f 2-Br cPr 2,3-di-F U-4g 2-OCF₃-5-Cl
U-4f 2-Me cPr 2-F-3-Cl U-4g 2-OCF₃-5-Br
U-4f 2-CF₃ cPr 2-F-3-Br U-4g 2-OCF₃-5-Me
U-4f 2-OMe cPr 2-F-3-Me U-4g 2-OCF₃-5-CF₃
U-4f 2-OCF₃ cPr 2-F-3-CF₃ U-4g 2-OCF₃-5-OMe
U-4f 3-F cPr 2-F-3-OMe U-4g 2,5-di-OCF₃
U-4f 3-Cl cPr 2-F-3-OCF₃ U-4g 3,4-di-F
U-4f 3-Br cPr 2-Cl-3-F U-4g 3-F-4-Cl
U-4f 3-Me cPr 2,3-di-Cl U-4g 3-F-4-Br
U-4f 3-CF₃ cPr 2-Cl-3-Br U-4g 3-F-4-Me
U-4f 3-OMe cPr 2-Cl-3-Me U-4g 3-F-4-CF₃
U-4f 3-OCF₃ cPr 2-Cl-3-CF₃ U-4g 3-F-4-OMe
U-4f 4-F cPr 2-Cl-3-OMe U-4g 3-F-4-OCF₃
U-4f 4-Cl cPr 2-Cl-3-OCF₃ U-4g 3-Cl-4-F
U-4f 4-Br cPr 2-Br-3-F U-4g 3,4-di-Cl
U-4f 4-Me cPr 2-Br-3-Cl U-4g 3-Cl-4-Br
U-4f 4-CF₃ cPr 2,3-di-Br U-4g 3-Cl-4-Me
U-4f 4-OMe cPr 2-Br-3-Me U-4g 3-Cl-4-CF₃
U-4f 4-OCF₃ cPr 2-Br-3-CF₃ U-4g 3-Cl-4-OMe
U-4f 5-F cPr 2-Br-3-OMe U-4g 3-Cl-4-OCF₃
U-4f 5-Cl cPr 2-Br-3-OCF₃ U-4g 3-Br-4-F
U-4f 5-Br cPr 2-Me-3-F U-4g 3-Br-4-Cl
U-4f 5-Me cPr 2-Me-3-Cl U-4g 3,4-di-Br
U-4f 5-CF₃ cPr 2-Me-3-Br U-4g 3-Br-4-Me
U-4f 5-OMe cPr 2,3-di-Me U-4g 3-Br-4-CF₃
U-4f 5-OCF₃ cPr 2-Me-3-CF₃ U-4g 3-Br-4-OMe
U-4g 2-F cPr 2-Me-3-OMe U-4g 3-Br-4-OCF₃
U-4g 2-Cl cPr 2-Me-3-OCF₃ U-4g 3-Me-4-F
U-4g 2-Br cPr 2-CF₃-3-F U-4g 3-Me-4-Cl
U-4g 2-Me cPr 2-CF₃-3-Cl U-4g 3-Me-4-Br
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
U-4g 2-CF₃ cPr 2-CF₃-3-Br U-4g 3,4-di-Me
U-4g 2-OMe cPr 2-CF₃-3-Me U-4g 3-Me-4-CF₃
U-4g 2-OCF₃ cPr 2,3-di-CF₃ U-4g 3-Me-4-OMe
U-4g 3-F cPr 2-CF₃-3-OMe U-4g 3-Me-4-OCF₃
U-4g 3-Cl cPr 2-CF₃-3-OCF₃ U-4g 3-CF₃-4-F
U-4g 3-Br cPr 2-OMe-3-F U-4g 3-CF₃-4-Cl
U-4g 3-Me cPr 2-OMe-3-Cl U-4g 3-CF₃-4-Br
U-4g 3-CF₃ cPr 2-OMe-3-Br U-4g 3-CF₃-4-Me
U-4g 3-OMe cPr 2-OMe-3-Me U-4g 3,4-di-CF₃
U-4g 3-OCF₃ cPr 2-OMe-3-CF₃ U-4g 3-CF₃-4-OMe
U-4g 4-F cPr 2,3-di-OMe U-4g 3-CF₃-4-OCF₃
U-4g 4-Cl cPr 2-OMe-3-OCF₃ U-4g 3-OMe-4-F
U-4g 4-Br cPr 2-OCF₃-3-F U-4g 3-OMe-4-Cl
U-4g 4-Me cPr 2-OCF₃-3-Cl U-4g 3-OMe-4-Br
U-4g 4-CF₃ cPr 2-OCF₃-3-Br U-4g 3-OMe-4-Me
U-4g 4-OMe cPr 2-OCF₃-3-Me U-4g 3-OMe-4-CF₃
U-4g 4-OCF₃ cPr 2-OCF₃-3-CF₃ U-4g 3,4-di-OMe
U-4g 5-F cPr 2-OCF₃-3-OMe U-4g 3-OMe-4-OCF₃
U-4g 5-Cl cPr 2,3-di-OCF₃ U-4g 3-OCF₃-4-F
U-4g 5-Br cPr 2,4-di-F U-4g 3-OCF₃-4-Cl
U-4g 5-Me cPr 2-F-4-Cl U-4g 3-OCF₃-4-Br
U-4g 5-CF₃ cPr 2-F-4-Br U-4g 3-OCF₃-4-Me
U-4g 5-OMe cPr 2-F-4-Me U-4g 3-OCF₃-4-CF₃
U-4g 5-OCF₃ cPr 2-F-4-CF₃ U-4g 3-OCF₃-4-OMe
OMe 2-F cPr 2-F-4-OMe U-4g 3,4-di-OCF₃
OMe 2-Cl cPr 2-F-4-OCF₃ U-4g 3,5-di-F
OMe 2-Br cPr 2-Cl-4-F U-4g 3-F-5-Cl
OMe 2-Me cPr 2,4-di-Cl U-4g 3-F-5-Br
OMe 2-CF₃ cPr 2-Cl-4-Br U-4g 3-F-5-Me
OMe 2-OMe cPr 2-Cl-4-Me U-4g 3-F-5-CF₃
OMe 2-OCF₃ cPr 2-Cl-4-CF₃ U-4g 3-F-5-OMe
OMe 3-F cPr 2-Cl-4-OMe U-4g 3-F-5-OCF₃
OMe 3-Cl cPr 2-Cl-4-OCF₃ U-4g 3-Cl-5-F
OMe 3-Br cPr 2-Br-4-F U-4g 3,5-di-Cl
OMe 3-Me cPr 2-Br-4-Cl U-4g 3-Cl-5-Br
OMe 3-CF₃ cPr 2,4-di-Br U-4g 3-Cl-5-Me
OMe 3-OMe cPr 2-Br-4-Me U-4g 3-Cl-5-CF₃
OMe 3-OCF₃ cPr 2-Br-4-CF₃ U-4g 3-Cl-5-OMe
OMe 4-F cPr 2-Br-4-OMe U-4g 3-Cl-5-OCF₃
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
OMe 4-Cl cPr 2-Br-4-OCF₃ U-4g 3-Br-5-F
OMe 4-Br cPr 2-Me-4-F U-4g 3-Br-5-Cl
OMe 4-Me cPr 2-Me-4-Cl U-4g 3,5-di-Br
OMe 4-CF₃ cPr 2-Me-4-Br U-4g 3-Br-5-Me
OMe 4-OMe cPr 2,4-di-Me U-4g 3-Br-5-CF₃
OMe 4-OCF₃ cPr 2-Me-4-CF₃ U-4g 3-Br-5-OMe
OMe 5-F cPr 2-Me-4-OMe U-4g 3-Br-5-OCF₃
OMe 5-Cl cPr 2-Me-4-OCF₃ U-4g 3-Me-5-F
OMe 5-Br cPr 2-CF₃-4-F U-4g 3-Me-5-Cl
OMe 5-Me cPr 2-CF₃-4-Cl U-4g 3-Me-5-Br
OMe 5-CF₃ cPr 2-CF₃-4-Br U-4g 3,5-di-Me
OMe 5-OMe cPr 2-CF₃-4-Me U-4g 3-Me-5-CF₃
OMe 5-OCF₃ cPr 2,4-di-CF₃ U-4g 3-Me-5-OMe
SMe 2-F cPr 2-CF₃-4-OMe U-4g 3-Me-5-OCF₃
SMe 2-Cl cPr 2-CF₃-4-OCF₃ U-4g 3-CF₃-5-F
SMe 2-Br cPr 2-OMe-4-F U-4g 3-CF₃-5-Cl
SMe 2-Me cPr 2-OMe-4-Cl U-4g 3-CF₃-5-Br
SMe 2-CF₃ cPr 2-OMe-4-Br U-4g 3-CF₃-5-Me
SMe 2-OMe cPr 2-OMe-4-Me U-4g 3,5-di-CF₃
SMe 2-OCF₃ cPr 2-OMe-4-CF₃ U-4g 3-CF₃-5-OMe
SMe 3-F cPr 2,4-di-OMe U-4g 3-CF₃-5-OCF₃
SMe 3-Cl cPr 2-OMe-4-OCF₃ U-4g 3-OMe-5-F
SMe 3-Br cPr 2-OCF₃-4-F U-4g 3-OMe-5-Cl
SMe 3-Me cPr 2-OCF₃-4-Cl U-4g 3-OMe-5-Br
SMe 3-CF₃ cPr 2-OCF₃-4-Br U-4g 3-OMe-5-Me
SMe 3-OMe cPr 2-OCF₃-4-Me U-4g 3-OMe-5-CF₃
SMe 3-OCF₃ cPr 2-OCF₃-4-CF₃ U-4g 3,5-di-OMe
SMe 4-F cPr 2-OCF₃-4-OMe U-4g 3-OMe-5-OCF₃
SMe 4-Cl cPr 2,4-di-OCF₃ U-4g 3-OCF₃-5-F
SMe 4-Br cPr 2,5-di-F U-4g 3-OCF₃-5-Cl
SMe 4-Me cPr 2-F-5-Cl U-4g 3-OCF₃-5-Br
SMe 4-CF₃ cPr 2-F-5-Br U-4g 3-OCF₃-5-Me
SMe 4-OMe cPr 2-F-5-Me U-4g 3-OCF₃-5-CF₃
SMe 4-OCF₃ cPr 2-F-5-CF₃ U-4g 3-OCF₃-5-OMe
SMe 5-F cPr 2-F-5-OMe U-4g 3,5-di-OCF₃
SMe 5-Cl cPr 2-F-5-OCF₃ OMe 2,3-di-F
SMe 5-Br cPr 2-Cl-5-F OMe 2-F-3-Cl
SMe 5-Me cPr 2,5-di-Cl OMe 2-F-3-Br
SMe 5-CF₃ cPr 2-Cl-5-Br OMe 2-F-3-Me
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
SMe 5-OMe cPr 2-Cl-5-Me OMe 2-F-3-CF₃
SMe 5-OCF₃ cPr 2-Cl-5-CF₃ OMe 2-F-3-OMe
Ac 2-F cPr 2-Cl-5-OMe OMe 2-F-3-OCF₃
Ac 2-Cl cPr 2-Cl-5-OCF₃ OMe 2-Cl-3-F
Ac 2-Br cPr 2-Br-5-F OMe 2,3-di-Cl
Ac 2-Me cPr 2-Br-5-Cl OMe 2-Cl-3-Br
Ac 2-CF₃ cPr 2,5-di-Br OMe 2-Cl-3-Me
Ac 2-OMe cPr 2-Br-5-Me OMe 2-Cl-3-CF₃
Ac 2-OCF₃ cPr 2-Br-5-CF₃ OMe 2-Cl-3-OMe
Ac 3-F cPr 2-Br-5-OMe OMe 2-Cl-3-OCF₃
Ac 3-Cl cPr 2-Br-5-OCF₃ OMe 2-Br-3-F
Ac 3-Br cPr 2-Me-5-F OMe 2-Br-3-Cl
Ac 3-Me cPr 2-Me-5-Cl OMe 2,3-di-Br
Ac 3-CF₃ cPr 2-Me-5-Br OMe 2-Br-3-Me
Ac 3-OMe cPr 2,5-di-Me OMe 2-Br-3-CF₃
Ac 3-OCF₃ cPr 2-Me-5-CF₃ OMe 2-Br-3-OMe
Ac 4-F cPr 2-Me-5-OMe OMe 2-Br-3-OCF₃
Ac 4-Cl cPr 2-Me-5-OCF₃ OMe 2-Me-3-F
Ac 4-Br cPr 2-CF₃-5-F OMe 2-Me-3-Cl
Ac 4-Me cPr 2-CF₃-5-Cl OMe 2-Me-3-Br
Ac 4-CF₃ cPr 2-CF₃-5-Br OMe 2,3-di-Me
Ac 4-OMe cPr 2-CF₃-5-Me OMe 2-Me-3-CF₃
Ac 4-OCF₃ cPr 2,5-di-CF₃ OMe 2-Me-3-OMe
Ac 5-F cPr 2-CF₃-5-OMe OMe 2-Me-3-OCF₃
Ac 5-Cl cPr 2-CF₃-5-OCF₃ OMe 2-CF₃-3-F
Ac 5-Br cPr 2-OMe-5-F OMe 2-CF₃-3-Cl
Ac 5-Me cPr 2-OMe-5-Cl OMe 2-CF₃-3-Br
Ac 5-CF₃ cPr 2-OMe-5-Br OMe 2-CF₃-3-Me
Ac 5-OMe cPr 2-OMe-5-Me OMe 2,3-di-CF₃
Ac 5-OCF₃ cPr 2-OMe-5-CF₃ OMe 2-CF₃-3-OMe
cPen 2-F cPr 2,5-di-OMe OMe 2-CF₃-3-OCF₃
cPen 2-Cl cPr 2-OMe-5-OCF₃ OMe 2-OMe-3-F
cPen 2-Br cPr 2-OCF₃-5-F OMe 2-OMe-3-Cl
cPen 2-Me cPr 2-OCF₃-5-Cl OMe 2-OMe-3-Br
cPen 2-CF₃ cPr 2-OCF₃-5-Br OMe 2-OMe-3-Me
cPen 2-OMe cPr 2-OCF₃-5-Me OMe 2-OMe-3-CF₃
cPen 2-OCF₃ cPr 2-OCF₃-5-CF₃ OMe 2,3-di-OMe
cPen 3-F cPr 2-OCF₃-5-OMe OMe 2-OMe-3-OCF₃
cPen 3-Cl cPr 2,5-di-OCF₃ OMe 2-OCF₃-3-F
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
cPen 3-Br cPr 3,4-di-F OMe 2-OCF₃-3-Cl
cPen 3-Me cPr 3-F-4-Cl OMe 2-OCF₃-3-Br
cPen 3-CF₃ cPr 3-F-4-Br OMe 2-OCF₃-3-Me
cPen 3-OMe cPr 3-F-4-Me OMe 2-OCF₃-3-CF₃
cPen 3-OCF₃ cPr 3-F-4-CF₃ OMe 2-OCF₃-3-OMe
cPen 4-F cPr 3-F-4-OMe OMe 2,3-di-OCF₃
cPen 4-Cl cPr 3-F-4-OCF₃ OMe 2,4-di-F
cPen 4-Br cPr 3-Cl-4-F OMe 2-F-4-Cl
cPen 4-Me cPr 3,4-di-Cl OMe 2-F-4-Br
cPen 4-CF₃ cPr 3-Cl-4-Br OMe 2-F-4-Me
cPen 4-OMe cPr 3-Cl-4-Me OMe 2-F-4-CF₃
cPen 4-OCF₃ cPr 3-Cl-4-CF₃ OMe 2-F-4-OMe
cPen 5-F cPr 3-Cl-4-OMe OMe 2-F-4-OCF₃
cPen 5-Cl cPr 3-Cl-4-OCF₃ OMe 2-Cl-4-F
cPen 5-Br cPr 3-Br-4-F OMe 2,4-di-Cl
cPen 5-Me cPr 3-Br-4-Cl OMe 2-Cl-4-Br
cPen 5-CF₃ cPr 3,4-di-Br OMe 2-Cl-4-Me
cPen 5-OMe cPr 3-Br-4-Me OMe 2-Cl-4-CF₃
cPen 5-OCF₃ cPr 3-Br-4-CF₃ OMe 2-Cl-4-OMe
U-1e 2-F cPr 3-Br-4-OMe OMe 2-Cl-4-OCF₃
U-1e 2-Cl cPr 3-Br-4-OCF₃ OMe 2-Br-4-F
U-1e 2-Br cPr 3-Me-4-F OMe 2-Br-4-Cl
U-1e 2-Me cPr 3-Me-4-Cl OMe 2,4-di-Br
U-1e 2-CF₃ cPr 3-Me-4-Br OMe 2-Br-4-Me
U-1e 2-OMe cPr 3,4-di-Me OMe 2-Br-4-CF₃
U-1e 2-OCF₃ cPr 3-Me-4-CF₃ OMe 2-Br-4-OMe
U-1e 3-F cPr 3-Me-4-OMe OMe 2-Br-4-OCF₃
U-1e 3-Cl cPr 3-Me-4-OCF₃ OMe 2-Me-4-F
U-1e 3-Br cPr 3-CF₃-4-F OMe 2-Me-4-Cl
U-1e 3-Me cPr 3-CF₃-4-Cl OMe 2-Me-4-Br
U-1e 3-CF₃ cPr 3-CF₃-4-Br OMe 2,4-di-Me
U-1e 3-OMe cPr 3-CF₃-4-Me OMe 2-Me-4-CF₃
U-1e 3-OCF₃ cPr 3,4-di-CF₃ OMe 2-Me-4-OMe
U-1e 4-F cPr 3-CF₃-4-OMe OMe 2-Me-4-OCF₃
U-1e 4-Cl cPr 3-CF₃-4-OCF₃ OMe 2-CF₃-4-F
U-1e 4-Br cPr 3-OMe-4-F OMe 2-CF₃-4-Cl
U-1e 4-Me cPr 3-OMe-4-Cl OMe 2-CF₃-4-Br
U-1e 4-CF₃ cPr 3-OMe-4-Br OMe 2-CF₃-4-Me
U-1e 4-OMe cPr 3-OMe-4-Me OMe 2,4-di-CF₃
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
U-1e 4-OCF₃ cPr 3-OMe-4-CF₃ OMe 2-CF₃-4-OMe
U-1e 5-F cPr 3,4-di-OMe OMe 2-CF₃-4-OCF₃
U-1e 5-Cl cPr 3-OMe-4-OCF₃ OMe 2-OMe-4-F
U-1e 5-Br cPr 3-OCF₃-4-F OMe 2-OMe-4-Cl
U-1e 5-Me cPr 3-OCF₃-4-Cl OMe 2-OMe-4-Br
U-1e 5-CF₃ cPr 3-OCF₃-4-Br OMe 2-OMe-4-Me
U-1e 5-OMe cPr 3-OCF₃-4-Me OMe 2-OMe-4-CF₃
U-1e 5-OCF₃ cPr 3-OCF₃-4-CF₃ OMe 2,4-di-OMe
Me 2-Ac cPr 3-OCF₃-4-OMe OMe 2-OMe-4-OCF₃
Me 2-(U-3b) cPr 3,4-di-OCF₃ OMe 2-OCF₃-4-F
Me 2-CF₂H cPr 3,5-di-F OMe 2-OCF₃-4-Cl
Me 2-CN cPr 3-F-5-Cl OMe 2-OCF₃-4-Br
Me 2-Et cPr 3-F-5-Br OMe 2-OCF₃-4-Me
Me 2-OCF₂H cPr 3-F-5-Me OMe 2-OCF₃-4-CF₃
Me 2-OEt cPr 3-F-5-CF₃ OMe 2-OCF₃-4-OMe
Me 2-C(O)CF₃ cPr 3-F-5-OMe OMe 2,4-di-OCF₃
Me 3-Ac cPr 3-F-5-OCF₃ OMe 2,5-di-F
Me 3-(U-3b) cPr 3-Cl-5-F OMe 2-F-5-Cl
Me 3-CF₂H cPr 3,5-di-Cl OMe 2-F-5-Br
Me 3-CN cPr 3-Cl-5-Br OMe 2-F-5-Me
Me 3-Et cPr 3-Cl-5-Me OMe 2-F-5-CF₃
Me 3-OCF₂H cPr 3-Cl-5-CF₃ OMe 2-F-5-OMe
Me 3-OEt cPr 3-Cl-5-OMe OMe 2-F-5-OCF₃
Me 3-C(O)CF₃ cPr 3-Cl-5-OCF₃ OMe 2-Cl-5-F
Me 4-Ac cPr 3-Br-5-F OMe 2,5-di-Cl
Me 4-(U-3b) cPr 3-Br-5-Cl OMe 2-Cl-5-Br
Me 4-CF₂H cPr 3,5-di-Br OMe 2-Cl-5-Me
Me 4-CN cPr 3-Br-5-Me OMe 2-Cl-5-CF₃
Me 4-Et cPr 3-Br-5-CF₃ OMe 2-Cl-5-OMe
Me 4-OCF₂H cPr 3-Br-5-OMe OMe 2-Cl-5-OCF₃
Me 4-OEt cPr 3-Br-5-OCF₃ OMe 2-Br-5-F
Me 4-C(O)CF₃ cPr 3-Me-5-F OMe 2-Br-5-Cl
Me 5-Ac cPr 3-Me-5-Cl OMe 2,5-di-Br
Me 5-(U-3b) cPr 3-Me-5-Br OMe 2-Br-5-Me
Me 5-CF₂H cPr 3,5-di-Me OMe 2-Br-5-CF₃
Me 5-CN cPr 3-Me-5-CF₃ OMe 2-Br-5-OMe
Me 5-Et cPr 3-Me-5-OMe OMe 2-Br-5-OCF₃
Me 5-OCF₂H cPr 3-Me-5-OCF₃ OMe 2-Me-5-F
Me 5-OEt cPr 3-CF₃-5-F OMe 2-Me-5-Cl
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
Me 5-C(O)CF₃ cPr 3-CF₃-5-Cl OMe 2-Me-5-Br
Et 2-Ac cPr 3-CF₃-5-Br OMe 2,5-di-Me
Et 2-(U-3b) cPr 3-CF₃-5-Me OMe 2-Me-5-CF₃
Et 2-CF₂H cPr 3,5-di-CF₃ OMe 2-Me-5-OMe
Et 2-CN cPr 3-CF₃-5-OMe OMe 2-Me-5-OCF₃
Et 2-Et cPr 3-CF₃-5-OCF₃ OMe 2-CF₃-5-F
Et 2-OCF₂H cPr 3-OMe-5-F OMe 2-CF₃-5-Cl
Et 2-OEt cPr 3-OMe-5-Cl OMe 2-CF₃-5-Br
Et 2-C(O)CF₃ cPr 3-OMe-5-Br OMe 2-CF₃-5-Me
Et 3-Ac cPr 3-OMe-5-Me OMe 2,5-di-CF₃
Et 3-(U-3b) cPr 3-OMe-5-CF₃ OMe 2-CF₃-5-OMe
Et 3-CF₂H cPr 3,5-di-OMe OMe 2-CF₃-5-OCF₃
Et 3-CN cPr 3-OMe-5-OCF₃ OMe 2-OMe-5-F
Et 3-Et cPr 3-OCF₃-5-F OMe 2-OMe-5-Cl
Et 3-OCF₂H cPr 3-OCF₃-5-Cl OMe 2-OMe-5-Br
Et 3-OEt cPr 3-OCF₃-5-Br OMe 2-OMe-5-Me
Et 3-C(O)CF₃ cPr 3-OCF₃-5-Me OMe 2-OMe-5-CF₃
Et 4-Ac cPr 3-OCF₃-5-CF₃ OMe 2,5-di-OMe
Et 4-(U-3b) cPr 3-OCF₃-5-OMe OMe 2-OMe-5-OCF₃
Et 4-CF₂H cPr 3,5-di-OCF₃ OMe 2-OCF₃-5-F
Et 4-CN U-4b 2,3-di-F OMe 2-OCF₃-5-Cl
Et 4-Et U-4b 2-F-3-Cl OMe 2-OCF₃-5-Br
Et 4-OCF₂H U-4b 2-F-3-Br OMe 2-OCF₃-5-Me
Et 4-OEt U-4b 2-F-3-Me OMe 2-OCF₃-5-CF₃
Et 4-C(O)CF₃ U-4b 2-F-3-CF₃ OMe 2-OCF₃-5-OMe
Et 5-Ac U-4b 2-F-3-OMe OMe 2,5-di-OCF₃
Et 5-(U-3b) U-4b 2-F-3-OCF₃ OMe 3,4-di-F
Et 5-CF₂H U-4b 2-Cl-3-F OMe 3-F-4-Cl
Et 5-CN U-4b 2,3-di-Cl OMe 3-F-4-Br
Et 5-Et U-4b 2-Cl-3-Br OMe 3-F-4-Me
Et 5-OCF₂H U-4b 2-Cl-3-Me OMe 3-F-4-CF₃
Et 5-OEt U-4b 2-Cl-3-CF₃ OMe 3-F-4-OMe
Et 5-C(O)CF₃ U-4b 2-Cl-3-OMe OMe 3-F-4-OCF₃
iPr 2-Ac U-4b 2-Cl-3-OCF₃ OMe 3-Cl-4-F
iPr 2-(U-3b) U-4b 2-Br-3-F OMe 3,4-di-Cl
iPr 2-CF₂H U-4b 2-Br-3-Cl OMe 3-Cl-4-Br
iPr 2-CN U-4b 2,3-di-Br OMe 3-Cl-4-Me
iPr 2-Et U-4b 2-Br-3-Me OMe 3-Cl-4-CF₃
iPr 2-OCF₂H U-4b 2-Br-3-CF₃ OMe 3-Cl-4-OMe
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
iPr 2-OEt U-4b 2-Br-3-OMe OMe 3-Cl-4-OCF₃
iPr 2-C(O)CF₃ U-4b 2-Br-3-OCF₃ OMe 3-Br-4-F
iPr 3-Ac U-4b 2-Me-3-F OMe 3-Br-4-Cl
iPr 3-(U-3b) U-4b 2-Me-3-Cl OMe 3,4-di-Br
iPr 3-CF₂H U-4b 2-Me-3-Br OMe 3-Br-4-Me
iPr 3-CN U-4b 2,3-di-Me OMe 3-Br-4-CF₃
iPr 3-Et U-4b 2-Me-3-CF₃ OMe 3-Br-4-OMe
iPr 3-OCF₂H U-4b 2-Me-3-OMe OMe 3-Br-4-OCF₃
iPr 3-OEt U-4b 2-Me-3-OCF₃ OMe 3-Me-4-F
iPr 3-C(O)CF₃ U-4b 2-CF₃-3-F OMe 3-Me-4-Cl
iPr 4-Ac U-4b 2-CF₃-3-Cl OMe 3-Me-4-Br
iPr 4-(U-3b) U-4b 2-CF₃-3-Br OMe 3,4-di-Me
iPr 4-CF₂H U-4b 2-CF₃-3-Me OMe 3-Me-4-CF₃
iPr 4-CN U-4b 2,3-di-CF₃ OMe 3-Me-4-OMe
iPr 4-Et U-4b 2-CF₃-3-OMe OMe 3-Me-4-OCF₃
iPr 4-OCF₂H U-4b 2-CF₃-3-OCF₃ OMe 3-CF₃-4-F
iPr 4-OEt U-4b 2-OMe-3-F OMe 3-CF₃-4-Cl
iPr 4-C(O)CF₃ U-4b 2-OMe-3-Cl OMe 3-CF₃-4-Br
iPr 5-Ac U-4b 2-OMe-3-Br OMe 3-CF₃-4-Me
iPr 5-(U-3b) U-4b 2-OMe-3-Me OMe 3,4-di-CF₃
iPr 5-CF₂H U-4b 2-OMe-3-CF₃ OMe 3-CF₃-4-OMe
iPr 5-CN U-4b 2,3-di-OMe OMe 3-CF₃-4-OCF₃
iPr 5-Et U-4b 2-OMe-3-OCF₃ OMe 3-OMe-4-F
iPr 5-OCF₂H U-4b 2-OCF₃-3-F OMe 3-OMe-4-Cl
iPr 5-OEt U-4b 2-OCF₃-3-Cl OMe 3-OMe-4-Br
iPr 5-C(O)CF₃ U-4b 2-OCF₃-3-Br OMe 3-OMe-4-Me
U-4a 2-Ac U-4b 2-OCF₃-3-Me OMe 3-OMe-4-CF₃
U-4a 2-(U-3b) U-4b 2-OCF₃-3-CF₃ OMe 3,4-di-OMe
U-4a 2-CF₂H U-4b 2-OCF₃-3-OMe OMe 3-OMe-4-OCF₃
U-4a 2-CN U-4b 2,3-di-OCF₃ OMe 3-OCF₃-4-F
U-4a 2-Et U-4b 2,4-di-F OMe 3-OCF₃-4-Cl
U-4a 2-OCF₂H U-4b 2-F-4-Cl OMe 3-OCF₃-4-Br
U-4a 2-OEt U-4b 2-F-4-Br OMe 3-OCF₃-4-Me
U-4a 2-C(O)CF₃ U-4b 2-F-4-Me OMe 3-OCF₃-4-CF₃
U-4a 3-Ac U-4b 2-F-4-CF₃ OMe 3-OCF₃-4-OMe
U-4a 3-(U-3b) U-4b 2-F-4-OMe OMe 3,4-di-OCF₃
U-4a 3-CF₂H U-4b 2-F-4-OCF₃ OMe 3,5-di-F
U-4a 3-CN U-4b 2-Cl-4-F OMe 3-F-5-Cl
U-4a 3-Et U-4b 2,4-di-Cl OMe 3-F-5-Br
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
U-4a 3-OCF₂H U-4b 2-Cl-4-Br OMe 3-F-5-Me
U-4a 3-OEt U-4b 2-Cl-4-Me OMe 3-F-5-CF₃
U-4a 3-C(O)CF₃ U-4b 2-Cl-4-CF₃ OMe 3-F-5-OMe
U-4a 4-Ac U-4b 2-Cl-4-OMe OMe 3-F-5-OCF₃
U-4a 4-(U-3b) U-4b 2-Cl-4-OCF₃ OMe 3-Cl-5-F
U-4a 4-CF₂H U-4b 2-Br-4-F OMe 3,5-di-Cl
U-4a 4-CN U-4b 2-Br-4-Cl OMe 3-Cl-5-Br
U-4a 4-Et U-4b 2,4-di-Br OMe 3-Cl-5-Me
U-4a 4-OCF₂H U-4b 2-Br-4-Me OMe 3-Cl-5-CF₃
U-4a 4-OEt U-4b 2-Br-4-CF₃ OMe 3-Cl-5-OMe
U-4a 4-C(O)CF₃ U-4b 2-Br-4-OMe OMe 3-Cl-5-OCF₃
U-4a 5-Ac U-4b 2-Br-4-OCF₃ OMe 3-Br-5-F
U-4a 5-(U-3b) U-4b 2-Me-4-F OMe 3-Br-5-Cl
U-4a 5-CF₂H U-4b 2-Me-4-Cl OMe 3,5-di-Br
U-4a 5-CN U-4b 2-Me-4-Br OMe 3-Br-5-Me
U-4a 5-Et U-4b 2,4-di-Me OMe 3-Br-5-CF₃
U-4a 5-OCF₂H U-4b 2-Me-4-CF₃ OMe 3-Br-5-OMe
U-4a 5-OEt U-4b 2-Me-4-OMe OMe 3-Br-5-OCF₃
U-4a 5-C(O)CF₃ U-4b 2-Me-4-OCF₃ OMe 3-Me-5-F
CF₃ 2-Ac U-4b 2-CF₃-4-F OMe 3-Me-5-Cl
CF₃ 2-(U-3b) U-4b 2-CF₃-4-Cl OMe 3-Me-5-Br
CF₃ 2-CF₂H U-4b 2-CF₃-4-Br OMe 3,5-di-Me
CF₃ 2-CN U-4b 2-CF₃-4-Me OMe 3-Me-5-CF₃
CF₃ 2-Et U-4b 2,4-di-CF₃ OMe 3-Me-5-OMe
CF₃ 2-OCF₂H U-4b 2-CF₃-4-OMe OMe 3-Me-5-OCF₃
CF₃ 2-OEt U-4b 2-CF₃-4-OCF₃ OMe 3-CF₃-5-F
CF₃ 2-C(O)CF₃ U-4b 2-OMe-4-F OMe 3-CF₃-5-Cl
CF₃ 3-Ac U-4b 2-OMe-4-Cl OMe 3-CF₃-5-Br
CF₃ 3-(U-3b) U-4b 2-OMe-4-Br OMe 3-CF₃-5-Me
CF₃ 3-CF₂H U-4b 2-OMe-4-Me OMe 3,5-di-CF₃
CF₃ 3-CN U-4b 2-OMe-4-CF₃ OMe 3-CF₃-5-OMe
CF₃ 3-Et U-4b 2,4-di-OMe OMe 3-CF₃-5-OCF₃
CF₃ 3-OCF₂H U-4b 2-OMe-4-OCF₃ OMe 3-OMe-5-F
CF₃ 3-OEt U-4b 2-OCF₃-4-F OMe 3-OMe-5-Cl
CF₃ 3-C(O)CF₃ U-4b 2-OCF₃-4-Cl OMe 3-OMe-5-Br
CF₃ 4-Ac U-4b 2-OCF₃-4-Br OMe 3-OMe-5-Me
CF₃ 4-(U-3b) U-4b 2-OCF₃-4-Me OMe 3-OMe-5-CF₃
CF₃ 4-CF₂H U-4b 2-OCF₃-4-CF₃ OMe 3,5-di-OMe
CF₃ 4-CN U-4b 2-OCF₃-4-OMe OMe 3-OMe-5-OCF₃
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
CF₃ 4-Et U-4b 2,4-di-OCF₃ OMe 3-OCF₃-5-F
CF₃ 4-OCF₂H U-4b 2,5-di-F OMe 3-OCF₃-5-Cl
CF₃ 4-OEt U-4b 2-F-5-Cl OMe 3-OCF₃-5-Br
CF₃ 4-C(O)CF₃ U-4b 2-F-5-Br OMe 3-OCF₃-5-Me
CF₃ 5-Ac U-4b 2-F-5-Me OMe 3-OCF₃-5-CF₃
CF₃ 5-(U-3b) U-4b 2-F-5-CF₃ OMe 3-OCF₃-5-OMe
CF₃ 5-CF₂H U-4b 2-F-5-OMe OMe 3,5-di-OCF₃
CF₃ 5-CN U-4b 2-F-5-OCF₃ SMe 2,3-di-F
CF₃ 5-Et U-4b 2-Cl-5-F SMe 2-F-3-Cl
CF₃ 5-OCF₂H U-4b 2,5-di-Cl SMe 2-F-3-Br
CF₃ 5-OEt U-4b 2-Cl-5-Br SMe 2-F-3-Me
CF₃ 5-C(O)CF₃ U-4b 2-Cl-5-Me SMe 2-F-3-CF₃
cPr 2-Ac U-4b 2-Cl-5-CF₃ SMe 2-F-3-OMe
cPr 2-(U-3b) U-4b 2-Cl-5-OMe SMe 2-F-3-OCF₃
cPr 2-CF₂H U-4b 2-Cl-5-OCF₃ SMe 2-Cl-3-F
cPr 2-CN U-4b 2-Br-5-F SMe 2,3-di-Cl
cPr 2-Et U-4b 2-Br-5-Cl SMe 2-Cl-3-Br
cPr 2-OCF₂H U-4b 2,5-di-Br SMe 2-Cl-3-Me
cPr 2-OEt U-4b 2-Br-5-Me SMe 2-Cl-3-CF₃
cPr 2-C(O)CF₃ U-4b 2-Br-5-CF₃ SMe 2-Cl-3-OMe
cPr 3-Ac U-4b 2-Br-5-OMe SMe 2-Cl-3-OCF₃
cPr 3-(U-3b) U-4b 2-Br-5-OCF₃ SMe 2-Br-3-F
cPr 3-CF₂H U-4b 2-Me-5-F SMe 2-Br-3-Cl
cPr 3-CN U-4b 2-Me-5-Cl SMe 2,3-di-Br
cPr 3-Et U-4b 2-Me-5-Br SMe 2-Br-3-Me
cPr 3-OCF₂H U-4b 2,5-di-Me SMe 2-Br-3-CF₃
cPr 3-OEt U-4b 2-Me-5-CF₃ SMe 2-Br-3-OMe
cPr 3-C(O)CF₃ U-4b 2-Me-5-OMe SMe 2-Br-3-OCF₃
cPr 4-Ac U-4b 2-Me-5-OCF₃ SMe 2-Me-3-F
cPr 4-(U-3b) U-4b 2-CF₃-5-F SMe 2-Me-3-Cl
cPr 4-CF₂H U-4b 2-CF₃-5-Cl SMe 2-Me-3-Br
cPr 4-CN U-4b 2-CF₃-5-Br SMe 2,3-di-Me
cPr 4-Et U-4b 2-CF₃-5-Me SMe 2-Me-3-CF₃
cPr 4-OCF₂H U-4b 2,5-di-CF₃ SMe 2-Me-3-OMe
cPr 4-OEt U-4b 2-CF₃-5-OMe SMe 2-Me-3-OCF₃
cPr 4-C(O)CF₃ U-4b 2-CF₃-5-OCF₃ SMe 2-CF₃-3-F
cPr 5-Ac U-4b 2-OMe-5-F SMe 2-CF₃-3-Cl
cPr 5-(U-3b) U-4b 2-OMe-5-Cl SMe 2-CF₃-3-Br
cPr 5-CF₂H U-4b 2-OMe-5-Br SMe 2-CF₃-3-Me
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
cPr 5-CN U-4b 2-OMe-5-Me SMe 2,3-di-CF₃
cPr 5-Et U-4b 2-OMe-5-CF₃ SMe 2-CF₃-3-OMe
cPr 5-OCF₂H U-4b 2,5-di-OMe SMe 2-CF₃-3-OCF₃
cPr 5-OEt U-4b 2-OMe-5-OCF₃ SMe 2-OMe-3-F
cPr 5-C(O)CF₃ U-4b 2-OCF₃-5-F SMe 2-OMe-3-Cl
Me 2,3-di-F U-4b 2-OCF₃-5-Cl SMe 2-OMe-3-Br
Me 2-F-3-Cl U-4b 2-OCF₃-5-Br SMe 2-OMe-3-Me
Me 2-F-3-Br U-4b 2-OCF₃-5-Me SMe 2-OMe-3-CF₃
Me 2-F-3-Me U-4b 2-OCF₃-5-CF₃ SMe 2,3-di-OMe
Me 2-F-3-CF₃ U-4b 2-OCF₃-5-OMe SMe 2-OMe-3-OCF₃
Me 2-F-3-OMe U-4b 2,5-di-OCF₃ SMe 2-OCF₃-3-F
Me 2-F-3-OCF₃ U-4b 3,4-di-F SMe 2-OCF₃-3-Cl
Me 2-Cl-3-F U-4b 3-F-4-Cl SMe 2-OCF₃-3-Br
Me 2,3-di-Cl U-4b 3-F-4-Br SMe 2-OCF₃-3-Me
Me 2-Cl-3-Br U-4b 3-F-4-Me SMe 2-OCF₃-3-CF₃
Me 2-Cl-3-Me U-4b 3-F-4-CF₃ SMe 2-OCF₃-3-OMe
Me 2-Cl-3-CF₃ U-4b 3-F-4-OMe SMe 2,3-di-OCF₃
Me 2-Cl-3-OMe U-4b 3-F-4-OCF₃ SMe 2,4-di-F
Me 2-Cl-3-OCF₃ U-4b 3-Cl-4-F SMe 2-F-4-Cl
Me 2-Br-3-F U-4b 3,4-di-Cl SMe 2-F-4-Br
Me 2-Br-3-Cl U-4b 3-Cl-4-Br SMe 2-F-4-Me
Me 2,3-di-Br U-4b 3-Cl-4-Me SMe 2-F-4-CF₃
Me 2-Br-3-Me U-4b 3-Cl-4-CF₃ SMe 2-F-4-OMe
Me 2-Br-3-CF₃ U-4b 3-Cl-4-OMe SMe 2-F-4-OCF₃
Me 2-Br-3-OMe U-4b 3-Cl-4-OCF₃ SMe 2-Cl-4-F
Me 2-Br-3-OCF₃ U-4b 3-Br-4-F SMe 2,4-di-Cl
Me 2-Me-3-F U-4b 3-Br-4-Cl SMe 2-Cl-4-Br
Me 2-Me-3-Cl U-4b 3,4-di-Br SMe 2-Cl-4-Me
Me 2-Me-3-Br U-4b 3-Br-4-Me SMe 2-Cl-4-CF₃
Me 2,3-di-Me U-4b 3-Br-4-CF₃ SMe 2-Cl-4-OMe
Me 2-Me-3-CF₃ U-4b 3-Br-4-OMe SMe 2-Cl-4-OCF₃
Me 2-Me-3-OMe U-4b 3-Br-4-OCF₃ SMe 2-Br-4-F
Me 2-Me-3-OCF₃ U-4b 3-Me-4-F SMe 2-Br-4-Cl
Me 2-CF₃-3-F U-4b 3-Me-4-Cl SMe 2,4-di-Br
Me 2-CF₃-3-Cl U-4b 3-Me-4-Br SMe 2-Br-4-Me
Me 2-CF₃-3-Br U-4b 3,4-di-Me SMe 2-Br-4-CF₃
Me 2-CF₃-3-Me U-4b 3-Me-4-CF₃ SMe 2-Br-4-OMe
Me 2,3-di-CF₃ U-4b 3-Me-4-OMe SMe 2-Br-4-OCF₃
Me 2-CF₃-3-OMe U-4b 3-Me-4-OCF₃ SMe 2-Me-4-F
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
Me 2-CF₃-3-OCF₃ U-4b 3-CF₃-4-F SMe 2-Me-4-Cl
Me 2-OMe-3-F U-4b 3-CF₃-4-Cl SMe 2-Me-4-Br
Me 2-OMe-3-Cl U-4b 3-CF₃-4-Br SMe 2,4-di-Me
Me 2-OMe-3-Br U-4b 3-CF₃-4-Me SMe 2-Me-4-CF₃
Me 2-OMe-3-Me U-4b 3,4-di-CF₃ SMe 2-Me-4-OMe
Me 2-OMe-3-CF₃ U-4b 3-CF₃-4-OMe SMe 2-Me-4-OCF₃
Me 2,3-di-OMe U-4b 3-CF₃-4-OCF₃ SMe 2-CF₃-4-F
Me 2-OMe-3-OCF₃ U-4b 3-OMe-4-F SMe 2-CF₃-4-Cl
Me 2-OCF₃-3-F U-4b 3-OMe-4-Cl SMe 2-CF₃-4-Br
Me 2-OCF₃-3-Cl U-4b 3-OMe-4-Br SMe 2-CF₃-4-Me
Me 2-OCF₃-3-Br U-4b 3-OMe-4-Me SMe 2,4-di-CF₃
Me 2-OCF₃-3-Me U-4b 3-OMe-4-CF₃ SMe 2-CF₃-4-OMe
Me 2-OCF₃-3-CF₃ U-4b 3,4-di-OMe SMe 2-CF₃-4-OCF₃
Me 2-OCF₃-3-OMe U-4b 3-OMe-4-OCF₃ SMe 2-OMe-4-F
Me 2,3-di-OCF₃ U-4b 3-OCF₃-4-F SMe 2-OMe-4-Cl
Me 2,4-di-F U-4b 3-OCF₃-4-Cl SMe 2-OMe-4-Br
Me 2-F-4-Cl U-4b 3-OCF₃-4-Br SMe 2-OMe-4-Me
Me 2-F-4-Br U-4b 3-OCF₃-4-Me SMe 2-OMe-4-CF₃
Me 2-F-4-Me U-4b 3-OCF₃-4-CF₃ SMe 2,4-di-OMe
Me 2-F-4-CF₃ U-4b 3-OCF₃-4-OMe SMe 2-OMe-4-OCF₃
Me 2-F-4-OMe U-4b 3,4-di-OCF₃ SMe 2-OCF₃-4-F
Me 2-F-4-OCF₃ U-4b 3,5-di-F SMe 2-OCF₃-4-Cl
Me 2-Cl-4-F U-4b 3-F-5-Cl SMe 2-OCF₃-4-Br
Me 2,4-di-Cl U-4b 3-F-5-Br SMe 2-OCF₃-4-Me
Me 2-Cl-4-Br U-4b 3-F-5-Me SMe 2-OCF₃-4-CF₃
Me 2-Cl-4-Me U-4b 3-F-5-CF₃ SMe 2-OCF₃-4-OMe
Me 2-Cl-4-CF₃ U-4b 3-F-5-OMe SMe 2,4-di-OCF₃
Me 2-Cl-4-OMe U-4b 3-F-5-OCF₃ SMe 2,5-di-F
Me 2-Cl-4-OCF₃ U-4b 3-Cl-5-F SMe 2-F-5-Cl
Me 2-Br-4-F U-4b 3,5-di-Cl SMe 2-F-5-Br
Me 2-Br-4-Cl U-4b 3-Cl-5-Br SMe 2-F-5-Me
Me 2,4-di-Br U-4b 3-Cl-5-Me SMe 2-F-5-CF₃
Me 2-Br-4-Me U-4b 3-Cl-5-CF₃ SMe 2-F-5-OMe
Me 2-Br-4-CF₃ U-4b 3-Cl-5-OMe SMe 2-F-5-OCF₃
Me 2-Br-4-OMe U-4b 3-Cl-5-OCF₃ SMe 2-Cl-5-F
Me 2-Br-4-OCF₃ U-4b 3-Br-5-F SMe 2,5-di-Cl
Me 2-Me-4-F U-4b 3-Br-5-Cl SMe 2-Cl-5-Br
Me 2-Me-4-Cl U-4b 3,5-di-Br SMe 2-Cl-5-Me
Me 2-Me-4-Br U-4b 3-Br-5-Me SMe 2-Cl-5-CF₃
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
Me 2,4-di-Me U-4b 3-Br-5-CF₃ SMe 2-Cl-5-OMe
Me 2-Me-4-CF₃ U-4b 3-Br-5-OMe SMe 2-Cl-5-OCF₃
Me 2-Me-4-OMe U-4b 3-Br-5-OCF₃ SMe 2-Br-5-F
Me 2-Me-4-OCF₃ U-4b 3-Me-5-F SMe 2-Br-5-Cl
Me 2-CF₃-4-F U-4b 3-Me-5-Cl SMe 2,5-di-Br
Me 2-CF₃-4-Cl U-4b 3-Me-5-Br SMe 2-Br-5-Me
Me 2-CF₃-4-Br U-4b 3,5-di-Me SMe 2-Br-5-CF₃
Me 2-CF₃-4-Me U-4b 3-Me-5-CF₃ SMe 2-Br-5-OMe
Me 2,4-di-CF₃ U-4b 3-Me-5-OMe SMe 2-Br-5-OCF₃
Me 2-CF₃-4-OMe U-4b 3-Me-5-OCF₃ SMe 2-Me-5-F
Me 2-CF₃-4-OCF₃ U-4b 3-CF₃-5-F SMe 2-Me-5-Cl
Me 2-OMe-4-F U-4b 3-CF₃-5-Cl SMe 2-Me-5-Br
Me 2-OMe-4-Cl U-4b 3-CF₃-5-Br SMe 2,5-di-Me
Me 2-OMe-4-Br U-4b 3-CF₃-5-Me SMe 2-Me-5-CF₃
Me 2-OMe-4-Me U-4b 3,5-di-CF₃ SMe 2-Me-5-OMe
Me 2-OMe-4-CF₃ U-4b 3-CF₃-5-OMe SMe 2-Me-5-OCF₃
Me 2,4-di-OMe U-4b 3-CF₃-5-OCF₃ SMe 2-CF₃-5-F
Me 2-OMe-4-OCF₃ U-4b 3-OMe-5-F SMe 2-CF₃-5-Cl
Me 2-OCF₃-4-F U-4b 3-OMe-5-Cl SMe 2-CF₃-5-Br
Me 2-OCF₃-4-Cl U-4b 3-OMe-5-Br SMe 2-CF₃-5-Me
Me 2-OCF₃-4-Br U-4b 3-OMe-5-Me SMe 2,5-di-CF₃
Me 2-OCF₃-4-Me U-4b 3-OMe-5-CF₃ SMe 2-CF₃-5-OMe
Me 2-OCF₃-4-CF₃ U-4b 3,5-di-OMe SMe 2-CF₃-5-OCF₃
Me 2-OCF₃-4-OMe U-4b 3-OMe-5-OCF₃ SMe 2-OMe-5-F
Me 2,4-di-OCF₃ U-4b 3-OCF₃-5-F SMe 2-OMe-5-Cl
Me 2,5-di-F U-4b 3-OCF₃-5-Cl SMe 2-OMe-5-Br
Me 2-F-5-Cl U-4b 3-OCF₃-5-Br SMe 2-OMe-5-Me
Me 2-F-5-Br U-4b 3-OCF₃-5-Me SMe 2-OMe-5-CF₃
Me 2-F-5-Me U-4b 3-OCF₃-5-CF₃ SMe 2,5-di-OMe
Me 2-F-5-CF₃ U-4b 3-OCF₃-5-OMe SMe 2-OMe-5-OCF₃
Me 2-F-5-OMe U-4b 3,5-di-OCF₃ SMe 2-OCF₃-5-F
Me 2-F-5-OCF₃ U-4c 2,3-di-F SMe 2-OCF₃-5-Cl
Me 2-Cl-5-F U-4c 2-F-3-Cl SMe 2-OCF₃-5-Br
Me 2,5-di-Cl U-4c 2-F-3-Br SMe 2-OCF₃-5-Me
Me 2-Cl-5-Br U-4c 2-F-3-Me SMe 2-OCF₃-5-CF₃
Me 2-Cl-5-Me U-4c 2-F-3-CF₃ SMe 2-OCF₃-5-OMe
Me 2-Cl-5-CF₃ U-4c 2-F-3-OMe SMe 2,5-di-OCF₃
Me 2-Cl-5-OMe U-4c 2-F-3-OCF₃ SMe 3,4-di-F
Me 2-Cl-5-OCF₃ U-4c 2-Cl-3-F SMe 3-F-4-Cl
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
Me 2-Br-5-F U-4c 2,3-di-Cl SMe 3-F-4-Br
Me 2-Br-5-Cl U-4c 2-Cl-3-Br SMe 3-F-4-Me
Me 2,5-di-Br U-4c 2-Cl-3-Me SMe 3-F-4-CF₃
Me 2-Br-5-Me U-4c 2-Cl-3-CF₃ SMe 3-F-4-OMe
Me 2-Br-5-CF₃ U-4c 2-Cl-3-OMe SMe 3-F-4-OCF₃
Me 2-Br-5-OMe U-4c 2-Cl-3-OCF₃ SMe 3-Cl-4-F
Me 2-Br-5-OCF₃ U-4c 2-Br-3-F SMe 3,4-di-Cl
Me 2-Me-5-F U-4c 2-Br-3-Cl SMe 3-Cl-4-Br
Me 2-Me-5-Cl U-4c 2,3-di-Br SMe 3-Cl-4-Me
Me 2-Me-5-Br U-4c 2-Br-3-Me SMe 3-Cl-4-CF₃
Me 2,5-di-Me U-4c 2-Br-3-CF₃ SMe 3-Cl-4-OMe
Me 2-Me-5-CF₃ U-4c 2-Br-3-OMe SMe 3-Cl-4-OCF₃
Me 2-Me-5-OMe U-4c 2-Br-3-OCF₃ SMe 3-Br-4-F
Me 2-Me-5-OCF₃ U-4c 2-Me-3-F SMe 3-Br-4-Cl
Me 2-CF₃-5-F U-4c 2-Me-3-Cl SMe 3,4-di-Br
Me 2-CF₃-5-Cl U-4c 2-Me-3-Br SMe 3-Br-4-Me
Me 2-CF₃-5-Br U-4c 2,3-di-Me SMe 3-Br-4-CF₃
Me 2-CF₃-5-Me U-4c 2-Me-3-CF₃ SMe 3-Br-4-OMe
Me 2,5-di-CF₃ U-4c 2-Me-3-OMe SMe 3-Br-4-OCF₃
Me 2-CF₃-5-OMe U-4c 2-Me-3-OCF₃ SMe 3-Me-4-F
Me 2-CF₃-5-OCF₃ U-4c 2-CF₃-3-F SMe 3-Me-4-Cl
Me 2-OMe-5-F U-4c 2-CF₃-3-Cl SMe 3-Me-4-Br
Me 2-OMe-5-Cl U-4c 2-CF₃-3-Br SMe 3,4-di-Me
Me 2-OMe-5-Br U-4c 2-CF₃-3-Me SMe 3-Me-4-CF₃
Me 2-OMe-5-Me U-4c 2,3-di-CF₃ SMe 3-Me-4-OMe
Me 2-OMe-5-CF₃ U-4c 2-CF₃-3-OMe SMe 3-Me-4-OCF₃
Me 2,5-di-OMe U-4c 2-CF₃-3-OCF₃ SMe 3-CF₃-4-F
Me 2-OMe-5-OCF₃ U-4c 2-OMe-3-F SMe 3-CF₃-4-Cl
Me 2-OCF₃-5-F U-4c 2-OMe-3-Cl SMe 3-CF₃-4-Br
Me 2-OCF₃-5-Cl U-4c 2-OMe-3-Br SMe 3-CF₃-4-Me
Me 2-OCF₃-5-Br U-4c 2-OMe-3-Me SMe 3,4-di-CF₃
Me 2-OCF₃-5-Me U-4c 2-OMe-3-CF₃ SMe 3-CF₃-4-OMe
Me 2-OCF₃-5-CF₃ U-4c 2,3-di-OMe SMe 3-CF₃-4-OCF₃
Me 2-OCF₃-5-OMe U-4c 2-OMe-3-OCF₃ SMe 3-OMe-4-F
Me 2,5-di-OCF₃ U-4c 2-OCF₃-3-F SMe 3-OMe-4-Cl
Me 3,4-di-F U-4c 2-OCF₃-3-Cl SMe 3-OMe-4-Br
Me 3-F-4-Cl U-4c 2-OCF₃-3-Br SMe 3-OMe-4-Me
Me 3-F-4-Br U-4c 2-OCF₃-3-Me SMe 3-OMe-4-CF₃
Me 3-F-4-Me U-4c 2-OCF₃-3-CF₃ SMe 3,4-di-OMe
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
Me 3-F-4-CF₃ U-4c 2-OCF₃-3-OMe SMe 3-OMe-4-OCF₃
Me 3-F-4-OMe U-4c 2,3-di-OCF₃ SMe 3-OCF₃-4-F
Me 3-F-4-OCF₃ U-4c 2,4-di-F SMe 3-OCF₃-4-Cl
Me 3-Cl-4-F U-4c 2-F-4-Cl SMe 3-OCF₃-4-Br
Me 3,4-di-Cl U-4c 2-F-4-Br SMe 3-OCF₃-4-Me
Me 3-Cl-4-Br U-4c 2-F-4-Me SMe 3-OCF₃-4-CF₃
Me 3-Cl-4-Me U-4c 2-F-4-CF₃ SMe 3-OCF₃-4-OMe
Me 3-Cl-4-CF₃ U-4c 2-F-4-OMe SMe 3,4-di-OCF₃
Me 3-Cl-4-OMe U-4c 2-F-4-OCF₃ SMe 3,5-di-F
Me 3-Cl-4-OCF₃ U-4c 2-Cl-4-F SMe 3-F-5-Cl
Me 3-Br-4-F U-4c 2,4-di-Cl SMe 3-F-5-Br
Me 3-Br-4-Cl U-4c 2-Cl-4-Br SMe 3-F-5-Me
Me 3,4-di-Br U-4c 2-Cl-4-Me SMe 3-F-5-CF₃
Me 3-Br-4-Me U-4c 2-Cl-4-CF₃ SMe 3-F-5-OMe
Me 3-Br-4-CF₃ U-4c 2-Cl-4-OMe SMe 3-F-5-OCF₃
Me 3-Br-4-OMe U-4c 2-Cl-4-OCF₃ SMe 3-Cl-5-F
Me 3-Br-4-OCF₃ U-4c 2-Br-4-F SMe 3,5-di-Cl
Me 3-Me-4-F U-4c 2-Br-4-Cl SMe 3-Cl-5-Br
Me 3-Me-4-Cl U-4c 2,4-di-Br SMe 3-Cl-5-Me
Me 3-Me-4-Br U-4c 2-Br-4-Me SMe 3-Cl-5-CF₃
Me 3,4-di-Me U-4c 2-Br-4-CF₃ SMe 3-Cl-5-OMe
Me 3-Me-4-CF₃ U-4c 2-Br-4-OMe SMe 3-Cl-5-OCF₃
Me 3-Me-4-OMe U-4c 2-Br-4-OCF₃ SMe 3-Br-5-F
Me 3-Me-4-OCF₃ U-4c 2-Me-4-F SMe 3-Br-5-Cl
Me 3-CF₃-4-F U-4c 2-Me-4-Cl SMe 3,5-di-Br
Me 3-CF₃-4-Cl U-4c 2-Me-4-Br SMe 3-Br-5-Me
Me 3-CF₃-4-Br U-4c 2,4-di-Me SMe 3-Br-5-CF₃
Me 3-CF₃-4-Me U-4c 2-Me-4-CF₃ SMe 3-Br-5-OMe
Me 3,4-di-CF₃ U-4c 2-Me-4-OMe SMe 3-Br-5-OCF₃
Me 3-CF₃-4-OMe U-4c 2-Me-4-OCF₃ SMe 3-Me-5-F
Me 3-CF₃-4-OCF₃ U-4c 2-CF₃-4-F SMe 3-Me-5-Cl
Me 3-OMe-4-F U-4c 2-CF₃-4-Cl SMe 3-Me-5-Br
Me 3-OMe-4-Cl U-4c 2-CF₃-4-Br SMe 3,5-di-Me
Me 3-OMe-4-Br U-4c 2-CF₃-4-Me SMe 3-Me-5-CF₃
Me 3-OMe-4-Me U-4c 2,4-di-CF₃ SMe 3-Me-5-OMe
Me 3-OMe-4-CF₃ U-4c 2-CF₃-4-OMe SMe 3-Me-5-OCF₃
Me 3,4-di-OMe U-4c 2-CF₃-4-OCF₃ SMe 3-CF₃-5-F
Me 3-OMe-4-OCF₃ U-4c 2-OMe-4-F SMe 3-CF₃-5-Cl
Me 3-OCF₃-4-F U-4c 2-OMe-4-Cl SMe 3-CF₃-5-Br
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
Me 3-OCF₃-4-Cl U-4c 2-OMe-4-Br SMe 3-CF₃-5-Me
Me 3-OCF₃-4-Br U-4c 2-OMe-4-Me SMe 3,5-di-CF₃
Me 3-OCF₃-4-Me U-4c 2-OMe-4-CF₃ SMe 3-CF₃-5-OMe
Me 3-OCF₃-4-CF₃ U-4c 2,4-di-OMe SMe 3-CF₃-5-OCF₃
Me 3-OCF₃-4-OMe U-4c 2-OMe-4-OCF₃ SMe 3-OMe-5-F
Me 3,4-di-OCF₃ U-4c 2-OCF₃-4-F SMe 3-OMe-5-Cl
Me 3,5-di-F U-4c 2-OCF₃-4-Cl SMe 3-OMe-5-Br
Me 3-F-5-Cl U-4c 2-OCF₃-4-Br SMe 3-OMe-5-Me
Me 3-F-5-Br U-4c 2-OCF₃-4-Me SMe 3-OMe-5-CF₃
Me 3-F-5-Me U-4c 2-OCF₃-4-CF₃ SMe 3,5-di-OMe
Me 3-F-5-CF₃ U-4c 2-OCF₃-4-OMe SMe 3-OMe-5-OCF₃
Me 3-F-5-OMe U-4c 2,4-di-OCF₃ SMe 3-OCF₃-5-F
Me 3-F-5-OCF₃ U-4c 2,5-di-F SMe 3-OCF₃-5-Cl
Me 3-Cl-5-F U-4c 2-F-5-Cl SMe 3-OCF₃-5-Br
Me 3,5-di-Cl U-4c 2-F-5-Br SMe 3-OCF₃-5-Me
Me 3-Cl-5-Br U-4c 2-F-5-Me SMe 3-OCF₃-5-CF₃
Me 3-Cl-5-Me U-4c 2-F-5-CF₃ SMe 3-OCF₃-5-OMe
Me 3-Cl-5-CF₃ U-4c 2-F-5-OMe SMe 3,5-di-OCF₃
Me 3-Cl-5-OMe U-4c 2-F-5-OCF₃ Ac 2,3-di-F
Me 3-Cl-5-OCF₃ U-4c 2-Cl-5-F Ac 2-F-3-Cl
Me 3-Br-5-F U-4c 2,5-di-Cl Ac 2-F-3-Br
Me 3-Br-5-Cl U-4c 2-Cl-5-Br Ac 2-F-3-Me
Me 3,5-di-Br U-4c 2-Cl-5-Me Ac 2-F-3-CF₃
Me 3-Br-5-Me U-4c 2-Cl-5-CF₃ Ac 2-F-3-OMe
Me 3-Br-5-CF₃ U-4c 2-Cl-5-OMe Ac 2-F-3-OCF₃
Me 3-Br-5-OMe U-4c 2-Cl-5-OCF₃ Ac 2-Cl-3-F
Me 3-Br-5-OCF₃ U-4c 2-Br-5-F Ac 2,3-di-Cl
Me 3-Me-5-F U-4c 2-Br-5-Cl Ac 2-Cl-3-Br
Me 3-Me-5-Cl U-4c 2,5-di-Br Ac 2-Cl-3-Me
Me 3-Me-5-Br U-4c 2-Br-5-Me Ac 2-Cl-3-CF₃
Me 3,5-di-Me U-4c 2-Br-5-CF₃ Ac 2-Cl-3-OMe
Me 3-Me-5-CF₃ U-4c 2-Br-5-OMe Ac 2-Cl-3-OCF₃
Me 3-Me-5-OMe U-4c 2-Br-5-OCF₃ Ac 2-Br-3-F
Me 3-Me-5-OCF₃ U-4c 2-Me-5-F Ac 2-Br-3-Cl
Me 3-CF₃-5-F U-4c 2-Me-5-Cl Ac 2,3-di-Br
Me 3-CF₃-5-Cl U-4c 2-Me-5-Br Ac 2-Br-3-Me
Me 3-CF₃-5-Br U-4c 2,5-di-Me Ac 2-Br-3-CF₃
Me 3-CF₃-5-Me U-4c 2-Me-5-CF₃ Ac 2-Br-3-OMe
Me 3,5-di-CF₃ U-4c 2-Me-5-OMe Ac 2-Br-3-OCF₃
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
Me 3-CF₃-5-OMe U-4c 2-Me-5-OCF₃ Ac 2-Me-3-F
Me 3-CF₃-5-OCF₃ U-4c 2-CF₃-5-F Ac 2-Me-3-Cl
Me 3-OMe-5-F U-4c 2-CF₃-5-Cl Ac 2-Me-3-Br
Me 3-OMe-5-Cl U-4c 2-CF₃-5-Br Ac 2,3-di-Me
Me 3-OMe-5-Br U-4c 2-CF₃-5-Me Ac 2-Me-3-CF₃
Me 3-OMe-5-Me U-4c 2,5-di-CF₃ Ac 2-Me-3-OMe
Me 3-OMe-5-CF₃ U-4c 2-CF₃-5-OMe Ac 2-Me-3-OCF₃
Me 3,5-di-OMe U-4c 2-CF₃-5-OCF₃ Ac 2-CF₃-3-F
Me 3-OMe-5-OCF₃ U-4c 2-OMe-5-F Ac 2-CF₃-3-Cl
Me 3-OCF₃-5-F U-4c 2-OMe-5-Cl Ac 2-CF₃-3-Br
Me 3-OCF₃-5-Cl U-4c 2-OMe-5-Br Ac 2-CF₃-3-Me
Me 3-OCF₃-5-Br U-4c 2-OMe-5-Me Ac 2,3-di-CF₃
Me 3-OCF₃-5-Me U-4c 2-OMe-5-CF₃ Ac 2-CF₃-3-OMe
Me 3-OCF₃-5-CF₃ U-4c 2,5-di-OMe Ac 2-CF₃-3-OCF₃
Me 3-OCF₃-5-OMe U-4c 2-OMe-5-OCF₃ Ac 2-OMe-3-F
Me 3,5-di-OCF₃ U-4c 2-OCF₃-5-F Ac 2-OMe-3-Cl
Et 2,3-di-F U-4c 2-OCF₃-5-Cl Ac 2-OMe-3-Br
Et 2-F-3-Cl U-4c 2-OCF₃-5-Br Ac 2-OMe-3-Me
Et 2-F-3-Br U-4c 2-OCF₃-5-Me Ac 2-OMe-3-CF₃
Et 2-F-3-Me U-4c 2-OCF₃-5-CF₃ Ac 2,3-di-OMe
Et 2-F-3-CF₃ U-4c 2-OCF₃-5-OMe Ac 2-OMe-3-OCF₃
Et 2-F-3-OMe U-4c 2,5-di-OCF₃ Ac 2-OCF₃-3-F
Et 2-F-3-OCF₃ U-4c 3,4-di-F Ac 2-OCF₃-3-Cl
Et 2-Cl-3-F U-4c 3-F-4-Cl Ac 2-OCF₃-3-Br
Et 2,3-di-Cl U-4c 3-F-4-Br Ac 2-OCF₃-3-Me
Et 2-Cl-3-Br U-4c 3-F-4-Me Ac 2-OCF₃-3-CF₃
Et 2-Cl-3-Me U-4c 3-F-4-CF₃ Ac 2-OCF₃-3-OMe
Et 2-Cl-3-CF₃ U-4c 3-F-4-OMe Ac 2,3-di-OCF₃
Et 2-Cl-3-OMe U-4c 3-F-4-OCF₃ Ac 2,4-di-F
Et 2-Cl-3-OCF₃ U-4c 3-Cl-4-F Ac 2-F-4-Cl
Et 2-Br-3-F U-4c 3,4-di-Cl Ac 2-F-4-Br
Et 2-Br-3-Cl U-4c 3-Cl-4-Br Ac 2-F-4-Me
Et 2,3-di-Br U-4c 3-Cl-4-Me Ac 2-F-4-CF₃
Et 2-Br-3-Me U-4c 3-Cl-4-CF₃ Ac 2-F-4-OMe
Et 2-Br-3-CF₃ U-4c 3-Cl-4-OMe Ac 2-F-4-OCF₃
Et 2-Br-3-OMe U-4c 3-Cl-4-OCF₃ Ac 2-Cl-4-F
Et 2-Br-3-OCF₃ U-4c 3-Br-4-F Ac 2,4-di-Cl
Et 2-Me-3-F U-4c 3-Br-4-Cl Ac 2-Cl-4-Br
Et 2-Me-3-Cl U-4c 3,4-di-Br Ac 2-Cl-4-Me
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
Et 2-Me-3-Br U-4c 3-Br-4-Me Ac 2-Cl-4-CF₃
Et 2,3-di-Me U-4c 3-Br-4-CF₃ Ac 2-Cl-4-OMe
Et 2-Me-3-CF₃ U-4c 3-Br-4-OMe Ac 2-Cl-4-OCF₃
Et 2-Me-3-OMe U-4c 3-Br-4-OCF₃ Ac 2-Br-4-F
Et 2-Me-3-OCF₃ U-4c 3-Me-4-F Ac 2-Br-4-Cl
Et 2-CF₃-3-F U-4c 3-Me-4-Cl Ac 2,4-di-Br
Et 2-CF₃-3-Cl U-4c 3-Me-4-Br Ac 2-Br-4-Me
Et 2-CF₃-3-Br U-4c 3,4-di-Me Ac 2-Br-4-CF₃
Et 2-CF₃-3-Me U-4c 3-Me-4-CF₃ Ac 2-Br-4-OMe
Et 2,3-di-CF₃ U-4c 3-Me-4-OMe Ac 2-Br-4-OCF₃
Et 2-CF₃-3-OMe U-4c 3-Me-4-OCF₃ Ac 2-Me-4-F
Et 2-CF₃-3-OCF₃ U-4c 3-CF₃-4-F Ac 2-Me-4-Cl
Et 2-OMe-3-F U-4c 3-CF₃-4-Cl Ac 2-Me-4-Br
Et 2-OMe-3-Cl U-4c 3-CF₃-4-Br Ac 2,4-di-Me
Et 2-OMe-3-Br U-4c 3-CF₃-4-Me Ac 2-Me-4-CF₃
Et 2-OMe-3-Me U-4c 3,4-di-CF₃ Ac 2-Me-4-OMe
Et 2-OMe-3-CF₃ U-4c 3-CF₃-4-OMe Ac 2-Me-4-OCF₃
Et 2,3-di-OMe U-4c 3-CF₃-4-OCF₃ Ac 2-CF₃-4-F
Et 2-OMe-3-OCF₃ U-4c 3-OMe-4-F Ac 2-CF₃-4-Cl
Et 2-OCF₃-3-F U-4c 3-OMe-4-Cl Ac 2-CF₃-4-Br
Et 2-OCF₃-3-Cl U-4c 3-OMe-4-Br Ac 2-CF₃-4-Me
Et 2-OCF₃-3-Br U-4c 3-OMe-4-Me Ac 2,4-di-CF₃
Et 2-OCF₃-3-Me U-4c 3-OMe-4-CF₃ Ac 2-CF₃-4-OMe
Et 2-OCF₃-3-CF₃ U-4c 3,4-di-OMe Ac 2-CF₃-4-OCF₃
Et 2-OCF₃-3-OMe U-4c 3-OMe-4-OCF₃ Ac 2-OMe-4-F
Et 2,3-di-OCF₃ U-4c 3-OCF₃-4-F Ac 2-OMe-4-Cl
Et 2,4-di-F U-4c 3-OCF₃-4-Cl Ac 2-OMe-4-Br
Et 2-F-4-Cl U-4c 3-OCF₃-4-Br Ac 2-OMe-4-Me
Et 2-F-4-Br U-4c 3-OCF₃-4-Me Ac 2-OMe-4-CF₃
Et 2-F-4-Me U-4c 3-OCF₃-4-CF₃ Ac 2,4-di-OMe
Et 2-F-4-CF₃ U-4c 3-OCF₃-4-OMe Ac 2-OMe-4-OCF₃
Et 2-F-4-OMe U-4c 3,4-di-OCF₃ Ac 2-OCF₃-4-F
Et 2-F-4-OCF₃ U-4c 3,5-di-F Ac 2-OCF₃-4-Cl
Et 2-Cl-4-F U-4c 3-F-5-Cl Ac 2-OCF₃-4-Br
Et 2,4-di-Cl U-4c 3-F-5-Br Ac 2-OCF₃-4-Me
Et 2-Cl-4-Br U-4c 3-F-5-Me Ac 2-OCF₃-4-CF₃
Et 2-Cl-4-Me U-4c 3-F-5-CF₃ Ac 2-OCF₃-4-OMe
Et 2-Cl-4-CF₃ U-4c 3-F-5-OMe Ac 2,4-di-OCF₃
Et 2-Cl-4-OMe U-4c 3-F-5-OCF₃ Ac 2,5-di-F
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
Et 2-Cl-4-OCF₃ U-4c 3-Cl-5-F Ac 2-F-5-Cl
Et 2-Br-4-F U-4c 3,5-di-Cl Ac 2-F-5-Br
Et 2-Br-4-Cl U-4c 3-Cl-5-Br Ac 2-F-5-Me
Et 2,4-di-Br U-4c 3-Cl-5-Me Ac 2-F-5-CF₃
Et 2-Br-4-Me U-4c 3-Cl-5-CF₃ Ac 2-F-5-OMe
Et 2-Br-4-CF₃ U-4c 3-Cl-5-OMe Ac 2-F-5-OCF₃
Et 2-Br-4-OMe U-4c 3-Cl-5-OCF₃ Ac 2-Cl-5-F
Et 2-Br-4-OCF₃ U-4c 3-Br-5-F Ac 2,5-di-Cl
Et 2-Me-4-F U-4c 3-Br-5-Cl Ac 2-Cl-5-Br
Et 2-Me-4-Cl U-4c 3,5-di-Br Ac 2-Cl-5-Me
Et 2-Me-4-Br U-4c 3-Br-5-Me Ac 2-Cl-5-CF₃
Et 2,4-di-Me U-4c 3-Br-5-CF₃ Ac 2-Cl-5-OMe
Et 2-Me-4-CF₃ U-4c 3-Br-5-OMe Ac 2-Cl-5-OCF₃
Et 2-Me-4-OMe U-4c 3-Br-5-OCF₃ Ac 2-Br-5-F
Et 2-Me-4-OCF₃ U-4c 3-Me-5-F Ac 2-Br-5-Cl
Et 2-CF₃-4-F U-4c 3-Me-5-Cl Ac 2,5-di-Br
Et 2-CF₃-4-Cl U-4c 3-Me-5-Br Ac 2-Br-5-Me
Et 2-CF₃-4-Br U-4c 3,5-di-Me Ac 2-Br-5-CF₃
Et 2-CF₃-4-Me U-4c 3-Me-5-CF₃ Ac 2-Br-5-OMe
Et 2,4-di-CF₃ U-4c 3-Me-5-OMe Ac 2-Br-5-OCF₃
Et 2-CF₃-4-OMe U-4c 3-Me-5-OCF₃ Ac 2-Me-5-F
Et 2-CF₃-4-OCF₃ U-4c 3-CF₃-5-F Ac 2-Me-5-Cl
Et 2-OMe-4-F U-4c 3-CF₃-5-Cl Ac 2-Me-5-Br
Et 2-OMe-4-Cl U-4c 3-CF₃-5-Br Ac 2,5-di-Me
Et 2-OMe-4-Br U-4c 3-CF₃-5-Me Ac 2-Me-5-CF₃
Et 2-OMe-4-Me U-4c 3,5-di-CF₃ Ac 2-Me-5-OMe
Et 2-OMe-4-CF₃ U-4c 3-CF₃-5-OMe Ac 2-Me-5-OCF₃
Et 2,4-di-OMe U-4c 3-CF₃-5-OCF₃ Ac 2-CF₃-5-F
Et 2-OMe-4-OCF₃ U-4c 3-OMe-5-F Ac 2-CF₃-5-Cl
Et 2-OCF₃-4-F U-4c 3-OMe-5-Cl Ac 2-CF₃-5-Br
Et 2-OCF₃-4-Cl U-4c 3-OMe-5-Br Ac 2-CF₃-5-Me
Et 2-OCF₃-4-Br U-4c 3-OMe-5-Me Ac 2,5-di-CF₃
Et 2-OCF₃-4-Me U-4c 3-OMe-5-CF₃ Ac 2-CF₃-5-OMe
Et 2-OCF₃-4-CF₃ U-4c 3,5-di-OMe Ac 2-CF₃-5-OCF₃
Et 2-OCF₃-4-OMe U-4c 3-OMe-5-OCF₃ Ac 2-OMe-5-F
Et 2,4-di-OCF₃ U-4c 3-OCF₃-5-F Ac 2-OMe-5-Cl
Et 2,5-di-F U-4c 3-OCF₃-5-Cl Ac 2-OMe-5-Br
Et 2-F-5-Cl U-4c 3-OCF₃-5-Br Ac 2-OMe-5-Me
Et 2-F-5-Br U-4c 3-OCF₃-5-Me Ac 2-OMe-5-CF₃
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
Et 2-F-5-Me U-4c 3-OCF₃-5-CF₃ Ac 2,5-di-OMe
Et 2-F-5-CF₃ U-4c 3-OCF₃-5-OMe Ac 2-OMe-5-OCF₃
Et 2-F-5-OMe U-4c 3,5-di-OCF₃ Ac 2-OCF₃-5-F
Et 2-F-5-OCF₃ U-4d 2,3-di-F Ac 2-OCF₃-5-Cl
Et 2-Cl-5-F U-4d 2-F-3-Cl Ac 2-OCF₃-5-Br
Et 2,5-di-Cl U-4d 2-F-3-Br Ac 2-OCF₃-5-Me
Et 2-Cl-5-Br U-4d 2-F-3-Me Ac 2-OCF₃-5-CF₃
Et 2-Cl-5-Me U-4d 2-F-3-CF₃ Ac 2-OCF₃-5-OMe
Et 2-Cl-5-CF₃ U-4d 2-F-3-OMe Ac 2,5-di-OCF₃
Et 2-Cl-5-OMe U-4d 2-F-3-OCF₃ Ac 3,4-di-F
Et 2-Cl-5-OCF₃ U-4d 2-Cl-3-F Ac 3-F-4-Cl
Et 2-Br-5-F U-4d 2,3-di-Cl Ac 3-F-4-Br
Et 2-Br-5-Cl U-4d 2-Cl-3-Br Ac 3-F-4-Me
Et 2,5-di-Br U-4d 2-Cl-3-Me Ac 3-F-4-CF₃
Et 2-Br-5-Me U-4d 2-Cl-3-CF₃ Ac 3-F-4-OMe
Et 2-Br-5-CF₃ U-4d 2-Cl-3-OMe Ac 3-F-4-OCF₃
Et 2-Br-5-OMe U-4d 2-Cl-3-OCF₃ Ac 3-Cl-4-F
Et 2-Br-5-OCF₃ U-4d 2-Br-3-F Ac 3,4-di-Cl
Et 2-Me-5-F U-4d 2-Br-3-Cl Ac 3-Cl-4-Br
Et 2-Me-5-Cl U-4d 2,3-di-Br Ac 3-Cl-4-Me
Et 2-Me-5-Br U-4d 2-Br-3-Me Ac 3-Cl-4-CF₃
Et 2,5-di-Me U-4d 2-Br-3-CF₃ Ac 3-Cl-4-OMe
Et 2-Me-5-CF₃ U-4d 2-Br-3-OMe Ac 3-Cl-4-OCF₃
Et 2-Me-5-OMe U-4d 2-Br-3-OCF₃ Ac 3-Br-4-F
Et 2-Me-5-OCF₃ U-4d 2-Me-3-F Ac 3-Br-4-Cl
Et 2-CF₃-5-F U-4d 2-Me-3-Cl Ac 3,4-di-Br
Et 2-CF₃-5-Cl U-4d 2-Me-3-Br Ac 3-Br-4-Me
Et 2-CF₃-5-Br U-4d 2,3-di-Me Ac 3-Br-4-CF₃
Et 2-CF₃-5-Me U-4d 2-Me-3-CF₃ Ac 3-Br-4-OMe
Et 2,5-di-CF₃ U-4d 2-Me-3-OMe Ac 3-Br-4-OCF₃
Et 2-CF₃-5-OMe U-4d 2-Me-3-OCF₃ Ac 3-Me-4-F
Et 2-CF₃-5-OCF₃ U-4d 2-CF₃-3-F Ac 3-Me-4-Cl
Et 2-OMe-5-F U-4d 2-CF₃-3-Cl Ac 3-Me-4-Br
Et 2-OMe-5-Cl U-4d 2-CF₃-3-Br Ac 3,4-di-Me
Et 2-OMe-5-Br U-4d 2-CF₃-3-Me Ac 3-Me-4-CF₃
Et 2-OMe-5-Me U-4d 2,3-di-CF₃ Ac 3-Me-4-OMe
Et 2-OMe-5-CF₃ U-4d 2-CF₃-3-OMe Ac 3-Me-4-OCF₃
Et 2,5-di-OMe U-4d 2-CF₃-3-OCF₃ Ac 3-CF₃-4-F
Et 2-OMe-5-OCF₃ U-4d 2-OMe-3-F Ac 3-CF₃-4-Cl
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
Et 2-OCF₃-5-F U-4d 2-OMe-3-Cl Ac 3-CF₃-4-Br
Et 2-OCF₃-5-Cl U-4d 2-OMe-3-Br Ac 3-CF₃-4-Me
Et 2-OCF₃-5-Br U-4d 2-OMe-3-Me Ac 3,4-di-CF₃
Et 2-OCF₃-5-Me U-4d 2-OMe-3-CF₃ Ac 3-CF₃-4-OMe
Et 2-OCF₃-5-CF₃ U-4d 2,3-di-OMe Ac 3-CF₃-4-OCF₃
Et 2-OCF₃-5-OMe U-4d 2-OMe-3-OCF₃ Ac 3-OMe-4-F
Et 2,5-di-OCF₃ U-4d 2-OCF₃-3-F Ac 3-OMe-4-Cl
Et 3,4-di-F U-4d 2-OCF₃-3-Cl Ac 3-OMe-4-Br
Et 3-F-4-Cl U-4d 2-OCF₃-3-Br Ac 3-OMe-4-Me
Et 3-F-4-Br U-4d 2-OCF₃-3-Me Ac 3-OMe-4-CF₃
Et 3-F-4-Me U-4d 2-OCF₃-3-CF₃ Ac 3,4-di-OMe
Et 3-F-4-CF₃ U-4d 2-OCF₃-3-OMe Ac 3-OMe-4-OCF₃
Et 3-F-4-OMe U-4d 2,3-di-OCF₃ Ac 3-OCF₃-4-F
Et 3-F-4-OCF₃ U-4d 2,4-di-F Ac 3-OCF₃-4-Cl
Et 3-Cl-4-F U-4d 2-F-4-Cl Ac 3-OCF₃-4-Br
Et 3,4-di-Cl U-4d 2-F-4-Br Ac 3-OCF₃-4-Me
Et 3-Cl-4-Br U-4d 2-F-4-Me Ac 3-OCF₃-4-CF₃
Et 3-Cl-4-Me U-4d 2-F-4-CF₃ Ac 3-OCF₃-4-OMe
Et 3-Cl-4-CF₃ U-4d 2-F-4-OMe Ac 3,4-di-OCF₃
Et 3-Cl-4-OMe U-4d 2-F-4-OCF₃ Ac 3,5-di-F
Et 3-Cl-4-OCF₃ U-4d 2-Cl-4-F Ac 3-F-5-Cl
Et 3-Br-4-F U-4d 2,4-di-Cl Ac 3-F-5-Br
Et 3-Br-4-Cl U-4d 2-Cl-4-Br Ac 3-F-5-Me
Et 3,4-di-Br U-4d 2-Cl-4-Me Ac 3-F-5-CF₃
Et 3-Br-4-Me U-4d 2-Cl-4-CF₃ Ac 3-F-5-OMe
Et 3-Br-4-CF₃ U-4d 2-Cl-4-OMe Ac 3-F-5-OCF₃
Et 3-Br-4-OMe U-4d 2-Cl-4-OCF₃ Ac 3-Cl-5-F
Et 3-Br-4-OCF₃ U-4d 2-Br-4-F Ac 3,5-di-Cl
Et 3-Me-4-F U-4d 2-Br-4-Cl Ac 3-Cl-5-Br
Et 3-Me-4-Cl U-4d 2,4-di-Br Ac 3-Cl-5-Me
Et 3-Me-4-Br U-4d 2-Br-4-Me Ac 3-Cl-5-CF₃
Et 3,4-di-Me U-4d 2-Br-4-CF₃ Ac 3-Cl-5-OMe
Et 3-Me-4-CF₃ U-4d 2-Br-4-OMe Ac 3-Cl-5-OCF₃
Et 3-Me-4-OMe U-4d 2-Br-4-OCF₃ Ac 3-Br-5-F
Et 3-Me-4-OCF₃ U-4d 2-Me-4-F Ac 3-Br-5-Cl
Et 3-CF₃-4-F U-4d 2-Me-4-Cl Ac 3,5-di-Br
Et 3-CF₃-4-Cl U-4d 2-Me-4-Br Ac 3-Br-5-Me
Et 3-CF₃-4-Br U-4d 2,4-di-Me Ac 3-Br-5-CF₃
Et 3-CF₃-4-Me U-4d 2-Me-4-CF₃ Ac 3-Br-5-OMe
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
Et 3,4-di-CF₃ U-4d 2-Me-4-OMe Ac 3-Br-5-OCF₃
Et 3-CF₃-4-OMe U-4d 2-Me-4-OCF₃ Ac 3-Me-5-F
Et 3-CF₃-4-OCF₃ U-4d 2-CF₃-4-F Ac 3-Me-5-Cl
Et 3-OMe-4-F U-4d 2-CF₃-4-Cl Ac 3-Me-5-Br
Et 3-OMe-4-Cl U-4d 2-CF₃-4-Br Ac 3,5-di-Me
Et 3-OMe-4-Br U-4d 2-CF₃-4-Me Ac 3-Me-5-CF₃
Et 3-OMe-4-Me U-4d 2,4-di-CF₃ Ac 3-Me-5-OMe
Et 3-OMe-4-CF₃ U-4d 2-CF₃-4-OMe Ac 3-Me-5-OCF₃
Et 3,4-di-OMe U-4d 2-CF₃-4-OCF₃ Ac 3-CF₃-5-F
Et 3-OMe-4-OCF₃ U-4d 2-OMe-4-F Ac 3-CF₃-5-Cl
Et 3-OCF₃-4-F U-4d 2-OMe-4-Cl Ac 3-CF₃-5-Br
Et 3-OCF₃-4-Cl U-4d 2-OMe-4-Br Ac 3-CF₃-5-Me
Et 3-OCF₃-4-Br U-4d 2-OMe-4-Me Ac 3,5-di-CF₃
Et 3-OCF₃-4-Me U-4d 2-OMe-4-CF₃ Ac 3-CF₃-5-OMe
Et 3-OCF₃-4-CF₃ U-4d 2,4-di-OMe Ac 3-CF₃-5-OCF₃
Et 3-OCF₃-4-OMe U-4d 2-OMe-4-OCF₃ Ac 3-OMe-5-F
Et 3,4-di-OCF₃ U-4d 2-OCF₃-4-F Ac 3-OMe-5-Cl
Et 3,5-di-F U-4d 2-OCF₃-4-Cl Ac 3-OMe-5-Br
Et 3-F-5-Cl U-4d 2-OCF₃-4-Br Ac 3-OMe-5-Me
Et 3-F-5-Br U-4d 2-OCF₃-4-Me Ac 3-OMe-5-CF₃
Et 3-F-5-Me U-4d 2-OCF₃-4-CF₃ Ac 3,5-di-OMe
Et 3-F-5-CF₃ U-4d 2-OCF₃-4-OMe Ac 3-OMe-5-OCF₃
Et 3-F-5-OMe U-4d 2,4-di-OCF₃ Ac 3-OCF₃-5-F
Et 3-F-5-OCF₃ U-4d 2,5-di-F Ac 3-OCF₃-5-Cl
Et 3-Cl-5-F U-4d 2-F-5-Cl Ac 3-OCF₃-5-Br
Et 3,5-di-Cl U-4d 2-F-5-Br Ac 3-OCF₃-5-Me
Et 3-Cl-5-Br U-4d 2-F-5-Me Ac 3-OCF₃-5-CF₃
Et 3-Cl-5-Me U-4d 2-F-5-CF₃ Ac 3-OCF₃-5-OMe
Et 3-Cl-5-CF₃ U-4d 2-F-5-OMe Ac 3,5-di-OCF₃
Et 3-Cl-5-OMe U-4d 2-F-5-OCF₃ cPen 2,3-di-F
Et 3-Cl-5-OCF₃ U-4d 2-Cl-5-F cPen 2-F-3-Cl
Et 3-Br-5-F U-4d 2,5-di-Cl cPen 2-F-3-Br
Et 3-Br-5-Cl U-4d 2-Cl-5-Br cPen 2-F-3-Me
Et 3,5-di-Br U-4d 2-Cl-5-Me cPen 2-F-3-CF₃
Et 3-Br-5-Me U-4d 2-Cl-5-CF₃ cPen 2-F-3-OMe
Et 3-Br-5-CF₃ U-4d 2-Cl-5-OMe cPen 2-F-3-OCF₃
Et 3-Br-5-OMe U-4d 2-Cl-5-OCF₃ cPen 2-Cl-3-F
Et 3-Br-5-OCF₃ U-4d 2-Br-5-F cPen 2,3-di-Cl
Et 3-Me-5-F U-4d 2-Br-5-Cl cPen 2-Cl-3-Br
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
Et 3-Me-5-Cl U-4d 2,5-di-Br cPen 2-Cl-3-Me
Et 3-Me-5-Br U-4d 2-Br-5-Me cPen 2-Cl-3-CF₃
Et 3,5-di-Me U-4d 2-Br-5-CF₃ cPen 2-Cl-3-OMe
Et 3-Me-5-CF₃ U-4d 2-Br-5-OMe cPen 2-Cl-3-OCF₃
Et 3-Me-5-OMe U-4d 2-Br-5-OCF₃ cPen 2-Br-3-F
Et 3-Me-5-OCF₃ U-4d 2-Me-5-F cPen 2-Br-3-Cl
Et 3-CF₃-5-F U-4d 2-Me-5-Cl cPen 2,3-di-Br
Et 3-CF₃-5-Cl U-4d 2-Me-5-Br cPen 2-Br-3-Me
Et 3-CF₃-5-Br U-4d 2,5-di-Me cPen 2-Br-3-CF₃
Et 3-CF₃-5-Me U-4d 2-Me-5-CF₃ cPen 2-Br-3-OMe
Et 3,5-di-CF₃ U-4d 2-Me-5-OMe cPen 2-Br-3-OCF₃
Et 3-CF₃-5-OMe U-4d 2-Me-5-OCF₃ cPen 2-Me-3-F
Et 3-CF₃-5-OCF₃ U-4d 2-CF₃-5-F cPen 2-Me-3-Cl
Et 3-OMe-5-F U-4d 2-CF₃-5-Cl cPen 2-Me-3-Br
Et 3-OMe-5-Cl U-4d 2-CF₃-5-Br cPen 2,3-di-Me
Et 3-OMe-5-Br U-4d 2-CF₃-5-Me cPen 2-Me-3-CF₃
Et 3-OMe-5-Me U-4d 2,5-di-CF₃ cPen 2-Me-3-OMe
Et 3-OMe-5-CF₃ U-4d 2-CF₃-5-OMe cPen 2-Me-3-OCF₃
Et 3,5-di-OMe U-4d 2-CF₃-5-OCF₃ cPen 2-CF₃-3-F
Et 3-OMe-5-OCF₃ U-4d 2-OMe-5-F cPen 2-CF₃-3-Cl
Et 3-OCF₃-5-F U-4d 2-OMe-5-Cl cPen 2-CF₃-3-Br
Et 3-OCF₃-5-Cl U-4d 2-OMe-5-Br cPen 2-CF₃-3-Me
Et 3-OCF₃-5-Br U-4d 2-OMe-5-Me cPen 2,3-di-CF₃
Et 3-OCF₃-5-Me U-4d 2-OMe-5-CF₃ cPen 2-CF₃-3-OMe
Et 3-OCF₃-5-CF₃ U-4d 2,5-di-OMe cPen 2-CF₃-3-OCF₃
Et 3-OCF₃-5-OMe U-4d 2-OMe-5-OCF₃ cPen 2-OMe-3-F
Et 3,5-di-OCF₃ U-4d 2-OCF₃-5-F cPen 2-OMe-3-Cl
iPr 2,3-di-F U-4d 2-OCF₃-5-Cl cPen 2-OMe-3-Br
iPr 2-F-3-Cl U-4d 2-OCF₃-5-Br cPen 2-OMe-3-Me
iPr 2-F-3-Br U-4d 2-OCF₃-5-Me cPen 2-OMe-3-CF₃
iPr 2-F-3-Me U-4d 2-OCF₃-5-CF₃ cPen 2,3-di-OMe
iPr 2-F-3-CF₃ U-4d 2-OCF₃-5-OMe cPen 2-OMe-3-OCF₃
iPr 2-F-3-OMe U-4d 2,5-di-OCF₃ cPen 2-OCF₃-3-F
iPr 2-F-3-OCF₃ U-4d 3,4-di-F cPen 2-OCF₃-3-Cl
iPr 2-Cl-3-F U-4d 3-F-4-Cl cPen 2-OCF₃-3-Br
iPr 2,3-di-Cl U-4d 3-F-4-Br cPen 2-OCF₃-3-Me
iPr 2-Cl-3-Br U-4d 3-F-4-Me cPen 2-OCF₃-3-CF₃
iPr 2-Cl-3-Me U-4d 3-F-4-CF₃ cPen 2-OCF₃-3-OMe
iPr 2-Cl-3-CF₃ U-4d 3-F-4-OMe cPen 2,3-di-OCF₃
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
iPr 2-Cl-3-OMe U-4d 3-F-4-OCF₃ cPen 2,4-di-F
iPr 2-Cl-3-OCF₃ U-4d 3-Cl-4-F cPen 2-F-4-Cl
iPr 2-Br-3-F U-4d 3,4-di-Cl cPen 2-F-4-Br
iPr 2-Br-3-Cl U-4d 3-Cl-4-Br cPen 2-F-4-Me
iPr 2,3-di-Br U-4d 3-Cl-4-Me cPen 2-F-4-CF₃
iPr 2-Br-3-Me U-4d 3-Cl-4-CF₃ cPen 2-F-4-OMe
iPr 2-Br-3-CF₃ U-4d 3-Cl-4-OMe cPen 2-F-4-OCF₃
iPr 2-Br-3-OMe U-4d 3-Cl-4-OCF₃ cPen 2-Cl-4-F
iPr 2-Br-3-OCF₃ U-4d 3-Br-4-F cPen 2,4-di-Cl
iPr 2-Me-3-F U-4d 3-Br-4-Cl cPen 2-Cl-4-Br
iPr 2-Me-3-Cl U-4d 3,4-di-Br cPen 2-Cl-4-Me
iPr 2-Me-3-Br U-4d 3-Br-4-Me cPen 2-Cl-4-CF₃
iPr 2,3-di-Me U-4d 3-Br-4-CF₃ cPen 2-Cl-4-OMe
iPr 2-Me-3-CF₃ U-4d 3-Br-4-OMe cPen 2-Cl-4-OCF₃
iPr 2-Me-3-OMe U-4d 3-Br-4-OCF₃ cPen 2-Br-4-F
iPr 2-Me-3-OCF₃ U-4d 3-Me-4-F cPen 2-Br-4-Cl
iPr 2-CF₃-3-F U-4d 3-Me-4-Cl cPen 2,4-di-Br
iPr 2-CF₃-3-Cl U-4d 3-Me-4-Br cPen 2-Br-4-Me
iPr 2-CF₃-3-Br U-4d 3,4-di-Me cPen 2-Br-4-CF₃
iPr 2-CF₃-3-Me U-4d 3-Me-4-CF₃ cPen 2-Br-4-OMe
iPr 2,3-di-CF₃ U-4d 3-Me-4-OMe cPen 2-Br-4-OCF₃
iPr 2-CF₃-3-OMe U-4d 3-Me-4-OCF₃ cPen 2-Me-4-F
iPr 2-CF₃-3-OCF₃ U-4d 3-CF₃-4-F cPen 2-Me-4-Cl
iPr 2-OMe-3-F U-4d 3-CF₃-4-Cl cPen 2-Me-4-Br
iPr 2-OMe-3-Cl U-4d 3-CF₃-4-Br cPen 2,4-di-Me
iPr 2-OMe-3-Br U-4d 3-CF₃-4-Me cPen 2-Me-4-CF₃
iPr 2-OMe-3-Me U-4d 3,4-di-CF₃ cPen 2-Me-4-OMe
iPr 2-OMe-3-CF₃ U-4d 3-CF₃-4-OMe cPen 2-Me-4-OCF₃
iPr 2,3-di-OMe U-4d 3-CF₃-4-OCF₃ cPen 2-CF₃-4-F
iPr 2-OMe-3-OCF₃ U-4d 3-OMe-4-F cPen 2-CF₃-4-Cl
iPr 2-OCF₃-3-F U-4d 3-OMe-4-Cl cPen 2-CF₃-4-Br
iPr 2-OCF₃-3-Cl U-4d 3-OMe-4-Br cPen 2-CF₃-4-Me
iPr 2-OCF₃-3-Br U-4d 3-OMe-4-Me cPen 2,4-di-CF₃
iPr 2-OCF₃-3-Me U-4d 3-OMe-4-CF₃ cPen 2-CF₃-4-OMe
iPr 2-OCF₃-3-CF₃ U-4d 3,4-di-OMe cPen 2-CF₃-4-OCF₃
iPr 2-OCF₃-3-OMe U-4d 3-OMe-4-OCF₃ cPen 2-OMe-4-F
iPr 2,3-di-OCF₃ U-4d 3-OCF₃-4-F cPen 2-OMe-4-Cl
iPr 2,4-di-F U-4d 3-OCF₃-4-Cl cPen 2-OMe-4-Br
iPr 2-F-4-Cl U-4d 3-OCF₃-4-Br cPen 2-OMe-4-Me
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
iPr 2-F-4-Br U-4d 3-OCF₃-4-Me cPen 2-OMe-4-CF₃
iPr 2-F-4-Me U-4d 3-OCF₃-4-CF₃ cPen 2,4-di-OMe
iPr 2-F-4-CF₃ U-4d 3-OCF₃-4-OMe cPen 2-OMe-4-OCF₃
iPr 2-F-4-OMe U-4d 3,4-di-OCF₃ cPen 2-OCF₃-4-F
iPr 2-F-4-OCF₃ U-4d 3,5-di-F cPen 2-OCF₃-4-Cl
iPr 2-Cl-4-F U-4d 3-F-5-Cl cPen 2-OCF₃-4-Br
iPr 2,4-di-Cl U-4d 3-F-5-Br cPen 2-OCF₃-4-Me
iPr 2-Cl-4-Br U-4d 3-F-5-Me cPen 2-OCF₃-4-CF₃
iPr 2-Cl-4-Me U-4d 3-F-5-CF₃ cPen 2-OCF₃-4-OMe
iPr 2-Cl-4-CF₃ U-4d 3-F-5-OMe cPen 2,4-di-OCF₃
iPr 2-Cl-4-OMe U-4d 3-F-5-OCF₃ cPen 2,5-di-F
iPr 2-Cl-4-OCF₃ U-4d 3-Cl-5-F cPen 2-F-5-Cl
iPr 2-Br-4-F U-4d 3,5-di-Cl cPen 2-F-5-Br
iPr 2-Br-4-Cl U-4d 3-Cl-5-Br cPen 2-F-5-Me
iPr 2,4-di-Br U-4d 3-Cl-5-Me cPen 2-F-5-CF₃
iPr 2-Br-4-Me U-4d 3-Cl-5-CF₃ cPen 2-F-5-OMe
iPr 2-Br-4-CF₃ U-4d 3-Cl-5-OMe cPen 2-F-5-OCF₃
iPr 2-Br-4-OMe U-4d 3-Cl-5-OCF₃ cPen 2-Cl-5-F
iPr 2-Br-4-OCF₃ U-4d 3-Br-5-F cPen 2,5-di-Cl
iPr 2-Me-4-F U-4d 3-Br-5-Cl cPen 2-Cl-5-Br
iPr 2-Me-4-Cl U-4d 3,5-di-Br cPen 2-Cl-5-Me
iPr 2-Me-4-Br U-4d 3-Br-5-Me cPen 2-Cl-5-CF₃
iPr 2,4-di-Me U-4d 3-Br-5-CF₃ cPen 2-Cl-5-OMe
iPr 2-Me-4-CF₃ U-4d 3-Br-5-OMe cPen 2-Cl-5-OCF₃
iPr 2-Me-4-OMe U-4d 3-Br-5-OCF₃ cPen 2-Br-5-F
iPr 2-Me-4-OCF₃ U-4d 3-Me-5-F cPen 2-Br-5-Cl
iPr 2-CF₃-4-F U-4d 3-Me-5-Cl cPen 2,5-di-Br
iPr 2-CF₃-4-Cl U-4d 3-Me-5-Br cPen 2-Br-5-Me
iPr 2-CF₃-4-Br U-4d 3,5-di-Me cPen 2-Br-5-CF₃
iPr 2-CF₃-4-Me U-4d 3-Me-5-CF₃ cPen 2-Br-5-OMe
iPr 2,4-di-CF₃ U-4d 3-Me-5-OMe cPen 2-Br-5-OCF₃
iPr 2-CF₃-4-OMe U-4d 3-Me-5-OCF₃ cPen 2-Me-5-F
iPr 2-CF₃-4-OCF₃ U-4d 3-CF₃-5-F cPen 2-Me-5-Cl
iPr 2-OMe-4-F U-4d 3-CF₃-5-Cl cPen 2-Me-5-Br
iPr 2-OMe-4-Cl U-4d 3-CF₃-5-Br cPen 2,5-di-Me
iPr 2-OMe-4-Br U-4d 3-CF₃-5-Me cPen 2-Me-5-CF₃
iPr 2-OMe-4-Me U-4d 3,5-di-CF₃ cPen 2-Me-5-OMe
iPr 2-OMe-4-CF₃ U-4d 3-CF₃-5-OMe cPen 2-Me-5-OCF₃
iPr 2,4-di-OMe U-4d 3-CF₃-5-OCF₃ cPen 2-CF₃-5-F
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
iPr 2-OMe-4-OCF₃ U-4d 3-OMe-5-F cPen 2-CF₃-5-Cl
iPr 2-OCF₃-4-F U-4d 3-OMe-5-Cl cPen 2-CF₃-5-Br
iPr 2-OCF₃-4-Cl U-4d 3-OMe-5-Br cPen 2-CF₃-5-Me
iPr 2-OCF₃-4-Br U-4d 3-OMe-5-Me cPen 2,5-di-CF₃
iPr 2-OCF₃-4-Me U-4d 3-OMe-5-CF₃ cPen 2-CF₃-5-OMe
iPr 2-OCF₃-4-CF₃ U-4d 3,5-di-OMe cPen 2-CF₃-5-OCF₃
iPr 2-OCF₃-4-OMe U-4d 3-OMe-5-OCF₃ cPen 2-OMe-5-F
iPr 2,4-di-OCF₃ U-4d 3-OCF₃-5-F cPen 2-OMe-5-Cl
iPr 2,5-di-F U-4d 3-OCF₃-5-Cl cPen 2-OMe-5-Br
iPr 2-F-5-Cl U-4d 3-OCF₃-5-Br cPen 2-OMe-5-Me
iPr 2-F-5-Br U-4d 3-OCF₃-5-Me cPen 2-OMe-5-CF₃
iPr 2-F-5-Me U-4d 3-OCF₃-5-CF₃ cPen 2,5-di-OMe
iPr 2-F-5-CF₃ U-4d 3-OCF₃-5-OMe cPen 2-OMe-5-OCF₃
iPr 2-F-5-OMe U-4d 3,5-di-OCF₃ cPen 2-OCF₃-5-F
iPr 2-F-5-OCF₃ U-4e 2,3-di-F cPen 2-OCF₃-5-Cl
iPr 2-Cl-5-F U-4e 2-F-3-Cl cPen 2-OCF₃-5-Br
iPr 2,5-di-Cl U-4e 2-F-3-Br cPen 2-OCF₃-5-Me
iPr 2-Cl-5-Br U-4e 2-F-3-Me cPen 2-OCF₃-5-CF₃
iPr 2-Cl-5-Me U-4e 2-F-3-CF₃ cPen 2-OCF₃-5-OMe
iPr 2-Cl-5-CF₃ U-4e 2-F-3-OMe cPen 2,5-di-OCF₃
iPr 2-Cl-5-OMe U-4e 2-F-3-OCF₃ cPen 3,4-di-F
iPr 2-Cl-5-OCF₃ U-4e 2-Cl-3-F cPen 3-F-4-Cl
iPr 2-Br-5-F U-4e 2,3-di-Cl cPen 3-F-4-Br
iPr 2-Br-5-Cl U-4e 2-Cl-3-Br cPen 3-F-4-Me
iPr 2,5-di-Br U-4e 2-Cl-3-Me cPen 3-F-4-CF₃
iPr 2-Br-5-Me U-4e 2-Cl-3-CF₃ cPen 3-F-4-OMe
iPr 2-Br-5-CF₃ U-4e 2-Cl-3-OMe cPen 3-F-4-OCF₃
iPr 2-Br-5-OMe U-4e 2-Cl-3-OCF₃ cPen 3-Cl-4-F
iPr 2-Br-5-OCF₃ U-4e 2-Br-3-F cPen 3,4-di-Cl
iPr 2-Me-5-F U-4e 2-Br-3-Cl cPen 3-Cl-4-Br
iPr 2-Me-5-Cl U-4e 2,3-di-Br cPen 3-Cl-4-Me
iPr 2-Me-5-Br U-4e 2-Br-3-Me cPen 3-Cl-4-CF₃
iPr 2,5-di-Me U-4e 2-Br-3-CF₃ cPen 3-Cl-4-OMe
iPr 2-Me-5-CF₃ U-4e 2-Br-3-OMe cPen 3-Cl-4-OCF₃
iPr 2-Me-5-OMe U-4e 2-Br-3-OCF₃ cPen 3-Br-4-F
iPr 2-Me-5-OCF₃ U-4e 2-Me-3-F cPen 3-Br-4-Cl
iPr 2-CF₃-5-F U-4e 2-Me-3-Cl cPen 3,4-di-Br
iPr 2-CF₃-5-Cl U-4e 2-Me-3-Br cPen 3-Br-4-Me
iPr 2-CF₃-5-Br U-4e 2,3-di-Me cPen 3-Br-4-CF₃
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
iPr 2-CF₃-5-Me U-4e 2-Me-3-CF₃ cPen 3-Br-4-OMe
iPr 2,5-di-CF₃ U-4e 2-Me-3-OMe cPen 3-Br-4-OCF₃
iPr 2-CF₃-5-OMe U-4e 2-Me-3-OCF₃ cPen 3-Me-4-F
iPr 2-CF₃-5-OCF₃ U-4e 2-CF₃-3-F cPen 3-Me-4-Cl
iPr 2-OMe-5-F U-4e 2-CF₃-3-Cl cPen 3-Me-4-Br
iPr 2-OMe-5-Cl U-4e 2-CF₃-3-Br cPen 3,4-di-Me
iPr 2-OMe-5-Br U-4e 2-CF₃-3-Me cPen 3-Me-4-CF₃
iPr 2-OMe-5-Me U-4e 2,3-di-CF₃ cPen 3-Me-4-OMe
iPr 2-OMe-5-CF₃ U-4e 2-CF₃-3-OMe cPen 3-Me-4-OCF₃
iPr 2,5-di-OMe U-4e 2-CF₃-3-OCF₃ cPen 3-CF₃-4-F
iPr 2-OMe-5-OCF₃ U-4e 2-OMe-3-F cPen 3-CF₃-4-Cl
iPr 2-OCF₃-5-F U-4e 2-OMe-3-Cl cPen 3-CF₃-4-Br
iPr 2-OCF₃-5-Cl U-4e 2-OMe-3-Br cPen 3-CF₃-4-Me
iPr 2-OCF₃-5-Br U-4e 2-OMe-3-Me cPen 3,4-di-CF₃
iPr 2-OCF₃-5-Me U-4e 2-OMe-3-CF₃ cPen 3-CF₃-4-OMe
iPr 2-OCF₃-5-CF₃ U-4e 2,3-di-OMe cPen 3-CF₃-4-OCF₃
iPr 2-OCF₃-5-OMe U-4e 2-OMe-3-OCF₃ cPen 3-OMe-4-F
iPr 2,5-di-OCF₃ U-4e 2-OCF₃-3-F cPen 3-OMe-4-Cl
iPr 3,4-di-F U-4e 2-OCF₃-3-Cl cPen 3-OMe-4-Br
iPr 3-F-4-Cl U-4e 2-OCF₃-3-Br cPen 3-OMe-4-Me
iPr 3-F-4-Br U-4e 2-OCF₃-3-Me cPen 3-OMe-4-CF₃
iPr 3-F-4-Me U-4e 2-OCF₃-3-CF₃ cPen 3,4-di-OMe
iPr 3-F-4-CF₃ U-4e 2-OCF₃-3-OMe cPen 3-OMe-4-OCF₃
iPr 3-F-4-OMe U-4e 2,3-di-OCF₃ cPen 3-OCF₃-4-F
iPr 3-F-4-OCF₃ U-4e 2,4-di-F cPen 3-OCF₃-4-Cl
iPr 3-Cl-4-F U-4e 2-F-4-Cl cPen 3-OCF₃-4-Br
iPr 3,4-di-Cl U-4e 2-F-4-Br cPen 3-OCF₃-4-Me
iPr 3-Cl-4-Br U-4e 2-F-4-Me cPen 3-OCF₃-4-CF₃
iPr 3-Cl-4-Me U-4e 2-F-4-CF₃ cPen 3-OCF₃-4-OMe
iPr 3-Cl-4-CF₃ U-4e 2-F-4-OMe cPen 3,4-di-OCF₃
iPr 3-Cl-4-OMe U-4e 2-F-4-OCF₃ cPen 3,5-di-F
iPr 3-Cl-4-OCF₃ U-4e 2-Cl-4-F cPen 3-F-5-Cl
iPr 3-Br-4-F U-4e 2,4-di-Cl cPen 3-F-5-Br
iPr 3-Br-4-Cl U-4e 2-Cl-4-Br cPen 3-F-5-Me
iPr 3,4-di-Br U-4e 2-Cl-4-Me cPen 3-F-5-CF₃
iPr 3-Br-4-Me U-4e 2-Cl-4-CF₃ cPen 3-F-5-OMe
iPr 3-Br-4-CF₃ U-4e 2-Cl-4-OMe cPen 3-F-5-OCF₃
iPr 3-Br-4-OMe U-4e 2-Cl-4-OCF₃ cPen 3-Cl-5-F
iPr 3-Br-4-OCF₃ U-4e 2-Br-4-F cPen 3,5-di-Cl
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
iPr 3-Me-4-F U-4e 2-Br-4-Cl cPen 3-Cl-5-Br
iPr 3-Me-4-Cl U-4e 2,4-di-Br cPen 3-Cl-5-Me
iPr 3-Me-4-Br U-4e 2-Br-4-Me cPen 3-Cl-5-CF₃
iPr 3,4-di-Me U-4e 2-Br-4-CF₃ cPen 3-Cl-5-OMe
iPr 3-Me-4-CF₃ U-4e 2-Br-4-OMe cPen 3-Cl-5-OCF₃
iPr 3-Me-4-OMe U-4e 2-Br-4-OCF₃ cPen 3-Br-5-F
iPr 3-Me-4-OCF₃ U-4e 2-Me-4-F cPen 3-Br-5-Cl
iPr 3-CF₃-4-F U-4e 2-Me-4-Cl cPen 3,5-di-Br
iPr 3-CF₃-4-Cl U-4e 2-Me-4-Br cPen 3-Br-5-Me
iPr 3-CF₃-4-Br U-4e 2,4-di-Me cPen 3-Br-5-CF₃
iPr 3-CF₃-4-Me U-4e 2-Me-4-CF₃ cPen 3-Br-5-OMe
iPr 3,4-di-CF₃ U-4e 2-Me-4-OMe cPen 3-Br-5-OCF₃
iPr 3-CF₃-4-OMe U-4e 2-Me-4-OCF₃ cPen 3-Me-5-F
iPr 3-CF₃-4-OCF₃ U-4e 2-CF₃-4-F cPen 3-Me-5-Cl
iPr 3-OMe-4-F U-4e 2-CF₃-4-Cl cPen 3-Me-5-Br
iPr 3-OMe-4-Cl U-4e 2-CF₃-4-Br cPen 3,5-di-Me
iPr 3-OMe-4-Br U-4e 2-CF₃-4-Me cPen 3-Me-5-CF₃
iPr 3-OMe-4-Me U-4e 2,4-di-CF₃ cPen 3-Me-5-OMe
iPr 3-OMe-4-CF₃ U-4e 2-CF₃-4-OMe cPen 3-Me-5-OCF₃
iPr 3,4-di-OMe U-4e 2-CF₃-4-OCF₃ cPen 3-CF₃-5-F
iPr 3-OMe-4-OCF₃ U-4e 2-OMe-4-F cPen 3-CF₃-5-Cl
iPr 3-OCF₃-4-F U-4e 2-OMe-4-Cl cPen 3-CF₃-5-Br
iPr 3-OCF₃-4-Cl U-4e 2-OMe-4-Br cPen 3-CF₃-5-Me
iPr 3-OCF₃-4-Br U-4e 2-OMe-4-Me cPen 3,5-di-CF₃
iPr 3-OCF₃-4-Me U-4e 2-OMe-4-CF₃ cPen 3-CF₃-5-OMe
iPr 3-OCF₃-4-CF₃ U-4e 2,4-di-OMe cPen 3-CF₃-5-OCF₃
iPr 3-OCF₃-4-OMe U-4e 2-OMe-4-OCF₃ cPen 3-OMe-5-F
iPr 3,4-di-OCF₃ U-4e 2-OCF₃-4-F cPen 3-OMe-5-Cl
iPr 3,5-di-F U-4e 2-OCF₃-4-Cl cPen 3-OMe-5-Br
iPr 3-F-5-Cl U-4e 2-OCF₃-4-Br cPen 3-OMe-5-Me
iPr 3-F-5-Br U-4e 2-OCF₃-4-Me cPen 3-OMe-5-CF₃
iPr 3-F-5-Me U-4e 2-OCF₃-4-CF₃ cPen 3,5-di-OMe
iPr 3-F-5-CF₃ U-4e 2-OCF₃-4-OMe cPen 3-OMe-5-OCF₃
iPr 3-F-5-OMe U-4e 2,4-di-OCF₃ cPen 3-OCF₃-5-F
iPr 3-F-5-OCF₃ U-4e 2,5-di-F cPen 3-OCF₃-5-Cl
iPr 3-Cl-5-F U-4e 2-F-5-Cl cPen 3-OCF₃-5-Br
iPr 3,5-di-Cl U-4e 2-F-5-Br cPen 3-OCF₃-5-Me
iPr 3-Cl-5-Br U-4e 2-F-5-Me cPen 3-OCF₃-5-CF₃
iPr 3-Cl-5-Me U-4e 2-F-5-CF₃ cPen 3-OCF₃-5-OMe
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
iPr 3-Cl-5-CF₃ U-4e 2-F-5-OMe cPen 3,5-di-OCF₃
iPr 3-Cl-5-OMe U-4e 2-F-5-OCF₃ U-1e 2,3-di-F
iPr 3-Cl-5-OCF₃ U-4e 2-Cl-5-F U-1e 2-F-3-Cl
iPr 3-Br-5-F U-4e 2,5-di-Cl U-1e 2-F-3-Br
iPr 3-Br-5-Cl U-4e 2-Cl-5-Br U-1e 2-F-3-Me
iPr 3,5-di-Br U-4e 2-Cl-5-Me U-1e 2-F-3-CF₃
iPr 3-Br-5-Me U-4e 2-Cl-5-CF₃ U-1e 2-F-3-OMe
iPr 3-Br-5-CF₃ U-4e 2-Cl-5-OMe U-1e 2-F-3-OCF₃
iPr 3-Br-5-OMe U-4e 2-Cl-5-OCF₃ U-1e 2-Cl-3-F
iPr 3-Br-5-OCF₃ U-4e 2-Br-5-F U-1e 2,3-di-Cl
iPr 3-Me-5-F U-4e 2-Br-5-Cl U-1e 2-Cl-3-Br
iPr 3-Me-5-Cl U-4e 2,5-di-Br U-1e 2-Cl-3-Me
iPr 3-Me-5-Br U-4e 2-Br-5-Me U-1e 2-Cl-3-CF₃
iPr 3,5-di-Me U-4e 2-Br-5-CF₃ U-1e 2-Cl-3-OMe
iPr 3-Me-5-CF₃ U-4e 2-Br-5-OMe U-1e 2-Cl-3-OCF₃
iPr 3-Me-5-OMe U-4e 2-Br-5-OCF₃ U-1e 2-Br-3-F
iPr 3-Me-5-OCF₃ U-4e 2-Me-5-F U-1e 2-Br-3-Cl
iPr 3-CF₃-5-F U-4e 2-Me-5-Cl U-1e 2,3-di-Br
iPr 3-CF₃-5-Cl U-4e 2-Me-5-Br U-1e 2-Br-3-Me
iPr 3-CF₃-5-Br U-4e 2,5-di-Me U-1e 2-Br-3-CF₃
iPr 3-CF₃-5-Me U-4e 2-Me-5-CF₃ U-1e 2-Br-3-OMe
iPr 3,5-di-CF₃ U-4e 2-Me-5-OMe U-1e 2-Br-3-OCF₃
iPr 3-CF₃-5-OMe U-4e 2-Me-5-OCF₃ U-1e 2-Me-3-F
iPr 3-CF₃-5-OCF₃ U-4e 2-CF₃-5-F U-1e 2-Me-3-Cl
iPr 3-OMe-5-F U-4e 2-CF₃-5-Cl U-1e 2-Me-3-Br
iPr 3-OMe-5-Cl U-4e 2-CF₃-5-Br U-1e 2,3-di-Me
iPr 3-OMe-5-Br U-4e 2-CF₃-5-Me U-1e 2-Me-3-CF₃
iPr 3-OMe-5-Me U-4e 2,5-di-CF₃ U-1e 2-Me-3-OMe
iPr 3-OMe-5-CF₃ U-4e 2-CF₃-5-OMe U-1e 2-Me-3-OCF₃
iPr 3,5-di-OMe U-4e 2-CF₃-5-OCF₃ U-1e 2-CF₃-3-F
iPr 3-OMe-5-OCF₃ U-4e 2-OMe-5-F U-1e 2-CF₃-3-Cl
iPr 3-OCF₃-5-F U-4e 2-OMe-5-Cl U-1e 2-CF₃-3-Br
iPr 3-OCF₃-5-Cl U-4e 2-OMe-5-Br U-1e 2-CF₃-3-Me
iPr 3-OCF₃-5-Br U-4e 2-OMe-5-Me U-1e 2,3-di-CF₃
iPr 3-OCF₃-5-Me U-4e 2-OMe-5-CF₃ U-1e 2-CF₃-3-OMe
iPr 3-OCF₃-5-CF₃ U-4e 2,5-di-OMe U-1e 2-CF₃-3-OCF₃
iPr 3-OCF₃-5-OMe U-4e 2-OMe-5-OCF₃ U-1e 2-OMe-3-F
iPr 3,5-di-OCF₃ U-4e 2-OCF₃-5-F U-1e 2-OMe-3-Cl
U-4a 2,3-di-F U-4e 2-OCF₃-5-Cl U-1e 2-OMe-3-Br
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
U-4a 2-F-3-Cl U-4e 2-OCF₃-5-Br U-1e 2-OMe-3-Me
U-4a 2-F-3-Br U-4e 2-OCF₃-5-Me U-1e 2-OMe-3-CF₃
U-4a 2-F-3-Me U-4e 2-OCF₃-5-CF₃ U-1e 2,3-di-OMe
U-4a 2-F-3-CF₃ U-4e 2-OCF₃-5-OMe U-1e 2-OMe-3-OCF₃
U-4a 2-F-3-OMe U-4e 2,5-di-OCF₃ U-1e 2-OCF₃-3-F
U-4a 2-F-3-OCF₃ U-4e 3,4-di-F U-1e 2-OCF₃-3-Cl
U-4a 2-Cl-3-F U-4e 3-F-4-Cl U-1e 2-OCF₃-3-Br
U-4a 2,3-di-Cl U-4e 3-F-4-Br U-1e 2-OCF₃-3-Me
U-4a 2-Cl-3-Br U-4e 3-F-4-Me U-1e 2-OCF₃-3-CF₃
U-4a 2-Cl-3-Me U-4e 3-F-4-CF₃ U-1e 2-OCF₃-3-OMe
U-4a 2-Cl-3-CF₃ U-4e 3-F-4-OMe U-1e 2,3-di-OCF₃
U-4a 2-Cl-3-OMe U-4e 3-F-4-OCF₃ U-1e 2,4-di-F
U-4a 2-Cl-3-OCF₃ U-4e 3-Cl-4-F U-1e 2-F-4-Cl
U-4a 2-Br-3-F U-4e 3,4-di-Cl U-1e 2-F-4-Br
U-4a 2-Br-3-Cl U-4e 3-Cl-4-Br U-1e 2-F-4-Me
U-4a 2,3-di-Br U-4e 3-Cl-4-Me U-1e 2-F-4-CF₃
U-4a 2-Br-3-Me U-4e 3-Cl-4-CF₃ U-1e 2-F-4-OMe
U-4a 2-Br-3-CF₃ U-4e 3-Cl-4-OMe U-1e 2-F-4-OCF₃
U-4a 2-Br-3-OMe U-4e 3-Cl-4-OCF₃ U-1e 2-Cl-4-F
U-4a 2-Br-3-OCF₃ U-4e 3-Br-4-F U-1e 2,4-di-Cl
U-4a 2-Me-3-F U-4e 3-Br-4-Cl U-1e 2-Cl-4-Br
U-4a 2-Me-3-Cl U-4e 3,4-di-Br U-1e 2-Cl-4-Me
U-4a 2-Me-3-Br U-4e 3-Br-4-Me U-1e 2-Cl-4-CF₃
U-4a 2,3-di-Me U-4e 3-Br-4-CF₃ U-1e 2-Cl-4-OMe
U-4a 2-Me-3-CF₃ U-4e 3-Br-4-OMe U-1e 2-Cl-4-OCF₃
U-4a 2-Me-3-OMe U-4e 3-Br-4-OCF₃ U-1e 2-Br-4-F
U-4a 2-Me-3-OCF₃ U-4e 3-Me-4-F U-1e 2-Br-4-Cl
U-4a 2-CF₃-3-F U-4e 3-Me-4-Cl U-1e 2,4-di-Br
U-4a 2-CF₃-3-Cl U-4e 3-Me-4-Br U-1e 2-Br-4-Me
U-4a 2-CF₃-3-Br U-4e 3,4-di-Me U-1e 2-Br-4-CF₃
U-4a 2-CF₃-3-Me U-4e 3-Me-4-CF₃ U-1e 2-Br-4-OMe
U-4a 2,3-di-CF₃ U-4e 3-Me-4-OMe U-1e 2-Br-4-OCF₃
U-4a 2-CF₃-3-OMe U-4e 3-Me-4-OCF₃ U-1e 2-Me-4-F
U-4a 2-CF₃-3-OCF₃ U-4e 3-CF₃-4-F U-1e 2-Me-4-Cl
U-4a 2-OMe-3-F U-4e 3-CF₃-4-Cl U-1e 2-Me-4-Br
U-4a 2-OMe-3-Cl U-4e 3-CF₃-4-Br U-1e 2,4-di-Me
U-4a 2-OMe-3-Br U-4e 3-CF₃-4-Me U-1e 2-Me-4-CF₃
U-4a 2-OMe-3-Me U-4e 3,4-di-CF₃ U-1e 2-Me-4-OMe
U-4a 2-OMe-3-CF₃ U-4e 3-CF₃-4-OMe U-1e 2-Me-4-OCF₃
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
U-4a 2,3-di-OMe U-4e 3-CF₃-4-OCF₃ U-1e 2-CF₃-4-F
U-4a 2-OMe-3-OCF₃ U-4e 3-OMe-4-F U-1e 2-CF₃-4-Cl
U-4a 2-OCF₃-3-F U-4e 3-OMe-4-Cl U-1e 2-CF₃-4-Br
U-4a 2-OCF₃-3-Cl U-4e 3-OMe-4-Br U-1e 2-CF₃-4-Me
U-4a 2-OCF₃-3-Br U-4e 3-OMe-4-Me U-1e 2,4-di-CF₃
U-4a 2-OCF₃-3-Me U-4e 3-OMe-4-CF₃ U-1e 2-CF₃-4-OMe
U-4a 2-OCF₃-3-CF₃ U-4e 3,4-di-OMe U-1e 2-CF₃-4-OCF₃
U-4a 2-OCF₃-3-OMe U-4e 3-OMe-4-OCF₃ U-1e 2-OMe-4-F
U-4a 2,3-di-OCF₃ U-4e 3-OCF₃-4-F U-1e 2-OMe-4-Cl
U-4a 2,4-di-F U-4e 3-OCF₃-4-Cl U-1e 2-OMe-4-Br
U-4a 2-F-4-Cl U-4e 3-OCF₃-4-Br U-1e 2-OMe-4-Me
U-4a 2-F-4-Br U-4e 3-OCF₃-4-Me U-1e 2-OMe-4-CF₃
U-4a 2-F-4-Me U-4e 3-OCF₃-4-CF₃ U-1e 2,4-di-OMe
U-4a 2-F-4-CF₃ U-4e 3-OCF₃-4-OMe U-1e 2-OMe-4-OCF₃
U-4a 2-F-4-OMe U-4e 3,4-di-OCF₃ U-1e 2-OCF₃-4-F
U-4a 2-F-4-OCF₃ U-4e 3,5-di-F U-1e 2-OCF₃-4-Cl
U-4a 2-Cl-4-F U-4e 3-F-5-Cl U-1e 2-OCF₃-4-Br
U-4a 2,4-di-Cl U-4e 3-F-5-Br U-1e 2-OCF₃-4-Me
U-4a 2-Cl-4-Br U-4e 3-F-5-Me U-1e 2-OCF₃-4-CF₃
U-4a 2-Cl-4-Me U-4e 3-F-5-CF₃ U-1e 2-OCF₃-4-OMe
U-4a 2-Cl-4-CF₃ U-4e 3-F-5-OMe U-1e 2,4-di-OCF₃
U-4a 2-Cl-4-OMe U-4e 3-F-5-OCF₃ U-1e 2,5-di-F
U-4a 2-Cl-4-OCF₃ U-4e 3-Cl-5-F U-1e 2-F-5-Cl
U-4a 2-Br-4-F U-4e 3,5-di-Cl U-1e 2-F-5-Br
U-4a 2-Br-4-Cl U-4e 3-Cl-5-Br U-1e 2-F-5-Me
U-4a 2,4-di-Br U-4e 3-Cl-5-Me U-1e 2-F-5-CF₃
U-4a 2-Br-4-Me U-4e 3-Cl-5-CF₃ U-1e 2-F-5-OMe
U-4a 2-Br-4-CF₃ U-4e 3-Cl-5-OMe U-1e 2-F-5-OCF₃
U-4a 2-Br-4-OMe U-4e 3-Cl-5-OCF₃ U-1e 2-Cl-5-F
U-4a 2-Br-4-OCF₃ U-4e 3-Br-5-F U-1e 2,5-di-Cl
U-4a 2-Me-4-F U-4e 3-Br-5-Cl U-1e 2-Cl-5-Br
U-4a 2-Me-4-Cl U-4e 3,5-di-Br U-1e 2-Cl-5-Me
U-4a 2-Me-4-Br U-4e 3-Br-5-Me U-1e 2-Cl-5-CF₃
U-4a 2,4-di-Me U-4e 3-Br-5-CF₃ U-1e 2-Cl-5-OMe
U-4a 2-Me-4-CF₃ U-4e 3-Br-5-OMe U-1e 2-Cl-5-OCF₃
U-4a 2-Me-4-OMe U-4e 3-Br-5-OCF₃ U-1e 2-Br-5-F
U-4a 2-Me-4-OCF₃ U-4e 3-Me-5-F U-1e 2-Br-5-Cl
U-4a 2-CF₃-4-F U-4e 3-Me-5-Cl U-1e 2,5-di-Br
U-4a 2-CF₃-4-Cl U-4e 3-Me-5-Br U-1e 2-Br-5-Me
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
U-4a 2-CF₃-4-Br U-4e 3,5-di-Me U-1e 2-Br-5-CF₃
U-4a 2-CF₃-4-Me U-4e 3-Me-5-CF₃ U-1e 2-Br-5-OMe
U-4a 2,4-di-CF₃ U-4e 3-Me-5-OMe U-1e 2-Br-5-OCF₃
U-4a 2-CF₃-4-OMe U-4e 3-Me-5-OCF₃ U-1e 2-Me-5-F
U-4a 2-CF₃-4-OCF₃ U-4e 3-CF₃-5-F U-1e 2-Me-5-Cl
U-4a 2-OMe-4-F U-4e 3-CF₃-5-Cl U-1e 2-Me-5-Br
U-4a 2-OMe-4-Cl U-4e 3-CF₃-5-Br U-1e 2,5-di-Me
U-4a 2-OMe-4-Br U-4e 3-CF₃-5-Me U-1e 2-Me-5-CF₃
U-4a 2-OMe-4-Me U-4e 3,5-di-CF₃ U-1e 2-Me-5-OMe
U-4a 2-OMe-4-CF₃ U-4e 3-CF₃-5-OMe U-1e 2-Me-5-OCF₃
U-4a 2,4-di-OMe U-4e 3-CF₃-5-OCF₃ U-1e 2-CF₃-5-F
U-4a 2-OMe-4-OCF₃ U-4e 3-OMe-5-F U-1e 2-CF₃-5-Cl
U-4a 2-OCF₃-4-F U-4e 3-OMe-5-Cl U-1e 2-CF₃-5-Br
U-4a 2-OCF₃-4-Cl U-4e 3-OMe-5-Br U-1e 2-CF₃-5-Me
U-4a 2-OCF₃-4-Br U-4e 3-OMe-5-Me U-1e 2,5-di-CF₃
U-4a 2-OCF₃-4-Me U-4e 3-OMe-5-CF₃ U-1e 2-CF₃-5-OMe
U-4a 2-OCF₃-4-CF₃ U-4e 3,5-di-OMe U-1e 2-CF₃-5-OCF₃
U-4a 2-OCF₃-4-OMe U-4e 3-OMe-5-OCF₃ U-1e 2-OMe-5-F
U-4a 2,4-di-OCF₃ U-4e 3-OCF₃-5-F U-1e 2-OMe-5-Cl
U-4a 2,5-di-F U-4e 3-OCF₃-5-Cl U-1e 2-OMe-5-Br
U-4a 2-F-5-Cl U-4e 3-OCF₃-5-Br U-1e 2-OMe-5-Me
U-4a 2-F-5-Br U-4e 3-OCF₃-5-Me U-1e 2-OMe-5-CF₃
U-4a 2-F-5-Me U-4e 3-OCF₃-5-CF₃ U-1e 2,5-di-OMe
U-4a 2-F-5-CF₃ U-4e 3-OCF₃-5-OMe U-1e 2-OMe-5-OCF₃
U-4a 2-F-5-OMe U-4e 3,5-di-OCF₃ U-1e 2-OCF₃-5-F
U-4a 2-F-5-OCF₃ U-4f 2,3-di-F U-1e 2-OCF₃-5-Cl
U-4a 2-Cl-5-F U-4f 2-F-3-Cl U-1e 2-OCF₃-5-Br
U-4a 2,5-di-Cl U-4f 2-F-3-Br U-1e 2-OCF₃-5-Me
U-4a 2-Cl-5-Br U-4f 2-F-3-Me U-1e 2-OCF₃-5-CF₃
U-4a 2-Cl-5-Me U-4f 2-F-3-CF₃ U-1e 2-OCF₃-5-OMe
U-4a 2-Cl-5-CF₃ U-4f 2-F-3-OMe U-1e 2,5-di-OCF₃
U-4a 2-Cl-5-OMe U-4f 2-F-3-OCF₃ U-1e 3,4-di-F
U-4a 2-Cl-5-OCF₃ U-4f 2-Cl-3-F U-1e 3-F-4-Cl
U-4a 2-Br-5-F U-4f 2,3-di-Cl U-1e 3-F-4-Br
U-4a 2-Br-5-Cl U-4f 2-Cl-3-Br U-1e 3-F-4-Me
U-4a 2,5-di-Br U-4f 2-Cl-3-Me U-1e 3-F-4-CF₃
U-4a 2-Br-5-Me U-4f 2-Cl-3-CF₃ U-1e 3-F-4-OMe
U-4a 2-Br-5-CF₃ U-4f 2-Cl-3-OMe U-1e 3-F-4-OCF₃
U-4a 2-Br-5-OMe U-4f 2-Cl-3-OCF₃ U-1e 3-Cl-4-F
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
U-4a 2-Br-5-OCF₃ U-4f 2-Br-3-F U-1e 3,4-di-Cl
U-4a 2-Me-5-F U-4f 2-Br-3-Cl U-1e 3-Cl-4-Br
U-4a 2-Me-5-Cl U-4f 2,3-di-Br U-1e 3-Cl-4-Me
U-4a 2-Me-5-Br U-4f 2-Br-3-Me U-1e 3-Cl-4-CF₃
U-4a 2,5-di-Me U-4f 2-Br-3-CF₃ U-1e 3-Cl-4-OMe
U-4a 2-Me-5-CF₃ U-4f 2-Br-3-OMe U-1e 3-Cl-4-OCF₃
U-4a 2-Me-5-OMe U-4f 2-Br-3-OCF₃ U-1e 3-Br-4-F
U-4a 2-Me-5-OCF₃ U-4f 2-Me-3-F U-1e 3-Br-4-Cl
U-4a 2-CF₃-5-F U-4f 2-Me-3-Cl U-1e 3,4-di-Br
U-4a 2-CF₃-5-Cl U-4f 2-Me-3-Br U-1e 3-Br-4-Me
U-4a 2-CF₃-5-Br U-4f 2,3-di-Me U-1e 3-Br-4-CF₃
U-4a 2-CF₃-5-Me U-4f 2-Me-3-CF₃ U-1e 3-Br-4-OMe
U-4a 2,5-di-CF₃ U-4f 2-Me-3-OMe U-1e 3-Br-4-OCF₃
U-4a 2-CF₃-5-OMe U-4f 2-Me-3-OCF₃ U-1e 3-Me-4-F
U-4a 2-CF₃-5-OCF₃ U-4f 2-CF₃-3-F U-1e 3-Me-4-Cl
U-4a 2-OMe-5-F U-4f 2-CF₃-3-Cl U-1e 3-Me-4-Br
U-4a 2-OMe-5-Cl U-4f 2-CF₃-3-Br U-1e 3,4-di-Me
U-4a 2-OMe-5-Br U-4f 2-CF₃-3-Me U-1e 3-Me-4-CF₃
U-4a 2-OMe-5-Me U-4f 2,3-di-CF₃ U-1e 3-Me-4-OMe
U-4a 2-OMe-5-CF₃ U-4f 2-CF₃-3-OMe U-1e 3-Me-4-OCF₃
U-4a 2,5-di-OMe U-4f 2-CF₃-3-OCF₃ U-1e 3-CF₃-4-F
U-4a 2-OMe-5-OCF₃ U-4f 2-OMe-3-F U-1e 3-CF₃-4-Cl
U-4a 2-OCF₃-5-F U-4f 2-OMe-3-Cl U-1e 3-CF₃-4-Br
U-4a 2-OCF₃-5-Cl U-4f 2-OMe-3-Br U-1e 3-CF₃-4-Me
U-4a 2-OCF₃-5-Br U-4f 2-OMe-3-Me U-1e 3,4-di-CF₃
U-4a 2-OCF₃-5-Me U-4f 2-OMe-3-CF₃ U-1e 3-CF₃-4-OMe
U-4a 2-OCF₃-5-CF₃ U-4f 2,3-di-OMe U-1e 3-CF₃-4-OCF₃
U-4a 2-OCF₃-5-OMe U-4f 2-OMe-3-OCF₃ U-1e 3-OMe-4-F
U-4a 2,5-di-OCF₃ U-4f 2-OCF₃-3-F U-1e 3-OMe-4-Cl
U-4a 3,4-di-F U-4f 2-OCF₃-3-Cl U-1e 3-OMe-4-Br
U-4a 3-F-4-Cl U-4f 2-OCF₃-3-Br U-1e 3-OMe-4-Me
U-4a 3-F-4-Br U-4f 2-OCF₃-3-Me U-1e 3-OMe-4-CF₃
U-4a 3-F-4-Me U-4f 2-OCF₃-3-CF₃ U-1e 3,4-di-OMe
U-4a 3-F-4-CF₃ U-4f 2-OCF₃-3-OMe U-1e 3-OMe-4-OCF₃
U-4a 3-F-4-OMe U-4f 2,3-di-OCF₃ U-1e 3-OCF₃-4-F
U-4a 3-F-4-OCF₃ U-4f 2,4-di-F U-1e 3-OCF₃-4-Cl
U-4a 3-Cl-4-F U-4f 2-F-4-Cl U-1e 3-OCF₃-4-Br
U-4a 3,4-di-Cl U-4f 2-F-4-Br U-1e 3-OCF₃-4-Me
U-4a 3-Cl-4-Br U-4f 2-F-4-Me U-1e 3-OCF₃-4-CF₃
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
U-4a 3-Cl-4-Me U-4f 2-F-4-CF₃ U-1e 3-OCF₃-4-OMe
U-4a 3-Cl-4-CF₃ U-4f 2-F-4-OMe U-1e 3,4-di-OCF₃
U-4a 3-Cl-4-OMe U-4f 2-F-4-OCF₃ U-1e 3,5-di-F
U-4a 3-Cl-4-OCF₃ U-4f 2-Cl-4-F U-1e 3-F-5-Cl
U-4a 3-Br-4-F U-4f 2,4-di-Cl U-1e 3-F-5-Br
U-4a 3-Br-4-Cl U-4f 2-Cl-4-Br U-1e 3-F-5-Me
U-4a 3,4-di-Br U-4f 2-Cl-4-Me U-1e 3-F-5-CF₃
U-4a 3-Br-4-Me U-4f 2-Cl-4-CF₃ U-1e 3-F-5-OMe
U-4a 3-Br-4-CF₃ U-4f 2-Cl-4-OMe U-1e 3-F-5-OCF₃
U-4a 3-Br-4-OMe U-4f 2-Cl-4-OCF₃ U-1e 3-Cl-5-F
U-4a 3-Br-4-OCF₃ U-4f 2-Br-4-F U-1e 3,5-di-Cl
U-4a 3-Me-4-F U-4f 2-Br-4-Cl U-1e 3-Cl-5-Br
U-4a 3-Me-4-Cl U-4f 2,4-di-Br U-1e 3-Cl-5-Me
U-4a 3-Me-4-Br U-4f 2-Br-4-Me U-1e 3-Cl-5-CF₃
U-4a 3,4-di-Me U-4f 2-Br-4-CF₃ U-1e 3-Cl-5-OMe
U-4a 3-Me-4-CF₃ U-4f 2-Br-4-OMe U-1e 3-Cl-5-OCF₃
U-4a 3-Me-4-OMe U-4f 2-Br-4-OCF₃ U-1e 3-Br-5-F
U-4a 3-Me-4-OCF₃ U-4f 2-Me-4-F U-1e 3-Br-5-Cl
U-4a 3-CF₃-4-F U-4f 2-Me-4-Cl U-1e 3,5-di-Br
U-4a 3-CF₃-4-Cl U-4f 2-Me-4-Br U-1e 3-Br-5-Me
U-4a 3-CF₃-4-Br U-4f 2,4-di-Me U-1e 3-Br-5-CF₃
U-4a 3-CF₃-4-Me U-4f 2-Me-4-CF₃ U-1e 3-Br-5-OMe
U-4a 3,4-di-CF₃ U-4f 2-Me-4-OMe U-1e 3-Br-5-OCF₃
U-4a 3-CF₃-4-OMe U-4f 2-Me-4-OCF₃ U-1e 3-Me-5-F
U-4a 3-CF₃-4-OCF₃ U-4f 2-CF₃-4-F U-1e 3-Me-5-Cl
U-4a 3-OMe-4-F U-4f 2-CF₃-4-Cl U-1e 3-Me-5-Br
U-4a 3-OMe-4-Cl U-4f 2-CF₃-4-Br U-1e 3,5-di-Me
U-4a 3-OMe-4-Br U-4f 2-CF₃-4-Me U-1e 3-Me-5-CF₃
U-4a 3-OMe-4-Me U-4f 2,4-di-CF₃ U-1e 3-Me-5-OMe
U-4a 3-OMe-4-CF₃ U-4f 2-CF₃-4-OMe U-1e 3-Me-5-OCF₃
U-4a 3,4-di-OMe U-4f 2-CF₃-4-OCF₃ U-1e 3-CF₃-5-F
U-4a 3-OMe-4-OCF₃ U-4f 2-OMe-4-F U-1e 3-CF₃-5-Cl
U-4a 3-OCF₃-4-F U-4f 2-OMe-4-Cl U-1e 3-CF₃-5-Br
U-4a 3-OCF₃-4-Cl U-4f 2-OMe-4-Br U-1e 3-CF₃-5-Me
U-4a 3-OCF₃-4-Br U-4f 2-OMe-4-Me U-1e 3,5-di-CF₃
U-4a 3-OCF₃-4-Me U-4f 2-OMe-4-CF₃ U-1e 3-CF₃-5-OMe
U-4a 3-OCF₃-4-CF₃ U-4f 2,4-di-OMe U-1e 3-CF₃-5-OCF₃
U-4a 3-OCF₃-4-OMe U-4f 2-OMe-4-OCF₃ U-1e 3-OMe-5-F
U-4a 3,4-di-OCF₃ U-4f 2-OCF₃-4-F U-1e 3-OMe-5-Cl
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）［第１表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
U-4a 3,5-di-F U-4f 2-OCF₃-4-Cl U-1e 3-OMe-5-Br
U-4a 3-F-5-Cl U-4f 2-OCF₃-4-Br U-1e 3-OMe-5-Me
U-4a 3-F-5-Br U-4f 2-OCF₃-4-Me U-1e 3-OMe-5-CF₃
U-4a 3-F-5-Me U-4f 2-OCF₃-4-CF₃ U-1e 3,5-di-OMe
U-4a 3-F-5-CF₃ U-4f 2-OCF₃-4-OMe U-1e 3-OMe-5-OCF₃
U-4a 3-F-5-OMe U-4f 2,4-di-OCF₃ U-1e 3-OCF₃-5-F
U-4a 3-F-5-OCF₃ U-4f 2,5-di-F U-1e 3-OCF₃-5-Cl
U-4a 3-Cl-5-F U-4f 2-F-5-Cl U-1e 3-OCF₃-5-Br
U-4a 3,5-di-Cl U-4f 2-F-5-Br U-1e 3-OCF₃-5-Me
U-4a 3-Cl-5-Br U-4f 2-F-5-Me U-1e 3-OCF₃-5-CF₃
U-4a 3-Cl-5-Me U-4f 2-F-5-CF₃ U-1e 3-OCF₃-5-OMe
U-4a 3-Cl-5-CF₃ U-4f 2-F-5-OMe U-1e 3,5-di-OCF₃
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Me 2-F-3-Ac cPr 3-Cl-4-Ac
Me 2-F-3-(U-3b) cPr 3-Cl-4-(U-3b)
Me 2-F-3-CF₂H cPr 3-Cl-4-CF₂H
Me 2-F-3-CN cPr 3-Cl-4-CN
Me 2-F-3-Et cPr 3-Cl-4-Et
Me 2-F-3-OCF₂H cPr 3-Cl-4-OCF₂H
Me 2-F-3-OEt cPr 3-Cl-4-OEt
Me 2-F-3-C(O)CF₃ cPr 3-Cl-4-C(O)CF₃
Me 2-Cl-3-Ac cPr 3-Br-4-Ac
Me 2-Cl-3-(U-3b) cPr 3-Br-4-(U-3b)
Me 2-Cl-3-CF₂H cPr 3-Br-4-CF₂H
Me 2-Cl-3-CN cPr 3-Br-4-CN
Me 2-Cl-3-Et cPr 3-Br-4-Et
Me 2-Cl-3-OCF₂H cPr 3-Br-4-OCF₂H
Me 2-Cl-3-OEt cPr 3-Br-4-OEt
Me 2-Cl-3-C(O)CF₃ cPr 3-Br-4-C(O)CF₃
Me 2-Br-3-Ac cPr 3-Me-4-Ac
Me 2-Br-3-(U-3b) cPr 3-Me-4-(U-3b)
Me 2-Br-3-CF₂H cPr 3-Me-4-CF₂H
Me 2-Br-3-CN cPr 3-Me-4-CN
Me 2-Br-3-Et cPr 3-Me-4-Et
Me 2-Br-3-OCF₂H cPr 3-Me-4-OCF₂H
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Me 2-Br-3-OEt cPr 3-Me-4-OEt
Me 2-Br-3-C(O)CF₃ cPr 3-Me-4-C(O)CF₃
Me 2-Me-3-Ac cPr 3-CF₃-4-Ac
Me 2-Me-3-(U-3b) cPr 3-CF₃-4-(U-3b)
Me 2-Me-3-CF₂H cPr 3-CF₃-4-CF₂H
Me 2-Me-3-CN cPr 3-CF₃-4-CN
Me 2-Me-3-Et cPr 3-CF₃-4-Et
Me 2-Me-3-OCF₂H cPr 3-CF₃-4-OCF₂H
Me 2-Me-3-OEt cPr 3-CF₃-4-OEt
Me 2-Me-3-C(O)CF₃ cPr 3-CF₃-4-C(O)CF₃
Me 2-CF₃-3-Ac cPr 3-OMe-4-Ac
Me 2-CF₃-3-(U-3b) cPr 3-OMe-4-(U-3b)
Me 2-CF₃-3-CF₂H cPr 3-OMe-4-CF₂H
Me 2-CF₃-3-CN cPr 3-OMe-4-CN
Me 2-CF₃-3-Et cPr 3-OMe-4-Et
Me 2-CF₃-3-OCF₂H cPr 3-OMe-4-OCF₂H
Me 2-CF₃-3-OEt cPr 3-OMe-4-OEt
Me 2-CF₃-3-C(O)CF₃ cPr 3-OMe-4-C(O)CF₃
Me 2-OMe-3-Ac cPr 3-OCF₃-4-Ac
Me 2-OMe-3-(U-3b) cPr 3-OCF₃-4-(U-3b)
Me 2-OMe-3-CF₂H cPr 3-OCF₃-4-CF₂H
Me 2-OMe-3-CN cPr 3-OCF₃-4-CN
Me 2-OMe-3-Et cPr 3-OCF₃-4-Et
Me 2-OMe-3-OCF₂H cPr 3-OCF₃-4-OCF₂H
Me 2-OMe-3-OEt cPr 3-OCF₃-4-OEt
Me 2-OMe-3-C(O)CF₃ cPr 3-OCF₃-4-C(O)CF₃
Me 2-OCF₃-3-Ac cPr 3-F-5-Ac
Me 2-OCF₃-3-(U-3b) cPr 3-F-5-(U-3b)
Me 2-OCF₃-3-CF₂H cPr 3-F-5-CF₂H
Me 2-OCF₃-3-CN cPr 3-F-5-CN
Me 2-OCF₃-3-Et cPr 3-F-5-Et
Me 2-OCF₃-3-OCF₂H cPr 3-F-5-OCF₂H
Me 2-OCF₃-3-OEt cPr 3-F-5-OEt
Me 2-OCF₃-3-C(O)CF₃ cPr 3-F-5-C(O)CF₃
Me 2-F-4-Ac cPr 3-Cl-5-Ac
Me 2-F-4-(U-3b) cPr 3-Cl-5-(U-3b)
Me 2-F-4-CF₂H cPr 3-Cl-5-CF₂H
Me 2-F-4-CN cPr 3-Cl-5-CN
Me 2-F-4-Et cPr 3-Cl-5-Et
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Me 2-F-4-OCF₂H cPr 3-Cl-5-OCF₂H
Me 2-F-4-OEt cPr 3-Cl-5-OEt
Me 2-F-4-C(O)CF₃ cPr 3-Cl-5-C(O)CF₃
Me 2-Cl-4-Ac cPr 3-Br-5-Ac
Me 2-Cl-4-(U-3b) cPr 3-Br-5-(U-3b)
Me 2-Cl-4-CF₂H cPr 3-Br-5-CF₂H
Me 2-Cl-4-CN cPr 3-Br-5-CN
Me 2-Cl-4-Et cPr 3-Br-5-Et
Me 2-Cl-4-OCF₂H cPr 3-Br-5-OCF₂H
Me 2-Cl-4-OEt cPr 3-Br-5-OEt
Me 2-Cl-4-C(O)CF₃ cPr 3-Br-5-C(O)CF₃
Me 2-Br-4-Ac cPr 3-Me-5-Ac
Me 2-Br-4-(U-3b) cPr 3-Me-5-(U-3b)
Me 2-Br-4-CF₂H cPr 3-Me-5-CF₂H
Me 2-Br-4-CN cPr 3-Me-5-CN
Me 2-Br-4-Et cPr 3-Me-5-Et
Me 2-Br-4-OCF₂H cPr 3-Me-5-OCF₂H
Me 2-Br-4-OEt cPr 3-Me-5-OEt
Me 2-Br-4-C(O)CF₃ cPr 3-Me-5-C(O)CF₃
Me 2-Me-4-Ac cPr 3-CF₃-5-Ac
Me 2-Me-4-(U-3b) cPr 3-CF₃-5-(U-3b)
Me 2-Me-4-CF₂H cPr 3-CF₃-5-CF₂H
Me 2-Me-4-CN cPr 3-CF₃-5-CN
Me 2-Me-4-Et cPr 3-CF₃-5-Et
Me 2-Me-4-OCF₂H cPr 3-CF₃-5-OCF₂H
Me 2-Me-4-OEt cPr 3-CF₃-5-OEt
Me 2-Me-4-C(O)CF₃ cPr 3-CF₃-5-C(O)CF₃
Me 2-CF₃-4-Ac cPr 3-OMe-5-Ac
Me 2-CF₃-4-(U-3b) cPr 3-OMe-5-(U-3b)
Me 2-CF₃-4-CF₂H cPr 3-OMe-5-CF₂H
Me 2-CF₃-4-CN cPr 3-OMe-5-CN
Me 2-CF₃-4-Et cPr 3-OMe-5-Et
Me 2-CF₃-4-OCF₂H cPr 3-OMe-5-OCF₂H
Me 2-CF₃-4-OEt cPr 3-OMe-5-OEt
Me 2-CF₃-4-C(O)CF₃ cPr 3-OMe-5-C(O)CF₃
Me 2-OMe-4-Ac cPr 3-OCF₃-5-Ac
Me 2-OMe-4-(U-3b) cPr 3-OCF₃-5-(U-3b)
Me 2-OMe-4-CF₂H cPr 3-OCF₃-5-CF₂H
Me 2-OMe-4-CN cPr 3-OCF₃-5-CN
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Me 2-OMe-4-Et cPr 3-OCF₃-5-Et
Me 2-OMe-4-OCF₂H cPr 3-OCF₃-5-OCF₂H
Me 2-OMe-4-OEt cPr 3-OCF₃-5-OEt
Me 2-OMe-4-C(O)CF₃ cPr 3-OCF₃-5-C(O)CF₃
Me 2-OCF₃-4-Ac cPr 2-Ac-3-F
Me 2-OCF₃-4-(U-3b) cPr 2-Ac-3-Cl
Me 2-OCF₃-4-CF₂H cPr 2-Ac-3-Br
Me 2-OCF₃-4-CN cPr 2-Ac-3-Me
Me 2-OCF₃-4-Et cPr 2-Ac-3-CF₃
Me 2-OCF₃-4-OCF₂H cPr 2-Ac-3-OMe
Me 2-OCF₃-4-OEt cPr 2-Ac-3-OCF₃
Me 2-OCF₃-4-C(O)CF₃ cPr 2-(U-3b)-3-F
Me 2-F-5-Ac cPr 2-(U-3b)-3-Cl
Me 2-F-5-(U-3b) cPr 2-(U-3b)-3-Br
Me 2-F-5-CF₂H cPr 2-(U-3b)-3-Me
Me 2-F-5-CN cPr 2-(U-3b)-3-CF₃
Me 2-F-5-Et cPr 2-(U-3b)-3-OMe
Me 2-F-5-OCF₂H cPr 2-(U-3b)-3-OCF₃
Me 2-F-5-OEt cPr 2-CF₂H-3-F
Me 2-F-5-C(O)CF₃ cPr 2-CF₂H-3-Cl
Me 2-Cl-5-Ac cPr 2-CF₂H-3-Br
Me 2-Cl-5-(U-3b) cPr 2-CF₂H-3-Me
Me 2-Cl-5-CF₂H cPr 2-CF₂H-3-CF₃
Me 2-Cl-5-CN cPr 2-CF₂H-3-OMe
Me 2-Cl-5-Et cPr 2-CF₂H-3-OCF₃
Me 2-Cl-5-OCF₂H cPr 2-CN-3-F
Me 2-Cl-5-OEt cPr 2-CN-3-Cl
Me 2-Cl-5-C(O)CF₃ cPr 2-CN-3-Br
Me 2-Br-5-Ac cPr 2-CN-3-Me
Me 2-Br-5-(U-3b) cPr 2-CN-3-CF₃
Me 2-Br-5-CF₂H cPr 2-CN-3-OMe
Me 2-Br-5-CN cPr 2-CN-3-OCF₃
Me 2-Br-5-Et cPr 2-Et-3-F
Me 2-Br-5-OCF₂H cPr 2-Et-3-Cl
Me 2-Br-5-OEt cPr 2-Et-3-Br
Me 2-Br-5-C(O)CF₃ cPr 2-Et-3-Me
Me 2-Me-5-Ac cPr 2-Et-3-CF₃
Me 2-Me-5-(U-3b) cPr 2-Et-3-OMe
Me 2-Me-5-CF₂H cPr 2-Et-3-OCF₃
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Me 2-Me-5-CN cPr 2-OCF₂H-3-F
Me 2-Me-5-Et cPr 2-OCF₂H-3-Cl
Me 2-Me-5-OCF₂H cPr 2-OCF₂H-3-Br
Me 2-Me-5-OEt cPr 2-OCF₂H-3-Me
Me 2-Me-5-C(O)CF₃ cPr 2-OCF₂H-3-CF₃
Me 2-CF₃-5-Ac cPr 2-OCF₂H-3-OMe
Me 2-CF₃-5-(U-3b) cPr 2-OCF₂H-3-OCF₃
Me 2-CF₃-5-CF₂H cPr 2-OEt-3-F
Me 2-CF₃-5-CN cPr 2-OEt-3-Cl
Me 2-CF₃-5-Et cPr 2-OEt-3-Br
Me 2-CF₃-5-OCF₂H cPr 2-OEt-3-Me
Me 2-CF₃-5-OEt cPr 2-OEt-3-CF₃
Me 2-CF₃-5-C(O)CF₃ cPr 2-OEt-3-OMe
Me 2-OMe-5-Ac cPr 2-OEt-3-OCF₃
Me 2-OMe-5-(U-3b) cPr 2-C(O)CF₃-3-F
Me 2-OMe-5-CF₂H cPr 2-C(O)CF₃-3-Cl
Me 2-OMe-5-CN cPr 2-C(O)CF₃-3-Br
Me 2-OMe-5-Et cPr 2-C(O)CF₃-3-Me
Me 2-OMe-5-OCF₂H cPr 2-C(O)CF₃-3-CF₃
Me 2-OMe-5-OEt cPr 2-C(O)CF₃-3-OMe
Me 2-OMe-5-C(O)CF₃ cPr 2-C(O)CF₃-3-OCF₃
Me 2-OCF₃-5-Ac cPr 2-Ac-4-F
Me 2-OCF₃-5-(U-3b) cPr 2-Ac-4-Cl
Me 2-OCF₃-5-CF₂H cPr 2-Ac-4-Br
Me 2-OCF₃-5-CN cPr 2-Ac-4-Me
Me 2-OCF₃-5-Et cPr 2-Ac-4-CF₃
Me 2-OCF₃-5-OCF₂H cPr 2-Ac-4-OMe
Me 2-OCF₃-5-OEt cPr 2-Ac-4-OCF₃
Me 2-OCF₃-5-C(O)CF₃ cPr 2-(U-3b)-4-F
Me 3-F-4-Ac cPr 2-(U-3b)-4-Cl
Me 3-F-4-(U-3b) cPr 2-(U-3b)-4-Br
Me 3-F-4-CF₂H cPr 2-(U-3b)-4-Me
Me 3-F-4-CN cPr 2-(U-3b)-4-CF₃
Me 3-F-4-Et cPr 2-(U-3b)-4-OMe
Me 3-F-4-OCF₂H cPr 2-(U-3b)-4-OCF₃
Me 3-F-4-OEt cPr 2-CF₂H-4-F
Me 3-F-4-C(O)CF₃ cPr 2-CF₂H-4-Cl
Me 3-Cl-4-Ac cPr 2-CF₂H-4-Br
Me 3-Cl-4-(U-3b) cPr 2-CF₂H-4-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Me 3-Cl-4-CF₂H cPr 2-CF₂H-4-CF₃
Me 3-Cl-4-CN cPr 2-CF₂H-4-OMe
Me 3-Cl-4-Et cPr 2-CF₂H-4-OCF₃
Me 3-Cl-4-OCF₂H cPr 2-CN-4-F
Me 3-Cl-4-OEt cPr 2-CN-4-Cl
Me 3-Cl-4-C(O)CF₃ cPr 2-CN-4-Br
Me 3-Br-4-Ac cPr 2-CN-4-Me
Me 3-Br-4-(U-3b) cPr 2-CN-4-CF₃
Me 3-Br-4-CF₂H cPr 2-CN-4-OMe
Me 3-Br-4-CN cPr 2-CN-4-OCF₃
Me 3-Br-4-Et cPr 2-Et-4-F
Me 3-Br-4-OCF₂H cPr 2-Et-4-Cl
Me 3-Br-4-OEt cPr 2-Et-4-Br
Me 3-Br-4-C(O)CF₃ cPr 2-Et-4-Me
Me 3-Me-4-Ac cPr 2-Et-4-CF₃
Me 3-Me-4-(U-3b) cPr 2-Et-4-OMe
Me 3-Me-4-CF₂H cPr 2-Et-4-OCF₃
Me 3-Me-4-CN cPr 2-OCF₂H-4-F
Me 3-Me-4-Et cPr 2-OCF₂H-4-Cl
Me 3-Me-4-OCF₂H cPr 2-OCF₂H-4-Br
Me 3-Me-4-OEt cPr 2-OCF₂H-4-Me
Me 3-Me-4-C(O)CF₃ cPr 2-OCF₂H-4-CF₃
Me 3-CF₃-4-Ac cPr 2-OCF₂H-4-OMe
Me 3-CF₃-4-(U-3b) cPr 2-OCF₂H-4-OCF₃
Me 3-CF₃-4-CF₂H cPr 2-OEt-4-F
Me 3-CF₃-4-CN cPr 2-OEt-4-Cl
Me 3-CF₃-4-Et cPr 2-OEt-4-Br
Me 3-CF₃-4-OCF₂H cPr 2-OEt-4-Me
Me 3-CF₃-4-OEt cPr 2-OEt-4-CF₃
Me 3-CF₃-4-C(O)CF₃ cPr 2-OEt-4-OMe
Me 3-OMe-4-Ac cPr 2-OEt-4-OCF₃
Me 3-OMe-4-(U-3b) cPr 2-C(O)CF₃-4-F
Me 3-OMe-4-CF₂H cPr 2-C(O)CF₃-4-Cl
Me 3-OMe-4-CN cPr 2-C(O)CF₃-4-Br
Me 3-OMe-4-Et cPr 2-C(O)CF₃-4-Me
Me 3-OMe-4-OCF₂H cPr 2-C(O)CF₃-4-CF₃
Me 3-OMe-4-OEt cPr 2-C(O)CF₃-4-OMe
Me 3-OMe-4-C(O)CF₃ cPr 2-C(O)CF₃-4-OCF₃
Me 3-OCF₃-4-Ac cPr 2-Ac-5-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Me 3-OCF₃-4-(U-3b) cPr 2-Ac-5-Cl
Me 3-OCF₃-4-CF₂H cPr 2-Ac-5-Br
Me 3-OCF₃-4-CN cPr 2-Ac-5-Me
Me 3-OCF₃-4-Et cPr 2-Ac-5-CF₃
Me 3-OCF₃-4-OCF₂H cPr 2-Ac-5-OMe
Me 3-OCF₃-4-OEt cPr 2-Ac-5-OCF₃
Me 3-OCF₃-4-C(O)CF₃ cPr 2-(U-3b)-5-F
Me 3-F-5-Ac cPr 2-(U-3b)-5-Cl
Me 3-F-5-(U-3b) cPr 2-(U-3b)-5-Br
Me 3-F-5-CF₂H cPr 2-(U-3b)-5-Me
Me 3-F-5-CN cPr 2-(U-3b)-5-CF₃
Me 3-F-5-Et cPr 2-(U-3b)-5-OMe
Me 3-F-5-OCF₂H cPr 2-(U-3b)-5-OCF₃
Me 3-F-5-OEt cPr 2-CF₂H-5-F
Me 3-F-5-C(O)CF₃ cPr 2-CF₂H-5-Cl
Me 3-Cl-5-Ac cPr 2-CF₂H-5-Br
Me 3-Cl-5-(U-3b) cPr 2-CF₂H-5-Me
Me 3-Cl-5-CF₂H cPr 2-CF₂H-5-CF₃
Me 3-Cl-5-CN cPr 2-CF₂H-5-OMe
Me 3-Cl-5-Et cPr 2-CF₂H-5-OCF₃
Me 3-Cl-5-OCF₂H cPr 2-CN-5-F
Me 3-Cl-5-OEt cPr 2-CN-5-Cl
Me 3-Cl-5-C(O)CF₃ cPr 2-CN-5-Br
Me 3-Br-5-Ac cPr 2-CN-5-Me
Me 3-Br-5-(U-3b) cPr 2-CN-5-CF₃
Me 3-Br-5-CF₂H cPr 2-CN-5-OMe
Me 3-Br-5-CN cPr 2-CN-5-OCF₃
Me 3-Br-5-Et cPr 2-Et-5-F
Me 3-Br-5-OCF₂H cPr 2-Et-5-Cl
Me 3-Br-5-OEt cPr 2-Et-5-Br
Me 3-Br-5-C(O)CF₃ cPr 2-Et-5-Me
Me 3-Me-5-Ac cPr 2-Et-5-CF₃
Me 3-Me-5-(U-3b) cPr 2-Et-5-OMe
Me 3-Me-5-CF₂H cPr 2-Et-5-OCF₃
Me 3-Me-5-CN cPr 2-OCF₂H-5-F
Me 3-Me-5-Et cPr 2-OCF₂H-5-Cl
Me 3-Me-5-OCF₂H cPr 2-OCF₂H-5-Br
Me 3-Me-5-OEt cPr 2-OCF₂H-5-Me
Me 3-Me-5-C(O)CF₃ cPr 2-OCF₂H-5-CF₃
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Me 3-CF₃-5-Ac cPr 2-OCF₂H-5-OMe
Me 3-CF₃-5-(U-3b) cPr 2-OCF₂H-5-OCF₃
Me 3-CF₃-5-CF₂H cPr 2-OEt-5-F
Me 3-CF₃-5-CN cPr 2-OEt-5-Cl
Me 3-CF₃-5-Et cPr 2-OEt-5-Br
Me 3-CF₃-5-OCF₂H cPr 2-OEt-5-Me
Me 3-CF₃-5-OEt cPr 2-OEt-5-CF₃
Me 3-CF₃-5-C(O)CF₃ cPr 2-OEt-5-OMe
Me 3-OMe-5-Ac cPr 2-OEt-5-OCF₃
Me 3-OMe-5-(U-3b) cPr 2-C(O)CF₃-5-F
Me 3-OMe-5-CF₂H cPr 2-C(O)CF₃-5-Cl
Me 3-OMe-5-CN cPr 2-C(O)CF₃-5-Br
Me 3-OMe-5-Et cPr 2-C(O)CF₃-5-Me
Me 3-OMe-5-OCF₂H cPr 2-C(O)CF₃-5-CF₃
Me 3-OMe-5-OEt cPr 2-C(O)CF₃-5-OMe
Me 3-OMe-5-C(O)CF₃ cPr 2-C(O)CF₃-5-OCF₃
Me 3-OCF₃-5-Ac cPr 3-Ac-4-F
Me 3-OCF₃-5-(U-3b) cPr 3-Ac-4-Cl
Me 3-OCF₃-5-CF₂H cPr 3-Ac-4-Br
Me 3-OCF₃-5-CN cPr 3-Ac-4-Me
Me 3-OCF₃-5-Et cPr 3-Ac-4-CF₃
Me 3-OCF₃-5-OCF₂H cPr 3-Ac-4-OMe
Me 3-OCF₃-5-OEt cPr 3-Ac-4-OCF₃
Me 3-OCF₃-5-C(O)CF₃ cPr 3-(U-3b)-4-F
Me 2-Ac-3-F cPr 3-(U-3b)-4-Cl
Me 2-Ac-3-Cl cPr 3-(U-3b)-4-Br
Me 2-Ac-3-Br cPr 3-(U-3b)-4-Me
Me 2-Ac-3-Me cPr 3-(U-3b)-4-CF₃
Me 2-Ac-3-CF₃ cPr 3-(U-3b)-4-OMe
Me 2-Ac-3-OMe cPr 3-(U-3b)-4-OCF₃
Me 2-Ac-3-OCF₃ cPr 3-CF₂H-4-F
Me 2-(U-3b)-3-F cPr 3-CF₂H-4-Cl
Me 2-(U-3b)-3-Cl cPr 3-CF₂H-4-Br
Me 2-(U-3b)-3-Br cPr 3-CF₂H-4-Me
Me 2-(U-3b)-3-Me cPr 3-CF₂H-4-CF₃
Me 2-(U-3b)-3-CF₃ cPr 3-CF₂H-4-OMe
Me 2-(U-3b)-3-OMe cPr 3-CF₂H-4-OCF₃
Me 2-(U-3b)-3-OCF₃ cPr 3-CN-4-F
Me 2-CF₂H-3-F cPr 3-CN-4-Cl
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Me 2-CF₂H-3-Cl cPr 3-CN-4-Br
Me 2-CF₂H-3-Br cPr 3-CN-4-Me
Me 2-CF₂H-3-Me cPr 3-CN-4-CF₃
Me 2-CF₂H-3-CF₃ cPr 3-CN-4-OMe
Me 2-CF₂H-3-OMe cPr 3-CN-4-OCF₃
Me 2-CF₂H-3-OCF₃ cPr 3-Et-4-F
Me 2-CN-3-F cPr 3-Et-4-Cl
Me 2-CN-3-Cl cPr 3-Et-4-Br
Me 2-CN-3-Br cPr 3-Et-4-Me
Me 2-CN-3-Me cPr 3-Et-4-CF₃
Me 2-CN-3-CF₃ cPr 3-Et-4-OMe
Me 2-CN-3-OMe cPr 3-Et-4-OCF₃
Me 2-CN-3-OCF₃ cPr 3-OCF₂H-4-F
Me 2-Et-3-F cPr 3-OCF₂H-4-Cl
Me 2-Et-3-Cl cPr 3-OCF₂H-4-Br
Me 2-Et-3-Br cPr 3-OCF₂H-4-Me
Me 2-Et-3-Me cPr 3-OCF₂H-4-CF₃
Me 2-Et-3-CF₃ cPr 3-OCF₂H-4-OMe
Me 2-Et-3-OMe cPr 3-OCF₂H-4-OCF₃
Me 2-Et-3-OCF₃ cPr 3-OEt-4-F
Me 2-OCF₂H-3-F cPr 3-OEt-4-Cl
Me 2-OCF₂H-3-Cl cPr 3-OEt-4-Br
Me 2-OCF₂H-3-Br cPr 3-OEt-4-Me
Me 2-OCF₂H-3-Me cPr 3-OEt-4-CF₃
Me 2-OCF₂H-3-CF₃ cPr 3-OEt-4-OMe
Me 2-OCF₂H-3-OMe cPr 3-OEt-4-OCF₃
Me 2-OCF₂H-3-OCF₃ cPr 3-C(O)CF₃-4-F
Me 2-OEt-3-F cPr 3-C(O)CF₃-4-Cl
Me 2-OEt-3-Cl cPr 3-C(O)CF₃-4-Br
Me 2-OEt-3-Br cPr 3-C(O)CF₃-4-Me
Me 2-OEt-3-Me cPr 3-C(O)CF₃-4-CF₃
Me 2-OEt-3-CF₃ cPr 3-C(O)CF₃-4-OMe
Me 2-OEt-3-OMe cPr 3-C(O)CF₃-4-OCF₃
Me 2-OEt-3-OCF₃ cPr 3-Ac-5-F
Me 2-C(O)CF₃-3-F cPr 3-Ac-5-Cl
Me 2-C(O)CF₃-3-Cl cPr 3-Ac-5-Br
Me 2-C(O)CF₃-3-Br cPr 3-Ac-5-Me
Me 2-C(O)CF₃-3-Me cPr 3-Ac-5-CF₃
Me 2-C(O)CF₃-3-CF₃ cPr 3-Ac-5-OMe
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Me 2-C(O)CF₃-3-OMe cPr 3-Ac-5-OCF₃
Me 2-C(O)CF₃-3-OCF₃ cPr 3-(U-3b)-5-F
Me 2-Ac-4-F cPr 3-(U-3b)-5-Cl
Me 2-Ac-4-Cl cPr 3-(U-3b)-5-Br
Me 2-Ac-4-Br cPr 3-(U-3b)-5-Me
Me 2-Ac-4-Me cPr 3-(U-3b)-5-CF₃
Me 2-Ac-4-CF₃ cPr 3-(U-3b)-5-OMe
Me 2-Ac-4-OMe cPr 3-(U-3b)-5-OCF₃
Me 2-Ac-4-OCF₃ cPr 3-CF₂H-5-F
Me 2-(U-3b)-4-F cPr 3-CF₂H-5-Cl
Me 2-(U-3b)-4-Cl cPr 3-CF₂H-5-Br
Me 2-(U-3b)-4-Br cPr 3-CF₂H-5-Me
Me 2-(U-3b)-4-Me cPr 3-CF₂H-5-CF₃
Me 2-(U-3b)-4-CF₃ cPr 3-CF₂H-5-OMe
Me 2-(U-3b)-4-OMe cPr 3-CF₂H-5-OCF₃
Me 2-(U-3b)-4-OCF₃ cPr 3-CN-5-F
Me 2-CF₂H-4-F cPr 3-CN-5-Cl
Me 2-CF₂H-4-Cl cPr 3-CN-5-Br
Me 2-CF₂H-4-Br cPr 3-CN-5-Me
Me 2-CF₂H-4-Me cPr 3-CN-5-CF₃
Me 2-CF₂H-4-CF₃ cPr 3-CN-5-OMe
Me 2-CF₂H-4-OMe cPr 3-CN-5-OCF₃
Me 2-CF₂H-4-OCF₃ cPr 3-Et-5-F
Me 2-CN-4-F cPr 3-Et-5-Cl
Me 2-CN-4-Cl cPr 3-Et-5-Br
Me 2-CN-4-Br cPr 3-Et-5-Me
Me 2-CN-4-Me cPr 3-Et-5-CF₃
Me 2-CN-4-CF₃ cPr 3-Et-5-OMe
Me 2-CN-4-OMe cPr 3-Et-5-OCF₃
Me 2-CN-4-OCF₃ cPr 3-OCF₂H-5-F
Me 2-Et-4-F cPr 3-OCF₂H-5-Cl
Me 2-Et-4-Cl cPr 3-OCF₂H-5-Br
Me 2-Et-4-Br cPr 3-OCF₂H-5-Me
Me 2-Et-4-Me cPr 3-OCF₂H-5-CF₃
Me 2-Et-4-CF₃ cPr 3-OCF₂H-5-OMe
Me 2-Et-4-OMe cPr 3-OCF₂H-5-OCF₃
Me 2-Et-4-OCF₃ cPr 3-OEt-5-F
Me 2-OCF₂H-4-F cPr 3-OEt-5-Cl
Me 2-OCF₂H-4-Cl cPr 3-OEt-5-Br
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Me 2-OCF₂H-4-Br cPr 3-OEt-5-Me
Me 2-OCF₂H-4-Me cPr 3-OEt-5-CF₃
Me 2-OCF₂H-4-CF₃ cPr 3-OEt-5-OMe
Me 2-OCF₂H-4-OMe cPr 3-OEt-5-OCF₃
Me 2-OCF₂H-4-OCF₃ cPr 3-C(O)CF₃-5-F
Me 2-OEt-4-F cPr 3-C(O)CF₃-5-Cl
Me 2-OEt-4-Cl cPr 3-C(O)CF₃-5-Br
Me 2-OEt-4-Br cPr 3-C(O)CF₃-5-Me
Me 2-OEt-4-Me cPr 3-C(O)CF₃-5-CF₃
Me 2-OEt-4-CF₃ cPr 3-C(O)CF₃-5-OMe
Me 2-OEt-4-OMe cPr 3-C(O)CF₃-5-OCF₃
Me 2-OEt-4-OCF₃ Me 2,3,4-tri-F
Me 2-C(O)CF₃-4-F Me 2,3-di-F-4-Cl
Me 2-C(O)CF₃-4-Cl Me 2,3-di-F-4-Br
Me 2-C(O)CF₃-4-Br Me 2,3-di-F-4-Me
Me 2-C(O)CF₃-4-Me Me 2,3-di-F-4-CF₃
Me 2-C(O)CF₃-4-CF₃ Me 2,3-di-F-4-OMe
Me 2-C(O)CF₃-4-OMe Me 2,4-di-F-3-Cl
Me 2-C(O)CF₃-4-OCF₃ Me 2-F-3,4-di-Cl
Me 2-Ac-5-F Me 2-F-3-Cl-4-Br
Me 2-Ac-5-Cl Me 2-F-3-Cl-4-Me
Me 2-Ac-5-Br Me 2-F-3-Cl-4-CF₃
Me 2-Ac-5-Me Me 2-F-3-Cl-4-OMe
Me 2-Ac-5-CF₃ Me 2,4-di-F-3-Br
Me 2-Ac-5-OMe Me 2-F-3-Br-4-Cl
Me 2-Ac-5-OCF₃ Me 2-F-3,4-di-Br
Me 2-(U-3b)-5-F Me 2-F-3-Br-4-Me
Me 2-(U-3b)-5-Cl Me 2-F-3-Br-4-CF₃
Me 2-(U-3b)-5-Br Me 2-F-3-Br-4-OMe
Me 2-(U-3b)-5-Me Me 2,4-di-F-3-Me
Me 2-(U-3b)-5-CF₃ Me 2-F-3-Me-4-Cl
Me 2-(U-3b)-5-OMe Me 2-F-3-Me-4-Br
Me 2-(U-3b)-5-OCF₃ Me 2-F-3,4-di-Me
Me 2-CF₂H-5-F Me 2-F-3-Me-4-CF₃
Me 2-CF₂H-5-Cl Me 2-F-3-Me-4-OMe
Me 2-CF₂H-5-Br Me 2,4-di-F-3-CF₃
Me 2-CF₂H-5-Me Me 2-F-3-CF₃-4-Cl
Me 2-CF₂H-5-CF₃ Me 2-F-3-CF₃-4-Br
Me 2-CF₂H-5-OMe Me 2-F-3-CF₃-4-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Me 2-CF₂H-5-OCF₃ Me 2-F-3,4-di-CF₃
Me 2-CN-5-F Me 2-F-3-CF₃-4-OMe
Me 2-CN-5-Cl Me 2,4-di-F-3-OMe
Me 2-CN-5-Br Me 2-F-3-OMe-4-Cl
Me 2-CN-5-Me Me 2-F-3-OMe-4-Br
Me 2-CN-5-CF₃ Me 2-F-3-OMe-4-Me
Me 2-CN-5-OMe Me 2-F-3-OMe-4-CF₃
Me 2-CN-5-OCF₃ Me 2-F-3,4-di-OMe
Me 2-Et-5-F Me 2,3,5-tri-F
Me 2-Et-5-Cl Me 2,3-di-F-5-Cl
Me 2-Et-5-Br Me 2,3-di-F-5-Br
Me 2-Et-5-Me Me 2,3-di-F-5-Me
Me 2-Et-5-CF₃ Me 2,3-di-F-5-CF₃
Me 2-Et-5-OMe Me 2,3-di-F-5-OMe
Me 2-Et-5-OCF₃ Me 2,5-di-F-3-Cl
Me 2-OCF₂H-5-F Me 2-F-3,5-di-Cl
Me 2-OCF₂H-5-Cl Me 2-F-3-Cl-5-Br
Me 2-OCF₂H-5-Br Me 2-F-3-Cl-5-Me
Me 2-OCF₂H-5-Me Me 2-F-3-Cl-5-CF₃
Me 2-OCF₂H-5-CF₃ Me 2-F-3-Cl-5-OMe
Me 2-OCF₂H-5-OMe Me 2,5-di-F-3-Br
Me 2-OCF₂H-5-OCF₃ Me 2-F-3-Br-5-Cl
Me 2-OEt-5-F Me 2-F-3,5-di-Br
Me 2-OEt-5-Cl Me 2-F-3-Br-5-Me
Me 2-OEt-5-Br Me 2-F-3-Br-5-CF₃
Me 2-OEt-5-Me Me 2-F-3-Br-5-OMe
Me 2-OEt-5-CF₃ Me 2,5-di-F-3-Me
Me 2-OEt-5-OMe Me 2-F-3-Me-5-Cl
Me 2-OEt-5-OCF₃ Me 2-F-3-Me-5-Br
Me 2-C(O)CF₃-5-F Me 2-F-3,5-di-Me
Me 2-C(O)CF₃-5-Cl Me 2-F-3-Me-5-CF₃
Me 2-C(O)CF₃-5-Br Me 2-F-3-Me-5-OMe
Me 2-C(O)CF₃-5-Me Me 2,5-di-F-3-CF₃
Me 2-C(O)CF₃-5-CF₃ Me 2-F-3-CF₃-5-Cl
Me 2-C(O)CF₃-5-OMe Me 2-F-3-CF₃-5-Br
Me 2-C(O)CF₃-5-OCF₃ Me 2-F-3-CF₃-5-Me
Me 3-Ac-4-F Me 2-F-3,5-di-CF₃
Me 3-Ac-4-Cl Me 2-F-3-CF₃-5-OMe
Me 3-Ac-4-Br Me 2,5-di-F-3-OMe
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Me 3-Ac-4-Me Me 2-F-3-OMe-5-Cl
Me 3-Ac-4-CF₃ Me 2-F-3-OMe-5-Br
Me 3-Ac-4-OMe Me 2-F-3-OMe-5-Me
Me 3-Ac-4-OCF₃ Me 2-F-3-OMe-5-CF₃
Me 3-(U-3b)-4-F Me 2-F-3,5-di-OMe
Me 3-(U-3b)-4-Cl Me 2,4,5-tri-F
Me 3-(U-3b)-4-Br Me 2,4-di-F-5-Cl
Me 3-(U-3b)-4-Me Me 2,4-di-F-5-Br
Me 3-(U-3b)-4-CF₃ Me 2,4-di-F-5-Me
Me 3-(U-3b)-4-OMe Me 2,4-di-F-5-CF₃
Me 3-(U-3b)-4-OCF₃ Me 2,4-di-F-5-OMe
Me 3-CF₂H-4-F Me 2,5-di-F-4-Cl
Me 3-CF₂H-4-Cl Me 2-F-4,5-di-Cl
Me 3-CF₂H-4-Br Me 2-F-4-Cl-5-Br
Me 3-CF₂H-4-Me Me 2-F-4-Cl-5-Me
Me 3-CF₂H-4-CF₃ Me 2-F-4-Cl-5-CF₃
Me 3-CF₂H-4-OMe Me 2-F-4-Cl-5-OMe
Me 3-CF₂H-4-OCF₃ Me 2,5-di-F-4-Br
Me 3-CN-4-F Me 2-F-4-Br-5-Cl
Me 3-CN-4-Cl Me 2-F-4,5-di-Br
Me 3-CN-4-Br Me 2-F-4-Br-5-Me
Me 3-CN-4-Me Me 2-F-4-Br-5-CF₃
Me 3-CN-4-CF₃ Me 2-F-4-Br-5-OMe
Me 3-CN-4-OMe Me 2,5-di-F-4-Me
Me 3-CN-4-OCF₃ Me 2-F-4-Me-5-Cl
Me 3-Et-4-F Me 2-F-4-Me-5-Br
Me 3-Et-4-Cl Me 2-F-4,5-di-Me
Me 3-Et-4-Br Me 2-F-4-Me-5-CF₃
Me 3-Et-4-Me Me 2-F-4-Me-5-OMe
Me 3-Et-4-CF₃ Me 2,5-di-F-4-CF₃
Me 3-Et-4-OMe Me 2-F-4-CF₃-5-Cl
Me 3-Et-4-OCF₃ Me 2-F-4-CF₃-5-Br
Me 3-OCF₂H-4-F Me 2-F-4-CF₃-5-Me
Me 3-OCF₂H-4-Cl Me 2-F-4,5-di-CF₃
Me 3-OCF₂H-4-Br Me 2-F-4-CF₃-5-OMe
Me 3-OCF₂H-4-Me Me 2,5-di-F-4-OMe
Me 3-OCF₂H-4-CF₃ Me 2-F-4-OMe-5-Cl
Me 3-OCF₂H-4-OMe Me 2-F-4-OMe-5-Br
Me 3-OCF₂H-4-OCF₃ Me 2-F-4-OMe-5-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Me 3-OEt-4-F Me 2-F-4-OMe-5-CF₃
Me 3-OEt-4-Cl Me 2-F-4,5-di-OMe
Me 3-OEt-4-Br Me 3,4,5-tri-F
Me 3-OEt-4-Me Me 3,4-di-F-5-Cl
Me 3-OEt-4-CF₃ Me 3,4-di-F-5-Br
Me 3-OEt-4-OMe Me 3,4-di-F-5-Me
Me 3-OEt-4-OCF₃ Me 3,4-di-F-5-CF₃
Me 3-C(O)CF₃-4-F Me 3,4-di-F-5-OMe
Me 3-C(O)CF₃-4-Cl Me 3,5-di-F-4-Cl
Me 3-C(O)CF₃-4-Br Me 3-F-4,5-di-Cl
Me 3-C(O)CF₃-4-Me Me 3-F-4-Cl-5-Br
Me 3-C(O)CF₃-4-CF₃ Me 3-F-4-Cl-5-Me
Me 3-C(O)CF₃-4-OMe Me 3-F-4-Cl-5-CF₃
Me 3-C(O)CF₃-4-OCF₃ Me 3-F-4-Cl-5-OMe
Me 3-Ac-5-F Me 3,5-di-F-4-Br
Me 3-Ac-5-Cl Me 3-F-4-Br-5-Cl
Me 3-Ac-5-Br Me 3-F-4,5-di-Br
Me 3-Ac-5-Me Me 3-F-4-Br-5-Me
Me 3-Ac-5-CF₃ Me 3-F-4-Br-5-CF₃
Me 3-Ac-5-OMe Me 3-F-4-Br-5-OMe
Me 3-Ac-5-OCF₃ Me 3,5-di-F-4-Me
Me 3-(U-3b)-5-F Me 3-F-4-Me-5-Cl
Me 3-(U-3b)-5-Cl Me 3-F-4-Me-5-Br
Me 3-(U-3b)-5-Br Me 3-F-4,5-di-Me
Me 3-(U-3b)-5-Me Me 3-F-4-Me-5-CF₃
Me 3-(U-3b)-5-CF₃ Me 3-F-4-Me-5-OMe
Me 3-(U-3b)-5-OMe Me 3,5-di-F-4-CF₃
Me 3-(U-3b)-5-OCF₃ Me 3-F-4-CF₃-5-Cl
Me 3-CF₂H-5-F Me 3-F-4-CF₃-5-Br
Me 3-CF₂H-5-Cl Me 3-F-4-CF₃-5-Me
Me 3-CF₂H-5-Br Me 3-F-4,5-di-CF₃
Me 3-CF₂H-5-Me Me 3-F-4-CF₃-5-OMe
Me 3-CF₂H-5-CF₃ Me 3,5-di-F-4-OMe
Me 3-CF₂H-5-OMe Me 3-F-4-OMe-5-Cl
Me 3-CF₂H-5-OCF₃ Me 3-F-4-OMe-5-Br
Me 3-CN-5-F Me 3-F-4-OMe-5-Me
Me 3-CN-5-Cl Me 3-F-4-OMe-5-CF₃
Me 3-CN-5-Br Me 3-F-4,5-di-OMe
Me 3-CN-5-Me Me 2-Cl-3,4-di-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Me 3-CN-5-CF₃ Me 2,4-di-Cl-3-F
Me 3-CN-5-OMe Me 2-Cl-3-F-4-Br
Me 3-CN-5-OCF₃ Me 2-Cl-3-F-4-Me
Me 3-Et-5-F Me 2-Cl-3-F-4-CF₃
Me 3-Et-5-Cl Me 2-Cl-3-F-4-OMe
Me 3-Et-5-Br Me 2,3-di-Cl-4-F
Me 3-Et-5-Me Me 2,3,4-tri-Cl
Me 3-Et-5-CF₃ Me 2,3-di-Cl-4-Br
Me 3-Et-5-OMe Me 2,3-di-Cl-4-Me
Me 3-Et-5-OCF₃ Me 2,3-di-Cl-4-CF₃
Me 3-OCF₂H-5-F Me 2,3-di-Cl-4-OMe
Me 3-OCF₂H-5-Cl Me 2-Cl-3-Br-4-F
Me 3-OCF₂H-5-Br Me 2,4-di-Cl-3-Br
Me 3-OCF₂H-5-Me Me 2-Cl-3,4-di-Br
Me 3-OCF₂H-5-CF₃ Me 2-Cl-3-Br-4-Me
Me 3-OCF₂H-5-OMe Me 2-Cl-3-Br-4-CF₃
Me 3-OCF₂H-5-OCF₃ Me 2-Cl-3-Br-4-OMe
Me 3-OEt-5-F Me 2-Cl-3-Me-4-F
Me 3-OEt-5-Cl Me 2,4-di-Cl-3-Me
Me 3-OEt-5-Br Me 2-Cl-3-Me-4-Br
Me 3-OEt-5-Me Me 2-Cl-3,4-di-Me
Me 3-OEt-5-CF₃ Me 2-Cl-3-Me-4-CF₃
Me 3-OEt-5-OMe Me 2-Cl-3-Me-4-OMe
Me 3-OEt-5-OCF₃ Me 2-Cl-3-CF₃-4-F
Me 3-C(O)CF₃-5-F Me 2,4-di-Cl-3-CF₃
Me 3-C(O)CF₃-5-Cl Me 2-Cl-3-CF₃-4-Br
Me 3-C(O)CF₃-5-Br Me 2-Cl-3-CF₃-4-Me
Me 3-C(O)CF₃-5-Me Me 2-Cl-3,4-di-CF₃
Me 3-C(O)CF₃-5-CF₃ Me 2-Cl-3-CF₃-4-OMe
Me 3-C(O)CF₃-5-OMe Me 2-Cl-3-OMe-4-F
Me 3-C(O)CF₃-5-OCF₃ Me 2,4-di-Cl-3-OMe
Et 2-F-3-Ac Me 2-Cl-3-OMe-4-Br
Et 2-F-3-(U-3b) Me 2-Cl-3-OMe-4-Me
Et 2-F-3-CF₂H Me 2-Cl-3-OMe-4-CF₃
Et 2-F-3-CN Me 2-Cl-3,4-di-OMe
Et 2-F-3-Et Me 2-Cl-3,5-di-F
Et 2-F-3-OCF₂H Me 2,5-di-Cl-3-F
Et 2-F-3-OEt Me 2-Cl-3-F-5-Br
Et 2-F-3-C(O)CF₃ Me 2-Cl-3-F-5-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Et 2-Cl-3-Ac Me 2-Cl-3-F-5-CF₃
Et 2-Cl-3-(U-3b) Me 2-Cl-3-F-5-OMe
Et 2-Cl-3-CF₂H Me 2,3-di-Cl-5-F
Et 2-Cl-3-CN Me 2,3,5-tri-Cl
Et 2-Cl-3-Et Me 2,3-di-Cl-5-Br
Et 2-Cl-3-OCF₂H Me 2,3-di-Cl-5-Me
Et 2-Cl-3-OEt Me 2,3-di-Cl-5-CF₃
Et 2-Cl-3-C(O)CF₃ Me 2,3-di-Cl-5-OMe
Et 2-Br-3-Ac Me 2-Cl-3-Br-5-F
Et 2-Br-3-(U-3b) Me 2,5-di-Cl-3-Br
Et 2-Br-3-CF₂H Me 2-Cl-3,5-di-Br
Et 2-Br-3-CN Me 2-Cl-3-Br-5-Me
Et 2-Br-3-Et Me 2-Cl-3-Br-5-CF₃
Et 2-Br-3-OCF₂H Me 2-Cl-3-Br-5-OMe
Et 2-Br-3-OEt Me 2-Cl-3-Me-5-F
Et 2-Br-3-C(O)CF₃ Me 2,5-di-Cl-3-Me
Et 2-Me-3-Ac Me 2-Cl-3-Me-5-Br
Et 2-Me-3-(U-3b) Me 2-Cl-3,5-di-Me
Et 2-Me-3-CF₂H Me 2-Cl-3-Me-5-CF₃
Et 2-Me-3-CN Me 2-Cl-3-Me-5-OMe
Et 2-Me-3-Et Me 2-Cl-3-CF₃-5-F
Et 2-Me-3-OCF₂H Me 2,5-di-Cl-3-CF₃
Et 2-Me-3-OEt Me 2-Cl-3-CF₃-5-Br
Et 2-Me-3-C(O)CF₃ Me 2-Cl-3-CF₃-5-Me
Et 2-CF₃-3-Ac Me 2-Cl-3,5-di-CF₃
Et 2-CF₃-3-(U-3b) Me 2-Cl-3-CF₃-5-OMe
Et 2-CF₃-3-CF₂H Me 2-Cl-3-OMe-5-F
Et 2-CF₃-3-CN Me 2,5-di-Cl-3-OMe
Et 2-CF₃-3-Et Me 2-Cl-3-OMe-5-Br
Et 2-CF₃-3-OCF₂H Me 2-Cl-3-OMe-5-Me
Et 2-CF₃-3-OEt Me 2-Cl-3-OMe-5-CF₃
Et 2-CF₃-3-C(O)CF₃ Me 2-Cl-3,5-di-OMe
Et 2-OMe-3-Ac Me 2-Cl-4,5-di-F
Et 2-OMe-3-(U-3b) Me 2,5-di-Cl-4-F
Et 2-OMe-3-CF₂H Me 2-Cl-4-F-5-Br
Et 2-OMe-3-CN Me 2-Cl-4-F-5-Me
Et 2-OMe-3-Et Me 2-Cl-4-F-5-CF₃
Et 2-OMe-3-OCF₂H Me 2-Cl-4-F-5-OMe
Et 2-OMe-3-OEt Me 2,4-di-Cl-5-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Et 2-OMe-3-C(O)CF₃ Me 2,4,5-tri-Cl
Et 2-OCF₃-3-Ac Me 2,4-di-Cl-5-Br
Et 2-OCF₃-3-(U-3b) Me 2,4-di-Cl-5-Me
Et 2-OCF₃-3-CF₂H Me 2,4-di-Cl-5-CF₃
Et 2-OCF₃-3-CN Me 2,4-di-Cl-5-OMe
Et 2-OCF₃-3-Et Me 2-Cl-4-Br-5-F
Et 2-OCF₃-3-OCF₂H Me 2,5-di-Cl-4-Br
Et 2-OCF₃-3-OEt Me 2-Cl-4,5-di-Br
Et 2-OCF₃-3-C(O)CF₃ Me 2-Cl-4-Br-5-Me
Et 2-F-4-Ac Me 2-Cl-4-Br-5-CF₃
Et 2-F-4-(U-3b) Me 2-Cl-4-Br-5-OMe
Et 2-F-4-CF₂H Me 2-Cl-4-Me-5-F
Et 2-F-4-CN Me 2,5-di-Cl-4-Me
Et 2-F-4-Et Me 2-Cl-4-Me-5-Br
Et 2-F-4-OCF₂H Me 2-Cl-4,5-di-Me
Et 2-F-4-OEt Me 2-Cl-4-Me-5-CF₃
Et 2-F-4-C(O)CF₃ Me 2-Cl-4-Me-5-OMe
Et 2-Cl-4-Ac Me 2-Cl-4-CF₃-5-F
Et 2-Cl-4-(U-3b) Me 2,5-di-Cl-4-CF₃
Et 2-Cl-4-CF₂H Me 2-Cl-4-CF₃-5-Br
Et 2-Cl-4-CN Me 2-Cl-4-CF₃-5-Me
Et 2-Cl-4-Et Me 2-Cl-4,5-di-CF₃
Et 2-Cl-4-OCF₂H Me 2-Cl-4-CF₃-5-OMe
Et 2-Cl-4-OEt Me 2-Cl-4-OMe-5-F
Et 2-Cl-4-C(O)CF₃ Me 2,5-di-Cl-4-OMe
Et 2-Br-4-Ac Me 2-Cl-4-OMe-5-Br
Et 2-Br-4-(U-3b) Me 2-Cl-4-OMe-5-Me
Et 2-Br-4-CF₂H Me 2-Cl-4-OMe-5-CF₃
Et 2-Br-4-CN Me 2-Cl-4,5-di-OMe
Et 2-Br-4-Et Me 3-Cl-4,5-di-F
Et 2-Br-4-OCF₂H Me 3,5-di-Cl-4-F
Et 2-Br-4-OEt Me 3-Cl-4-F-5-Br
Et 2-Br-4-C(O)CF₃ Me 3-Cl-4-F-5-Me
Et 2-Me-4-Ac Me 3-Cl-4-F-5-CF₃
Et 2-Me-4-(U-3b) Me 3-Cl-4-F-5-OMe
Et 2-Me-4-CF₂H Me 3,4-di-Cl-5-F
Et 2-Me-4-CN Me 3,4,5-tri-Cl
Et 2-Me-4-Et Me 3,4-di-Cl-5-Br
Et 2-Me-4-OCF₂H Me 3,4-di-Cl-5-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Et 2-Me-4-OEt Me 3,4-di-Cl-5-CF₃
Et 2-Me-4-C(O)CF₃ Me 3,4-di-Cl-5-OMe
Et 2-CF₃-4-Ac Me 3-Cl-4-Br-5-F
Et 2-CF₃-4-(U-3b) Me 3,5-di-Cl-4-Br
Et 2-CF₃-4-CF₂H Me 3-Cl-4,5-di-Br
Et 2-CF₃-4-CN Me 3-Cl-4-Br-5-Me
Et 2-CF₃-4-Et Me 3-Cl-4-Br-5-CF₃
Et 2-CF₃-4-OCF₂H Me 3-Cl-4-Br-5-OMe
Et 2-CF₃-4-OEt Me 3-Cl-4-Me-5-F
Et 2-CF₃-4-C(O)CF₃ Me 3,5-di-Cl-4-Me
Et 2-OMe-4-Ac Me 3-Cl-4-Me-5-Br
Et 2-OMe-4-(U-3b) Me 3-Cl-4,5-di-Me
Et 2-OMe-4-CF₂H Me 3-Cl-4-Me-5-CF₃
Et 2-OMe-4-CN Me 3-Cl-4-Me-5-OMe
Et 2-OMe-4-Et Me 3-Cl-4-CF₃-5-F
Et 2-OMe-4-OCF₂H Me 3,5-di-Cl-4-CF₃
Et 2-OMe-4-OEt Me 3-Cl-4-CF₃-5-Br
Et 2-OMe-4-C(O)CF₃ Me 3-Cl-4-CF₃-5-Me
Et 2-OCF₃-4-Ac Me 3-Cl-4,5-di-CF₃
Et 2-OCF₃-4-(U-3b) Me 3-Cl-4-CF₃-5-OMe
Et 2-OCF₃-4-CF₂H Me 3-Cl-4-OMe-5-F
Et 2-OCF₃-4-CN Me 3,5-di-Cl-4-OMe
Et 2-OCF₃-4-Et Me 3-Cl-4-OMe-5-Br
Et 2-OCF₃-4-OCF₂H Me 3-Cl-4-OMe-5-Me
Et 2-OCF₃-4-OEt Me 3-Cl-4-OMe-5-CF₃
Et 2-OCF₃-4-C(O)CF₃ Me 3-Cl-4,5-di-OMe
Et 2-F-5-Ac Me 2-Br-3,4-di-F
Et 2-F-5-(U-3b) Me 2-Br-3-F-4-Cl
Et 2-F-5-CF₂H Me 2,4-di-Br-3-F
Et 2-F-5-CN Me 2-Br-3-F-4-Me
Et 2-F-5-Et Me 2-Br-3-F-4-CF₃
Et 2-F-5-OCF₂H Me 2-Br-3-F-4-OMe
Et 2-F-5-OEt Me 2-Br-3-Cl-4-F
Et 2-F-5-C(O)CF₃ Me 2-Br-3,4-di-Cl
Et 2-Cl-5-Ac Me 2,4-di-Br-3-Cl
Et 2-Cl-5-(U-3b) Me 2-Br-3-Cl-4-Me
Et 2-Cl-5-CF₂H Me 2-Br-3-Cl-4-CF₃
Et 2-Cl-5-CN Me 2-Br-3-Cl-4-OMe
Et 2-Cl-5-Et Me 2,3-di-Br-4-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Et 2-Cl-5-OCF₂H Me 2,3-di-Br-4-Cl
Et 2-Cl-5-OEt Me 2,3,4-tri-Br
Et 2-Cl-5-C(O)CF₃ Me 2,3-di-Br-4-Me
Et 2-Br-5-Ac Me 2,3-di-Br-4-CF₃
Et 2-Br-5-(U-3b) Me 2,3-di-Br-4-OMe
Et 2-Br-5-CF₂H Me 2-Br-3-Me-4-F
Et 2-Br-5-CN Me 2-Br-3-Me-4-Cl
Et 2-Br-5-Et Me 2,4-di-Br-3-Me
Et 2-Br-5-OCF₂H Me 2-Br-3,4-di-Me
Et 2-Br-5-OEt Me 2-Br-3-Me-4-CF₃
Et 2-Br-5-C(O)CF₃ Me 2-Br-3-Me-4-OMe
Et 2-Me-5-Ac Me 2-Br-3-CF₃-4-F
Et 2-Me-5-(U-3b) Me 2-Br-3-CF₃-4-Cl
Et 2-Me-5-CF₂H Me 2,4-di-Br-3-CF₃
Et 2-Me-5-CN Me 2-Br-3-CF₃-4-Me
Et 2-Me-5-Et Me 2-Br-3,4-di-CF₃
Et 2-Me-5-OCF₂H Me 2-Br-3-CF₃-4-OMe
Et 2-Me-5-OEt Me 2-Br-3-OMe-4-F
Et 2-Me-5-C(O)CF₃ Me 2-Br-3-OMe-4-Cl
Et 2-CF₃-5-Ac Me 2,4-di-Br-3-OMe
Et 2-CF₃-5-(U-3b) Me 2-Br-3-OMe-4-Me
Et 2-CF₃-5-CF₂H Me 2-Br-3-OMe-4-CF₃
Et 2-CF₃-5-CN Me 2-Br-3,4-di-OMe
Et 2-CF₃-5-Et Me 2-Br-3,5-di-F
Et 2-CF₃-5-OCF₂H Me 2-Br-3-F-5-Cl
Et 2-CF₃-5-OEt Me 2,5-di-Br-3-F
Et 2-CF₃-5-C(O)CF₃ Me 2-Br-3-F-5-Me
Et 2-OMe-5-Ac Me 2-Br-3-F-5-CF₃
Et 2-OMe-5-(U-3b) Me 2-Br-3-F-5-OMe
Et 2-OMe-5-CF₂H Me 2-Br-3-Cl-5-F
Et 2-OMe-5-CN Me 2-Br-3,5-di-Cl
Et 2-OMe-5-Et Me 2,5-di-Br-3-Cl
Et 2-OMe-5-OCF₂H Me 2-Br-3-Cl-5-Me
Et 2-OMe-5-OEt Me 2-Br-3-Cl-5-CF₃
Et 2-OMe-5-C(O)CF₃ Me 2-Br-3-Cl-5-OMe
Et 2-OCF₃-5-Ac Me 2,3-di-Br-5-F
Et 2-OCF₃-5-(U-3b) Me 2,3-di-Br-5-Cl
Et 2-OCF₃-5-CF₂H Me 2,3,5-tri-Br
Et 2-OCF₃-5-CN Me 2,3-di-Br-5-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Et 2-OCF₃-5-Et Me 2,3-di-Br-5-CF₃
Et 2-OCF₃-5-OCF₂H Me 2,3-di-Br-5-OMe
Et 2-OCF₃-5-OEt Me 2-Br-3-Me-5-F
Et 2-OCF₃-5-C(O)CF₃ Me 2-Br-3-Me-5-Cl
Et 3-F-4-Ac Me 2,5-di-Br-3-Me
Et 3-F-4-(U-3b) Me 2-Br-3,5-di-Me
Et 3-F-4-CF₂H Me 2-Br-3-Me-5-CF₃
Et 3-F-4-CN Me 2-Br-3-Me-5-OMe
Et 3-F-4-Et Me 2-Br-3-CF₃-5-F
Et 3-F-4-OCF₂H Me 2-Br-3-CF₃-5-Cl
Et 3-F-4-OEt Me 2,5-di-Br-3-CF₃
Et 3-F-4-C(O)CF₃ Me 2-Br-3-CF₃-5-Me
Et 3-Cl-4-Ac Me 2-Br-3,5-di-CF₃
Et 3-Cl-4-(U-3b) Me 2-Br-3-CF₃-5-OMe
Et 3-Cl-4-CF₂H Me 2-Br-3-OMe-5-F
Et 3-Cl-4-CN Me 2-Br-3-OMe-5-Cl
Et 3-Cl-4-Et Me 2,5-di-Br-3-OMe
Et 3-Cl-4-OCF₂H Me 2-Br-3-OMe-5-Me
Et 3-Cl-4-OEt Me 2-Br-3-OMe-5-CF₃
Et 3-Cl-4-C(O)CF₃ Me 2-Br-3,5-di-OMe
Et 3-Br-4-Ac Me 2-Br-4,5-di-F
Et 3-Br-4-(U-3b) Me 2-Br-4-F-5-Cl
Et 3-Br-4-CF₂H Me 2,5-di-Br-4-F
Et 3-Br-4-CN Me 2-Br-4-F-5-Me
Et 3-Br-4-Et Me 2-Br-4-F-5-CF₃
Et 3-Br-4-OCF₂H Me 2-Br-4-F-5-OMe
Et 3-Br-4-OEt Me 2-Br-4-Cl-5-F
Et 3-Br-4-C(O)CF₃ Me 2-Br-4,5-di-Cl
Et 3-Me-4-Ac Me 2,5-di-Br-4-Cl
Et 3-Me-4-(U-3b) Me 2-Br-4-Cl-5-Me
Et 3-Me-4-CF₂H Me 2-Br-4-Cl-5-CF₃
Et 3-Me-4-CN Me 2-Br-4-Cl-5-OMe
Et 3-Me-4-Et Me 2,4-di-Br-5-F
Et 3-Me-4-OCF₂H Me 2,4-di-Br-5-Cl
Et 3-Me-4-OEt Me 2,4,5-tri-Br
Et 3-Me-4-C(O)CF₃ Me 2,4-di-Br-5-Me
Et 3-CF₃-4-Ac Me 2,4-di-Br-5-CF₃
Et 3-CF₃-4-(U-3b) Me 2,4-di-Br-5-OMe
Et 3-CF₃-4-CF₂H Me 2-Br-4-Me-5-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Et 3-CF₃-4-CN Me 2-Br-4-Me-5-Cl
Et 3-CF₃-4-Et Me 2,5-di-Br-4-Me
Et 3-CF₃-4-OCF₂H Me 2-Br-4,5-di-Me
Et 3-CF₃-4-OEt Me 2-Br-4-Me-5-CF₃
Et 3-CF₃-4-C(O)CF₃ Me 2-Br-4-Me-5-OMe
Et 3-OMe-4-Ac Me 2-Br-4-CF₃-5-F
Et 3-OMe-4-(U-3b) Me 2-Br-4-CF₃-5-Cl
Et 3-OMe-4-CF₂H Me 2,5-di-Br-4-CF₃
Et 3-OMe-4-CN Me 2-Br-4-CF₃-5-Me
Et 3-OMe-4-Et Me 2-Br-4,5-di-CF₃
Et 3-OMe-4-OCF₂H Me 2-Br-4-CF₃-5-OMe
Et 3-OMe-4-OEt Me 2-Br-4-OMe-5-F
Et 3-OMe-4-C(O)CF₃ Me 2-Br-4-OMe-5-Cl
Et 3-OCF₃-4-Ac Me 2,5-di-Br-4-OMe
Et 3-OCF₃-4-(U-3b) Me 2-Br-4-OMe-5-Me
Et 3-OCF₃-4-CF₂H Me 2-Br-4-OMe-5-CF₃
Et 3-OCF₃-4-CN Me 2-Br-4,5-di-OMe
Et 3-OCF₃-4-Et Me 3-Br-4,5-di-F
Et 3-OCF₃-4-OCF₂H Me 3-Br-4-F-5-Cl
Et 3-OCF₃-4-OEt Me 3,5-di-Br-4-F
Et 3-OCF₃-4-C(O)CF₃ Me 3-Br-4-F-5-Me
Et 3-F-5-Ac Me 3-Br-4-F-5-CF₃
Et 3-F-5-(U-3b) Me 3-Br-4-F-5-OMe
Et 3-F-5-CF₂H Me 3-Br-4-Cl-5-F
Et 3-F-5-CN Me 3-Br-4,5-di-Cl
Et 3-F-5-Et Me 3,5-di-Br-4-Cl
Et 3-F-5-OCF₂H Me 3-Br-4-Cl-5-Me
Et 3-F-5-OEt Me 3-Br-4-Cl-5-CF₃
Et 3-F-5-C(O)CF₃ Me 3-Br-4-Cl-5-OMe
Et 3-Cl-5-Ac Me 3,4-di-Br-5-F
Et 3-Cl-5-(U-3b) Me 3,4-di-Br-5-Cl
Et 3-Cl-5-CF₂H Me 3,4,5-tri-Br
Et 3-Cl-5-CN Me 3,4-di-Br-5-Me
Et 3-Cl-5-Et Me 3,4-di-Br-5-CF₃
Et 3-Cl-5-OCF₂H Me 3,4-di-Br-5-OMe
Et 3-Cl-5-OEt Me 3-Br-4-Me-5-F
Et 3-Cl-5-C(O)CF₃ Me 3-Br-4-Me-5-Cl
Et 3-Br-5-Ac Me 3,5-di-Br-4-Me
Et 3-Br-5-(U-3b) Me 3-Br-4,5-di-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Et 3-Br-5-CF₂H Me 3-Br-4-Me-5-CF₃
Et 3-Br-5-CN Me 3-Br-4-Me-5-OMe
Et 3-Br-5-Et Me 3-Br-4-CF₃-5-F
Et 3-Br-5-OCF₂H Me 3-Br-4-CF₃-5-Cl
Et 3-Br-5-OEt Me 3,5-di-Br-4-CF₃
Et 3-Br-5-C(O)CF₃ Me 3-Br-4-CF₃-5-Me
Et 3-Me-5-Ac Me 3-Br-4,5-di-CF₃
Et 3-Me-5-(U-3b) Me 3-Br-4-CF₃-5-OMe
Et 3-Me-5-CF₂H Me 3-Br-4-OMe-5-F
Et 3-Me-5-CN Me 3-Br-4-OMe-5-Cl
Et 3-Me-5-Et Me 3,5-di-Br-4-OMe
Et 3-Me-5-OCF₂H Me 3-Br-4-OMe-5-Me
Et 3-Me-5-OEt Me 3-Br-4-OMe-5-CF₃
Et 3-Me-5-C(O)CF₃ Me 3-Br-4,5-di-OMe
Et 3-CF₃-5-Ac Me 2-Me-3,4-di-F
Et 3-CF₃-5-(U-3b) Me 2-Me-3-F-4-Cl
Et 3-CF₃-5-CF₂H Me 2-Me-3-F-4-Br
Et 3-CF₃-5-CN Me 2,4-di-Me-3-F
Et 3-CF₃-5-Et Me 2-Me-3-F-4-CF₃
Et 3-CF₃-5-OCF₂H Me 2-Me-3-F-4-OMe
Et 3-CF₃-5-OEt Me 2-Me-3-Cl-4-F
Et 3-CF₃-5-C(O)CF₃ Me 2-Me-3,4-di-Cl
Et 3-OMe-5-Ac Me 2-Me-3-Cl-4-Br
Et 3-OMe-5-(U-3b) Me 2,4-di-Me-3-Cl
Et 3-OMe-5-CF₂H Me 2-Me-3-Cl-4-CF₃
Et 3-OMe-5-CN Me 2-Me-3-Cl-4-OMe
Et 3-OMe-5-Et Me 2-Me-3-Br-4-F
Et 3-OMe-5-OCF₂H Me 2-Me-3-Br-4-Cl
Et 3-OMe-5-OEt Me 2-Me-3,4-di-Br
Et 3-OMe-5-C(O)CF₃ Me 2,4-di-Me-3-Br
Et 3-OCF₃-5-Ac Me 2-Me-3-Br-4-CF₃
Et 3-OCF₃-5-(U-3b) Me 2-Me-3-Br-4-OMe
Et 3-OCF₃-5-CF₂H Me 2,3-di-Me-4-F
Et 3-OCF₃-5-CN Me 2,3-di-Me-4-Cl
Et 3-OCF₃-5-Et Me 2,3-di-Me-4-Br
Et 3-OCF₃-5-OCF₂H Me 2,3,4-tri-Me
Et 3-OCF₃-5-OEt Me 2,3-di-Me-4-CF₃
Et 3-OCF₃-5-C(O)CF₃ Me 2,3-di-Me-4-OMe
Et 2-Ac-3-F Me 2-Me-3-CF₃-4-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Et 2-Ac-3-Cl Me 2-Me-3-CF₃-4-Cl
Et 2-Ac-3-Br Me 2-Me-3-CF₃-4-Br
Et 2-Ac-3-Me Me 2,4-di-Me-3-CF₃
Et 2-Ac-3-CF₃ Me 2-Me-3,4-di-CF₃
Et 2-Ac-3-OMe Me 2-Me-3-CF₃-4-OMe
Et 2-Ac-3-OCF₃ Me 2-Me-3-OMe-4-F
Et 2-(U-3b)-3-F Me 2-Me-3-OMe-4-Cl
Et 2-(U-3b)-3-Cl Me 2-Me-3-OMe-4-Br
Et 2-(U-3b)-3-Br Me 2,4-di-Me-3-OMe
Et 2-(U-3b)-3-Me Me 2-Me-3-OMe-4-CF₃
Et 2-(U-3b)-3-CF₃ Me 2-Me-3,4-di-OMe
Et 2-(U-3b)-3-OMe Me 2-Me-3,5-di-F
Et 2-(U-3b)-3-OCF₃ Me 2-Me-3-F-5-Cl
Et 2-CF₂H-3-F Me 2-Me-3-F-5-Br
Et 2-CF₂H-3-Cl Me 2,5-di-Me-3-F
Et 2-CF₂H-3-Br Me 2-Me-3-F-5-CF₃
Et 2-CF₂H-3-Me Me 2-Me-3-F-5-OMe
Et 2-CF₂H-3-CF₃ Me 2-Me-3-Cl-5-F
Et 2-CF₂H-3-OMe Me 2-Me-3,5-di-Cl
Et 2-CF₂H-3-OCF₃ Me 2-Me-3-Cl-5-Br
Et 2-CN-3-F Me 2,5-di-Me-3-Cl
Et 2-CN-3-Cl Me 2-Me-3-Cl-5-CF₃
Et 2-CN-3-Br Me 2-Me-3-Cl-5-OMe
Et 2-CN-3-Me Me 2-Me-3-Br-5-F
Et 2-CN-3-CF₃ Me 2-Me-3-Br-5-Cl
Et 2-CN-3-OMe Me 2-Me-3,5-di-Br
Et 2-CN-3-OCF₃ Me 2,5-di-Me-3-Br
Et 2-Et-3-F Me 2-Me-3-Br-5-CF₃
Et 2-Et-3-Cl Me 2-Me-3-Br-5-OMe
Et 2-Et-3-Br Me 2,3-di-Me-5-F
Et 2-Et-3-Me Me 2,3-di-Me-5-Cl
Et 2-Et-3-CF₃ Me 2,3-di-Me-5-Br
Et 2-Et-3-OMe Me 2,3,5-tri-Me
Et 2-Et-3-OCF₃ Me 2,3-di-Me-5-CF₃
Et 2-OCF₂H-3-F Me 2,3-di-Me-5-OMe
Et 2-OCF₂H-3-Cl Me 2-Me-3-CF₃-5-F
Et 2-OCF₂H-3-Br Me 2-Me-3-CF₃-5-Cl
Et 2-OCF₂H-3-Me Me 2-Me-3-CF₃-5-Br
Et 2-OCF₂H-3-CF₃ Me 2,5-di-Me-3-CF₃
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Et 2-OCF₂H-3-OMe Me 2-Me-3,5-di-CF₃
Et 2-OCF₂H-3-OCF₃ Me 2-Me-3-CF₃-5-OMe
Et 2-OEt-3-F Me 2-Me-3-OMe-5-F
Et 2-OEt-3-Cl Me 2-Me-3-OMe-5-Cl
Et 2-OEt-3-Br Me 2-Me-3-OMe-5-Br
Et 2-OEt-3-Me Me 2,5-di-Me-3-OMe
Et 2-OEt-3-CF₃ Me 2-Me-3-OMe-5-CF₃
Et 2-OEt-3-OMe Me 2-Me-3,5-di-OMe
Et 2-OEt-3-OCF₃ Me 2-Me-4,5-di-F
Et 2-C(O)CF₃-3-F Me 2-Me-4-F-5-Cl
Et 2-C(O)CF₃-3-Cl Me 2-Me-4-F-5-Br
Et 2-C(O)CF₃-3-Br Me 2,5-di-Me-4-F
Et 2-C(O)CF₃-3-Me Me 2-Me-4-F-5-CF₃
Et 2-C(O)CF₃-3-CF₃ Me 2-Me-4-F-5-OMe
Et 2-C(O)CF₃-3-OMe Me 2-Me-4-Cl-5-F
Et 2-C(O)CF₃-3-OCF₃ Me 2-Me-4,5-di-Cl
Et 2-Ac-4-F Me 2-Me-4-Cl-5-Br
Et 2-Ac-4-Cl Me 2,5-di-Me-4-Cl
Et 2-Ac-4-Br Me 2-Me-4-Cl-5-CF₃
Et 2-Ac-4-Me Me 2-Me-4-Cl-5-OMe
Et 2-Ac-4-CF₃ Me 2-Me-4-Br-5-F
Et 2-Ac-4-OMe Me 2-Me-4-Br-5-Cl
Et 2-Ac-4-OCF₃ Me 2-Me-4,5-di-Br
Et 2-(U-3b)-4-F Me 2,5-di-Me-4-Br
Et 2-(U-3b)-4-Cl Me 2-Me-4-Br-5-CF₃
Et 2-(U-3b)-4-Br Me 2-Me-4-Br-5-OMe
Et 2-(U-3b)-4-Me Me 2,4-di-Me-5-F
Et 2-(U-3b)-4-CF₃ Me 2,4-di-Me-5-Cl
Et 2-(U-3b)-4-OMe Me 2,4-di-Me-5-Br
Et 2-(U-3b)-4-OCF₃ Me 2,4,5-tri-Me
Et 2-CF₂H-4-F Me 2,4-di-Me-5-CF₃
Et 2-CF₂H-4-Cl Me 2,4-di-Me-5-OMe
Et 2-CF₂H-4-Br Me 2-Me-4-CF₃-5-F
Et 2-CF₂H-4-Me Me 2-Me-4-CF₃-5-Cl
Et 2-CF₂H-4-CF₃ Me 2-Me-4-CF₃-5-Br
Et 2-CF₂H-4-OMe Me 2,5-di-Me-4-CF₃
Et 2-CF₂H-4-OCF₃ Me 2-Me-4,5-di-CF₃
Et 2-CN-4-F Me 2-Me-4-CF₃-5-OMe
Et 2-CN-4-Cl Me 2-Me-4-OMe-5-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Et 2-CN-4-Br Me 2-Me-4-OMe-5-Cl
Et 2-CN-4-Me Me 2-Me-4-OMe-5-Br
Et 2-CN-4-CF₃ Me 2,5-di-Me-4-OMe
Et 2-CN-4-OMe Me 2-Me-4-OMe-5-CF₃
Et 2-CN-4-OCF₃ Me 2-Me-4,5-di-OMe
Et 2-Et-4-F Me 3-Me-4,5-di-F
Et 2-Et-4-Cl Me 3-Me-4-F-5-Cl
Et 2-Et-4-Br Me 3-Me-4-F-5-Br
Et 2-Et-4-Me Me 3,5-di-Me-4-F
Et 2-Et-4-CF₃ Me 3-Me-4-F-5-CF₃
Et 2-Et-4-OMe Me 3-Me-4-F-5-OMe
Et 2-Et-4-OCF₃ Me 3-Me-4-Cl-5-F
Et 2-OCF₂H-4-F Me 3-Me-4,5-di-Cl
Et 2-OCF₂H-4-Cl Me 3-Me-4-Cl-5-Br
Et 2-OCF₂H-4-Br Me 3,5-di-Me-4-Cl
Et 2-OCF₂H-4-Me Me 3-Me-4-Cl-5-CF₃
Et 2-OCF₂H-4-CF₃ Me 3-Me-4-Cl-5-OMe
Et 2-OCF₂H-4-OMe Me 3-Me-4-Br-5-F
Et 2-OCF₂H-4-OCF₃ Me 3-Me-4-Br-5-Cl
Et 2-OEt-4-F Me 3-Me-4,5-di-Br
Et 2-OEt-4-Cl Me 3,5-di-Me-4-Br
Et 2-OEt-4-Br Me 3-Me-4-Br-5-CF₃
Et 2-OEt-4-Me Me 3-Me-4-Br-5-OMe
Et 2-OEt-4-CF₃ Me 3,4-di-Me-5-F
Et 2-OEt-4-OMe Me 3,4-di-Me-5-Cl
Et 2-OEt-4-OCF₃ Me 3,4-di-Me-5-Br
Et 2-C(O)CF₃-4-F Me 3,4,5-tri-Me
Et 2-C(O)CF₃-4-Cl Me 3,4-di-Me-5-CF₃
Et 2-C(O)CF₃-4-Br Me 3,4-di-Me-5-OMe
Et 2-C(O)CF₃-4-Me Me 3-Me-4-CF₃-5-F
Et 2-C(O)CF₃-4-CF₃ Me 3-Me-4-CF₃-5-Cl
Et 2-C(O)CF₃-4-OMe Me 3-Me-4-CF₃-5-Br
Et 2-C(O)CF₃-4-OCF₃ Me 3,5-di-Me-4-CF₃
Et 2-Ac-5-F Me 3-Me-4,5-di-CF₃
Et 2-Ac-5-Cl Me 3-Me-4-CF₃-5-OMe
Et 2-Ac-5-Br Me 3-Me-4-OMe-5-F
Et 2-Ac-5-Me Me 3-Me-4-OMe-5-Cl
Et 2-Ac-5-CF₃ Me 3-Me-4-OMe-5-Br
Et 2-Ac-5-OMe Me 3,5-di-Me-4-OMe
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Et 2-Ac-5-OCF₃ Me 3-Me-4-OMe-5-CF₃
Et 2-(U-3b)-5-F Me 3-Me-4,5-di-OMe
Et 2-(U-3b)-5-Cl Me 2-CF₃-3,4-di-F
Et 2-(U-3b)-5-Br Me 2-CF₃-3-F-4-Cl
Et 2-(U-3b)-5-Me Me 2-CF₃-3-F-4-Br
Et 2-(U-3b)-5-CF₃ Me 2-CF₃-3-F-4-Me
Et 2-(U-3b)-5-OMe Me 2,4-di-CF₃-3-F
Et 2-(U-3b)-5-OCF₃ Me 2-CF₃-3-F-4-OMe
Et 2-CF₂H-5-F Me 2-CF₃-3-Cl-4-F
Et 2-CF₂H-5-Cl Me 2-CF₃-3,4-di-Cl
Et 2-CF₂H-5-Br Me 2-CF₃-3-Cl-4-Br
Et 2-CF₂H-5-Me Me 2-CF₃-3-Cl-4-Me
Et 2-CF₂H-5-CF₃ Me 2,4-di-CF₃-3-Cl
Et 2-CF₂H-5-OMe Me 2-CF₃-3-Cl-4-OMe
Et 2-CF₂H-5-OCF₃ Me 2-CF₃-3-Br-4-F
Et 2-CN-5-F Me 2-CF₃-3-Br-4-Cl
Et 2-CN-5-Cl Me 2-CF₃-3,4-di-Br
Et 2-CN-5-Br Me 2-CF₃-3-Br-4-Me
Et 2-CN-5-Me Me 2,4-di-CF₃-3-Br
Et 2-CN-5-CF₃ Me 2-CF₃-3-Br-4-OMe
Et 2-CN-5-OMe Me 2-CF₃-3-Me-4-F
Et 2-CN-5-OCF₃ Me 2-CF₃-3-Me-4-Cl
Et 2-Et-5-F Me 2-CF₃-3-Me-4-Br
Et 2-Et-5-Cl Me 2-CF₃-3,4-di-Me
Et 2-Et-5-Br Me 2,4-di-CF₃-3-Me
Et 2-Et-5-Me Me 2-CF₃-3-Me-4-OMe
Et 2-Et-5-CF₃ Me 2,3-di-CF₃-4-F
Et 2-Et-5-OMe Me 2,3-di-CF₃-4-Cl
Et 2-Et-5-OCF₃ Me 2,3-di-CF₃-4-Br
Et 2-OCF₂H-5-F Me 2,3-di-CF₃-4-Me
Et 2-OCF₂H-5-Cl Me 2,3,4-tri-CF₃
Et 2-OCF₂H-5-Br Me 2,3-di-CF₃-4-OMe
Et 2-OCF₂H-5-Me Me 2-CF₃-3-OMe-4-F
Et 2-OCF₂H-5-CF₃ Me 2-CF₃-3-OMe-4-Cl
Et 2-OCF₂H-5-OMe Me 2-CF₃-3-OMe-4-Br
Et 2-OCF₂H-5-OCF₃ Me 2-CF₃-3-OMe-4-Me
Et 2-OEt-5-F Me 2,4-di-CF₃-3-OMe
Et 2-OEt-5-Cl Me 2-CF₃-3,4-di-OMe
Et 2-OEt-5-Br Me 2-CF₃-3,5-di-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Et 2-OEt-5-Me Me 2-CF₃-3-F-5-Cl
Et 2-OEt-5-CF₃ Me 2-CF₃-3-F-5-Br
Et 2-OEt-5-OMe Me 2-CF₃-3-F-5-Me
Et 2-OEt-5-OCF₃ Me 2,5-di-CF₃-3-F
Et 2-C(O)CF₃-5-F Me 2-CF₃-3-F-5-OMe
Et 2-C(O)CF₃-5-Cl Me 2-CF₃-3-Cl-5-F
Et 2-C(O)CF₃-5-Br Me 2-CF₃-3,5-di-Cl
Et 2-C(O)CF₃-5-Me Me 2-CF₃-3-Cl-5-Br
Et 2-C(O)CF₃-5-CF₃ Me 2-CF₃-3-Cl-5-Me
Et 2-C(O)CF₃-5-OMe Me 2,5-di-CF₃-3-Cl
Et 2-C(O)CF₃-5-OCF₃ Me 2-CF₃-3-Cl-5-OMe
Et 3-Ac-4-F Me 2-CF₃-3-Br-5-F
Et 3-Ac-4-Cl Me 2-CF₃-3-Br-5-Cl
Et 3-Ac-4-Br Me 2-CF₃-3,5-di-Br
Et 3-Ac-4-Me Me 2-CF₃-3-Br-5-Me
Et 3-Ac-4-CF₃ Me 2,5-di-CF₃-3-Br
Et 3-Ac-4-OMe Me 2-CF₃-3-Br-5-OMe
Et 3-Ac-4-OCF₃ Me 2-CF₃-3-Me-5-F
Et 3-(U-3b)-4-F Me 2-CF₃-3-Me-5-Cl
Et 3-(U-3b)-4-Cl Me 2-CF₃-3-Me-5-Br
Et 3-(U-3b)-4-Br Me 2-CF₃-3,5-di-Me
Et 3-(U-3b)-4-Me Me 2,5-di-CF₃-3-Me
Et 3-(U-3b)-4-CF₃ Me 2-CF₃-3-Me-5-OMe
Et 3-(U-3b)-4-OMe Me 2,3-di-CF₃-5-F
Et 3-(U-3b)-4-OCF₃ Me 2,3-di-CF₃-5-Cl
Et 3-CF₂H-4-F Me 2,3-di-CF₃-5-Br
Et 3-CF₂H-4-Cl Me 2,3-di-CF₃-5-Me
Et 3-CF₂H-4-Br Me 2,3,5-tri-CF₃
Et 3-CF₂H-4-Me Me 2,3-di-CF₃-5-OMe
Et 3-CF₂H-4-CF₃ Me 2-CF₃-3-OMe-5-F
Et 3-CF₂H-4-OMe Me 2-CF₃-3-OMe-5-Cl
Et 3-CF₂H-4-OCF₃ Me 2-CF₃-3-OMe-5-Br
Et 3-CN-4-F Me 2-CF₃-3-OMe-5-Me
Et 3-CN-4-Cl Me 2,5-di-CF₃-3-OMe
Et 3-CN-4-Br Me 2-CF₃-3,5-di-OMe
Et 3-CN-4-Me Me 2-CF₃-4,5-di-F
Et 3-CN-4-CF₃ Me 2-CF₃-4-F-5-Cl
Et 3-CN-4-OMe Me 2-CF₃-4-F-5-Br
Et 3-CN-4-OCF₃ Me 2-CF₃-4-F-5-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Et 3-Et-4-F Me 2,5-di-CF₃-4-F
Et 3-Et-4-Cl Me 2-CF₃-4-F-5-OMe
Et 3-Et-4-Br Me 2-CF₃-4-Cl-5-F
Et 3-Et-4-Me Me 2-CF₃-4,5-di-Cl
Et 3-Et-4-CF₃ Me 2-CF₃-4-Cl-5-Br
Et 3-Et-4-OMe Me 2-CF₃-4-Cl-5-Me
Et 3-Et-4-OCF₃ Me 2,5-di-CF₃-4-Cl
Et 3-OCF₂H-4-F Me 2-CF₃-4-Cl-5-OMe
Et 3-OCF₂H-4-Cl Me 2-CF₃-4-Br-5-F
Et 3-OCF₂H-4-Br Me 2-CF₃-4-Br-5-Cl
Et 3-OCF₂H-4-Me Me 2-CF₃-4,5-di-Br
Et 3-OCF₂H-4-CF₃ Me 2-CF₃-4-Br-5-Me
Et 3-OCF₂H-4-OMe Me 2,5-di-CF₃-4-Br
Et 3-OCF₂H-4-OCF₃ Me 2-CF₃-4-Br-5-OMe
Et 3-OEt-4-F Me 2-CF₃-4-Me-5-F
Et 3-OEt-4-Cl Me 2-CF₃-4-Me-5-Cl
Et 3-OEt-4-Br Me 2-CF₃-4-Me-5-Br
Et 3-OEt-4-Me Me 2-CF₃-4,5-di-Me
Et 3-OEt-4-CF₃ Me 2,5-di-CF₃-4-Me
Et 3-OEt-4-OMe Me 2-CF₃-4-Me-5-OMe
Et 3-OEt-4-OCF₃ Me 2,4-di-CF₃-5-F
Et 3-C(O)CF₃-4-F Me 2,4-di-CF₃-5-Cl
Et 3-C(O)CF₃-4-Cl Me 2,4-di-CF₃-5-Br
Et 3-C(O)CF₃-4-Br Me 2,4-di-CF₃-5-Me
Et 3-C(O)CF₃-4-Me Me 2,4,5-tri-CF₃
Et 3-C(O)CF₃-4-CF₃ Me 2,4-di-CF₃-5-OMe
Et 3-C(O)CF₃-4-OMe Me 2-CF₃-4-OMe-5-F
Et 3-C(O)CF₃-4-OCF₃ Me 2-CF₃-4-OMe-5-Cl
Et 3-Ac-5-F Me 2-CF₃-4-OMe-5-Br
Et 3-Ac-5-Cl Me 2-CF₃-4-OMe-5-Me
Et 3-Ac-5-Br Me 2,5-di-CF₃-4-OMe
Et 3-Ac-5-Me Me 2-CF₃-4,5-di-OMe
Et 3-Ac-5-CF₃ Me 3-CF₃-4,5-di-F
Et 3-Ac-5-OMe Me 3-CF₃-4-F-5-Cl
Et 3-Ac-5-OCF₃ Me 3-CF₃-4-F-5-Br
Et 3-(U-3b)-5-F Me 3-CF₃-4-F-5-Me
Et 3-(U-3b)-5-Cl Me 3,5-di-CF₃-4-F
Et 3-(U-3b)-5-Br Me 3-CF₃-4-F-5-OMe
Et 3-(U-3b)-5-Me Me 3-CF₃-4-Cl-5-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Et 3-(U-3b)-5-CF₃ Me 3-CF₃-4,5-di-Cl
Et 3-(U-3b)-5-OMe Me 3-CF₃-4-Cl-5-Br
Et 3-(U-3b)-5-OCF₃ Me 3-CF₃-4-Cl-5-Me
Et 3-CF₂H-5-F Me 3,5-di-CF₃-4-Cl
Et 3-CF₂H-5-Cl Me 3-CF₃-4-Cl-5-OMe
Et 3-CF₂H-5-Br Me 3-CF₃-4-Br-5-F
Et 3-CF₂H-5-Me Me 3-CF₃-4-Br-5-Cl
Et 3-CF₂H-5-CF₃ Me 3-CF₃-4,5-di-Br
Et 3-CF₂H-5-OMe Me 3-CF₃-4-Br-5-Me
Et 3-CF₂H-5-OCF₃ Me 3,5-di-CF₃-4-Br
Et 3-CN-5-F Me 3-CF₃-4-Br-5-OMe
Et 3-CN-5-Cl Me 3-CF₃-4-Me-5-F
Et 3-CN-5-Br Me 3-CF₃-4-Me-5-Cl
Et 3-CN-5-Me Me 3-CF₃-4-Me-5-Br
Et 3-CN-5-CF₃ Me 3-CF₃-4,5-di-Me
Et 3-CN-5-OMe Me 3,5-di-CF₃-4-Me
Et 3-CN-5-OCF₃ Me 3-CF₃-4-Me-5-OMe
Et 3-Et-5-F Me 3,4-di-CF₃-5-F
Et 3-Et-5-Cl Me 3,4-di-CF₃-5-Cl
Et 3-Et-5-Br Me 3,4-di-CF₃-5-Br
Et 3-Et-5-Me Me 3,4-di-CF₃-5-Me
Et 3-Et-5-CF₃ Me 3,4,5-tri-CF₃
Et 3-Et-5-OMe Me 3,4-di-CF₃-5-OMe
Et 3-Et-5-OCF₃ Me 3-CF₃-4-OMe-5-F
Et 3-OCF₂H-5-F Me 3-CF₃-4-OMe-5-Cl
Et 3-OCF₂H-5-Cl Me 3-CF₃-4-OMe-5-Br
Et 3-OCF₂H-5-Br Me 3-CF₃-4-OMe-5-Me
Et 3-OCF₂H-5-Me Me 3,5-di-CF₃-4-OMe
Et 3-OCF₂H-5-CF₃ Me 3-CF₃-4,5-di-OMe
Et 3-OCF₂H-5-OMe Me 2-OMe-3,4-di-F
Et 3-OCF₂H-5-OCF₃ Me 2-OMe-3-F-4-Cl
Et 3-OEt-5-F Me 2-OMe-3-F-4-Br
Et 3-OEt-5-Cl Me 2-OMe-3-F-4-Me
Et 3-OEt-5-Br Me 2-OMe-3-F-4-CF₃
Et 3-OEt-5-Me Me 2,4-di-OMe-3-F
Et 3-OEt-5-CF₃ Me 2-OMe-3-Cl-4-F
Et 3-OEt-5-OMe Me 2-OMe-3,4-di-Cl
Et 3-OEt-5-OCF₃ Me 2-OMe-3-Cl-4-Br
Et 3-C(O)CF₃-5-F Me 2-OMe-3-Cl-4-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
Et 3-C(O)CF₃-5-Cl Me 2-OMe-3-Cl-4-CF₃
Et 3-C(O)CF₃-5-Br Me 2,4-di-OMe-3-Cl
Et 3-C(O)CF₃-5-Me Me 2-OMe-3-Br-4-F
Et 3-C(O)CF₃-5-CF₃ Me 2-OMe-3-Br-4-Cl
Et 3-C(O)CF₃-5-OMe Me 2-OMe-3,4-di-Br
Et 3-C(O)CF₃-5-OCF₃ Me 2-OMe-3-Br-4-Me
iPr 2-F-3-Ac Me 2-OMe-3-Br-4-CF₃
iPr 2-F-3-(U-3b) Me 2,4-di-OMe-3-Br
iPr 2-F-3-CF₂H Me 2-OMe-3-Me-4-F
iPr 2-F-3-CN Me 2-OMe-3-Me-4-Cl
iPr 2-F-3-Et Me 2-OMe-3-Me-4-Br
iPr 2-F-3-OCF₂H Me 2-OMe-3,4-di-Me
iPr 2-F-3-OEt Me 2-OMe-3-Me-4-CF₃
iPr 2-F-3-C(O)CF₃ Me 2,4-di-OMe-3-Me
iPr 2-Cl-3-Ac Me 2-OMe-3-CF₃-4-F
iPr 2-Cl-3-(U-3b) Me 2-OMe-3-CF₃-4-Cl
iPr 2-Cl-3-CF₂H Me 2-OMe-3-CF₃-4-Br
iPr 2-Cl-3-CN Me 2-OMe-3-CF₃-4-Me
iPr 2-Cl-3-Et Me 2-OMe-3,4-di-CF₃
iPr 2-Cl-3-OCF₂H Me 2,4-di-OMe-3-CF₃
iPr 2-Cl-3-OEt Me 2,3-di-OMe-4-F
iPr 2-Cl-3-C(O)CF₃ Me 2,3-di-OMe-4-Cl
iPr 2-Br-3-Ac Me 2,3-di-OMe-4-Br
iPr 2-Br-3-(U-3b) Me 2,3-di-OMe-4-Me
iPr 2-Br-3-CF₂H Me 2,3-di-OMe-4-CF₃
iPr 2-Br-3-CN Me 2,3,4-tri-OMe
iPr 2-Br-3-Et Me 2-OMe-3,5-di-F
iPr 2-Br-3-OCF₂H Me 2-OMe-3-F-5-Cl
iPr 2-Br-3-OEt Me 2-OMe-3-F-5-Br
iPr 2-Br-3-C(O)CF₃ Me 2-OMe-3-F-5-Me
iPr 2-Me-3-Ac Me 2-OMe-3-F-5-CF₃
iPr 2-Me-3-(U-3b) Me 2,5-di-OMe-3-F
iPr 2-Me-3-CF₂H Me 2-OMe-3-Cl-5-F
iPr 2-Me-3-CN Me 2-OMe-3,5-di-Cl
iPr 2-Me-3-Et Me 2-OMe-3-Cl-5-Br
iPr 2-Me-3-OCF₂H Me 2-OMe-3-Cl-5-Me
iPr 2-Me-3-OEt Me 2-OMe-3-Cl-5-CF₃
iPr 2-Me-3-C(O)CF₃ Me 2,5-di-OMe-3-Cl
iPr 2-CF₃-3-Ac Me 2-OMe-3-Br-5-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
iPr 2-CF₃-3-(U-3b) Me 2-OMe-3-Br-5-Cl
iPr 2-CF₃-3-CF₂H Me 2-OMe-3,5-di-Br
iPr 2-CF₃-3-CN Me 2-OMe-3-Br-5-Me
iPr 2-CF₃-3-Et Me 2-OMe-3-Br-5-CF₃
iPr 2-CF₃-3-OCF₂H Me 2,5-di-OMe-3-Br
iPr 2-CF₃-3-OEt Me 2-OMe-3-Me-5-F
iPr 2-CF₃-3-C(O)CF₃ Me 2-OMe-3-Me-5-Cl
iPr 2-OMe-3-Ac Me 2-OMe-3-Me-5-Br
iPr 2-OMe-3-(U-3b) Me 2-OMe-3,5-di-Me
iPr 2-OMe-3-CF₂H Me 2-OMe-3-Me-5-CF₃
iPr 2-OMe-3-CN Me 2,5-di-OMe-3-Me
iPr 2-OMe-3-Et Me 2-OMe-3-CF₃-5-F
iPr 2-OMe-3-OCF₂H Me 2-OMe-3-CF₃-5-Cl
iPr 2-OMe-3-OEt Me 2-OMe-3-CF₃-5-Br
iPr 2-OMe-3-C(O)CF₃ Me 2-OMe-3-CF₃-5-Me
iPr 2-OCF₃-3-Ac Me 2-OMe-3,5-di-CF₃
iPr 2-OCF₃-3-(U-3b) Me 2,5-di-OMe-3-CF₃
iPr 2-OCF₃-3-CF₂H Me 2,3-di-OMe-5-F
iPr 2-OCF₃-3-CN Me 2,3-di-OMe-5-Cl
iPr 2-OCF₃-3-Et Me 2,3-di-OMe-5-Br
iPr 2-OCF₃-3-OCF₂H Me 2,3-di-OMe-5-Me
iPr 2-OCF₃-3-OEt Me 2,3-di-OMe-5-CF₃
iPr 2-OCF₃-3-C(O)CF₃ Me 2,3,5-tri-OMe
iPr 2-F-4-Ac Me 2-OMe-4,5-di-F
iPr 2-F-4-(U-3b) Me 2-OMe-4-F-5-Cl
iPr 2-F-4-CF₂H Me 2-OMe-4-F-5-Br
iPr 2-F-4-CN Me 2-OMe-4-F-5-Me
iPr 2-F-4-Et Me 2-OMe-4-F-5-CF₃
iPr 2-F-4-OCF₂H Me 2,5-di-OMe-4-F
iPr 2-F-4-OEt Me 2-OMe-4-Cl-5-F
iPr 2-F-4-C(O)CF₃ Me 2-OMe-4,5-di-Cl
iPr 2-Cl-4-Ac Me 2-OMe-4-Cl-5-Br
iPr 2-Cl-4-(U-3b) Me 2-OMe-4-Cl-5-Me
iPr 2-Cl-4-CF₂H Me 2-OMe-4-Cl-5-CF₃
iPr 2-Cl-4-CN Me 2,5-di-OMe-4-Cl
iPr 2-Cl-4-Et Me 2-OMe-4-Br-5-F
iPr 2-Cl-4-OCF₂H Me 2-OMe-4-Br-5-Cl
iPr 2-Cl-4-OEt Me 2-OMe-4,5-di-Br
iPr 2-Cl-4-C(O)CF₃ Me 2-OMe-4-Br-5-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
iPr 2-Br-4-Ac Me 2-OMe-4-Br-5-CF₃
iPr 2-Br-4-(U-3b) Me 2,5-di-OMe-4-Br
iPr 2-Br-4-CF₂H Me 2-OMe-4-Me-5-F
iPr 2-Br-4-CN Me 2-OMe-4-Me-5-Cl
iPr 2-Br-4-Et Me 2-OMe-4-Me-5-Br
iPr 2-Br-4-OCF₂H Me 2-OMe-4,5-di-Me
iPr 2-Br-4-OEt Me 2-OMe-4-Me-5-CF₃
iPr 2-Br-4-C(O)CF₃ Me 2,5-di-OMe-4-Me
iPr 2-Me-4-Ac Me 2-OMe-4-CF₃-5-F
iPr 2-Me-4-(U-3b) Me 2-OMe-4-CF₃-5-Cl
iPr 2-Me-4-CF₂H Me 2-OMe-4-CF₃-5-Br
iPr 2-Me-4-CN Me 2-OMe-4-CF₃-5-Me
iPr 2-Me-4-Et Me 2-OMe-4,5-di-CF₃
iPr 2-Me-4-OCF₂H Me 2,5-di-OMe-4-CF₃
iPr 2-Me-4-OEt Me 2,4-di-OMe-5-F
iPr 2-Me-4-C(O)CF₃ Me 2,4-di-OMe-5-Cl
iPr 2-CF₃-4-Ac Me 2,4-di-OMe-5-Br
iPr 2-CF₃-4-(U-3b) Me 2,4-di-OMe-5-Me
iPr 2-CF₃-4-CF₂H Me 2,4-di-OMe-5-CF₃
iPr 2-CF₃-4-CN Me 2,4,5-tri-OMe
iPr 2-CF₃-4-Et Me 3-OMe-4,5-di-F
iPr 2-CF₃-4-OCF₂H Me 3-OMe-4-F-5-Cl
iPr 2-CF₃-4-OEt Me 3-OMe-4-F-5-Br
iPr 2-CF₃-4-C(O)CF₃ Me 3-OMe-4-F-5-Me
iPr 2-OMe-4-Ac Me 3-OMe-4-F-5-CF₃
iPr 2-OMe-4-(U-3b) Me 3,5-di-OMe-4-F
iPr 2-OMe-4-CF₂H Me 3-OMe-4-Cl-5-F
iPr 2-OMe-4-CN Me 3-OMe-4,5-di-Cl
iPr 2-OMe-4-Et Me 3-OMe-4-Cl-5-Br
iPr 2-OMe-4-OCF₂H Me 3-OMe-4-Cl-5-Me
iPr 2-OMe-4-OEt Me 3-OMe-4-Cl-5-CF₃
iPr 2-OMe-4-C(O)CF₃ Me 3,5-di-OMe-4-Cl
iPr 2-OCF₃-4-Ac Me 3-OMe-4-Br-5-F
iPr 2-OCF₃-4-(U-3b) Me 3-OMe-4-Br-5-Cl
iPr 2-OCF₃-4-CF₂H Me 3-OMe-4,5-di-Br
iPr 2-OCF₃-4-CN Me 3-OMe-4-Br-5-Me
iPr 2-OCF₃-4-Et Me 3-OMe-4-Br-5-CF₃
iPr 2-OCF₃-4-OCF₂H Me 3,5-di-OMe-4-Br
iPr 2-OCF₃-4-OEt Me 3-OMe-4-Me-5-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
iPr 2-OCF₃-4-C(O)CF₃ Me 3-OMe-4-Me-5-Cl
iPr 2-F-5-Ac Me 3-OMe-4-Me-5-Br
iPr 2-F-5-(U-3b) Me 3-OMe-4,5-di-Me
iPr 2-F-5-CF₂H Me 3-OMe-4-Me-5-CF₃
iPr 2-F-5-CN Me 3,5-di-OMe-4-Me
iPr 2-F-5-Et Me 3-OMe-4-CF₃-5-F
iPr 2-F-5-OCF₂H Me 3-OMe-4-CF₃-5-Cl
iPr 2-F-5-OEt Me 3-OMe-4-CF₃-5-Br
iPr 2-F-5-C(O)CF₃ Me 3-OMe-4-CF₃-5-Me
iPr 2-Cl-5-Ac Me 3-OMe-4,5-di-CF₃
iPr 2-Cl-5-(U-3b) Me 3,5-di-OMe-4-CF₃
iPr 2-Cl-5-CF₂H Me 3,4-di-OMe-5-F
iPr 2-Cl-5-CN Me 3,4-di-OMe-5-Cl
iPr 2-Cl-5-Et Me 3,4-di-OMe-5-Br
iPr 2-Cl-5-OCF₂H Me 3,4-di-OMe-5-Me
iPr 2-Cl-5-OEt Me 3,4-di-OMe-5-CF₃
iPr 2-Cl-5-C(O)CF₃ Me 3,4,5-tri-OMe
iPr 2-Br-5-Ac Et 2,3,4-tri-F
iPr 2-Br-5-(U-3b) Et 2,3-di-F-4-Cl
iPr 2-Br-5-CF₂H Et 2,3-di-F-4-Br
iPr 2-Br-5-CN Et 2,3-di-F-4-Me
iPr 2-Br-5-Et Et 2,3-di-F-4-CF₃
iPr 2-Br-5-OCF₂H Et 2,3-di-F-4-OMe
iPr 2-Br-5-OEt Et 2,4-di-F-3-Cl
iPr 2-Br-5-C(O)CF₃ Et 2-F-3,4-di-Cl
iPr 2-Me-5-Ac Et 2-F-3-Cl-4-Br
iPr 2-Me-5-(U-3b) Et 2-F-3-Cl-4-Me
iPr 2-Me-5-CF₂H Et 2-F-3-Cl-4-CF₃
iPr 2-Me-5-CN Et 2-F-3-Cl-4-OMe
iPr 2-Me-5-Et Et 2,4-di-F-3-Br
iPr 2-Me-5-OCF₂H Et 2-F-3-Br-4-Cl
iPr 2-Me-5-OEt Et 2-F-3,4-di-Br
iPr 2-Me-5-C(O)CF₃ Et 2-F-3-Br-4-Me
iPr 2-CF₃-5-Ac Et 2-F-3-Br-4-CF₃
iPr 2-CF₃-5-(U-3b) Et 2-F-3-Br-4-OMe
iPr 2-CF₃-5-CF₂H Et 2,4-di-F-3-Me
iPr 2-CF₃-5-CN Et 2-F-3-Me-4-Cl
iPr 2-CF₃-5-Et Et 2-F-3-Me-4-Br
iPr 2-CF₃-5-OCF₂H Et 2-F-3,4-di-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
iPr 2-CF₃-5-OEt Et 2-F-3-Me-4-CF₃
iPr 2-CF₃-5-C(O)CF₃ Et 2-F-3-Me-4-OMe
iPr 2-OMe-5-Ac Et 2,4-di-F-3-CF₃
iPr 2-OMe-5-(U-3b) Et 2-F-3-CF₃-4-Cl
iPr 2-OMe-5-CF₂H Et 2-F-3-CF₃-4-Br
iPr 2-OMe-5-CN Et 2-F-3-CF₃-4-Me
iPr 2-OMe-5-Et Et 2-F-3,4-di-CF₃
iPr 2-OMe-5-OCF₂H Et 2-F-3-CF₃-4-OMe
iPr 2-OMe-5-OEt Et 2,4-di-F-3-OMe
iPr 2-OMe-5-C(O)CF₃ Et 2-F-3-OMe-4-Cl
iPr 2-OCF₃-5-Ac Et 2-F-3-OMe-4-Br
iPr 2-OCF₃-5-(U-3b) Et 2-F-3-OMe-4-Me
iPr 2-OCF₃-5-CF₂H Et 2-F-3-OMe-4-CF₃
iPr 2-OCF₃-5-CN Et 2-F-3,4-di-OMe
iPr 2-OCF₃-5-Et Et 2,3,5-tri-F
iPr 2-OCF₃-5-OCF₂H Et 2,3-di-F-5-Cl
iPr 2-OCF₃-5-OEt Et 2,3-di-F-5-Br
iPr 2-OCF₃-5-C(O)CF₃ Et 2,3-di-F-5-Me
iPr 3-F-4-Ac Et 2,3-di-F-5-CF₃
iPr 3-F-4-(U-3b) Et 2,3-di-F-5-OMe
iPr 3-F-4-CF₂H Et 2,5-di-F-3-Cl
iPr 3-F-4-CN Et 2-F-3,5-di-Cl
iPr 3-F-4-Et Et 2-F-3-Cl-5-Br
iPr 3-F-4-OCF₂H Et 2-F-3-Cl-5-Me
iPr 3-F-4-OEt Et 2-F-3-Cl-5-CF₃
iPr 3-F-4-C(O)CF₃ Et 2-F-3-Cl-5-OMe
iPr 3-Cl-4-Ac Et 2,5-di-F-3-Br
iPr 3-Cl-4-(U-3b) Et 2-F-3-Br-5-Cl
iPr 3-Cl-4-CF₂H Et 2-F-3,5-di-Br
iPr 3-Cl-4-CN Et 2-F-3-Br-5-Me
iPr 3-Cl-4-Et Et 2-F-3-Br-5-CF₃
iPr 3-Cl-4-OCF₂H Et 2-F-3-Br-5-OMe
iPr 3-Cl-4-OEt Et 2,5-di-F-3-Me
iPr 3-Cl-4-C(O)CF₃ Et 2-F-3-Me-5-Cl
iPr 3-Br-4-Ac Et 2-F-3-Me-5-Br
iPr 3-Br-4-(U-3b) Et 2-F-3,5-di-Me
iPr 3-Br-4-CF₂H Et 2-F-3-Me-5-CF₃
iPr 3-Br-4-CN Et 2-F-3-Me-5-OMe
iPr 3-Br-4-Et Et 2,5-di-F-3-CF₃
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
iPr 3-Br-4-OCF₂H Et 2-F-3-CF₃-5-Cl
iPr 3-Br-4-OEt Et 2-F-3-CF₃-5-Br
iPr 3-Br-4-C(O)CF₃ Et 2-F-3-CF₃-5-Me
iPr 3-Me-4-Ac Et 2-F-3,5-di-CF₃
iPr 3-Me-4-(U-3b) Et 2-F-3-CF₃-5-OMe
iPr 3-Me-4-CF₂H Et 2,5-di-F-3-OMe
iPr 3-Me-4-CN Et 2-F-3-OMe-5-Cl
iPr 3-Me-4-Et Et 2-F-3-OMe-5-Br
iPr 3-Me-4-OCF₂H Et 2-F-3-OMe-5-Me
iPr 3-Me-4-OEt Et 2-F-3-OMe-5-CF₃
iPr 3-Me-4-C(O)CF₃ Et 2-F-3,5-di-OMe
iPr 3-CF₃-4-Ac Et 2,4,5-tri-F
iPr 3-CF₃-4-(U-3b) Et 2,4-di-F-5-Cl
iPr 3-CF₃-4-CF₂H Et 2,4-di-F-5-Br
iPr 3-CF₃-4-CN Et 2,4-di-F-5-Me
iPr 3-CF₃-4-Et Et 2,4-di-F-5-CF₃
iPr 3-CF₃-4-OCF₂H Et 2,4-di-F-5-OMe
iPr 3-CF₃-4-OEt Et 2,5-di-F-4-Cl
iPr 3-CF₃-4-C(O)CF₃ Et 2-F-4,5-di-Cl
iPr 3-OMe-4-Ac Et 2-F-4-Cl-5-Br
iPr 3-OMe-4-(U-3b) Et 2-F-4-Cl-5-Me
iPr 3-OMe-4-CF₂H Et 2-F-4-Cl-5-CF₃
iPr 3-OMe-4-CN Et 2-F-4-Cl-5-OMe
iPr 3-OMe-4-Et Et 2,5-di-F-4-Br
iPr 3-OMe-4-OCF₂H Et 2-F-4-Br-5-Cl
iPr 3-OMe-4-OEt Et 2-F-4,5-di-Br
iPr 3-OMe-4-C(O)CF₃ Et 2-F-4-Br-5-Me
iPr 3-OCF₃-4-Ac Et 2-F-4-Br-5-CF₃
iPr 3-OCF₃-4-(U-3b) Et 2-F-4-Br-5-OMe
iPr 3-OCF₃-4-CF₂H Et 2,5-di-F-4-Me
iPr 3-OCF₃-4-CN Et 2-F-4-Me-5-Cl
iPr 3-OCF₃-4-Et Et 2-F-4-Me-5-Br
iPr 3-OCF₃-4-OCF₂H Et 2-F-4,5-di-Me
iPr 3-OCF₃-4-OEt Et 2-F-4-Me-5-CF₃
iPr 3-OCF₃-4-C(O)CF₃ Et 2-F-4-Me-5-OMe
iPr 3-F-5-Ac Et 2,5-di-F-4-CF₃
iPr 3-F-5-(U-3b) Et 2-F-4-CF₃-5-Cl
iPr 3-F-5-CF₂H Et 2-F-4-CF₃-5-Br
iPr 3-F-5-CN Et 2-F-4-CF₃-5-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
iPr 3-F-5-Et Et 2-F-4,5-di-CF₃
iPr 3-F-5-OCF₂H Et 2-F-4-CF₃-5-OMe
iPr 3-F-5-OEt Et 2,5-di-F-4-OMe
iPr 3-F-5-C(O)CF₃ Et 2-F-4-OMe-5-Cl
iPr 3-Cl-5-Ac Et 2-F-4-OMe-5-Br
iPr 3-Cl-5-(U-3b) Et 2-F-4-OMe-5-Me
iPr 3-Cl-5-CF₂H Et 2-F-4-OMe-5-CF₃
iPr 3-Cl-5-CN Et 2-F-4,5-di-OMe
iPr 3-Cl-5-Et Et 3,4,5-tri-F
iPr 3-Cl-5-OCF₂H Et 3,4-di-F-5-Cl
iPr 3-Cl-5-OEt Et 3,4-di-F-5-Br
iPr 3-Cl-5-C(O)CF₃ Et 3,4-di-F-5-Me
iPr 3-Br-5-Ac Et 3,4-di-F-5-CF₃
iPr 3-Br-5-(U-3b) Et 3,4-di-F-5-OMe
iPr 3-Br-5-CF₂H Et 3,5-di-F-4-Cl
iPr 3-Br-5-CN Et 3-F-4,5-di-Cl
iPr 3-Br-5-Et Et 3-F-4-Cl-5-Br
iPr 3-Br-5-OCF₂H Et 3-F-4-Cl-5-Me
iPr 3-Br-5-OEt Et 3-F-4-Cl-5-CF₃
iPr 3-Br-5-C(O)CF₃ Et 3-F-4-Cl-5-OMe
iPr 3-Me-5-Ac Et 3,5-di-F-4-Br
iPr 3-Me-5-(U-3b) Et 3-F-4-Br-5-Cl
iPr 3-Me-5-CF₂H Et 3-F-4,5-di-Br
iPr 3-Me-5-CN Et 3-F-4-Br-5-Me
iPr 3-Me-5-Et Et 3-F-4-Br-5-CF₃
iPr 3-Me-5-OCF₂H Et 3-F-4-Br-5-OMe
iPr 3-Me-5-OEt Et 3,5-di-F-4-Me
iPr 3-Me-5-C(O)CF₃ Et 3-F-4-Me-5-Cl
iPr 3-CF₃-5-Ac Et 3-F-4-Me-5-Br
iPr 3-CF₃-5-(U-3b) Et 3-F-4,5-di-Me
iPr 3-CF₃-5-CF₂H Et 3-F-4-Me-5-CF₃
iPr 3-CF₃-5-CN Et 3-F-4-Me-5-OMe
iPr 3-CF₃-5-Et Et 3,5-di-F-4-CF₃
iPr 3-CF₃-5-OCF₂H Et 3-F-4-CF₃-5-Cl
iPr 3-CF₃-5-OEt Et 3-F-4-CF₃-5-Br
iPr 3-CF₃-5-C(O)CF₃ Et 3-F-4-CF₃-5-Me
iPr 3-OMe-5-Ac Et 3-F-4,5-di-CF₃
iPr 3-OMe-5-(U-3b) Et 3-F-4-CF₃-5-OMe
iPr 3-OMe-5-CF₂H Et 3,5-di-F-4-OMe
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
iPr 3-OMe-5-CN Et 3-F-4-OMe-5-Cl
iPr 3-OMe-5-Et Et 3-F-4-OMe-5-Br
iPr 3-OMe-5-OCF₂H Et 3-F-4-OMe-5-Me
iPr 3-OMe-5-OEt Et 3-F-4-OMe-5-CF₃
iPr 3-OMe-5-C(O)CF₃ Et 3-F-4,5-di-OMe
iPr 3-OCF₃-5-Ac Et 2-Cl-3,4-di-F
iPr 3-OCF₃-5-(U-3b) Et 2,4-di-Cl-3-F
iPr 3-OCF₃-5-CF₂H Et 2-Cl-3-F-4-Br
iPr 3-OCF₃-5-CN Et 2-Cl-3-F-4-Me
iPr 3-OCF₃-5-Et Et 2-Cl-3-F-4-CF₃
iPr 3-OCF₃-5-OCF₂H Et 2-Cl-3-F-4-OMe
iPr 3-OCF₃-5-OEt Et 2,3-di-Cl-4-F
iPr 3-OCF₃-5-C(O)CF₃ Et 2,3,4-tri-Cl
iPr 2-Ac-3-F Et 2,3-di-Cl-4-Br
iPr 2-Ac-3-Cl Et 2,3-di-Cl-4-Me
iPr 2-Ac-3-Br Et 2,3-di-Cl-4-CF₃
iPr 2-Ac-3-Me Et 2,3-di-Cl-4-OMe
iPr 2-Ac-3-CF₃ Et 2-Cl-3-Br-4-F
iPr 2-Ac-3-OMe Et 2,4-di-Cl-3-Br
iPr 2-Ac-3-OCF₃ Et 2-Cl-3,4-di-Br
iPr 2-(U-3b)-3-F Et 2-Cl-3-Br-4-Me
iPr 2-(U-3b)-3-Cl Et 2-Cl-3-Br-4-CF₃
iPr 2-(U-3b)-3-Br Et 2-Cl-3-Br-4-OMe
iPr 2-(U-3b)-3-Me Et 2-Cl-3-Me-4-F
iPr 2-(U-3b)-3-CF₃ Et 2,4-di-Cl-3-Me
iPr 2-(U-3b)-3-OMe Et 2-Cl-3-Me-4-Br
iPr 2-(U-3b)-3-OCF₃ Et 2-Cl-3,4-di-Me
iPr 2-CF₂H-3-F Et 2-Cl-3-Me-4-CF₃
iPr 2-CF₂H-3-Cl Et 2-Cl-3-Me-4-OMe
iPr 2-CF₂H-3-Br Et 2-Cl-3-CF₃-4-F
iPr 2-CF₂H-3-Me Et 2,4-di-Cl-3-CF₃
iPr 2-CF₂H-3-CF₃ Et 2-Cl-3-CF₃-4-Br
iPr 2-CF₂H-3-OMe Et 2-Cl-3-CF₃-4-Me
iPr 2-CF₂H-3-OCF₃ Et 2-Cl-3,4-di-CF₃
iPr 2-CN-3-F Et 2-Cl-3-CF₃-4-OMe
iPr 2-CN-3-Cl Et 2-Cl-3-OMe-4-F
iPr 2-CN-3-Br Et 2,4-di-Cl-3-OMe
iPr 2-CN-3-Me Et 2-Cl-3-OMe-4-Br
iPr 2-CN-3-CF₃ Et 2-Cl-3-OMe-4-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
iPr 2-CN-3-OMe Et 2-Cl-3-OMe-4-CF₃
iPr 2-CN-3-OCF₃ Et 2-Cl-3,4-di-OMe
iPr 2-Et-3-F Et 2-Cl-3,5-di-F
iPr 2-Et-3-Cl Et 2,5-di-Cl-3-F
iPr 2-Et-3-Br Et 2-Cl-3-F-5-Br
iPr 2-Et-3-Me Et 2-Cl-3-F-5-Me
iPr 2-Et-3-CF₃ Et 2-Cl-3-F-5-CF₃
iPr 2-Et-3-OMe Et 2-Cl-3-F-5-OMe
iPr 2-Et-3-OCF₃ Et 2,3-di-Cl-5-F
iPr 2-OCF₂H-3-F Et 2,3,5-tri-Cl
iPr 2-OCF₂H-3-Cl Et 2,3-di-Cl-5-Br
iPr 2-OCF₂H-3-Br Et 2,3-di-Cl-5-Me
iPr 2-OCF₂H-3-Me Et 2,3-di-Cl-5-CF₃
iPr 2-OCF₂H-3-CF₃ Et 2,3-di-Cl-5-OMe
iPr 2-OCF₂H-3-OMe Et 2-Cl-3-Br-5-F
iPr 2-OCF₂H-3-OCF₃ Et 2,5-di-Cl-3-Br
iPr 2-OEt-3-F Et 2-Cl-3,5-di-Br
iPr 2-OEt-3-Cl Et 2-Cl-3-Br-5-Me
iPr 2-OEt-3-Br Et 2-Cl-3-Br-5-CF₃
iPr 2-OEt-3-Me Et 2-Cl-3-Br-5-OMe
iPr 2-OEt-3-CF₃ Et 2-Cl-3-Me-5-F
iPr 2-OEt-3-OMe Et 2,5-di-Cl-3-Me
iPr 2-OEt-3-OCF₃ Et 2-Cl-3-Me-5-Br
iPr 2-C(O)CF₃-3-F Et 2-Cl-3,5-di-Me
iPr 2-C(O)CF₃-3-Cl Et 2-Cl-3-Me-5-CF₃
iPr 2-C(O)CF₃-3-Br Et 2-Cl-3-Me-5-OMe
iPr 2-C(O)CF₃-3-Me Et 2-Cl-3-CF₃-5-F
iPr 2-C(O)CF₃-3-CF₃ Et 2,5-di-Cl-3-CF₃
iPr 2-C(O)CF₃-3-OMe Et 2-Cl-3-CF₃-5-Br
iPr 2-C(O)CF₃-3-OCF₃ Et 2-Cl-3-CF₃-5-Me
iPr 2-Ac-4-F Et 2-Cl-3,5-di-CF₃
iPr 2-Ac-4-Cl Et 2-Cl-3-CF₃-5-OMe
iPr 2-Ac-4-Br Et 2-Cl-3-OMe-5-F
iPr 2-Ac-4-Me Et 2,5-di-Cl-3-OMe
iPr 2-Ac-4-CF₃ Et 2-Cl-3-OMe-5-Br
iPr 2-Ac-4-OMe Et 2-Cl-3-OMe-5-Me
iPr 2-Ac-4-OCF₃ Et 2-Cl-3-OMe-5-CF₃
iPr 2-(U-3b)-4-F Et 2-Cl-3,5-di-OMe
iPr 2-(U-3b)-4-Cl Et 2-Cl-4,5-di-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
iPr 2-(U-3b)-4-Br Et 2,5-di-Cl-4-F
iPr 2-(U-3b)-4-Me Et 2-Cl-4-F-5-Br
iPr 2-(U-3b)-4-CF₃ Et 2-Cl-4-F-5-Me
iPr 2-(U-3b)-4-OMe Et 2-Cl-4-F-5-CF₃
iPr 2-(U-3b)-4-OCF₃ Et 2-Cl-4-F-5-OMe
iPr 2-CF₂H-4-F Et 2,4-di-Cl-5-F
iPr 2-CF₂H-4-Cl Et 2,4,5-tri-Cl
iPr 2-CF₂H-4-Br Et 2,4-di-Cl-5-Br
iPr 2-CF₂H-4-Me Et 2,4-di-Cl-5-Me
iPr 2-CF₂H-4-CF₃ Et 2,4-di-Cl-5-CF₃
iPr 2-CF₂H-4-OMe Et 2,4-di-Cl-5-OMe
iPr 2-CF₂H-4-OCF₃ Et 2-Cl-4-Br-5-F
iPr 2-CN-4-F Et 2,5-di-Cl-4-Br
iPr 2-CN-4-Cl Et 2-Cl-4,5-di-Br
iPr 2-CN-4-Br Et 2-Cl-4-Br-5-Me
iPr 2-CN-4-Me Et 2-Cl-4-Br-5-CF₃
iPr 2-CN-4-CF₃ Et 2-Cl-4-Br-5-OMe
iPr 2-CN-4-OMe Et 2-Cl-4-Me-5-F
iPr 2-CN-4-OCF₃ Et 2,5-di-Cl-4-Me
iPr 2-Et-4-F Et 2-Cl-4-Me-5-Br
iPr 2-Et-4-Cl Et 2-Cl-4,5-di-Me
iPr 2-Et-4-Br Et 2-Cl-4-Me-5-CF₃
iPr 2-Et-4-Me Et 2-Cl-4-Me-5-OMe
iPr 2-Et-4-CF₃ Et 2-Cl-4-CF₃-5-F
iPr 2-Et-4-OMe Et 2,5-di-Cl-4-CF₃
iPr 2-Et-4-OCF₃ Et 2-Cl-4-CF₃-5-Br
iPr 2-OCF₂H-4-F Et 2-Cl-4-CF₃-5-Me
iPr 2-OCF₂H-4-Cl Et 2-Cl-4,5-di-CF₃
iPr 2-OCF₂H-4-Br Et 2-Cl-4-CF₃-5-OMe
iPr 2-OCF₂H-4-Me Et 2-Cl-4-OMe-5-F
iPr 2-OCF₂H-4-CF₃ Et 2,5-di-Cl-4-OMe
iPr 2-OCF₂H-4-OMe Et 2-Cl-4-OMe-5-Br
iPr 2-OCF₂H-4-OCF₃ Et 2-Cl-4-OMe-5-Me
iPr 2-OEt-4-F Et 2-Cl-4-OMe-5-CF₃
iPr 2-OEt-4-Cl Et 2-Cl-4,5-di-OMe
iPr 2-OEt-4-Br Et 3-Cl-4,5-di-F
iPr 2-OEt-4-Me Et 3,5-di-Cl-4-F
iPr 2-OEt-4-CF₃ Et 3-Cl-4-F-5-Br
iPr 2-OEt-4-OMe Et 3-Cl-4-F-5-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
iPr 2-OEt-4-OCF₃ Et 3-Cl-4-F-5-CF₃
iPr 2-C(O)CF₃-4-F Et 3-Cl-4-F-5-OMe
iPr 2-C(O)CF₃-4-Cl Et 3,4-di-Cl-5-F
iPr 2-C(O)CF₃-4-Br Et 3,4,5-tri-Cl
iPr 2-C(O)CF₃-4-Me Et 3,4-di-Cl-5-Br
iPr 2-C(O)CF₃-4-CF₃ Et 3,4-di-Cl-5-Me
iPr 2-C(O)CF₃-4-OMe Et 3,4-di-Cl-5-CF₃
iPr 2-C(O)CF₃-4-OCF₃ Et 3,4-di-Cl-5-OMe
iPr 2-Ac-5-F Et 3-Cl-4-Br-5-F
iPr 2-Ac-5-Cl Et 3,5-di-Cl-4-Br
iPr 2-Ac-5-Br Et 3-Cl-4,5-di-Br
iPr 2-Ac-5-Me Et 3-Cl-4-Br-5-Me
iPr 2-Ac-5-CF₃ Et 3-Cl-4-Br-5-CF₃
iPr 2-Ac-5-OMe Et 3-Cl-4-Br-5-OMe
iPr 2-Ac-5-OCF₃ Et 3-Cl-4-Me-5-F
iPr 2-(U-3b)-5-F Et 3,5-di-Cl-4-Me
iPr 2-(U-3b)-5-Cl Et 3-Cl-4-Me-5-Br
iPr 2-(U-3b)-5-Br Et 3-Cl-4,5-di-Me
iPr 2-(U-3b)-5-Me Et 3-Cl-4-Me-5-CF₃
iPr 2-(U-3b)-5-CF₃ Et 3-Cl-4-Me-5-OMe
iPr 2-(U-3b)-5-OMe Et 3-Cl-4-CF₃-5-F
iPr 2-(U-3b)-5-OCF₃ Et 3,5-di-Cl-4-CF₃
iPr 2-CF₂H-5-F Et 3-Cl-4-CF₃-5-Br
iPr 2-CF₂H-5-Cl Et 3-Cl-4-CF₃-5-Me
iPr 2-CF₂H-5-Br Et 3-Cl-4,5-di-CF₃
iPr 2-CF₂H-5-Me Et 3-Cl-4-CF₃-5-OMe
iPr 2-CF₂H-5-CF₃ Et 3-Cl-4-OMe-5-F
iPr 2-CF₂H-5-OMe Et 3,5-di-Cl-4-OMe
iPr 2-CF₂H-5-OCF₃ Et 3-Cl-4-OMe-5-Br
iPr 2-CN-5-F Et 3-Cl-4-OMe-5-Me
iPr 2-CN-5-Cl Et 3-Cl-4-OMe-5-CF₃
iPr 2-CN-5-Br Et 3-Cl-4,5-di-OMe
iPr 2-CN-5-Me Et 2-Br-3,4-di-F
iPr 2-CN-5-CF₃ Et 2-Br-3-F-4-Cl
iPr 2-CN-5-OMe Et 2,4-di-Br-3-F
iPr 2-CN-5-OCF₃ Et 2-Br-3-F-4-Me
iPr 2-Et-5-F Et 2-Br-3-F-4-CF₃
iPr 2-Et-5-Cl Et 2-Br-3-F-4-OMe
iPr 2-Et-5-Br Et 2-Br-3-Cl-4-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
iPr 2-Et-5-Me Et 2-Br-3,4-di-Cl
iPr 2-Et-5-CF₃ Et 2,4-di-Br-3-Cl
iPr 2-Et-5-OMe Et 2-Br-3-Cl-4-Me
iPr 2-Et-5-OCF₃ Et 2-Br-3-Cl-4-CF₃
iPr 2-OCF₂H-5-F Et 2-Br-3-Cl-4-OMe
iPr 2-OCF₂H-5-Cl Et 2,3-di-Br-4-F
iPr 2-OCF₂H-5-Br Et 2,3-di-Br-4-Cl
iPr 2-OCF₂H-5-Me Et 2,3,4-tri-Br
iPr 2-OCF₂H-5-CF₃ Et 2,3-di-Br-4-Me
iPr 2-OCF₂H-5-OMe Et 2,3-di-Br-4-CF₃
iPr 2-OCF₂H-5-OCF₃ Et 2,3-di-Br-4-OMe
iPr 2-OEt-5-F Et 2-Br-3-Me-4-F
iPr 2-OEt-5-Cl Et 2-Br-3-Me-4-Cl
iPr 2-OEt-5-Br Et 2,4-di-Br-3-Me
iPr 2-OEt-5-Me Et 2-Br-3,4-di-Me
iPr 2-OEt-5-CF₃ Et 2-Br-3-Me-4-CF₃
iPr 2-OEt-5-OMe Et 2-Br-3-Me-4-OMe
iPr 2-OEt-5-OCF₃ Et 2-Br-3-CF₃-4-F
iPr 2-C(O)CF₃-5-F Et 2-Br-3-CF₃-4-Cl
iPr 2-C(O)CF₃-5-Cl Et 2,4-di-Br-3-CF₃
iPr 2-C(O)CF₃-5-Br Et 2-Br-3-CF₃-4-Me
iPr 2-C(O)CF₃-5-Me Et 2-Br-3,4-di-CF₃
iPr 2-C(O)CF₃-5-CF₃ Et 2-Br-3-CF₃-4-OMe
iPr 2-C(O)CF₃-5-OMe Et 2-Br-3-OMe-4-F
iPr 2-C(O)CF₃-5-OCF₃ Et 2-Br-3-OMe-4-Cl
iPr 3-Ac-4-F Et 2,4-di-Br-3-OMe
iPr 3-Ac-4-Cl Et 2-Br-3-OMe-4-Me
iPr 3-Ac-4-Br Et 2-Br-3-OMe-4-CF₃
iPr 3-Ac-4-Me Et 2-Br-3,4-di-OMe
iPr 3-Ac-4-CF₃ Et 2-Br-3,5-di-F
iPr 3-Ac-4-OMe Et 2-Br-3-F-5-Cl
iPr 3-Ac-4-OCF₃ Et 2,5-di-Br-3-F
iPr 3-(U-3b)-4-F Et 2-Br-3-F-5-Me
iPr 3-(U-3b)-4-Cl Et 2-Br-3-F-5-CF₃
iPr 3-(U-3b)-4-Br Et 2-Br-3-F-5-OMe
iPr 3-(U-3b)-4-Me Et 2-Br-3-Cl-5-F
iPr 3-(U-3b)-4-CF₃ Et 2-Br-3,5-di-Cl
iPr 3-(U-3b)-4-OMe Et 2,5-di-Br-3-Cl
iPr 3-(U-3b)-4-OCF₃ Et 2-Br-3-Cl-5-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
iPr 3-CF₂H-4-F Et 2-Br-3-Cl-5-CF₃
iPr 3-CF₂H-4-Cl Et 2-Br-3-Cl-5-OMe
iPr 3-CF₂H-4-Br Et 2,3-di-Br-5-F
iPr 3-CF₂H-4-Me Et 2,3-di-Br-5-Cl
iPr 3-CF₂H-4-CF₃ Et 2,3,5-tri-Br
iPr 3-CF₂H-4-OMe Et 2,3-di-Br-5-Me
iPr 3-CF₂H-4-OCF₃ Et 2,3-di-Br-5-CF₃
iPr 3-CN-4-F Et 2,3-di-Br-5-OMe
iPr 3-CN-4-Cl Et 2-Br-3-Me-5-F
iPr 3-CN-4-Br Et 2-Br-3-Me-5-Cl
iPr 3-CN-4-Me Et 2,5-di-Br-3-Me
iPr 3-CN-4-CF₃ Et 2-Br-3,5-di-Me
iPr 3-CN-4-OMe Et 2-Br-3-Me-5-CF₃
iPr 3-CN-4-OCF₃ Et 2-Br-3-Me-5-OMe
iPr 3-Et-4-F Et 2-Br-3-CF₃-5-F
iPr 3-Et-4-Cl Et 2-Br-3-CF₃-5-Cl
iPr 3-Et-4-Br Et 2,5-di-Br-3-CF₃
iPr 3-Et-4-Me Et 2-Br-3-CF₃-5-Me
iPr 3-Et-4-CF₃ Et 2-Br-3,5-di-CF₃
iPr 3-Et-4-OMe Et 2-Br-3-CF₃-5-OMe
iPr 3-Et-4-OCF₃ Et 2-Br-3-OMe-5-F
iPr 3-OCF₂H-4-F Et 2-Br-3-OMe-5-Cl
iPr 3-OCF₂H-4-Cl Et 2,5-di-Br-3-OMe
iPr 3-OCF₂H-4-Br Et 2-Br-3-OMe-5-Me
iPr 3-OCF₂H-4-Me Et 2-Br-3-OMe-5-CF₃
iPr 3-OCF₂H-4-CF₃ Et 2-Br-3,5-di-OMe
iPr 3-OCF₂H-4-OMe Et 2-Br-4,5-di-F
iPr 3-OCF₂H-4-OCF₃ Et 2-Br-4-F-5-Cl
iPr 3-OEt-4-F Et 2,5-di-Br-4-F
iPr 3-OEt-4-Cl Et 2-Br-4-F-5-Me
iPr 3-OEt-4-Br Et 2-Br-4-F-5-CF₃
iPr 3-OEt-4-Me Et 2-Br-4-F-5-OMe
iPr 3-OEt-4-CF₃ Et 2-Br-4-Cl-5-F
iPr 3-OEt-4-OMe Et 2-Br-4,5-di-Cl
iPr 3-OEt-4-OCF₃ Et 2,5-di-Br-4-Cl
iPr 3-C(O)CF₃-4-F Et 2-Br-4-Cl-5-Me
iPr 3-C(O)CF₃-4-Cl Et 2-Br-4-Cl-5-CF₃
iPr 3-C(O)CF₃-4-Br Et 2-Br-4-Cl-5-OMe
iPr 3-C(O)CF₃-4-Me Et 2,4-di-Br-5-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
iPr 3-C(O)CF₃-4-CF₃ Et 2,4-di-Br-5-Cl
iPr 3-C(O)CF₃-4-OMe Et 2,4,5-tri-Br
iPr 3-C(O)CF₃-4-OCF₃ Et 2,4-di-Br-5-Me
iPr 3-Ac-5-F Et 2,4-di-Br-5-CF₃
iPr 3-Ac-5-Cl Et 2,4-di-Br-5-OMe
iPr 3-Ac-5-Br Et 2-Br-4-Me-5-F
iPr 3-Ac-5-Me Et 2-Br-4-Me-5-Cl
iPr 3-Ac-5-CF₃ Et 2,5-di-Br-4-Me
iPr 3-Ac-5-OMe Et 2-Br-4,5-di-Me
iPr 3-Ac-5-OCF₃ Et 2-Br-4-Me-5-CF₃
iPr 3-(U-3b)-5-F Et 2-Br-4-Me-5-OMe
iPr 3-(U-3b)-5-Cl Et 2-Br-4-CF₃-5-F
iPr 3-(U-3b)-5-Br Et 2-Br-4-CF₃-5-Cl
iPr 3-(U-3b)-5-Me Et 2,5-di-Br-4-CF₃
iPr 3-(U-3b)-5-CF₃ Et 2-Br-4-CF₃-5-Me
iPr 3-(U-3b)-5-OMe Et 2-Br-4,5-di-CF₃
iPr 3-(U-3b)-5-OCF₃ Et 2-Br-4-CF₃-5-OMe
iPr 3-CF₂H-5-F Et 2-Br-4-OMe-5-F
iPr 3-CF₂H-5-Cl Et 2-Br-4-OMe-5-Cl
iPr 3-CF₂H-5-Br Et 2,5-di-Br-4-OMe
iPr 3-CF₂H-5-Me Et 2-Br-4-OMe-5-Me
iPr 3-CF₂H-5-CF₃ Et 2-Br-4-OMe-5-CF₃
iPr 3-CF₂H-5-OMe Et 2-Br-4,5-di-OMe
iPr 3-CF₂H-5-OCF₃ Et 3-Br-4,5-di-F
iPr 3-CN-5-F Et 3-Br-4-F-5-Cl
iPr 3-CN-5-Cl Et 3,5-di-Br-4-F
iPr 3-CN-5-Br Et 3-Br-4-F-5-Me
iPr 3-CN-5-Me Et 3-Br-4-F-5-CF₃
iPr 3-CN-5-CF₃ Et 3-Br-4-F-5-OMe
iPr 3-CN-5-OMe Et 3-Br-4-Cl-5-F
iPr 3-CN-5-OCF₃ Et 3-Br-4,5-di-Cl
iPr 3-Et-5-F Et 3,5-di-Br-4-Cl
iPr 3-Et-5-Cl Et 3-Br-4-Cl-5-Me
iPr 3-Et-5-Br Et 3-Br-4-Cl-5-CF₃
iPr 3-Et-5-Me Et 3-Br-4-Cl-5-OMe
iPr 3-Et-5-CF₃ Et 3,4-di-Br-5-F
iPr 3-Et-5-OMe Et 3,4-di-Br-5-Cl
iPr 3-Et-5-OCF₃ Et 3,4,5-tri-Br
iPr 3-OCF₂H-5-F Et 3,4-di-Br-5-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
iPr 3-OCF₂H-5-Cl Et 3,4-di-Br-5-CF₃
iPr 3-OCF₂H-5-Br Et 3,4-di-Br-5-OMe
iPr 3-OCF₂H-5-Me Et 3-Br-4-Me-5-F
iPr 3-OCF₂H-5-CF₃ Et 3-Br-4-Me-5-Cl
iPr 3-OCF₂H-5-OMe Et 3,5-di-Br-4-Me
iPr 3-OCF₂H-5-OCF₃ Et 3-Br-4,5-di-Me
iPr 3-OEt-5-F Et 3-Br-4-Me-5-CF₃
iPr 3-OEt-5-Cl Et 3-Br-4-Me-5-OMe
iPr 3-OEt-5-Br Et 3-Br-4-CF₃-5-F
iPr 3-OEt-5-Me Et 3-Br-4-CF₃-5-Cl
iPr 3-OEt-5-CF₃ Et 3,5-di-Br-4-CF₃
iPr 3-OEt-5-OMe Et 3-Br-4-CF₃-5-Me
iPr 3-OEt-5-OCF₃ Et 3-Br-4,5-di-CF₃
iPr 3-C(O)CF₃-5-F Et 3-Br-4-CF₃-5-OMe
iPr 3-C(O)CF₃-5-Cl Et 3-Br-4-OMe-5-F
iPr 3-C(O)CF₃-5-Br Et 3-Br-4-OMe-5-Cl
iPr 3-C(O)CF₃-5-Me Et 3,5-di-Br-4-OMe
iPr 3-C(O)CF₃-5-CF₃ Et 3-Br-4-OMe-5-Me
iPr 3-C(O)CF₃-5-OMe Et 3-Br-4-OMe-5-CF₃
iPr 3-C(O)CF₃-5-OCF₃ Et 3-Br-4,5-di-OMe
U-4a 2-F-3-Ac Et 2-Me-3,4-di-F
U-4a 2-F-3-(U-3b) Et 2-Me-3-F-4-Cl
U-4a 2-F-3-CF₂H Et 2-Me-3-F-4-Br
U-4a 2-F-3-CN Et 2,4-di-Me-3-F
U-4a 2-F-3-Et Et 2-Me-3-F-4-CF₃
U-4a 2-F-3-OCF₂H Et 2-Me-3-F-4-OMe
U-4a 2-F-3-OEt Et 2-Me-3-Cl-4-F
U-4a 2-F-3-C(O)CF₃ Et 2-Me-3,4-di-Cl
U-4a 2-Cl-3-Ac Et 2-Me-3-Cl-4-Br
U-4a 2-Cl-3-(U-3b) Et 2,4-di-Me-3-Cl
U-4a 2-Cl-3-CF₂H Et 2-Me-3-Cl-4-CF₃
U-4a 2-Cl-3-CN Et 2-Me-3-Cl-4-OMe
U-4a 2-Cl-3-Et Et 2-Me-3-Br-4-F
U-4a 2-Cl-3-OCF₂H Et 2-Me-3-Br-4-Cl
U-4a 2-Cl-3-OEt Et 2-Me-3,4-di-Br
U-4a 2-Cl-3-C(O)CF₃ Et 2,4-di-Me-3-Br
U-4a 2-Br-3-Ac Et 2-Me-3-Br-4-CF₃
U-4a 2-Br-3-(U-3b) Et 2-Me-3-Br-4-OMe
U-4a 2-Br-3-CF₂H Et 2,3-di-Me-4-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
U-4a 2-Br-3-CN Et 2,3-di-Me-4-Cl
U-4a 2-Br-3-Et Et 2,3-di-Me-4-Br
U-4a 2-Br-3-OCF₂H Et 2,3,4-tri-Me
U-4a 2-Br-3-OEt Et 2,3-di-Me-4-CF₃
U-4a 2-Br-3-C(O)CF₃ Et 2,3-di-Me-4-OMe
U-4a 2-Me-3-Ac Et 2-Me-3-CF₃-4-F
U-4a 2-Me-3-(U-3b) Et 2-Me-3-CF₃-4-Cl
U-4a 2-Me-3-CF₂H Et 2-Me-3-CF₃-4-Br
U-4a 2-Me-3-CN Et 2,4-di-Me-3-CF₃
U-4a 2-Me-3-Et Et 2-Me-3,4-di-CF₃
U-4a 2-Me-3-OCF₂H Et 2-Me-3-CF₃-4-OMe
U-4a 2-Me-3-OEt Et 2-Me-3-OMe-4-F
U-4a 2-Me-3-C(O)CF₃ Et 2-Me-3-OMe-4-Cl
U-4a 2-CF₃-3-Ac Et 2-Me-3-OMe-4-Br
U-4a 2-CF₃-3-(U-3b) Et 2,4-di-Me-3-OMe
U-4a 2-CF₃-3-CF₂H Et 2-Me-3-OMe-4-CF₃
U-4a 2-CF₃-3-CN Et 2-Me-3,4-di-OMe
U-4a 2-CF₃-3-Et Et 2-Me-3,5-di-F
U-4a 2-CF₃-3-OCF₂H Et 2-Me-3-F-5-Cl
U-4a 2-CF₃-3-OEt Et 2-Me-3-F-5-Br
U-4a 2-CF₃-3-C(O)CF₃ Et 2,5-di-Me-3-F
U-4a 2-OMe-3-Ac Et 2-Me-3-F-5-CF₃
U-4a 2-OMe-3-(U-3b) Et 2-Me-3-F-5-OMe
U-4a 2-OMe-3-CF₂H Et 2-Me-3-Cl-5-F
U-4a 2-OMe-3-CN Et 2-Me-3,5-di-Cl
U-4a 2-OMe-3-Et Et 2-Me-3-Cl-5-Br
U-4a 2-OMe-3-OCF₂H Et 2,5-di-Me-3-Cl
U-4a 2-OMe-3-OEt Et 2-Me-3-Cl-5-CF₃
U-4a 2-OMe-3-C(O)CF₃ Et 2-Me-3-Cl-5-OMe
U-4a 2-OCF₃-3-Ac Et 2-Me-3-Br-5-F
U-4a 2-OCF₃-3-(U-3b) Et 2-Me-3-Br-5-Cl
U-4a 2-OCF₃-3-CF₂H Et 2-Me-3,5-di-Br
U-4a 2-OCF₃-3-CN Et 2,5-di-Me-3-Br
U-4a 2-OCF₃-3-Et Et 2-Me-3-Br-5-CF₃
U-4a 2-OCF₃-3-OCF₂H Et 2-Me-3-Br-5-OMe
U-4a 2-OCF₃-3-OEt Et 2,3-di-Me-5-F
U-4a 2-OCF₃-3-C(O)CF₃ Et 2,3-di-Me-5-Cl
U-4a 2-F-4-Ac Et 2,3-di-Me-5-Br
U-4a 2-F-4-(U-3b) Et 2,3,5-tri-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
U-4a 2-F-4-CF₂H Et 2,3-di-Me-5-CF₃
U-4a 2-F-4-CN Et 2,3-di-Me-5-OMe
U-4a 2-F-4-Et Et 2-Me-3-CF₃-5-F
U-4a 2-F-4-OCF₂H Et 2-Me-3-CF₃-5-Cl
U-4a 2-F-4-OEt Et 2-Me-3-CF₃-5-Br
U-4a 2-F-4-C(O)CF₃ Et 2,5-di-Me-3-CF₃
U-4a 2-Cl-4-Ac Et 2-Me-3,5-di-CF₃
U-4a 2-Cl-4-(U-3b) Et 2-Me-3-CF₃-5-OMe
U-4a 2-Cl-4-CF₂H Et 2-Me-3-OMe-5-F
U-4a 2-Cl-4-CN Et 2-Me-3-OMe-5-Cl
U-4a 2-Cl-4-Et Et 2-Me-3-OMe-5-Br
U-4a 2-Cl-4-OCF₂H Et 2,5-di-Me-3-OMe
U-4a 2-Cl-4-OEt Et 2-Me-3-OMe-5-CF₃
U-4a 2-Cl-4-C(O)CF₃ Et 2-Me-3,5-di-OMe
U-4a 2-Br-4-Ac Et 2-Me-4,5-di-F
U-4a 2-Br-4-(U-3b) Et 2-Me-4-F-5-Cl
U-4a 2-Br-4-CF₂H Et 2-Me-4-F-5-Br
U-4a 2-Br-4-CN Et 2,5-di-Me-4-F
U-4a 2-Br-4-Et Et 2-Me-4-F-5-CF₃
U-4a 2-Br-4-OCF₂H Et 2-Me-4-F-5-OMe
U-4a 2-Br-4-OEt Et 2-Me-4-Cl-5-F
U-4a 2-Br-4-C(O)CF₃ Et 2-Me-4,5-di-Cl
U-4a 2-Me-4-Ac Et 2-Me-4-Cl-5-Br
U-4a 2-Me-4-(U-3b) Et 2,5-di-Me-4-Cl
U-4a 2-Me-4-CF₂H Et 2-Me-4-Cl-5-CF₃
U-4a 2-Me-4-CN Et 2-Me-4-Cl-5-OMe
U-4a 2-Me-4-Et Et 2-Me-4-Br-5-F
U-4a 2-Me-4-OCF₂H Et 2-Me-4-Br-5-Cl
U-4a 2-Me-4-OEt Et 2-Me-4,5-di-Br
U-4a 2-Me-4-C(O)CF₃ Et 2,5-di-Me-4-Br
U-4a 2-CF₃-4-Ac Et 2-Me-4-Br-5-CF₃
U-4a 2-CF₃-4-(U-3b) Et 2-Me-4-Br-5-OMe
U-4a 2-CF₃-4-CF₂H Et 2,4-di-Me-5-F
U-4a 2-CF₃-4-CN Et 2,4-di-Me-5-Cl
U-4a 2-CF₃-4-Et Et 2,4-di-Me-5-Br
U-4a 2-CF₃-4-OCF₂H Et 2,4,5-tri-Me
U-4a 2-CF₃-4-OEt Et 2,4-di-Me-5-CF₃
U-4a 2-CF₃-4-C(O)CF₃ Et 2,4-di-Me-5-OMe
U-4a 2-OMe-4-Ac Et 2-Me-4-CF₃-5-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
U-4a 2-OMe-4-(U-3b) Et 2-Me-4-CF₃-5-Cl
U-4a 2-OMe-4-CF₂H Et 2-Me-4-CF₃-5-Br
U-4a 2-OMe-4-CN Et 2,5-di-Me-4-CF₃
U-4a 2-OMe-4-Et Et 2-Me-4,5-di-CF₃
U-4a 2-OMe-4-OCF₂H Et 2-Me-4-CF₃-5-OMe
U-4a 2-OMe-4-OEt Et 2-Me-4-OMe-5-F
U-4a 2-OMe-4-C(O)CF₃ Et 2-Me-4-OMe-5-Cl
U-4a 2-OCF₃-4-Ac Et 2-Me-4-OMe-5-Br
U-4a 2-OCF₃-4-(U-3b) Et 2,5-di-Me-4-OMe
U-4a 2-OCF₃-4-CF₂H Et 2-Me-4-OMe-5-CF₃
U-4a 2-OCF₃-4-CN Et 2-Me-4,5-di-OMe
U-4a 2-OCF₃-4-Et Et 3-Me-4,5-di-F
U-4a 2-OCF₃-4-OCF₂H Et 3-Me-4-F-5-Cl
U-4a 2-OCF₃-4-OEt Et 3-Me-4-F-5-Br
U-4a 2-OCF₃-4-C(O)CF₃ Et 3,5-di-Me-4-F
U-4a 2-F-5-Ac Et 3-Me-4-F-5-CF₃
U-4a 2-F-5-(U-3b) Et 3-Me-4-F-5-OMe
U-4a 2-F-5-CF₂H Et 3-Me-4-Cl-5-F
U-4a 2-F-5-CN Et 3-Me-4,5-di-Cl
U-4a 2-F-5-Et Et 3-Me-4-Cl-5-Br
U-4a 2-F-5-OCF₂H Et 3,5-di-Me-4-Cl
U-4a 2-F-5-OEt Et 3-Me-4-Cl-5-CF₃
U-4a 2-F-5-C(O)CF₃ Et 3-Me-4-Cl-5-OMe
U-4a 2-Cl-5-Ac Et 3-Me-4-Br-5-F
U-4a 2-Cl-5-(U-3b) Et 3-Me-4-Br-5-Cl
U-4a 2-Cl-5-CF₂H Et 3-Me-4,5-di-Br
U-4a 2-Cl-5-CN Et 3,5-di-Me-4-Br
U-4a 2-Cl-5-Et Et 3-Me-4-Br-5-CF₃
U-4a 2-Cl-5-OCF₂H Et 3-Me-4-Br-5-OMe
U-4a 2-Cl-5-OEt Et 3,4-di-Me-5-F
U-4a 2-Cl-5-C(O)CF₃ Et 3,4-di-Me-5-Cl
U-4a 2-Br-5-Ac Et 3,4-di-Me-5-Br
U-4a 2-Br-5-(U-3b) Et 3,4,5-tri-Me
U-4a 2-Br-5-CF₂H Et 3,4-di-Me-5-CF₃
U-4a 2-Br-5-CN Et 3,4-di-Me-5-OMe
U-4a 2-Br-5-Et Et 3-Me-4-CF₃-5-F
U-4a 2-Br-5-OCF₂H Et 3-Me-4-CF₃-5-Cl
U-4a 2-Br-5-OEt Et 3-Me-4-CF₃-5-Br
U-4a 2-Br-5-C(O)CF₃ Et 3,5-di-Me-4-CF₃
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
U-4a 2-Me-5-Ac Et 3-Me-4,5-di-CF₃
U-4a 2-Me-5-(U-3b) Et 3-Me-4-CF₃-5-OMe
U-4a 2-Me-5-CF₂H Et 3-Me-4-OMe-5-F
U-4a 2-Me-5-CN Et 3-Me-4-OMe-5-Cl
U-4a 2-Me-5-Et Et 3-Me-4-OMe-5-Br
U-4a 2-Me-5-OCF₂H Et 3,5-di-Me-4-OMe
U-4a 2-Me-5-OEt Et 3-Me-4-OMe-5-CF₃
U-4a 2-Me-5-C(O)CF₃ Et 3-Me-4,5-di-OMe
U-4a 2-CF₃-5-Ac Et 2-CF₃-3,4-di-F
U-4a 2-CF₃-5-(U-3b) Et 2-CF₃-3-F-4-Cl
U-4a 2-CF₃-5-CF₂H Et 2-CF₃-3-F-4-Br
U-4a 2-CF₃-5-CN Et 2-CF₃-3-F-4-Me
U-4a 2-CF₃-5-Et Et 2,4-di-CF₃-3-F
U-4a 2-CF₃-5-OCF₂H Et 2-CF₃-3-F-4-OMe
U-4a 2-CF₃-5-OEt Et 2-CF₃-3-Cl-4-F
U-4a 2-CF₃-5-C(O)CF₃ Et 2-CF₃-3,4-di-Cl
U-4a 2-OMe-5-Ac Et 2-CF₃-3-Cl-4-Br
U-4a 2-OMe-5-(U-3b) Et 2-CF₃-3-Cl-4-Me
U-4a 2-OMe-5-CF₂H Et 2,4-di-CF₃-3-Cl
U-4a 2-OMe-5-CN Et 2-CF₃-3-Cl-4-OMe
U-4a 2-OMe-5-Et Et 2-CF₃-3-Br-4-F
U-4a 2-OMe-5-OCF₂H Et 2-CF₃-3-Br-4-Cl
U-4a 2-OMe-5-OEt Et 2-CF₃-3,4-di-Br
U-4a 2-OMe-5-C(O)CF₃ Et 2-CF₃-3-Br-4-Me
U-4a 2-OCF₃-5-Ac Et 2,4-di-CF₃-3-Br
U-4a 2-OCF₃-5-(U-3b) Et 2-CF₃-3-Br-4-OMe
U-4a 2-OCF₃-5-CF₂H Et 2-CF₃-3-Me-4-F
U-4a 2-OCF₃-5-CN Et 2-CF₃-3-Me-4-Cl
U-4a 2-OCF₃-5-Et Et 2-CF₃-3-Me-4-Br
U-4a 2-OCF₃-5-OCF₂H Et 2-CF₃-3,4-di-Me
U-4a 2-OCF₃-5-OEt Et 2,4-di-CF₃-3-Me
U-4a 2-OCF₃-5-C(O)CF₃ Et 2-CF₃-3-Me-4-OMe
U-4a 3-F-4-Ac Et 2,3-di-CF₃-4-F
U-4a 3-F-4-(U-3b) Et 2,3-di-CF₃-4-Cl
U-4a 3-F-4-CF₂H Et 2,3-di-CF₃-4-Br
U-4a 3-F-4-CN Et 2,3-di-CF₃-4-Me
U-4a 3-F-4-Et Et 2,3,4-tri-CF₃
U-4a 3-F-4-OCF₂H Et 2,3-di-CF₃-4-OMe
U-4a 3-F-4-OEt Et 2-CF₃-3-OMe-4-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
U-4a 3-F-4-C(O)CF₃ Et 2-CF₃-3-OMe-4-Cl
U-4a 3-Cl-4-Ac Et 2-CF₃-3-OMe-4-Br
U-4a 3-Cl-4-(U-3b) Et 2-CF₃-3-OMe-4-Me
U-4a 3-Cl-4-CF₂H Et 2,4-di-CF₃-3-OMe
U-4a 3-Cl-4-CN Et 2-CF₃-3,4-di-OMe
U-4a 3-Cl-4-Et Et 2-CF₃-3,5-di-F
U-4a 3-Cl-4-OCF₂H Et 2-CF₃-3-F-5-Cl
U-4a 3-Cl-4-OEt Et 2-CF₃-3-F-5-Br
U-4a 3-Cl-4-C(O)CF₃ Et 2-CF₃-3-F-5-Me
U-4a 3-Br-4-Ac Et 2,5-di-CF₃-3-F
U-4a 3-Br-4-(U-3b) Et 2-CF₃-3-F-5-OMe
U-4a 3-Br-4-CF₂H Et 2-CF₃-3-Cl-5-F
U-4a 3-Br-4-CN Et 2-CF₃-3,5-di-Cl
U-4a 3-Br-4-Et Et 2-CF₃-3-Cl-5-Br
U-4a 3-Br-4-OCF₂H Et 2-CF₃-3-Cl-5-Me
U-4a 3-Br-4-OEt Et 2,5-di-CF₃-3-Cl
U-4a 3-Br-4-C(O)CF₃ Et 2-CF₃-3-Cl-5-OMe
U-4a 3-Me-4-Ac Et 2-CF₃-3-Br-5-F
U-4a 3-Me-4-(U-3b) Et 2-CF₃-3-Br-5-Cl
U-4a 3-Me-4-CF₂H Et 2-CF₃-3,5-di-Br
U-4a 3-Me-4-CN Et 2-CF₃-3-Br-5-Me
U-4a 3-Me-4-Et Et 2,5-di-CF₃-3-Br
U-4a 3-Me-4-OCF₂H Et 2-CF₃-3-Br-5-OMe
U-4a 3-Me-4-OEt Et 2-CF₃-3-Me-5-F
U-4a 3-Me-4-C(O)CF₃ Et 2-CF₃-3-Me-5-Cl
U-4a 3-CF₃-4-Ac Et 2-CF₃-3-Me-5-Br
U-4a 3-CF₃-4-(U-3b) Et 2-CF₃-3,5-di-Me
U-4a 3-CF₃-4-CF₂H Et 2,5-di-CF₃-3-Me
U-4a 3-CF₃-4-CN Et 2-CF₃-3-Me-5-OMe
U-4a 3-CF₃-4-Et Et 2,3-di-CF₃-5-F
U-4a 3-CF₃-4-OCF₂H Et 2,3-di-CF₃-5-Cl
U-4a 3-CF₃-4-OEt Et 2,3-di-CF₃-5-Br
U-4a 3-CF₃-4-C(O)CF₃ Et 2,3-di-CF₃-5-Me
U-4a 3-OMe-4-Ac Et 2,3,5-tri-CF₃
U-4a 3-OMe-4-(U-3b) Et 2,3-di-CF₃-5-OMe
U-4a 3-OMe-4-CF₂H Et 2-CF₃-3-OMe-5-F
U-4a 3-OMe-4-CN Et 2-CF₃-3-OMe-5-Cl
U-4a 3-OMe-4-Et Et 2-CF₃-3-OMe-5-Br
U-4a 3-OMe-4-OCF₂H Et 2-CF₃-3-OMe-5-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
U-4a 3-OMe-4-OEt Et 2,5-di-CF₃-3-OMe
U-4a 3-OMe-4-C(O)CF₃ Et 2-CF₃-3,5-di-OMe
U-4a 3-OCF₃-4-Ac Et 2-CF₃-4,5-di-F
U-4a 3-OCF₃-4-(U-3b) Et 2-CF₃-4-F-5-Cl
U-4a 3-OCF₃-4-CF₂H Et 2-CF₃-4-F-5-Br
U-4a 3-OCF₃-4-CN Et 2-CF₃-4-F-5-Me
U-4a 3-OCF₃-4-Et Et 2,5-di-CF₃-4-F
U-4a 3-OCF₃-4-OCF₂H Et 2-CF₃-4-F-5-OMe
U-4a 3-OCF₃-4-OEt Et 2-CF₃-4-Cl-5-F
U-4a 3-OCF₃-4-C(O)CF₃ Et 2-CF₃-4,5-di-Cl
U-4a 3-F-5-Ac Et 2-CF₃-4-Cl-5-Br
U-4a 3-F-5-(U-3b) Et 2-CF₃-4-Cl-5-Me
U-4a 3-F-5-CF₂H Et 2,5-di-CF₃-4-Cl
U-4a 3-F-5-CN Et 2-CF₃-4-Cl-5-OMe
U-4a 3-F-5-Et Et 2-CF₃-4-Br-5-F
U-4a 3-F-5-OCF₂H Et 2-CF₃-4-Br-5-Cl
U-4a 3-F-5-OEt Et 2-CF₃-4,5-di-Br
U-4a 3-F-5-C(O)CF₃ Et 2-CF₃-4-Br-5-Me
U-4a 3-Cl-5-Ac Et 2,5-di-CF₃-4-Br
U-4a 3-Cl-5-(U-3b) Et 2-CF₃-4-Br-5-OMe
U-4a 3-Cl-5-CF₂H Et 2-CF₃-4-Me-5-F
U-4a 3-Cl-5-CN Et 2-CF₃-4-Me-5-Cl
U-4a 3-Cl-5-Et Et 2-CF₃-4-Me-5-Br
U-4a 3-Cl-5-OCF₂H Et 2-CF₃-4,5-di-Me
U-4a 3-Cl-5-OEt Et 2,5-di-CF₃-4-Me
U-4a 3-Cl-5-C(O)CF₃ Et 2-CF₃-4-Me-5-OMe
U-4a 3-Br-5-Ac Et 2,4-di-CF₃-5-F
U-4a 3-Br-5-(U-3b) Et 2,4-di-CF₃-5-Cl
U-4a 3-Br-5-CF₂H Et 2,4-di-CF₃-5-Br
U-4a 3-Br-5-CN Et 2,4-di-CF₃-5-Me
U-4a 3-Br-5-Et Et 2,4,5-tri-CF₃
U-4a 3-Br-5-OCF₂H Et 2,4-di-CF₃-5-OMe
U-4a 3-Br-5-OEt Et 2-CF₃-4-OMe-5-F
U-4a 3-Br-5-C(O)CF₃ Et 2-CF₃-4-OMe-5-Cl
U-4a 3-Me-5-Ac Et 2-CF₃-4-OMe-5-Br
U-4a 3-Me-5-(U-3b) Et 2-CF₃-4-OMe-5-Me
U-4a 3-Me-5-CF₂H Et 2,5-di-CF₃-4-OMe
U-4a 3-Me-5-CN Et 2-CF₃-4,5-di-OMe
U-4a 3-Me-5-Et Et 3-CF₃-4,5-di-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
U-4a 3-Me-5-OCF₂H Et 3-CF₃-4-F-5-Cl
U-4a 3-Me-5-OEt Et 3-CF₃-4-F-5-Br
U-4a 3-Me-5-C(O)CF₃ Et 3-CF₃-4-F-5-Me
U-4a 3-CF₃-5-Ac Et 3,5-di-CF₃-4-F
U-4a 3-CF₃-5-(U-3b) Et 3-CF₃-4-F-5-OMe
U-4a 3-CF₃-5-CF₂H Et 3-CF₃-4-Cl-5-F
U-4a 3-CF₃-5-CN Et 3-CF₃-4,5-di-Cl
U-4a 3-CF₃-5-Et Et 3-CF₃-4-Cl-5-Br
U-4a 3-CF₃-5-OCF₂H Et 3-CF₃-4-Cl-5-Me
U-4a 3-CF₃-5-OEt Et 3,5-di-CF₃-4-Cl
U-4a 3-CF₃-5-C(O)CF₃ Et 3-CF₃-4-Cl-5-OMe
U-4a 3-OMe-5-Ac Et 3-CF₃-4-Br-5-F
U-4a 3-OMe-5-(U-3b) Et 3-CF₃-4-Br-5-Cl
U-4a 3-OMe-5-CF₂H Et 3-CF₃-4,5-di-Br
U-4a 3-OMe-5-CN Et 3-CF₃-4-Br-5-Me
U-4a 3-OMe-5-Et Et 3,5-di-CF₃-4-Br
U-4a 3-OMe-5-OCF₂H Et 3-CF₃-4-Br-5-OMe
U-4a 3-OMe-5-OEt Et 3-CF₃-4-Me-5-F
U-4a 3-OMe-5-C(O)CF₃ Et 3-CF₃-4-Me-5-Cl
U-4a 3-OCF₃-5-Ac Et 3-CF₃-4-Me-5-Br
U-4a 3-OCF₃-5-(U-3b) Et 3-CF₃-4,5-di-Me
U-4a 3-OCF₃-5-CF₂H Et 3,5-di-CF₃-4-Me
U-4a 3-OCF₃-5-CN Et 3-CF₃-4-Me-5-OMe
U-4a 3-OCF₃-5-Et Et 3,4-di-CF₃-5-F
U-4a 3-OCF₃-5-OCF₂H Et 3,4-di-CF₃-5-Cl
U-4a 3-OCF₃-5-OEt Et 3,4-di-CF₃-5-Br
U-4a 3-OCF₃-5-C(O)CF₃ Et 3,4-di-CF₃-5-Me
U-4a 2-Ac-3-F Et 3,4,5-tri-CF₃
U-4a 2-Ac-3-Cl Et 3,4-di-CF₃-5-OMe
U-4a 2-Ac-3-Br Et 3-CF₃-4-OMe-5-F
U-4a 2-Ac-3-Me Et 3-CF₃-4-OMe-5-Cl
U-4a 2-Ac-3-CF₃ Et 3-CF₃-4-OMe-5-Br
U-4a 2-Ac-3-OMe Et 3-CF₃-4-OMe-5-Me
U-4a 2-Ac-3-OCF₃ Et 3,5-di-CF₃-4-OMe
U-4a 2-(U-3b)-3-F Et 3-CF₃-4,5-di-OMe
U-4a 2-(U-3b)-3-Cl Et 2-OMe-3,4-di-F
U-4a 2-(U-3b)-3-Br Et 2-OMe-3-F-4-Cl
U-4a 2-(U-3b)-3-Me Et 2-OMe-3-F-4-Br
U-4a 2-(U-3b)-3-CF₃ Et 2-OMe-3-F-4-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
U-4a 2-(U-3b)-3-OMe Et 2-OMe-3-F-4-CF₃
U-4a 2-(U-3b)-3-OCF₃ Et 2,4-di-OMe-3-F
U-4a 2-CF₂H-3-F Et 2-OMe-3-Cl-4-F
U-4a 2-CF₂H-3-Cl Et 2-OMe-3,4-di-Cl
U-4a 2-CF₂H-3-Br Et 2-OMe-3-Cl-4-Br
U-4a 2-CF₂H-3-Me Et 2-OMe-3-Cl-4-Me
U-4a 2-CF₂H-3-CF₃ Et 2-OMe-3-Cl-4-CF₃
U-4a 2-CF₂H-3-OMe Et 2,4-di-OMe-3-Cl
U-4a 2-CF₂H-3-OCF₃ Et 2-OMe-3-Br-4-F
U-4a 2-CN-3-F Et 2-OMe-3-Br-4-Cl
U-4a 2-CN-3-Cl Et 2-OMe-3,4-di-Br
U-4a 2-CN-3-Br Et 2-OMe-3-Br-4-Me
U-4a 2-CN-3-Me Et 2-OMe-3-Br-4-CF₃
U-4a 2-CN-3-CF₃ Et 2,4-di-OMe-3-Br
U-4a 2-CN-3-OMe Et 2-OMe-3-Me-4-F
U-4a 2-CN-3-OCF₃ Et 2-OMe-3-Me-4-Cl
U-4a 2-Et-3-F Et 2-OMe-3-Me-4-Br
U-4a 2-Et-3-Cl Et 2-OMe-3,4-di-Me
U-4a 2-Et-3-Br Et 2-OMe-3-Me-4-CF₃
U-4a 2-Et-3-Me Et 2,4-di-OMe-3-Me
U-4a 2-Et-3-CF₃ Et 2-OMe-3-CF₃-4-F
U-4a 2-Et-3-OMe Et 2-OMe-3-CF₃-4-Cl
U-4a 2-Et-3-OCF₃ Et 2-OMe-3-CF₃-4-Br
U-4a 2-OCF₂H-3-F Et 2-OMe-3-CF₃-4-Me
U-4a 2-OCF₂H-3-Cl Et 2-OMe-3,4-di-CF₃
U-4a 2-OCF₂H-3-Br Et 2,4-di-OMe-3-CF₃
U-4a 2-OCF₂H-3-Me Et 2,3-di-OMe-4-F
U-4a 2-OCF₂H-3-CF₃ Et 2,3-di-OMe-4-Cl
U-4a 2-OCF₂H-3-OMe Et 2,3-di-OMe-4-Br
U-4a 2-OCF₂H-3-OCF₃ Et 2,3-di-OMe-4-Me
U-4a 2-OEt-3-F Et 2,3-di-OMe-4-CF₃
U-4a 2-OEt-3-Cl Et 2,3,4-tri-OMe
U-4a 2-OEt-3-Br Et 2-OMe-3,5-di-F
U-4a 2-OEt-3-Me Et 2-OMe-3-F-5-Cl
U-4a 2-OEt-3-CF₃ Et 2-OMe-3-F-5-Br
U-4a 2-OEt-3-OMe Et 2-OMe-3-F-5-Me
U-4a 2-OEt-3-OCF₃ Et 2-OMe-3-F-5-CF₃
U-4a 2-C(O)CF₃-3-F Et 2,5-di-OMe-3-F
U-4a 2-C(O)CF₃-3-Cl Et 2-OMe-3-Cl-5-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
U-4a 2-C(O)CF₃-3-Br Et 2-OMe-3,5-di-Cl
U-4a 2-C(O)CF₃-3-Me Et 2-OMe-3-Cl-5-Br
U-4a 2-C(O)CF₃-3-CF₃ Et 2-OMe-3-Cl-5-Me
U-4a 2-C(O)CF₃-3-OMe Et 2-OMe-3-Cl-5-CF₃
U-4a 2-C(O)CF₃-3-OCF₃ Et 2,5-di-OMe-3-Cl
U-4a 2-Ac-4-F Et 2-OMe-3-Br-5-F
U-4a 2-Ac-4-Cl Et 2-OMe-3-Br-5-Cl
U-4a 2-Ac-4-Br Et 2-OMe-3,5-di-Br
U-4a 2-Ac-4-Me Et 2-OMe-3-Br-5-Me
U-4a 2-Ac-4-CF₃ Et 2-OMe-3-Br-5-CF₃
U-4a 2-Ac-4-OMe Et 2,5-di-OMe-3-Br
U-4a 2-Ac-4-OCF₃ Et 2-OMe-3-Me-5-F
U-4a 2-(U-3b)-4-F Et 2-OMe-3-Me-5-Cl
U-4a 2-(U-3b)-4-Cl Et 2-OMe-3-Me-5-Br
U-4a 2-(U-3b)-4-Br Et 2-OMe-3,5-di-Me
U-4a 2-(U-3b)-4-Me Et 2-OMe-3-Me-5-CF₃
U-4a 2-(U-3b)-4-CF₃ Et 2,5-di-OMe-3-Me
U-4a 2-(U-3b)-4-OMe Et 2-OMe-3-CF₃-5-F
U-4a 2-(U-3b)-4-OCF₃ Et 2-OMe-3-CF₃-5-Cl
U-4a 2-CF₂H-4-F Et 2-OMe-3-CF₃-5-Br
U-4a 2-CF₂H-4-Cl Et 2-OMe-3-CF₃-5-Me
U-4a 2-CF₂H-4-Br Et 2-OMe-3,5-di-CF₃
U-4a 2-CF₂H-4-Me Et 2,5-di-OMe-3-CF₃
U-4a 2-CF₂H-4-CF₃ Et 2,3-di-OMe-5-F
U-4a 2-CF₂H-4-OMe Et 2,3-di-OMe-5-Cl
U-4a 2-CF₂H-4-OCF₃ Et 2,3-di-OMe-5-Br
U-4a 2-CN-4-F Et 2,3-di-OMe-5-Me
U-4a 2-CN-4-Cl Et 2,3-di-OMe-5-CF₃
U-4a 2-CN-4-Br Et 2,3,5-tri-OMe
U-4a 2-CN-4-Me Et 2-OMe-4,5-di-F
U-4a 2-CN-4-CF₃ Et 2-OMe-4-F-5-Cl
U-4a 2-CN-4-OMe Et 2-OMe-4-F-5-Br
U-4a 2-CN-4-OCF₃ Et 2-OMe-4-F-5-Me
U-4a 2-Et-4-F Et 2-OMe-4-F-5-CF₃
U-4a 2-Et-4-Cl Et 2,5-di-OMe-4-F
U-4a 2-Et-4-Br Et 2-OMe-4-Cl-5-F
U-4a 2-Et-4-Me Et 2-OMe-4,5-di-Cl
U-4a 2-Et-4-CF₃ Et 2-OMe-4-Cl-5-Br
U-4a 2-Et-4-OMe Et 2-OMe-4-Cl-5-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
U-4a 2-Et-4-OCF₃ Et 2-OMe-4-Cl-5-CF₃
U-4a 2-OCF₂H-4-F Et 2,5-di-OMe-4-Cl
U-4a 2-OCF₂H-4-Cl Et 2-OMe-4-Br-5-F
U-4a 2-OCF₂H-4-Br Et 2-OMe-4-Br-5-Cl
U-4a 2-OCF₂H-4-Me Et 2-OMe-4,5-di-Br
U-4a 2-OCF₂H-4-CF₃ Et 2-OMe-4-Br-5-Me
U-4a 2-OCF₂H-4-OMe Et 2-OMe-4-Br-5-CF₃
U-4a 2-OCF₂H-4-OCF₃ Et 2,5-di-OMe-4-Br
U-4a 2-OEt-4-F Et 2-OMe-4-Me-5-F
U-4a 2-OEt-4-Cl Et 2-OMe-4-Me-5-Cl
U-4a 2-OEt-4-Br Et 2-OMe-4-Me-5-Br
U-4a 2-OEt-4-Me Et 2-OMe-4,5-di-Me
U-4a 2-OEt-4-CF₃ Et 2-OMe-4-Me-5-CF₃
U-4a 2-OEt-4-OMe Et 2,5-di-OMe-4-Me
U-4a 2-OEt-4-OCF₃ Et 2-OMe-4-CF₃-5-F
U-4a 2-C(O)CF₃-4-F Et 2-OMe-4-CF₃-5-Cl
U-4a 2-C(O)CF₃-4-Cl Et 2-OMe-4-CF₃-5-Br
U-4a 2-C(O)CF₃-4-Br Et 2-OMe-4-CF₃-5-Me
U-4a 2-C(O)CF₃-4-Me Et 2-OMe-4,5-di-CF₃
U-4a 2-C(O)CF₃-4-CF₃ Et 2,5-di-OMe-4-CF₃
U-4a 2-C(O)CF₃-4-OMe Et 2,4-di-OMe-5-F
U-4a 2-C(O)CF₃-4-OCF₃ Et 2,4-di-OMe-5-Cl
U-4a 2-Ac-5-F Et 2,4-di-OMe-5-Br
U-4a 2-Ac-5-Cl Et 2,4-di-OMe-5-Me
U-4a 2-Ac-5-Br Et 2,4-di-OMe-5-CF₃
U-4a 2-Ac-5-Me Et 2,4,5-tri-OMe
U-4a 2-Ac-5-CF₃ Et 3-OMe-4,5-di-F
U-4a 2-Ac-5-OMe Et 3-OMe-4-F-5-Cl
U-4a 2-Ac-5-OCF₃ Et 3-OMe-4-F-5-Br
U-4a 2-(U-3b)-5-F Et 3-OMe-4-F-5-Me
U-4a 2-(U-3b)-5-Cl Et 3-OMe-4-F-5-CF₃
U-4a 2-(U-3b)-5-Br Et 3,5-di-OMe-4-F
U-4a 2-(U-3b)-5-Me Et 3-OMe-4-Cl-5-F
U-4a 2-(U-3b)-5-CF₃ Et 3-OMe-4,5-di-Cl
U-4a 2-(U-3b)-5-OMe Et 3-OMe-4-Cl-5-Br
U-4a 2-(U-3b)-5-OCF₃ Et 3-OMe-4-Cl-5-Me
U-4a 2-CF₂H-5-F Et 3-OMe-4-Cl-5-CF₃
U-4a 2-CF₂H-5-Cl Et 3,5-di-OMe-4-Cl
U-4a 2-CF₂H-5-Br Et 3-OMe-4-Br-5-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
U-4a 2-CF₂H-5-Me Et 3-OMe-4-Br-5-Cl
U-4a 2-CF₂H-5-CF₃ Et 3-OMe-4,5-di-Br
U-4a 2-CF₂H-5-OMe Et 3-OMe-4-Br-5-Me
U-4a 2-CF₂H-5-OCF₃ Et 3-OMe-4-Br-5-CF₃
U-4a 2-CN-5-F Et 3,5-di-OMe-4-Br
U-4a 2-CN-5-Cl Et 3-OMe-4-Me-5-F
U-4a 2-CN-5-Br Et 3-OMe-4-Me-5-Cl
U-4a 2-CN-5-Me Et 3-OMe-4-Me-5-Br
U-4a 2-CN-5-CF₃ Et 3-OMe-4,5-di-Me
U-4a 2-CN-5-OMe Et 3-OMe-4-Me-5-CF₃
U-4a 2-CN-5-OCF₃ Et 3,5-di-OMe-4-Me
U-4a 2-Et-5-F Et 3-OMe-4-CF₃-5-F
U-4a 2-Et-5-Cl Et 3-OMe-4-CF₃-5-Cl
U-4a 2-Et-5-Br Et 3-OMe-4-CF₃-5-Br
U-4a 2-Et-5-Me Et 3-OMe-4-CF₃-5-Me
U-4a 2-Et-5-CF₃ Et 3-OMe-4,5-di-CF₃
U-4a 2-Et-5-OMe Et 3,5-di-OMe-4-CF₃
U-4a 2-Et-5-OCF₃ Et 3,4-di-OMe-5-F
U-4a 2-OCF₂H-5-F Et 3,4-di-OMe-5-Cl
U-4a 2-OCF₂H-5-Cl Et 3,4-di-OMe-5-Br
U-4a 2-OCF₂H-5-Br Et 3,4-di-OMe-5-Me
U-4a 2-OCF₂H-5-Me Et 3,4-di-OMe-5-CF₃
U-4a 2-OCF₂H-5-CF₃ Et 3,4,5-tri-OMe
U-4a 2-OCF₂H-5-OMe cPr 2,3,4-tri-F
U-4a 2-OCF₂H-5-OCF₃ cPr 2,3-di-F-4-Cl
U-4a 2-OEt-5-F cPr 2,3-di-F-4-Br
U-4a 2-OEt-5-Cl cPr 2,3-di-F-4-Me
U-4a 2-OEt-5-Br cPr 2,3-di-F-4-CF₃
U-4a 2-OEt-5-Me cPr 2,3-di-F-4-OMe
U-4a 2-OEt-5-CF₃ cPr 2,4-di-F-3-Cl
U-4a 2-OEt-5-OMe cPr 2-F-3,4-di-Cl
U-4a 2-OEt-5-OCF₃ cPr 2-F-3-Cl-4-Br
U-4a 2-C(O)CF₃-5-F cPr 2-F-3-Cl-4-Me
U-4a 2-C(O)CF₃-5-Cl cPr 2-F-3-Cl-4-CF₃
U-4a 2-C(O)CF₃-5-Br cPr 2-F-3-Cl-4-OMe
U-4a 2-C(O)CF₃-5-Me cPr 2,4-di-F-3-Br
U-4a 2-C(O)CF₃-5-CF₃ cPr 2-F-3-Br-4-Cl
U-4a 2-C(O)CF₃-5-OMe cPr 2-F-3,4-di-Br
U-4a 2-C(O)CF₃-5-OCF₃ cPr 2-F-3-Br-4-Me
U-4a 3-Ac-4-F cPr 2-F-3-Br-4-CF₃
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
U-4a 3-Ac-4-Cl cPr 2-F-3-Br-4-OMe
U-4a 3-Ac-4-Br cPr 2,4-di-F-3-Me
U-4a 3-Ac-4-Me cPr 2-F-3-Me-4-Cl
U-4a 3-Ac-4-CF₃ cPr 2-F-3-Me-4-Br
U-4a 3-Ac-4-OMe cPr 2-F-3,4-di-Me
U-4a 3-Ac-4-OCF₃ cPr 2-F-3-Me-4-CF₃
U-4a 3-(U-3b)-4-F cPr 2-F-3-Me-4-OMe
U-4a 3-(U-3b)-4-Cl cPr 2,4-di-F-3-CF₃
U-4a 3-(U-3b)-4-Br cPr 2-F-3-CF₃-4-Cl
U-4a 3-(U-3b)-4-Me cPr 2-F-3-CF₃-4-Br
U-4a 3-(U-3b)-4-CF₃ cPr 2-F-3-CF₃-4-Me
U-4a 3-(U-3b)-4-OMe cPr 2-F-3,4-di-CF₃
U-4a 3-(U-3b)-4-OCF₃ cPr 2-F-3-CF₃-4-OMe
U-4a 3-CF₂H-4-F cPr 2,4-di-F-3-OMe
U-4a 3-CF₂H-4-Cl cPr 2-F-3-OMe-4-Cl
U-4a 3-CF₂H-4-Br cPr 2-F-3-OMe-4-Br
U-4a 3-CF₂H-4-Me cPr 2-F-3-OMe-4-Me
U-4a 3-CF₂H-4-CF₃ cPr 2-F-3-OMe-4-CF₃
U-4a 3-CF₂H-4-OMe cPr 2-F-3,4-di-OMe
U-4a 3-CF₂H-4-OCF₃ cPr 2,3,5-tri-F
U-4a 3-CN-4-F cPr 2,3-di-F-5-Cl
U-4a 3-CN-4-Cl cPr 2,3-di-F-5-Br
U-4a 3-CN-4-Br cPr 2,3-di-F-5-Me
U-4a 3-CN-4-Me cPr 2,3-di-F-5-CF₃
U-4a 3-CN-4-CF₃ cPr 2,3-di-F-5-OMe
U-4a 3-CN-4-OMe cPr 2,5-di-F-3-Cl
U-4a 3-CN-4-OCF₃ cPr 2-F-3,5-di-Cl
U-4a 3-Et-4-F cPr 2-F-3-Cl-5-Br
U-4a 3-Et-4-Cl cPr 2-F-3-Cl-5-Me
U-4a 3-Et-4-Br cPr 2-F-3-Cl-5-CF₃
U-4a 3-Et-4-Me cPr 2-F-3-Cl-5-OMe
U-4a 3-Et-4-CF₃ cPr 2,5-di-F-3-Br
U-4a 3-Et-4-OMe cPr 2-F-3-Br-5-Cl
U-4a 3-Et-4-OCF₃ cPr 2-F-3,5-di-Br
U-4a 3-OCF₂H-4-F cPr 2-F-3-Br-5-Me
U-4a 3-OCF₂H-4-Cl cPr 2-F-3-Br-5-CF₃
U-4a 3-OCF₂H-4-Br cPr 2-F-3-Br-5-OMe
U-4a 3-OCF₂H-4-Me cPr 2,5-di-F-3-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
U-4a 3-OCF₂H-4-CF₃ cPr 2-F-3-Me-5-Cl
U-4a 3-OCF₂H-4-OMe cPr 2-F-3-Me-5-Br
U-4a 3-OCF₂H-4-OCF₃ cPr 2-F-3,5-di-Me
U-4a 3-OEt-4-F cPr 2-F-3-Me-5-CF₃
U-4a 3-OEt-4-Cl cPr 2-F-3-Me-5-OMe
U-4a 3-OEt-4-Br cPr 2,5-di-F-3-CF₃
U-4a 3-OEt-4-Me cPr 2-F-3-CF₃-5-Cl
U-4a 3-OEt-4-CF₃ cPr 2-F-3-CF₃-5-Br
U-4a 3-OEt-4-OMe cPr 2-F-3-CF₃-5-Me
U-4a 3-OEt-4-OCF₃ cPr 2-F-3,5-di-CF₃
U-4a 3-C(O)CF₃-4-F cPr 2-F-3-CF₃-5-OMe
U-4a 3-C(O)CF₃-4-Cl cPr 2,5-di-F-3-OMe
U-4a 3-C(O)CF₃-4-Br cPr 2-F-3-OMe-5-Cl
U-4a 3-C(O)CF₃-4-Me cPr 2-F-3-OMe-5-Br
U-4a 3-C(O)CF₃-4-CF₃ cPr 2-F-3-OMe-5-Me
U-4a 3-C(O)CF₃-4-OMe cPr 2-F-3-OMe-5-CF₃
U-4a 3-C(O)CF₃-4-OCF₃ cPr 2-F-3,5-di-OMe
U-4a 3-Ac-5-F cPr 2,4,5-tri-F
U-4a 3-Ac-5-Cl cPr 2,4-di-F-5-Cl
U-4a 3-Ac-5-Br cPr 2,4-di-F-5-Br
U-4a 3-Ac-5-Me cPr 2,4-di-F-5-Me
U-4a 3-Ac-5-CF₃ cPr 2,4-di-F-5-CF₃
U-4a 3-Ac-5-OMe cPr 2,4-di-F-5-OMe
U-4a 3-Ac-5-OCF₃ cPr 2,5-di-F-4-Cl
U-4a 3-(U-3b)-5-F cPr 2-F-4,5-di-Cl
U-4a 3-(U-3b)-5-Cl cPr 2-F-4-Cl-5-Br
U-4a 3-(U-3b)-5-Br cPr 2-F-4-Cl-5-Me
U-4a 3-(U-3b)-5-Me cPr 2-F-4-Cl-5-CF₃
U-4a 3-(U-3b)-5-CF₃ cPr 2-F-4-Cl-5-OMe
U-4a 3-(U-3b)-5-OMe cPr 2,5-di-F-4-Br
U-4a 3-(U-3b)-5-OCF₃ cPr 2-F-4-Br-5-Cl
U-4a 3-CF₂H-5-F cPr 2-F-4,5-di-Br
U-4a 3-CF₂H-5-Cl cPr 2-F-4-Br-5-Me
U-4a 3-CF₂H-5-Br cPr 2-F-4-Br-5-CF₃
U-4a 3-CF₂H-5-Me cPr 2-F-4-Br-5-OMe
U-4a 3-CF₂H-5-CF₃ cPr 2,5-di-F-4-Me
U-4a 3-CF₂H-5-OMe cPr 2-F-4-Me-5-Cl
U-4a 3-CF₂H-5-OCF₃ cPr 2-F-4-Me-5-Br
U-4a 3-CN-5-F cPr 2-F-4,5-di-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
U-4a 3-CN-5-Cl cPr 2-F-4-Me-5-CF₃
U-4a 3-CN-5-Br cPr 2-F-4-Me-5-OMe
U-4a 3-CN-5-Me cPr 2,5-di-F-4-CF₃
U-4a 3-CN-5-CF₃ cPr 2-F-4-CF₃-5-Cl
U-4a 3-CN-5-OMe cPr 2-F-4-CF₃-5-Br
U-4a 3-CN-5-OCF₃ cPr 2-F-4-CF₃-5-Me
U-4a 3-Et-5-F cPr 2-F-4,5-di-CF₃
U-4a 3-Et-5-Cl cPr 2-F-4-CF₃-5-OMe
U-4a 3-Et-5-Br cPr 2,5-di-F-4-OMe
U-4a 3-Et-5-Me cPr 2-F-4-OMe-5-Cl
U-4a 3-Et-5-CF₃ cPr 2-F-4-OMe-5-Br
U-4a 3-Et-5-OMe cPr 2-F-4-OMe-5-Me
U-4a 3-Et-5-OCF₃ cPr 2-F-4-OMe-5-CF₃
U-4a 3-OCF₂H-5-F cPr 2-F-4,5-di-OMe
U-4a 3-OCF₂H-5-Cl cPr 3,4,5-tri-F
U-4a 3-OCF₂H-5-Br cPr 3,4-di-F-5-Cl
U-4a 3-OCF₂H-5-Me cPr 3,4-di-F-5-Br
U-4a 3-OCF₂H-5-CF₃ cPr 3,4-di-F-5-Me
U-4a 3-OCF₂H-5-OMe cPr 3,4-di-F-5-CF₃
U-4a 3-OCF₂H-5-OCF₃ cPr 3,4-di-F-5-OMe
U-4a 3-OEt-5-F cPr 3,5-di-F-4-Cl
U-4a 3-OEt-5-Cl cPr 3-F-4,5-di-Cl
U-4a 3-OEt-5-Br cPr 3-F-4-Cl-5-Br
U-4a 3-OEt-5-Me cPr 3-F-4-Cl-5-Me
U-4a 3-OEt-5-CF₃ cPr 3-F-4-Cl-5-CF₃
U-4a 3-OEt-5-OMe cPr 3-F-4-Cl-5-OMe
U-4a 3-OEt-5-OCF₃ cPr 3,5-di-F-4-Br
U-4a 3-C(O)CF₃-5-F cPr 3-F-4-Br-5-Cl
U-4a 3-C(O)CF₃-5-Cl cPr 3-F-4,5-di-Br
U-4a 3-C(O)CF₃-5-Br cPr 3-F-4-Br-5-Me
U-4a 3-C(O)CF₃-5-Me cPr 3-F-4-Br-5-CF₃
U-4a 3-C(O)CF₃-5-CF₃ cPr 3-F-4-Br-5-OMe
U-4a 3-C(O)CF₃-5-OMe cPr 3,5-di-F-4-Me
U-4a 3-C(O)CF₃-5-OCF₃ cPr 3-F-4-Me-5-Cl
CF₃ 2-F-3-Ac cPr 3-F-4-Me-5-Br
CF₃ 2-F-3-(U-3b) cPr 3-F-4,5-di-Me
CF₃ 2-F-3-CF₂H cPr 3-F-4-Me-5-CF₃
CF₃ 2-F-3-CN cPr 3-F-4-Me-5-OMe
CF₃ 2-F-3-Et cPr 3,5-di-F-4-CF₃
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
CF₃ 2-F-3-OCF₂H cPr 3-F-4-CF₃-5-Cl
CF₃ 2-F-3-OEt cPr 3-F-4-CF₃-5-Br
CF₃ 2-F-3-C(O)CF₃ cPr 3-F-4-CF₃-5-Me
CF₃ 2-Cl-3-Ac cPr 3-F-4,5-di-CF₃
CF₃ 2-Cl-3-(U-3b) cPr 3-F-4-CF₃-5-OMe
CF₃ 2-Cl-3-CF₂H cPr 3,5-di-F-4-OMe
CF₃ 2-Cl-3-CN cPr 3-F-4-OMe-5-Cl
CF₃ 2-Cl-3-Et cPr 3-F-4-OMe-5-Br
CF₃ 2-Cl-3-OCF₂H cPr 3-F-4-OMe-5-Me
CF₃ 2-Cl-3-OEt cPr 3-F-4-OMe-5-CF₃
CF₃ 2-Cl-3-C(O)CF₃ cPr 3-F-4,5-di-OMe
CF₃ 2-Br-3-Ac cPr 2-Cl-3,4-di-F
CF₃ 2-Br-3-(U-3b) cPr 2,4-di-Cl-3-F
CF₃ 2-Br-3-CF₂H cPr 2-Cl-3-F-4-Br
CF₃ 2-Br-3-CN cPr 2-Cl-3-F-4-Me
CF₃ 2-Br-3-Et cPr 2-Cl-3-F-4-CF₃
CF₃ 2-Br-3-OCF₂H cPr 2-Cl-3-F-4-OMe
CF₃ 2-Br-3-OEt cPr 2,3-di-Cl-4-F
CF₃ 2-Br-3-C(O)CF₃ cPr 2,3,4-tri-Cl
CF₃ 2-Me-3-Ac cPr 2,3-di-Cl-4-Br
CF₃ 2-Me-3-(U-3b) cPr 2,3-di-Cl-4-Me
CF₃ 2-Me-3-CF₂H cPr 2,3-di-Cl-4-CF₃
CF₃ 2-Me-3-CN cPr 2,3-di-Cl-4-OMe
CF₃ 2-Me-3-Et cPr 2-Cl-3-Br-4-F
CF₃ 2-Me-3-OCF₂H cPr 2,4-di-Cl-3-Br
CF₃ 2-Me-3-OEt cPr 2-Cl-3,4-di-Br
CF₃ 2-Me-3-C(O)CF₃ cPr 2-Cl-3-Br-4-Me
CF₃ 2-CF₃-3-Ac cPr 2-Cl-3-Br-4-CF₃
CF₃ 2-CF₃-3-(U-3b) cPr 2-Cl-3-Br-4-OMe
CF₃ 2-CF₃-3-CF₂H cPr 2-Cl-3-Me-4-F
CF₃ 2-CF₃-3-CN cPr 2,4-di-Cl-3-Me
CF₃ 2-CF₃-3-Et cPr 2-Cl-3-Me-4-Br
CF₃ 2-CF₃-3-OCF₂H cPr 2-Cl-3,4-di-Me
CF₃ 2-CF₃-3-OEt cPr 2-Cl-3-Me-4-CF₃
CF₃ 2-CF₃-3-C(O)CF₃ cPr 2-Cl-3-Me-4-OMe
CF₃ 2-OMe-3-Ac cPr 2-Cl-3-CF₃-4-F
CF₃ 2-OMe-3-(U-3b) cPr 2,4-di-Cl-3-CF₃
CF₃ 2-OMe-3-CF₂H cPr 2-Cl-3-CF₃-4-Br
CF₃ 2-OMe-3-CN cPr 2-Cl-3-CF₃-4-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
CF₃ 2-OMe-3-Et cPr 2-Cl-3,4-di-CF₃
CF₃ 2-OMe-3-OCF₂H cPr 2-Cl-3-CF₃-4-OMe
CF₃ 2-OMe-3-OEt cPr 2-Cl-3-OMe-4-F
CF₃ 2-OMe-3-C(O)CF₃ cPr 2,4-di-Cl-3-OMe
CF₃ 2-OCF₃-3-Ac cPr 2-Cl-3-OMe-4-Br
CF₃ 2-OCF₃-3-(U-3b) cPr 2-Cl-3-OMe-4-Me
CF₃ 2-OCF₃-3-CF₂H cPr 2-Cl-3-OMe-4-CF₃
CF₃ 2-OCF₃-3-CN cPr 2-Cl-3,4-di-OMe
CF₃ 2-OCF₃-3-Et cPr 2-Cl-3,5-di-F
CF₃ 2-OCF₃-3-OCF₂H cPr 2,5-di-Cl-3-F
CF₃ 2-OCF₃-3-OEt cPr 2-Cl-3-F-5-Br
CF₃ 2-OCF₃-3-C(O)CF₃ cPr 2-Cl-3-F-5-Me
CF₃ 2-F-4-Ac cPr 2-Cl-3-F-5-CF₃
CF₃ 2-F-4-(U-3b) cPr 2-Cl-3-F-5-OMe
CF₃ 2-F-4-CF₂H cPr 2,3-di-Cl-5-F
CF₃ 2-F-4-CN cPr 2,3,5-tri-Cl
CF₃ 2-F-4-Et cPr 2,3-di-Cl-5-Br
CF₃ 2-F-4-OCF₂H cPr 2,3-di-Cl-5-Me
CF₃ 2-F-4-OEt cPr 2,3-di-Cl-5-CF₃
CF₃ 2-F-4-C(O)CF₃ cPr 2,3-di-Cl-5-OMe
CF₃ 2-Cl-4-Ac cPr 2-Cl-3-Br-5-F
CF₃ 2-Cl-4-(U-3b) cPr 2,5-di-Cl-3-Br
CF₃ 2-Cl-4-CF₂H cPr 2-Cl-3,5-di-Br
CF₃ 2-Cl-4-CN cPr 2-Cl-3-Br-5-Me
CF₃ 2-Cl-4-Et cPr 2-Cl-3-Br-5-CF₃
CF₃ 2-Cl-4-OCF₂H cPr 2-Cl-3-Br-5-OMe
CF₃ 2-Cl-4-OEt cPr 2-Cl-3-Me-5-F
CF₃ 2-Cl-4-C(O)CF₃ cPr 2,5-di-Cl-3-Me
CF₃ 2-Br-4-Ac cPr 2-Cl-3-Me-5-Br
CF₃ 2-Br-4-(U-3b) cPr 2-Cl-3,5-di-Me
CF₃ 2-Br-4-CF₂H cPr 2-Cl-3-Me-5-CF₃
CF₃ 2-Br-4-CN cPr 2-Cl-3-Me-5-OMe
CF₃ 2-Br-4-Et cPr 2-Cl-3-CF₃-5-F
CF₃ 2-Br-4-OCF₂H cPr 2,5-di-Cl-3-CF₃
CF₃ 2-Br-4-OEt cPr 2-Cl-3-CF₃-5-Br
CF₃ 2-Br-4-C(O)CF₃ cPr 2-Cl-3-CF₃-5-Me
CF₃ 2-Me-4-Ac cPr 2-Cl-3,5-di-CF₃
CF₃ 2-Me-4-(U-3b) cPr 2-Cl-3-CF₃-5-OMe
CF₃ 2-Me-4-CF₂H cPr 2-Cl-3-OMe-5-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
CF₃ 2-Me-4-CN cPr 2,5-di-Cl-3-OMe
CF₃ 2-Me-4-Et cPr 2-Cl-3-OMe-5-Br
CF₃ 2-Me-4-OCF₂H cPr 2-Cl-3-OMe-5-Me
CF₃ 2-Me-4-OEt cPr 2-Cl-3-OMe-5-CF₃
CF₃ 2-Me-4-C(O)CF₃ cPr 2-Cl-3,5-di-OMe
CF₃ 2-CF₃-4-Ac cPr 2-Cl-4,5-di-F
CF₃ 2-CF₃-4-(U-3b) cPr 2,5-di-Cl-4-F
CF₃ 2-CF₃-4-CF₂H cPr 2-Cl-4-F-5-Br
CF₃ 2-CF₃-4-CN cPr 2-Cl-4-F-5-Me
CF₃ 2-CF₃-4-Et cPr 2-Cl-4-F-5-CF₃
CF₃ 2-CF₃-4-OCF₂H cPr 2-Cl-4-F-5-OMe
CF₃ 2-CF₃-4-OEt cPr 2,4-di-Cl-5-F
CF₃ 2-CF₃-4-C(O)CF₃ cPr 2,4,5-tri-Cl
CF₃ 2-OMe-4-Ac cPr 2,4-di-Cl-5-Br
CF₃ 2-OMe-4-(U-3b) cPr 2,4-di-Cl-5-Me
CF₃ 2-OMe-4-CF₂H cPr 2,4-di-Cl-5-CF₃
CF₃ 2-OMe-4-CN cPr 2,4-di-Cl-5-OMe
CF₃ 2-OMe-4-Et cPr 2-Cl-4-Br-5-F
CF₃ 2-OMe-4-OCF₂H cPr 2,5-di-Cl-4-Br
CF₃ 2-OMe-4-OEt cPr 2-Cl-4,5-di-Br
CF₃ 2-OMe-4-C(O)CF₃ cPr 2-Cl-4-Br-5-Me
CF₃ 2-OCF₃-4-Ac cPr 2-Cl-4-Br-5-CF₃
CF₃ 2-OCF₃-4-(U-3b) cPr 2-Cl-4-Br-5-OMe
CF₃ 2-OCF₃-4-CF₂H cPr 2-Cl-4-Me-5-F
CF₃ 2-OCF₃-4-CN cPr 2,5-di-Cl-4-Me
CF₃ 2-OCF₃-4-Et cPr 2-Cl-4-Me-5-Br
CF₃ 2-OCF₃-4-OCF₂H cPr 2-Cl-4,5-di-Me
CF₃ 2-OCF₃-4-OEt cPr 2-Cl-4-Me-5-CF₃
CF₃ 2-OCF₃-4-C(O)CF₃ cPr 2-Cl-4-Me-5-OMe
CF₃ 2-F-5-Ac cPr 2-Cl-4-CF₃-5-F
CF₃ 2-F-5-(U-3b) cPr 2,5-di-Cl-4-CF₃
CF₃ 2-F-5-CF₂H cPr 2-Cl-4-CF₃-5-Br
CF₃ 2-F-5-CN cPr 2-Cl-4-CF₃-5-Me
CF₃ 2-F-5-Et cPr 2-Cl-4,5-di-CF₃
CF₃ 2-F-5-OCF₂H cPr 2-Cl-4-CF₃-5-OMe
CF₃ 2-F-5-OEt cPr 2-Cl-4-OMe-5-F
CF₃ 2-F-5-C(O)CF₃ cPr 2,5-di-Cl-4-OMe
CF₃ 2-Cl-5-Ac cPr 2-Cl-4-OMe-5-Br
CF₃ 2-Cl-5-(U-3b) cPr 2-Cl-4-OMe-5-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
CF₃ 2-Cl-5-CF₂H cPr 2-Cl-4-OMe-5-CF₃
CF₃ 2-Cl-5-CN cPr 2-Cl-4,5-di-OMe
CF₃ 2-Cl-5-Et cPr 3-Cl-4,5-di-F
CF₃ 2-Cl-5-OCF₂H cPr 3,5-di-Cl-4-F
CF₃ 2-Cl-5-OEt cPr 3-Cl-4-F-5-Br
CF₃ 2-Cl-5-C(O)CF₃ cPr 3-Cl-4-F-5-Me
CF₃ 2-Br-5-Ac cPr 3-Cl-4-F-5-CF₃
CF₃ 2-Br-5-(U-3b) cPr 3-Cl-4-F-5-OMe
CF₃ 2-Br-5-CF₂H cPr 3,4-di-Cl-5-F
CF₃ 2-Br-5-CN cPr 3,4,5-tri-Cl
CF₃ 2-Br-5-Et cPr 3,4-di-Cl-5-Br
CF₃ 2-Br-5-OCF₂H cPr 3,4-di-Cl-5-Me
CF₃ 2-Br-5-OEt cPr 3,4-di-Cl-5-CF₃
CF₃ 2-Br-5-C(O)CF₃ cPr 3,4-di-Cl-5-OMe
CF₃ 2-Me-5-Ac cPr 3-Cl-4-Br-5-F
CF₃ 2-Me-5-(U-3b) cPr 3,5-di-Cl-4-Br
CF₃ 2-Me-5-CF₂H cPr 3-Cl-4,5-di-Br
CF₃ 2-Me-5-CN cPr 3-Cl-4-Br-5-Me
CF₃ 2-Me-5-Et cPr 3-Cl-4-Br-5-CF₃
CF₃ 2-Me-5-OCF₂H cPr 3-Cl-4-Br-5-OMe
CF₃ 2-Me-5-OEt cPr 3-Cl-4-Me-5-F
CF₃ 2-Me-5-C(O)CF₃ cPr 3,5-di-Cl-4-Me
CF₃ 2-CF₃-5-Ac cPr 3-Cl-4-Me-5-Br
CF₃ 2-CF₃-5-(U-3b) cPr 3-Cl-4,5-di-Me
CF₃ 2-CF₃-5-CF₂H cPr 3-Cl-4-Me-5-CF₃
CF₃ 2-CF₃-5-CN cPr 3-Cl-4-Me-5-OMe
CF₃ 2-CF₃-5-Et cPr 3-Cl-4-CF₃-5-F
CF₃ 2-CF₃-5-OCF₂H cPr 3,5-di-Cl-4-CF₃
CF₃ 2-CF₃-5-OEt cPr 3-Cl-4-CF₃-5-Br
CF₃ 2-CF₃-5-C(O)CF₃ cPr 3-Cl-4-CF₃-5-Me
CF₃ 2-OMe-5-Ac cPr 3-Cl-4,5-di-CF₃
CF₃ 2-OMe-5-(U-3b) cPr 3-Cl-4-CF₃-5-OMe
CF₃ 2-OMe-5-CF₂H cPr 3-Cl-4-OMe-5-F
CF₃ 2-OMe-5-CN cPr 3,5-di-Cl-4-OMe
CF₃ 2-OMe-5-Et cPr 3-Cl-4-OMe-5-Br
CF₃ 2-OMe-5-OCF₂H cPr 3-Cl-4-OMe-5-Me
CF₃ 2-OMe-5-OEt cPr 3-Cl-4-OMe-5-CF₃
CF₃ 2-OMe-5-C(O)CF₃ cPr 3-Cl-4,5-di-OMe
CF₃ 2-OCF₃-5-Ac cPr 2-Br-3,4-di-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
CF₃ 2-OCF₃-5-(U-3b) cPr 2-Br-3-F-4-Cl
CF₃ 2-OCF₃-5-CF₂H cPr 2,4-di-Br-3-F
CF₃ 2-OCF₃-5-CN cPr 2-Br-3-F-4-Me
CF₃ 2-OCF₃-5-Et cPr 2-Br-3-F-4-CF₃
CF₃ 2-OCF₃-5-OCF₂H cPr 2-Br-3-F-4-OMe
CF₃ 2-OCF₃-5-OEt cPr 2-Br-3-Cl-4-F
CF₃ 2-OCF₃-5-C(O)CF₃ cPr 2-Br-3,4-di-Cl
CF₃ 3-F-4-Ac cPr 2,4-di-Br-3-Cl
CF₃ 3-F-4-(U-3b) cPr 2-Br-3-Cl-4-Me
CF₃ 3-F-4-CF₂H cPr 2-Br-3-Cl-4-CF₃
CF₃ 3-F-4-CN cPr 2-Br-3-Cl-4-OMe
CF₃ 3-F-4-Et cPr 2,3-di-Br-4-F
CF₃ 3-F-4-OCF₂H cPr 2,3-di-Br-4-Cl
CF₃ 3-F-4-OEt cPr 2,3,4-tri-Br
CF₃ 3-F-4-C(O)CF₃ cPr 2,3-di-Br-4-Me
CF₃ 3-Cl-4-Ac cPr 2,3-di-Br-4-CF₃
CF₃ 3-Cl-4-(U-3b) cPr 2,3-di-Br-4-OMe
CF₃ 3-Cl-4-CF₂H cPr 2-Br-3-Me-4-F
CF₃ 3-Cl-4-CN cPr 2-Br-3-Me-4-Cl
CF₃ 3-Cl-4-Et cPr 2,4-di-Br-3-Me
CF₃ 3-Cl-4-OCF₂H cPr 2-Br-3,4-di-Me
CF₃ 3-Cl-4-OEt cPr 2-Br-3-Me-4-CF₃
CF₃ 3-Cl-4-C(O)CF₃ cPr 2-Br-3-Me-4-OMe
CF₃ 3-Br-4-Ac cPr 2-Br-3-CF₃-4-F
CF₃ 3-Br-4-(U-3b) cPr 2-Br-3-CF₃-4-Cl
CF₃ 3-Br-4-CF₂H cPr 2,4-di-Br-3-CF₃
CF₃ 3-Br-4-CN cPr 2-Br-3-CF₃-4-Me
CF₃ 3-Br-4-Et cPr 2-Br-3,4-di-CF₃
CF₃ 3-Br-4-OCF₂H cPr 2-Br-3-CF₃-4-OMe
CF₃ 3-Br-4-OEt cPr 2-Br-3-OMe-4-F
CF₃ 3-Br-4-C(O)CF₃ cPr 2-Br-3-OMe-4-Cl
CF₃ 3-Me-4-Ac cPr 2,4-di-Br-3-OMe
CF₃ 3-Me-4-(U-3b) cPr 2-Br-3-OMe-4-Me
CF₃ 3-Me-4-CF₂H cPr 2-Br-3-OMe-4-CF₃
CF₃ 3-Me-4-CN cPr 2-Br-3,4-di-OMe
CF₃ 3-Me-4-Et cPr 2-Br-3,5-di-F
CF₃ 3-Me-4-OCF₂H cPr 2-Br-3-F-5-Cl
CF₃ 3-Me-4-OEt cPr 2,5-di-Br-3-F
CF₃ 3-Me-4-C(O)CF₃ cPr 2-Br-3-F-5-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
CF₃ 3-CF₃-4-Ac cPr 2-Br-3-F-5-CF₃
CF₃ 3-CF₃-4-(U-3b) cPr 2-Br-3-F-5-OMe
CF₃ 3-CF₃-4-CF₂H cPr 2-Br-3-Cl-5-F
CF₃ 3-CF₃-4-CN cPr 2-Br-3,5-di-Cl
CF₃ 3-CF₃-4-Et cPr 2,5-di-Br-3-Cl
CF₃ 3-CF₃-4-OCF₂H cPr 2-Br-3-Cl-5-Me
CF₃ 3-CF₃-4-OEt cPr 2-Br-3-Cl-5-CF₃
CF₃ 3-CF₃-4-C(O)CF₃ cPr 2-Br-3-Cl-5-OMe
CF₃ 3-OMe-4-Ac cPr 2,3-di-Br-5-F
CF₃ 3-OMe-4-(U-3b) cPr 2,3-di-Br-5-Cl
CF₃ 3-OMe-4-CF₂H cPr 2,3,5-tri-Br
CF₃ 3-OMe-4-CN cPr 2,3-di-Br-5-Me
CF₃ 3-OMe-4-Et cPr 2,3-di-Br-5-CF₃
CF₃ 3-OMe-4-OCF₂H cPr 2,3-di-Br-5-OMe
CF₃ 3-OMe-4-OEt cPr 2-Br-3-Me-5-F
CF₃ 3-OMe-4-C(O)CF₃ cPr 2-Br-3-Me-5-Cl
CF₃ 3-OCF₃-4-Ac cPr 2,5-di-Br-3-Me
CF₃ 3-OCF₃-4-(U-3b) cPr 2-Br-3,5-di-Me
CF₃ 3-OCF₃-4-CF₂H cPr 2-Br-3-Me-5-CF₃
CF₃ 3-OCF₃-4-CN cPr 2-Br-3-Me-5-OMe
CF₃ 3-OCF₃-4-Et cPr 2-Br-3-CF₃-5-F
CF₃ 3-OCF₃-4-OCF₂H cPr 2-Br-3-CF₃-5-Cl
CF₃ 3-OCF₃-4-OEt cPr 2,5-di-Br-3-CF₃
CF₃ 3-OCF₃-4-C(O)CF₃ cPr 2-Br-3-CF₃-5-Me
CF₃ 3-F-5-Ac cPr 2-Br-3,5-di-CF₃
CF₃ 3-F-5-(U-3b) cPr 2-Br-3-CF₃-5-OMe
CF₃ 3-F-5-CF₂H cPr 2-Br-3-OMe-5-F
CF₃ 3-F-5-CN cPr 2-Br-3-OMe-5-Cl
CF₃ 3-F-5-Et cPr 2,5-di-Br-3-OMe
CF₃ 3-F-5-OCF₂H cPr 2-Br-3-OMe-5-Me
CF₃ 3-F-5-OEt cPr 2-Br-3-OMe-5-CF₃
CF₃ 3-F-5-C(O)CF₃ cPr 2-Br-3,5-di-OMe
CF₃ 3-Cl-5-Ac cPr 2-Br-4,5-di-F
CF₃ 3-Cl-5-(U-3b) cPr 2-Br-4-F-5-Cl
CF₃ 3-Cl-5-CF₂H cPr 2,5-di-Br-4-F
CF₃ 3-Cl-5-CN cPr 2-Br-4-F-5-Me
CF₃ 3-Cl-5-Et cPr 2-Br-4-F-5-CF₃
CF₃ 3-Cl-5-OCF₂H cPr 2-Br-4-F-5-OMe
CF₃ 3-Cl-5-OEt cPr 2-Br-4-Cl-5-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
CF₃ 3-Cl-5-C(O)CF₃ cPr 2-Br-4,5-di-Cl
CF₃ 3-Br-5-Ac cPr 2,5-di-Br-4-Cl
CF₃ 3-Br-5-(U-3b) cPr 2-Br-4-Cl-5-Me
CF₃ 3-Br-5-CF₂H cPr 2-Br-4-Cl-5-CF₃
CF₃ 3-Br-5-CN cPr 2-Br-4-Cl-5-OMe
CF₃ 3-Br-5-Et cPr 2,4-di-Br-5-F
CF₃ 3-Br-5-OCF₂H cPr 2,4-di-Br-5-Cl
CF₃ 3-Br-5-OEt cPr 2,4,5-tri-Br
CF₃ 3-Br-5-C(O)CF₃ cPr 2,4-di-Br-5-Me
CF₃ 3-Me-5-Ac cPr 2,4-di-Br-5-CF₃
CF₃ 3-Me-5-(U-3b) cPr 2,4-di-Br-5-OMe
CF₃ 3-Me-5-CF₂H cPr 2-Br-4-Me-5-F
CF₃ 3-Me-5-CN cPr 2-Br-4-Me-5-Cl
CF₃ 3-Me-5-Et cPr 2,5-di-Br-4-Me
CF₃ 3-Me-5-OCF₂H cPr 2-Br-4,5-di-Me
CF₃ 3-Me-5-OEt cPr 2-Br-4-Me-5-CF₃
CF₃ 3-Me-5-C(O)CF₃ cPr 2-Br-4-Me-5-OMe
CF₃ 3-CF₃-5-Ac cPr 2-Br-4-CF₃-5-F
CF₃ 3-CF₃-5-(U-3b) cPr 2-Br-4-CF₃-5-Cl
CF₃ 3-CF₃-5-CF₂H cPr 2,5-di-Br-4-CF₃
CF₃ 3-CF₃-5-CN cPr 2-Br-4-CF₃-5-Me
CF₃ 3-CF₃-5-Et cPr 2-Br-4,5-di-CF₃
CF₃ 3-CF₃-5-OCF₂H cPr 2-Br-4-CF₃-5-OMe
CF₃ 3-CF₃-5-OEt cPr 2-Br-4-OMe-5-F
CF₃ 3-CF₃-5-C(O)CF₃ cPr 2-Br-4-OMe-5-Cl
CF₃ 3-OMe-5-Ac cPr 2,5-di-Br-4-OMe
CF₃ 3-OMe-5-(U-3b) cPr 2-Br-4-OMe-5-Me
CF₃ 3-OMe-5-CF₂H cPr 2-Br-4-OMe-5-CF₃
CF₃ 3-OMe-5-CN cPr 2-Br-4,5-di-OMe
CF₃ 3-OMe-5-Et cPr 3-Br-4,5-di-F
CF₃ 3-OMe-5-OCF₂H cPr 3-Br-4-F-5-Cl
CF₃ 3-OMe-5-OEt cPr 3,5-di-Br-4-F
CF₃ 3-OMe-5-C(O)CF₃ cPr 3-Br-4-F-5-Me
CF₃ 3-OCF₃-5-Ac cPr 3-Br-4-F-5-CF₃
CF₃ 3-OCF₃-5-(U-3b) cPr 3-Br-4-F-5-OMe
CF₃ 3-OCF₃-5-CF₂H cPr 3-Br-4-Cl-5-F
CF₃ 3-OCF₃-5-CN cPr 3-Br-4,5-di-Cl
CF₃ 3-OCF₃-5-Et cPr 3,5-di-Br-4-Cl
CF₃ 3-OCF₃-5-OCF₂H cPr 3-Br-4-Cl-5-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
CF₃ 3-OCF₃-5-OEt cPr 3-Br-4-Cl-5-CF₃
CF₃ 3-OCF₃-5-C(O)CF₃ cPr 3-Br-4-Cl-5-OMe
CF₃ 2-Ac-3-F cPr 3,4-di-Br-5-F
CF₃ 2-Ac-3-Cl cPr 3,4-di-Br-5-Cl
CF₃ 2-Ac-3-Br cPr 3,4,5-tri-Br
CF₃ 2-Ac-3-Me cPr 3,4-di-Br-5-Me
CF₃ 2-Ac-3-CF₃ cPr 3,4-di-Br-5-CF₃
CF₃ 2-Ac-3-OMe cPr 3,4-di-Br-5-OMe
CF₃ 2-Ac-3-OCF₃ cPr 3-Br-4-Me-5-F
CF₃ 2-(U-3b)-3-F cPr 3-Br-4-Me-5-Cl
CF₃ 2-(U-3b)-3-Cl cPr 3,5-di-Br-4-Me
CF₃ 2-(U-3b)-3-Br cPr 3-Br-4,5-di-Me
CF₃ 2-(U-3b)-3-Me cPr 3-Br-4-Me-5-CF₃
CF₃ 2-(U-3b)-3-CF₃ cPr 3-Br-4-Me-5-OMe
CF₃ 2-(U-3b)-3-OMe cPr 3-Br-4-CF₃-5-F
CF₃ 2-(U-3b)-3-OCF₃ cPr 3-Br-4-CF₃-5-Cl
CF₃ 2-CF₂H-3-F cPr 3,5-di-Br-4-CF₃
CF₃ 2-CF₂H-3-Cl cPr 3-Br-4-CF₃-5-Me
CF₃ 2-CF₂H-3-Br cPr 3-Br-4,5-di-CF₃
CF₃ 2-CF₂H-3-Me cPr 3-Br-4-CF₃-5-OMe
CF₃ 2-CF₂H-3-CF₃ cPr 3-Br-4-OMe-5-F
CF₃ 2-CF₂H-3-OMe cPr 3-Br-4-OMe-5-Cl
CF₃ 2-CF₂H-3-OCF₃ cPr 3,5-di-Br-4-OMe
CF₃ 2-CN-3-F cPr 3-Br-4-OMe-5-Me
CF₃ 2-CN-3-Cl cPr 3-Br-4-OMe-5-CF₃
CF₃ 2-CN-3-Br cPr 3-Br-4,5-di-OMe
CF₃ 2-CN-3-Me cPr 2-Me-3,4-di-F
CF₃ 2-CN-3-CF₃ cPr 2-Me-3-F-4-Cl
CF₃ 2-CN-3-OMe cPr 2-Me-3-F-4-Br
CF₃ 2-CN-3-OCF₃ cPr 2,4-di-Me-3-F
CF₃ 2-Et-3-F cPr 2-Me-3-F-4-CF₃
CF₃ 2-Et-3-Cl cPr 2-Me-3-F-4-OMe
CF₃ 2-Et-3-Br cPr 2-Me-3-Cl-4-F
CF₃ 2-Et-3-Me cPr 2-Me-3,4-di-Cl
CF₃ 2-Et-3-CF₃ cPr 2-Me-3-Cl-4-Br
CF₃ 2-Et-3-OMe cPr 2,4-di-Me-3-Cl
CF₃ 2-Et-3-OCF₃ cPr 2-Me-3-Cl-4-CF₃
CF₃ 2-OCF₂H-3-F cPr 2-Me-3-Cl-4-OMe
CF₃ 2-OCF₂H-3-Cl cPr 2-Me-3-Br-4-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
CF₃ 2-OCF₂H-3-Br cPr 2-Me-3-Br-4-Cl
CF₃ 2-OCF₂H-3-Me cPr 2-Me-3,4-di-Br
CF₃ 2-OCF₂H-3-CF₃ cPr 2,4-di-Me-3-Br
CF₃ 2-OCF₂H-3-OMe cPr 2-Me-3-Br-4-CF₃
CF₃ 2-OCF₂H-3-OCF₃ cPr 2-Me-3-Br-4-OMe
CF₃ 2-OEt-3-F cPr 2,3-di-Me-4-F
CF₃ 2-OEt-3-Cl cPr 2,3-di-Me-4-Cl
CF₃ 2-OEt-3-Br cPr 2,3-di-Me-4-Br
CF₃ 2-OEt-3-Me cPr 2,3,4-tri-Me
CF₃ 2-OEt-3-CF₃ cPr 2,3-di-Me-4-CF₃
CF₃ 2-OEt-3-OMe cPr 2,3-di-Me-4-OMe
CF₃ 2-OEt-3-OCF₃ cPr 2-Me-3-CF₃-4-F
CF₃ 2-C(O)CF₃-3-F cPr 2-Me-3-CF₃-4-Cl
CF₃ 2-C(O)CF₃-3-Cl cPr 2-Me-3-CF₃-4-Br
CF₃ 2-C(O)CF₃-3-Br cPr 2,4-di-Me-3-CF₃
CF₃ 2-C(O)CF₃-3-Me cPr 2-Me-3,4-di-CF₃
CF₃ 2-C(O)CF₃-3-CF₃ cPr 2-Me-3-CF₃-4-OMe
CF₃ 2-C(O)CF₃-3-OMe cPr 2-Me-3-OMe-4-F
CF₃ 2-C(O)CF₃-3-OCF₃ cPr 2-Me-3-OMe-4-Cl
CF₃ 2-Ac-4-F cPr 2-Me-3-OMe-4-Br
CF₃ 2-Ac-4-Cl cPr 2,4-di-Me-3-OMe
CF₃ 2-Ac-4-Br cPr 2-Me-3-OMe-4-CF₃
CF₃ 2-Ac-4-Me cPr 2-Me-3,4-di-OMe
CF₃ 2-Ac-4-CF₃ cPr 2-Me-3,5-di-F
CF₃ 2-Ac-4-OMe cPr 2-Me-3-F-5-Cl
CF₃ 2-Ac-4-OCF₃ cPr 2-Me-3-F-5-Br
CF₃ 2-(U-3b)-4-F cPr 2,5-di-Me-3-F
CF₃ 2-(U-3b)-4-Cl cPr 2-Me-3-F-5-CF₃
CF₃ 2-(U-3b)-4-Br cPr 2-Me-3-F-5-OMe
CF₃ 2-(U-3b)-4-Me cPr 2-Me-3-Cl-5-F
CF₃ 2-(U-3b)-4-CF₃ cPr 2-Me-3,5-di-Cl
CF₃ 2-(U-3b)-4-OMe cPr 2-Me-3-Cl-5-Br
CF₃ 2-(U-3b)-4-OCF₃ cPr 2,5-di-Me-3-Cl
CF₃ 2-CF₂H-4-F cPr 2-Me-3-Cl-5-CF₃
CF₃ 2-CF₂H-4-Cl cPr 2-Me-3-Cl-5-OMe
CF₃ 2-CF₂H-4-Br cPr 2-Me-3-Br-5-F
CF₃ 2-CF₂H-4-Me cPr 2-Me-3-Br-5-Cl
CF₃ 2-CF₂H-4-CF₃ cPr 2-Me-3,5-di-Br
CF₃ 2-CF₂H-4-OMe cPr 2,5-di-Me-3-Br
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
CF₃ 2-CF₂H-4-OCF₃ cPr 2-Me-3-Br-5-CF₃
CF₃ 2-CN-4-F cPr 2-Me-3-Br-5-OMe
CF₃ 2-CN-4-Cl cPr 2,3-di-Me-5-F
CF₃ 2-CN-4-Br cPr 2,3-di-Me-5-Cl
CF₃ 2-CN-4-Me cPr 2,3-di-Me-5-Br
CF₃ 2-CN-4-CF₃ cPr 2,3,5-tri-Me
CF₃ 2-CN-4-OMe cPr 2,3-di-Me-5-CF₃
CF₃ 2-CN-4-OCF₃ cPr 2,3-di-Me-5-OMe
CF₃ 2-Et-4-F cPr 2-Me-3-CF₃-5-F
CF₃ 2-Et-4-Cl cPr 2-Me-3-CF₃-5-Cl
CF₃ 2-Et-4-Br cPr 2-Me-3-CF₃-5-Br
CF₃ 2-Et-4-Me cPr 2,5-di-Me-3-CF₃
CF₃ 2-Et-4-CF₃ cPr 2-Me-3,5-di-CF₃
CF₃ 2-Et-4-OMe cPr 2-Me-3-CF₃-5-OMe
CF₃ 2-Et-4-OCF₃ cPr 2-Me-3-OMe-5-F
CF₃ 2-OCF₂H-4-F cPr 2-Me-3-OMe-5-Cl
CF₃ 2-OCF₂H-4-Cl cPr 2-Me-3-OMe-5-Br
CF₃ 2-OCF₂H-4-Br cPr 2,5-di-Me-3-OMe
CF₃ 2-OCF₂H-4-Me cPr 2-Me-3-OMe-5-CF₃
CF₃ 2-OCF₂H-4-CF₃ cPr 2-Me-3,5-di-OMe
CF₃ 2-OCF₂H-4-OMe cPr 2-Me-4,5-di-F
CF₃ 2-OCF₂H-4-OCF₃ cPr 2-Me-4-F-5-Cl
CF₃ 2-OEt-4-F cPr 2-Me-4-F-5-Br
CF₃ 2-OEt-4-Cl cPr 2,5-di-Me-4-F
CF₃ 2-OEt-4-Br cPr 2-Me-4-F-5-CF₃
CF₃ 2-OEt-4-Me cPr 2-Me-4-F-5-OMe
CF₃ 2-OEt-4-CF₃ cPr 2-Me-4-Cl-5-F
CF₃ 2-OEt-4-OMe cPr 2-Me-4,5-di-Cl
CF₃ 2-OEt-4-OCF₃ cPr 2-Me-4-Cl-5-Br
CF₃ 2-C(O)CF₃-4-F cPr 2,5-di-Me-4-Cl
CF₃ 2-C(O)CF₃-4-Cl cPr 2-Me-4-Cl-5-CF₃
CF₃ 2-C(O)CF₃-4-Br cPr 2-Me-4-Cl-5-OMe
CF₃ 2-C(O)CF₃-4-Me cPr 2-Me-4-Br-5-F
CF₃ 2-C(O)CF₃-4-CF₃ cPr 2-Me-4-Br-5-Cl
CF₃ 2-C(O)CF₃-4-OMe cPr 2-Me-4,5-di-Br
CF₃ 2-C(O)CF₃-4-OCF₃ cPr 2,5-di-Me-4-Br
CF₃ 2-Ac-5-F cPr 2-Me-4-Br-5-CF₃
CF₃ 2-Ac-5-Cl cPr 2-Me-4-Br-5-OMe
CF₃ 2-Ac-5-Br cPr 2,4-di-Me-5-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
CF₃ 2-Ac-5-Me cPr 2,4-di-Me-5-Cl
CF₃ 2-Ac-5-CF₃ cPr 2,4-di-Me-5-Br
CF₃ 2-Ac-5-OMe cPr 2,4,5-tri-Me
CF₃ 2-Ac-5-OCF₃ cPr 2,4-di-Me-5-CF₃
CF₃ 2-(U-3b)-5-F cPr 2,4-di-Me-5-OMe
CF₃ 2-(U-3b)-5-Cl cPr 2-Me-4-CF₃-5-F
CF₃ 2-(U-3b)-5-Br cPr 2-Me-4-CF₃-5-Cl
CF₃ 2-(U-3b)-5-Me cPr 2-Me-4-CF₃-5-Br
CF₃ 2-(U-3b)-5-CF₃ cPr 2,5-di-Me-4-CF₃
CF₃ 2-(U-3b)-5-OMe cPr 2-Me-4,5-di-CF₃
CF₃ 2-(U-3b)-5-OCF₃ cPr 2-Me-4-CF₃-5-OMe
CF₃ 2-CF₂H-5-F cPr 2-Me-4-OMe-5-F
CF₃ 2-CF₂H-5-Cl cPr 2-Me-4-OMe-5-Cl
CF₃ 2-CF₂H-5-Br cPr 2-Me-4-OMe-5-Br
CF₃ 2-CF₂H-5-Me cPr 2,5-di-Me-4-OMe
CF₃ 2-CF₂H-5-CF₃ cPr 2-Me-4-OMe-5-CF₃
CF₃ 2-CF₂H-5-OMe cPr 2-Me-4,5-di-OMe
CF₃ 2-CF₂H-5-OCF₃ cPr 3-Me-4,5-di-F
CF₃ 2-CN-5-F cPr 3-Me-4-F-5-Cl
CF₃ 2-CN-5-Cl cPr 3-Me-4-F-5-Br
CF₃ 2-CN-5-Br cPr 3,5-di-Me-4-F
CF₃ 2-CN-5-Me cPr 3-Me-4-F-5-CF₃
CF₃ 2-CN-5-CF₃ cPr 3-Me-4-F-5-OMe
CF₃ 2-CN-5-OMe cPr 3-Me-4-Cl-5-F
CF₃ 2-CN-5-OCF₃ cPr 3-Me-4,5-di-Cl
CF₃ 2-Et-5-F cPr 3-Me-4-Cl-5-Br
CF₃ 2-Et-5-Cl cPr 3,5-di-Me-4-Cl
CF₃ 2-Et-5-Br cPr 3-Me-4-Cl-5-CF₃
CF₃ 2-Et-5-Me cPr 3-Me-4-Cl-5-OMe
CF₃ 2-Et-5-CF₃ cPr 3-Me-4-Br-5-F
CF₃ 2-Et-5-OMe cPr 3-Me-4-Br-5-Cl
CF₃ 2-Et-5-OCF₃ cPr 3-Me-4,5-di-Br
CF₃ 2-OCF₂H-5-F cPr 3,5-di-Me-4-Br
CF₃ 2-OCF₂H-5-Cl cPr 3-Me-4-Br-5-CF₃
CF₃ 2-OCF₂H-5-Br cPr 3-Me-4-Br-5-OMe
CF₃ 2-OCF₂H-5-Me cPr 3,4-di-Me-5-F
CF₃ 2-OCF₂H-5-CF₃ cPr 3,4-di-Me-5-Cl
CF₃ 2-OCF₂H-5-OMe cPr 3,4-di-Me-5-Br
CF₃ 2-OCF₂H-5-OCF₃ cPr 3,4,5-tri-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
CF₃ 2-OEt-5-F cPr 3,4-di-Me-5-CF₃
CF₃ 2-OEt-5-Cl cPr 3,4-di-Me-5-OMe
CF₃ 2-OEt-5-Br cPr 3-Me-4-CF₃-5-F
CF₃ 2-OEt-5-Me cPr 3-Me-4-CF₃-5-Cl
CF₃ 2-OEt-5-CF₃ cPr 3-Me-4-CF₃-5-Br
CF₃ 2-OEt-5-OMe cPr 3,5-di-Me-4-CF₃
CF₃ 2-OEt-5-OCF₃ cPr 3-Me-4,5-di-CF₃
CF₃ 2-C(O)CF₃-5-F cPr 3-Me-4-CF₃-5-OMe
CF₃ 2-C(O)CF₃-5-Cl cPr 3-Me-4-OMe-5-F
CF₃ 2-C(O)CF₃-5-Br cPr 3-Me-4-OMe-5-Cl
CF₃ 2-C(O)CF₃-5-Me cPr 3-Me-4-OMe-5-Br
CF₃ 2-C(O)CF₃-5-CF₃ cPr 3,5-di-Me-4-OMe
CF₃ 2-C(O)CF₃-5-OMe cPr 3-Me-4-OMe-5-CF₃
CF₃ 2-C(O)CF₃-5-OCF₃ cPr 3-Me-4,5-di-OMe
CF₃ 3-Ac-4-F cPr 2-CF₃-3,4-di-F
CF₃ 3-Ac-4-Cl cPr 2-CF₃-3-F-4-Cl
CF₃ 3-Ac-4-Br cPr 2-CF₃-3-F-4-Br
CF₃ 3-Ac-4-Me cPr 2-CF₃-3-F-4-Me
CF₃ 3-Ac-4-CF₃ cPr 2,4-di-CF₃-3-F
CF₃ 3-Ac-4-OMe cPr 2-CF₃-3-F-4-OMe
CF₃ 3-Ac-4-OCF₃ cPr 2-CF₃-3-Cl-4-F
CF₃ 3-(U-3b)-4-F cPr 2-CF₃-3,4-di-Cl
CF₃ 3-(U-3b)-4-Cl cPr 2-CF₃-3-Cl-4-Br
CF₃ 3-(U-3b)-4-Br cPr 2-CF₃-3-Cl-4-Me
CF₃ 3-(U-3b)-4-Me cPr 2,4-di-CF₃-3-Cl
CF₃ 3-(U-3b)-4-CF₃ cPr 2-CF₃-3-Cl-4-OMe
CF₃ 3-(U-3b)-4-OMe cPr 2-CF₃-3-Br-4-F
CF₃ 3-(U-3b)-4-OCF₃ cPr 2-CF₃-3-Br-4-Cl
CF₃ 3-CF₂H-4-F cPr 2-CF₃-3,4-di-Br
CF₃ 3-CF₂H-4-Cl cPr 2-CF₃-3-Br-4-Me
CF₃ 3-CF₂H-4-Br cPr 2,4-di-CF₃-3-Br
CF₃ 3-CF₂H-4-Me cPr 2-CF₃-3-Br-4-OMe
CF₃ 3-CF₂H-4-CF₃ cPr 2-CF₃-3-Me-4-F
CF₃ 3-CF₂H-4-OMe cPr 2-CF₃-3-Me-4-Cl
CF₃ 3-CF₂H-4-OCF₃ cPr 2-CF₃-3-Me-4-Br
CF₃ 3-CN-4-F cPr 2-CF₃-3,4-di-Me
CF₃ 3-CN-4-Cl cPr 2,4-di-CF₃-3-Me
CF₃ 3-CN-4-Br cPr 2-CF₃-3-Me-4-OMe
CF₃ 3-CN-4-Me cPr 2,3-di-CF₃-4-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
CF₃ 3-CN-4-CF₃ cPr 2,3-di-CF₃-4-Cl
CF₃ 3-CN-4-OMe cPr 2,3-di-CF₃-4-Br
CF₃ 3-CN-4-OCF₃ cPr 2,3-di-CF₃-4-Me
CF₃ 3-Et-4-F cPr 2,3,4-tri-CF₃
CF₃ 3-Et-4-Cl cPr 2,3-di-CF₃-4-OMe
CF₃ 3-Et-4-Br cPr 2-CF₃-3-OMe-4-F
CF₃ 3-Et-4-Me cPr 2-CF₃-3-OMe-4-Cl
CF₃ 3-Et-4-CF₃ cPr 2-CF₃-3-OMe-4-Br
CF₃ 3-Et-4-OMe cPr 2-CF₃-3-OMe-4-Me
CF₃ 3-Et-4-OCF₃ cPr 2,4-di-CF₃-3-OMe
CF₃ 3-OCF₂H-4-F cPr 2-CF₃-3,4-di-OMe
CF₃ 3-OCF₂H-4-Cl cPr 2-CF₃-3,5-di-F
CF₃ 3-OCF₂H-4-Br cPr 2-CF₃-3-F-5-Cl
CF₃ 3-OCF₂H-4-Me cPr 2-CF₃-3-F-5-Br
CF₃ 3-OCF₂H-4-CF₃ cPr 2-CF₃-3-F-5-Me
CF₃ 3-OCF₂H-4-OMe cPr 2,5-di-CF₃-3-F
CF₃ 3-OCF₂H-4-OCF₃ cPr 2-CF₃-3-F-5-OMe
CF₃ 3-OEt-4-F cPr 2-CF₃-3-Cl-5-F
CF₃ 3-OEt-4-Cl cPr 2-CF₃-3,5-di-Cl
CF₃ 3-OEt-4-Br cPr 2-CF₃-3-Cl-5-Br
CF₃ 3-OEt-4-Me cPr 2-CF₃-3-Cl-5-Me
CF₃ 3-OEt-4-CF₃ cPr 2,5-di-CF₃-3-Cl
CF₃ 3-OEt-4-OMe cPr 2-CF₃-3-Cl-5-OMe
CF₃ 3-OEt-4-OCF₃ cPr 2-CF₃-3-Br-5-F
CF₃ 3-C(O)CF₃-4-F cPr 2-CF₃-3-Br-5-Cl
CF₃ 3-C(O)CF₃-4-Cl cPr 2-CF₃-3,5-di-Br
CF₃ 3-C(O)CF₃-4-Br cPr 2-CF₃-3-Br-5-Me
CF₃ 3-C(O)CF₃-4-Me cPr 2,5-di-CF₃-3-Br
CF₃ 3-C(O)CF₃-4-CF₃ cPr 2-CF₃-3-Br-5-OMe
CF₃ 3-C(O)CF₃-4-OMe cPr 2-CF₃-3-Me-5-F
CF₃ 3-C(O)CF₃-4-OCF₃ cPr 2-CF₃-3-Me-5-Cl
CF₃ 3-Ac-5-F cPr 2-CF₃-3-Me-5-Br
CF₃ 3-Ac-5-Cl cPr 2-CF₃-3,5-di-Me
CF₃ 3-Ac-5-Br cPr 2,5-di-CF₃-3-Me
CF₃ 3-Ac-5-Me cPr 2-CF₃-3-Me-5-OMe
CF₃ 3-Ac-5-CF₃ cPr 2,3-di-CF₃-5-F
CF₃ 3-Ac-5-OMe cPr 2,3-di-CF₃-5-Cl
CF₃ 3-Ac-5-OCF₃ cPr 2,3-di-CF₃-5-Br
CF₃ 3-(U-3b)-5-F cPr 2,3-di-CF₃-5-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
CF₃ 3-(U-3b)-5-Cl cPr 2,3,5-tri-CF₃
CF₃ 3-(U-3b)-5-Br cPr 2,3-di-CF₃-5-OMe
CF₃ 3-(U-3b)-5-Me cPr 2-CF₃-3-OMe-5-F
CF₃ 3-(U-3b)-5-CF₃ cPr 2-CF₃-3-OMe-5-Cl
CF₃ 3-(U-3b)-5-OMe cPr 2-CF₃-3-OMe-5-Br
CF₃ 3-(U-3b)-5-OCF₃ cPr 2-CF₃-3-OMe-5-Me
CF₃ 3-CF₂H-5-F cPr 2,5-di-CF₃-3-OMe
CF₃ 3-CF₂H-5-Cl cPr 2-CF₃-3,5-di-OMe
CF₃ 3-CF₂H-5-Br cPr 2-CF₃-4,5-di-F
CF₃ 3-CF₂H-5-Me cPr 2-CF₃-4-F-5-Cl
CF₃ 3-CF₂H-5-CF₃ cPr 2-CF₃-4-F-5-Br
CF₃ 3-CF₂H-5-OMe cPr 2-CF₃-4-F-5-Me
CF₃ 3-CF₂H-5-OCF₃ cPr 2,5-di-CF₃-4-F
CF₃ 3-CN-5-F cPr 2-CF₃-4-F-5-OMe
CF₃ 3-CN-5-Cl cPr 2-CF₃-4-Cl-5-F
CF₃ 3-CN-5-Br cPr 2-CF₃-4,5-di-Cl
CF₃ 3-CN-5-Me cPr 2-CF₃-4-Cl-5-Br
CF₃ 3-CN-5-CF₃ cPr 2-CF₃-4-Cl-5-Me
CF₃ 3-CN-5-OMe cPr 2,5-di-CF₃-4-Cl
CF₃ 3-CN-5-OCF₃ cPr 2-CF₃-4-Cl-5-OMe
CF₃ 3-Et-5-F cPr 2-CF₃-4-Br-5-F
CF₃ 3-Et-5-Cl cPr 2-CF₃-4-Br-5-Cl
CF₃ 3-Et-5-Br cPr 2-CF₃-4,5-di-Br
CF₃ 3-Et-5-Me cPr 2-CF₃-4-Br-5-Me
CF₃ 3-Et-5-CF₃ cPr 2,5-di-CF₃-4-Br
CF₃ 3-Et-5-OMe cPr 2-CF₃-4-Br-5-OMe
CF₃ 3-Et-5-OCF₃ cPr 2-CF₃-4-Me-5-F
CF₃ 3-OCF₂H-5-F cPr 2-CF₃-4-Me-5-Cl
CF₃ 3-OCF₂H-5-Cl cPr 2-CF₃-4-Me-5-Br
CF₃ 3-OCF₂H-5-Br cPr 2-CF₃-4,5-di-Me
CF₃ 3-OCF₂H-5-Me cPr 2,5-di-CF₃-4-Me
CF₃ 3-OCF₂H-5-CF₃ cPr 2-CF₃-4-Me-5-OMe
CF₃ 3-OCF₂H-5-OMe cPr 2,4-di-CF₃-5-F
CF₃ 3-OCF₂H-5-OCF₃ cPr 2,4-di-CF₃-5-Cl
CF₃ 3-OEt-5-F cPr 2,4-di-CF₃-5-Br
CF₃ 3-OEt-5-Cl cPr 2,4-di-CF₃-5-Me
CF₃ 3-OEt-5-Br cPr 2,4,5-tri-CF₃
CF₃ 3-OEt-5-Me cPr 2,4-di-CF₃-5-OMe
CF₃ 3-OEt-5-CF₃ cPr 2-CF₃-4-OMe-5-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
CF₃ 3-OEt-5-OMe cPr 2-CF₃-4-OMe-5-Cl
CF₃ 3-OEt-5-OCF₃ cPr 2-CF₃-4-OMe-5-Br
CF₃ 3-C(O)CF₃-5-F cPr 2-CF₃-4-OMe-5-Me
CF₃ 3-C(O)CF₃-5-Cl cPr 2,5-di-CF₃-4-OMe
CF₃ 3-C(O)CF₃-5-Br cPr 2-CF₃-4,5-di-OMe
CF₃ 3-C(O)CF₃-5-Me cPr 3-CF₃-4,5-di-F
CF₃ 3-C(O)CF₃-5-CF₃ cPr 3-CF₃-4-F-5-Cl
CF₃ 3-C(O)CF₃-5-OMe cPr 3-CF₃-4-F-5-Br
CF₃ 3-C(O)CF₃-5-OCF₃ cPr 3-CF₃-4-F-5-Me
cPr 2-F-3-Ac cPr 3,5-di-CF₃-4-F
cPr 2-F-3-(U-3b) cPr 3-CF₃-4-F-5-OMe
cPr 2-F-3-CF₂H cPr 3-CF₃-4-Cl-5-F
cPr 2-F-3-CN cPr 3-CF₃-4,5-di-Cl
cPr 2-F-3-Et cPr 3-CF₃-4-Cl-5-Br
cPr 2-F-3-OCF₂H cPr 3-CF₃-4-Cl-5-Me
cPr 2-F-3-OEt cPr 3,5-di-CF₃-4-Cl
cPr 2-F-3-C(O)CF₃ cPr 3-CF₃-4-Cl-5-OMe
cPr 2-Cl-3-Ac cPr 3-CF₃-4-Br-5-F
cPr 2-Cl-3-(U-3b) cPr 3-CF₃-4-Br-5-Cl
cPr 2-Cl-3-CF₂H cPr 3-CF₃-4,5-di-Br
cPr 2-Cl-3-CN cPr 3-CF₃-4-Br-5-Me
cPr 2-Cl-3-Et cPr 3,5-di-CF₃-4-Br
cPr 2-Cl-3-OCF₂H cPr 3-CF₃-4-Br-5-OMe
cPr 2-Cl-3-OEt cPr 3-CF₃-4-Me-5-F
cPr 2-Cl-3-C(O)CF₃ cPr 3-CF₃-4-Me-5-Cl
cPr 2-Br-3-Ac cPr 3-CF₃-4-Me-5-Br
cPr 2-Br-3-(U-3b) cPr 3-CF₃-4,5-di-Me
cPr 2-Br-3-CF₂H cPr 3,5-di-CF₃-4-Me
cPr 2-Br-3-CN cPr 3-CF₃-4-Me-5-OMe
cPr 2-Br-3-Et cPr 3,4-di-CF₃-5-F
cPr 2-Br-3-OCF₂H cPr 3,4-di-CF₃-5-Cl
cPr 2-Br-3-OEt cPr 3,4-di-CF₃-5-Br
cPr 2-Br-3-C(O)CF₃ cPr 3,4-di-CF₃-5-Me
cPr 2-Me-3-Ac cPr 3,4,5-tri-CF₃
cPr 2-Me-3-(U-3b) cPr 3,4-di-CF₃-5-OMe
cPr 2-Me-3-CF₂H cPr 3-CF₃-4-OMe-5-F
cPr 2-Me-3-CN cPr 3-CF₃-4-OMe-5-Cl
cPr 2-Me-3-Et cPr 3-CF₃-4-OMe-5-Br
cPr 2-Me-3-OCF₂H cPr 3-CF₃-4-OMe-5-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
cPr 2-Me-3-OEt cPr 3,5-di-CF₃-4-OMe
cPr 2-Me-3-C(O)CF₃ cPr 3-CF₃-4,5-di-OMe
cPr 2-CF₃-3-Ac cPr 2-OMe-3,4-di-F
cPr 2-CF₃-3-(U-3b) cPr 2-OMe-3-F-4-Cl
cPr 2-CF₃-3-CF₂H cPr 2-OMe-3-F-4-Br
cPr 2-CF₃-3-CN cPr 2-OMe-3-F-4-Me
cPr 2-CF₃-3-Et cPr 2-OMe-3-F-4-CF₃
cPr 2-CF₃-3-OCF₂H cPr 2,4-di-OMe-3-F
cPr 2-CF₃-3-OEt cPr 2-OMe-3-Cl-4-F
cPr 2-CF₃-3-C(O)CF₃ cPr 2-OMe-3,4-di-Cl
cPr 2-OMe-3-Ac cPr 2-OMe-3-Cl-4-Br
cPr 2-OMe-3-(U-3b) cPr 2-OMe-3-Cl-4-Me
cPr 2-OMe-3-CF₂H cPr 2-OMe-3-Cl-4-CF₃
cPr 2-OMe-3-CN cPr 2,4-di-OMe-3-Cl
cPr 2-OMe-3-Et cPr 2-OMe-3-Br-4-F
cPr 2-OMe-3-OCF₂H cPr 2-OMe-3-Br-4-Cl
cPr 2-OMe-3-OEt cPr 2-OMe-3,4-di-Br
cPr 2-OMe-3-C(O)CF₃ cPr 2-OMe-3-Br-4-Me
cPr 2-OCF₃-3-Ac cPr 2-OMe-3-Br-4-CF₃
cPr 2-OCF₃-3-(U-3b) cPr 2,4-di-OMe-3-Br
cPr 2-OCF₃-3-CF₂H cPr 2-OMe-3-Me-4-F
cPr 2-OCF₃-3-CN cPr 2-OMe-3-Me-4-Cl
cPr 2-OCF₃-3-Et cPr 2-OMe-3-Me-4-Br
cPr 2-OCF₃-3-OCF₂H cPr 2-OMe-3,4-di-Me
cPr 2-OCF₃-3-OEt cPr 2-OMe-3-Me-4-CF₃
cPr 2-OCF₃-3-C(O)CF₃ cPr 2,4-di-OMe-3-Me
cPr 2-F-4-Ac cPr 2-OMe-3-CF₃-4-F
cPr 2-F-4-(U-3b) cPr 2-OMe-3-CF₃-4-Cl
cPr 2-F-4-CF₂H cPr 2-OMe-3-CF₃-4-Br
cPr 2-F-4-CN cPr 2-OMe-3-CF₃-4-Me
cPr 2-F-4-Et cPr 2-OMe-3,4-di-CF₃
cPr 2-F-4-OCF₂H cPr 2,4-di-OMe-3-CF₃
cPr 2-F-4-OEt cPr 2,3-di-OMe-4-F
cPr 2-F-4-C(O)CF₃ cPr 2,3-di-OMe-4-Cl
cPr 2-Cl-4-Ac cPr 2,3-di-OMe-4-Br
cPr 2-Cl-4-(U-3b) cPr 2,3-di-OMe-4-Me
cPr 2-Cl-4-CF₂H cPr 2,3-di-OMe-4-CF₃
cPr 2-Cl-4-CN cPr 2,3,4-tri-OMe
cPr 2-Cl-4-Et cPr 2-OMe-3,5-di-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
cPr 2-Cl-4-OCF₂H cPr 2-OMe-3-F-5-Cl
cPr 2-Cl-4-OEt cPr 2-OMe-3-F-5-Br
cPr 2-Cl-4-C(O)CF₃ cPr 2-OMe-3-F-5-Me
cPr 2-Br-4-Ac cPr 2-OMe-3-F-5-CF₃
cPr 2-Br-4-(U-3b) cPr 2,5-di-OMe-3-F
cPr 2-Br-4-CF₂H cPr 2-OMe-3-Cl-5-F
cPr 2-Br-4-CN cPr 2-OMe-3,5-di-Cl
cPr 2-Br-4-Et cPr 2-OMe-3-Cl-5-Br
cPr 2-Br-4-OCF₂H cPr 2-OMe-3-Cl-5-Me
cPr 2-Br-4-OEt cPr 2-OMe-3-Cl-5-CF₃
cPr 2-Br-4-C(O)CF₃ cPr 2,5-di-OMe-3-Cl
cPr 2-Me-4-Ac cPr 2-OMe-3-Br-5-F
cPr 2-Me-4-(U-3b) cPr 2-OMe-3-Br-5-Cl
cPr 2-Me-4-CF₂H cPr 2-OMe-3,5-di-Br
cPr 2-Me-4-CN cPr 2-OMe-3-Br-5-Me
cPr 2-Me-4-Et cPr 2-OMe-3-Br-5-CF₃
cPr 2-Me-4-OCF₂H cPr 2,5-di-OMe-3-Br
cPr 2-Me-4-OEt cPr 2-OMe-3-Me-5-F
cPr 2-Me-4-C(O)CF₃ cPr 2-OMe-3-Me-5-Cl
cPr 2-CF₃-4-Ac cPr 2-OMe-3-Me-5-Br
cPr 2-CF₃-4-(U-3b) cPr 2-OMe-3,5-di-Me
cPr 2-CF₃-4-CF₂H cPr 2-OMe-3-Me-5-CF₃
cPr 2-CF₃-4-CN cPr 2,5-di-OMe-3-Me
cPr 2-CF₃-4-Et cPr 2-OMe-3-CF₃-5-F
cPr 2-CF₃-4-OCF₂H cPr 2-OMe-3-CF₃-5-Cl
cPr 2-CF₃-4-OEt cPr 2-OMe-3-CF₃-5-Br
cPr 2-CF₃-4-C(O)CF₃ cPr 2-OMe-3-CF₃-5-Me
cPr 2-OMe-4-Ac cPr 2-OMe-3,5-di-CF₃
cPr 2-OMe-4-(U-3b) cPr 2,5-di-OMe-3-CF₃
cPr 2-OMe-4-CF₂H cPr 2,3-di-OMe-5-F
cPr 2-OMe-4-CN cPr 2,3-di-OMe-5-Cl
cPr 2-OMe-4-Et cPr 2,3-di-OMe-5-Br
cPr 2-OMe-4-OCF₂H cPr 2,3-di-OMe-5-Me
cPr 2-OMe-4-OEt cPr 2,3-di-OMe-5-CF₃
cPr 2-OMe-4-C(O)CF₃ cPr 2,3,5-tri-OMe
cPr 2-OCF₃-4-Ac cPr 2-OMe-4,5-di-F
cPr 2-OCF₃-4-(U-3b) cPr 2-OMe-4-F-5-Cl
cPr 2-OCF₃-4-CF₂H cPr 2-OMe-4-F-5-Br
cPr 2-OCF₃-4-CN cPr 2-OMe-4-F-5-Me
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
cPr 2-OCF₃-4-Et cPr 2-OMe-4-F-5-CF₃
cPr 2-OCF₃-4-OCF₂H cPr 2,5-di-OMe-4-F
cPr 2-OCF₃-4-OEt cPr 2-OMe-4-Cl-5-F
cPr 2-OCF₃-4-C(O)CF₃ cPr 2-OMe-4,5-di-Cl
cPr 2-F-5-Ac cPr 2-OMe-4-Cl-5-Br
cPr 2-F-5-(U-3b) cPr 2-OMe-4-Cl-5-Me
cPr 2-F-5-CF₂H cPr 2-OMe-4-Cl-5-CF₃
cPr 2-F-5-CN cPr 2,5-di-OMe-4-Cl
cPr 2-F-5-Et cPr 2-OMe-4-Br-5-F
cPr 2-F-5-OCF₂H cPr 2-OMe-4-Br-5-Cl
cPr 2-F-5-OEt cPr 2-OMe-4,5-di-Br
cPr 2-F-5-C(O)CF₃ cPr 2-OMe-4-Br-5-Me
cPr 2-Cl-5-Ac cPr 2-OMe-4-Br-5-CF₃
cPr 2-Cl-5-(U-3b) cPr 2,5-di-OMe-4-Br
cPr 2-Cl-5-CF₂H cPr 2-OMe-4-Me-5-F
cPr 2-Cl-5-CN cPr 2-OMe-4-Me-5-Cl
cPr 2-Cl-5-Et cPr 2-OMe-4-Me-5-Br
cPr 2-Cl-5-OCF₂H cPr 2-OMe-4,5-di-Me
cPr 2-Cl-5-OEt cPr 2-OMe-4-Me-5-CF₃
cPr 2-Cl-5-C(O)CF₃ cPr 2,5-di-OMe-4-Me
cPr 2-Br-5-Ac cPr 2-OMe-4-CF₃-5-F
cPr 2-Br-5-(U-3b) cPr 2-OMe-4-CF₃-5-Cl
cPr 2-Br-5-CF₂H cPr 2-OMe-4-CF₃-5-Br
cPr 2-Br-5-CN cPr 2-OMe-4-CF₃-5-Me
cPr 2-Br-5-Et cPr 2-OMe-4,5-di-CF₃
cPr 2-Br-5-OCF₂H cPr 2,5-di-OMe-4-CF₃
cPr 2-Br-5-OEt cPr 2,4-di-OMe-5-F
cPr 2-Br-5-C(O)CF₃ cPr 2,4-di-OMe-5-Cl
cPr 2-Me-5-Ac cPr 2,4-di-OMe-5-Br
cPr 2-Me-5-(U-3b) cPr 2,4-di-OMe-5-Me
cPr 2-Me-5-CF₂H cPr 2,4-di-OMe-5-CF₃
cPr 2-Me-5-CN cPr 2,4,5-tri-OMe
cPr 2-Me-5-Et cPr 3-OMe-4,5-di-F
cPr 2-Me-5-OCF₂H cPr 3-OMe-4-F-5-Cl
cPr 2-Me-5-OEt cPr 3-OMe-4-F-5-Br
cPr 2-Me-5-C(O)CF₃ cPr 3-OMe-4-F-5-Me
cPr 2-CF₃-5-Ac cPr 3-OMe-4-F-5-CF₃
cPr 2-CF₃-5-(U-3b) cPr 3,5-di-OMe-4-F
cPr 2-CF₃-5-CF₂H cPr 3-OMe-4-Cl-5-F
−−−−−−−−−−− −−−−−−−−−−−−−
［第１表］（続き）［第１表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−
cPr 2-CF₃-5-CN cPr 3-OMe-4,5-di-Cl
cPr 2-CF₃-5-Et cPr 3-OMe-4-Cl-5-Br
cPr 2-CF₃-5-OCF₂H cPr 3-OMe-4-Cl-5-Me
cPr 2-CF₃-5-OEt cPr 3-OMe-4-Cl-5-CF₃
cPr 2-CF₃-5-C(O)CF₃ cPr 3,5-di-OMe-4-Cl
cPr 2-OMe-5-Ac cPr 3-OMe-4-Br-5-F
cPr 2-OMe-5-(U-3b) cPr 3-OMe-4-Br-5-Cl
cPr 2-OMe-5-CF₂H cPr 3-OMe-4,5-di-Br
cPr 2-OMe-5-CN cPr 3-OMe-4-Br-5-Me
cPr 2-OMe-5-Et cPr 3-OMe-4-Br-5-CF₃
cPr 2-OMe-5-OCF₂H cPr 3,5-di-OMe-4-Br
cPr 2-OMe-5-OEt cPr 3-OMe-4-Me-5-F
cPr 2-OMe-5-C(O)CF₃ cPr 3-OMe-4-Me-5-Cl
cPr 2-OCF₃-5-Ac cPr 3-OMe-4-Me-5-Br
cPr 2-OCF₃-5-(U-3b) cPr 3-OMe-4,5-di-Me
cPr 2-OCF₃-5-CF₂H cPr 3-OMe-4-Me-5-CF₃
cPr 2-OCF₃-5-CN cPr 3,5-di-OMe-4-Me
cPr 2-OCF₃-5-Et cPr 3-OMe-4-CF₃-5-F
cPr 2-OCF₃-5-OCF₂H cPr 3-OMe-4-CF₃-5-Cl
cPr 2-OCF₃-5-OEt cPr 3-OMe-4-CF₃-5-Br
cPr 2-OCF₃-5-C(O)CF₃ cPr 3-OMe-4-CF₃-5-Me
cPr 3-F-4-Ac cPr 3-OMe-4,5-di-CF₃
cPr 3-F-4-(U-3b) cPr 3,5-di-OMe-4-CF₃
cPr 3-F-4-CF₂H cPr 3,4-di-OMe-5-F
cPr 3-F-4-CN cPr 3,4-di-OMe-5-Cl
cPr 3-F-4-Et cPr 3,4-di-OMe-5-Br
cPr 3-F-4-OCF₂H cPr 3,4-di-OMe-5-Me
cPr 3-F-4-OEt cPr 3,4-di-OMe-5-CF₃
cPr 3-F-4-C(O)CF₃ cPr 3,4,5-tri-OMe
−−−−−−−−−−− −−−−−−−−−−−−−
［第２表］ [Table 1] [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
Me 2-F U-4a 3-Cl-5-OMe U-4f 2-F-5-OCF_Three
Me 2-Cl U-4a 3-Cl-5-OCF_Three    U-4f 2-Cl-5-F
Me 2-Br U-4a 3-Br-5-F U-4f 2,5-di-Cl
Me 2-Me U-4a 3-Br-5-Cl U-4f 2-Cl-5-Br
Me 2-CF_Three          U-4a 3,5-di-Br U-4f 2-Cl-5-Me
Me 2-OMe U-4a 3-Br-5-Me U-4f 2-Cl-5-CF_Three
Me 2-OCF_Three         U-4a 3-Br-5-CF_Three     U-4f 2-Cl-5-OMe
Me 3-F U-4a 3-Br-5-OMe U-4f 2-Cl-5-OCF_Three
Me 3-Cl U-4a 3-Br-5-OCF_Three    U-4f 2-Br-5-F
Me 3-Br U-4a 3-Me-5-F U-4f 2-Br-5-Cl
Me 3-Me U-4a 3-Me-5-Cl U-4f 2,5-di-Br
Me 3-CF_Three          U-4a 3-Me-5-Br U-4f 2-Br-5-Me
Me 3-OMe U-4a 3,5-di-Me U-4f 2-Br-5-CF_Three
Me 3-OCF_Three         U-4a 3-Me-5-CF_Three     U-4f 2-Br-5-OMe
Me 4-F U-4a 3-Me-5-OMe U-4f 2-Br-5-OCF_Three
Me 4-Cl U-4a 3-Me-5-OCF_Three    U-4f 2-Me-5-F
Me 4-Br U-4a 3-CF_Three-5-F U-4f 2-Me-5-Cl
Me 4-Me U-4a 3-CF_Three-5-Cl U-4f 2-Me-5-Br
Me 4-CF_Three          U-4a 3-CF_Three-5-Br U-4f 2,5-di-Me
Me 4-OMe U-4a 3-CF_Three-5-Me U-4f 2-Me-5-CF_Three
Me 4-OCF_Three         U-4a 3,5-di-CF_Three     U-4f 2-Me-5-OMe
Me 5-F U-4a 3-CF_Three-5-OMe U-4f 2-Me-5-OCF_Three
Me 5-Cl U-4a 3-CF_Three-5-OCF_Three   U-4f 2-CF_Three-5-F
Me 5-Br U-4a 3-OMe-5-F U-4f 2-CF_Three-5-Cl
Me 5-Me U-4a 3-OMe-5-Cl U-4f 2-CF_Three-5-Br
Me 5-CF_Three          U-4a 3-OMe-5-Br U-4f 2-CF_Three-5-Me
Me 5-OMe U-4a 3-OMe-5-Me U-4f 2,5-di-CF_Three
Me 5-OCF_Three         U-4a 3-OMe-5-CF_Three    U-4f 2-CF_Three-5-OMe
Et 2-F U-4a 3,5-di-OMe U-4f 2-CF_Three-5-OCF_Three
Et 2-Cl U-4a 3-OMe-5-OCF_Three   U-4f 2-OMe-5-F
Et 2-Br U-4a 3-OCF_Three-5-F U-4f 2-OMe-5-Cl
Et 2-Me U-4a 3-OCF_Three-5-Cl U-4f 2-OMe-5-Br
Et 2-CF_Three          U-4a 3-OCF_Three-5-Br U-4f 2-OMe-5-Me
Et 2-OMe U-4a 3-OCF_Three-5-Me U-4f 2-OMe-5-CF_Three
Et 2-OCF_Three         U-4a 3-OCF_Three-5-CF_Three   U-4f 2,5-di-OMe
Et 3-F U-4a 3-OCF_Three-5-OMe U-4f 2-OMe-5-OCF_Three
Et 3-Cl U-4a 3,5-di-OCF_Three    U-4f 2-OCF_Three-5-F
Et 3-Br CF_Three   2,3-di-F U-4f 2-OCF_Three-5-Cl
Et 3-Me CF_Three   2-F-3-Cl U-4f 2-OCF_Three-5-Br
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
Et 3-CF_Three          CF_Three   2-F-3-Br U-4f 2-OCF_Three-5-Me
Et 3-OMe CF_Three   2-F-3-Me U-4f 2-OCF_Three-5-CF_Three
Et 3-OCF_Three         CF_Three   2-F-3-CF_Three      U-4f 2-OCF_Three-5-OMe
Et 4-F CF_Three   2-F-3-OMe U-4f 2,5-di-OCF_Three
Et 4-Cl CF_Three   2-F-3-OCF_Three     U-4f 3,4-di-F
Et 4-Br CF_Three   2-Cl-3-F U-4f 3-F-4-Cl
Et 4-Me CF_Three   2,3-di-Cl U-4f 3-F-4-Br
Et 4-CF_Three          CF_Three   2-Cl-3-Br U-4f 3-F-4-Me
Et 4-OMe CF_Three   2-Cl-3-Me U-4f 3-F-4-CF_Three
Et 4-OCF_Three         CF_Three   2-Cl-3-CF_Three     U-4f 3-F-4-OMe
Et 5-F CF_Three   2-Cl-3-OMe U-4f 3-F-4-OCF_Three
Et 5-Cl CF_Three   2-Cl-3-OCF_Three    U-4f 3-Cl-4-F
Et 5-Br CF_Three   2-Br-3-F U-4f 3,4-di-Cl
Et 5-Me CF_Three   2-Br-3-Cl U-4f 3-Cl-4-Br
Et 5-CF_Three          CF_Three   2,3-di-Br U-4f 3-Cl-4-Me
Et 5-OMe CF_Three   2-Br-3-Me U-4f 3-Cl-4-CF_Three
Et 5-OCF_Three         CF_Three   2-Br-3-CF_Three     U-4f 3-Cl-4-OMe
iPr 2-F CF_Three   2-Br-3-OMe U-4f 3-Cl-4-OCF_Three
iPr 2-Cl CF_Three   2-Br-3-OCF_Three    U-4f 3-Br-4-F
iPr 2-Br CF_Three   2-Me-3-F U-4f 3-Br-4-Cl
iPr 2-Me CF_Three   2-Me-3-Cl U-4f 3,4-di-Br
iPr 2-CF_Three          CF_Three   2-Me-3-Br U-4f 3-Br-4-Me
iPr 2-OMe CF_Three   2,3-di-Me U-4f 3-Br-4-CF_Three
iPr 2-OCF_Three         CF_Three   2-Me-3-CF_Three     U-4f 3-Br-4-OMe
iPr 3-F CF_Three   2-Me-3-OMe U-4f 3-Br-4-OCF_Three
iPr 3-Cl CF_Three   2-Me-3-OCF_Three    U-4f 3-Me-4-F
iPr 3-Br CF_Three   2-CF_Three-3-F U-4f 3-Me-4-Cl
iPr 3-Me CF_Three   2-CF_Three-3-Cl U-4f 3-Me-4-Br
iPr 3-CF_Three          CF_Three   2-CF_Three-3-Br U-4f 3,4-di-Me
iPr 3-OMe CF_Three   2-CF_Three-3-Me U-4f 3-Me-4-CF_Three
iPr 3-OCF_Three         CF_Three   2,3-di-CF_Three     U-4f 3-Me-4-OMe
iPr 4-F CF_Three   2-CF_Three-3-OMe U-4f 3-Me-4-OCF_Three
iPr 4-Cl CF_Three   2-CF_Three-3-OCF_Three   U-4f 3-CF_Three-4-F
iPr 4-Br CF_Three   2-OMe-3-F U-4f 3-CF_Three-4-Cl
iPr 4-Me CF_Three   2-OMe-3-Cl U-4f 3-CF_Three-4-Br
iPr 4-CF_Three          CF_Three   2-OMe-3-Br U-4f 3-CF_Three-4-Me
iPr 4-OMe CF_Three   2-OMe-3-Me U-4f 3,4-di-CF_Three
iPr 4-OCF_Three         CF_Three   2-OMe-3-CF_Three    U-4f 3-CF_Three-4-OMe
iPr 5-F CF_Three   2,3-di-OMe U-4f 3-CF_Three-4-OCF_Three
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
iPr 5-Cl CF_Three   2-OMe-3-OCF_Three   U-4f 3-OMe-4-F
iPr 5-Br CF_Three   2-OCF_Three-3-F U-4f 3-OMe-4-Cl
iPr 5-Me CF_Three   2-OCF_Three-3-Cl U-4f 3-OMe-4-Br
iPr 5-CF_Three          CF_Three   2-OCF_Three-3-Br U-4f 3-OMe-4-Me
iPr 5-OMe CF_Three   2-OCF_Three-3-Me U-4f 3-OMe-4-CF_Three
iPr 5-OCF_Three         CF_Three   2-OCF_Three-3-CF_Three   U-4f 3,4-di-OMe
U-4a 2-F CF_Three   2-OCF_Three-3-OMe U-4f 3-OMe-4-OCF_Three
U-4a 2-Cl CF_Three   2,3-di-OCF_Three    U-4f 3-OCF_Three-4-F
U-4a 2-Br CF_Three   2,4-di-F U-4f 3-OCF_Three-4-Cl
U-4a 2-Me CF_Three   2-F-4-Cl U-4f 3-OCF_Three-4-Br
U-4a 2-CF_Three          CF_Three   2-F-4-Br U-4f 3-OCF_Three-4-Me
U-4a 2-OMe CF_Three   2-F-4-Me U-4f 3-OCF_Three-4-CF_Three
U-4a 2-OCF_Three         CF_Three   2-F-4-CF_Three      U-4f 3-OCF_Three-4-OMe
U-4a 3-F CF_Three   2-F-4-OMe U-4f 3,4-di-OCF_Three
U-4a 3-Cl CF_Three   2-F-4-OCF_Three     U-4f 3,5-di-F
U-4a 3-Br CF_Three   2-Cl-4-F U-4f 3-F-5-Cl
U-4a 3-Me CF_Three   2,4-di-Cl U-4f 3-F-5-Br
U-4a 3-CF_Three          CF_Three   2-Cl-4-Br U-4f 3-F-5-Me
U-4a 3-OMe CF_Three   2-Cl-4-Me U-4f 3-F-5-CF_Three
U-4a 3-OCF_Three         CF_Three   2-Cl-4-CF_Three     U-4f 3-F-5-OMe
U-4a 4-F CF_Three   2-Cl-4-OMe U-4f 3-F-5-OCF_Three
U-4a 4-Cl CF_Three   2-Cl-4-OCF_Three    U-4f 3-Cl-5-F
U-4a 4-Br CF_Three   2-Br-4-F U-4f 3,5-di-Cl
U-4a 4-Me CF_Three   2-Br-4-Cl U-4f 3-Cl-5-Br
U-4a 4-CF_Three          CF_Three   2,4-di-Br U-4f 3-Cl-5-Me
U-4a 4-OMe CF_Three   2-Br-4-Me U-4f 3-Cl-5-CF_Three
U-4a 4-OCF_Three         CF_Three   2-Br-4-CF_Three     U-4f 3-Cl-5-OMe
U-4a 5-F CF_Three   2-Br-4-OMe U-4f 3-Cl-5-OCF_Three
U-4a 5-Cl CF_Three   2-Br-4-OCF_Three    U-4f 3-Br-5-F
U-4a 5-Br CF_Three   2-Me-4-F U-4f 3-Br-5-Cl
U-4a 5-Me CF_Three   2-Me-4-Cl U-4f 3,5-di-Br
U-4a 5-CF_Three          CF_Three   2-Me-4-Br U-4f 3-Br-5-Me
U-4a 5-OMe CF_Three   2,4-di-Me U-4f 3-Br-5-CF_Three
U-4a 5-OCF_Three         CF_Three   2-Me-4-CF_Three     U-4f 3-Br-5-OMe
CF_Three   2-F CF_Three   2-Me-4-OMe U-4f 3-Br-5-OCF_Three
CF_Three   2-Cl CF_Three   2-Me-4-OCF_Three    U-4f 3-Me-5-F
CF_Three   2-Br CF_Three   2-CF_Three-4-F U-4f 3-Me-5-Cl
CF_Three   2-Me CF_Three   2-CF_Three-4-Cl U-4f 3-Me-5-Br
CF_Three   2-CF_Three          CF_Three   2-CF_Three-4-Br U-4f 3,5-di-Me
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
CF_Three   2-OMe CF_Three   2-CF_Three-4-Me U-4f 3-Me-5-CF_Three
CF_Three   2-OCF_Three         CF_Three   2,4-di-CF_Three     U-4f 3-Me-5-OMe
CF_Three   3-F CF_Three   2-CF_Three-4-OMe U-4f 3-Me-5-OCF_Three
CF_Three   3-Cl CF_Three   2-CF_Three-4-OCF_Three   U-4f 3-CF_Three-5-F
CF_Three   3-Br CF_Three   2-OMe-4-F U-4f 3-CF_Three-5-Cl
CF_Three   3-Me CF_Three   2-OMe-4-Cl U-4f 3-CF_Three-5-Br
CF_Three   3-CF_Three          CF_Three   2-OMe-4-Br U-4f 3-CF_Three-5-Me
CF_Three   3-OMe CF_Three   2-OMe-4-Me U-4f 3,5-di-CF_Three
CF_Three   3-OCF_Three         CF_Three   2-OMe-4-CF_Three    U-4f 3-CF_Three-5-OMe
CF_Three   4-F CF_Three   2,4-di-OMe U-4f 3-CF_Three-5-OCF_Three
CF_Three   4-Cl CF_Three   2-OMe-4-OCF_Three   U-4f 3-OMe-5-F
CF_Three   4-Br CF_Three   2-OCF_Three-4-F U-4f 3-OMe-5-Cl
CF_Three   4-Me CF_Three   2-OCF_Three-4-Cl U-4f 3-OMe-5-Br
CF_Three   4-CF_Three          CF_Three   2-OCF_Three-4-Br U-4f 3-OMe-5-Me
CF_Three   4-OMe CF_Three   2-OCF_Three-4-Me U-4f 3-OMe-5-CF_Three
CF_Three   4-OCF_Three         CF_Three   2-OCF_Three-4-CF_Three   U-4f 3,5-di-OMe
CF_Three   5-F CF_Three   2-OCF_Three-4-OMe U-4f 3-OMe-5-OCF_Three
CF_Three   5-Cl CF_Three   2,4-di-OCF_Three    U-4f 3-OCF_Three-5-F
CF_Three   5-Br CF_Three   2,5-di-F U-4f 3-OCF_Three-5-Cl
CF_Three   5-Me CF_Three   2-F-5-Cl U-4f 3-OCF_Three-5-Br
CF_Three   5-CF_Three          CF_Three   2-F-5-Br U-4f 3-OCF_Three-5-Me
CF_Three   5-OMe CF_Three   2-F-5-Me U-4f 3-OCF_Three-5-CF_Three
CF_Three   5-OCF_Three         CF_Three   2-F-5-CF_Three      U-4f 3-OCF_Three-5-OMe
cPr 2-F CF_Three   2-F-5-OMe U-4f 3,5-di-OCF_Three
cPr 2-Cl CF_Three   2-F-5-OCF_Three     U-4g 2,3-di-F
cPr 2-Br CF_Three   2-Cl-5-F U-4g 2-F-3-Cl
cPr 2-Me CF_Three   2,5-di-Cl U-4g 2-F-3-Br
cPr 2-CF_Three          CF_Three   2-Cl-5-Br U-4g 2-F-3-Me
cPr 2-OMe CF_Three   2-Cl-5-Me U-4g 2-F-3-CF_Three
cPr 2-OCF_Three         CF_Three   2-Cl-5-CF_Three     U-4g 2-F-3-OMe
cPr 3-F CF_Three   2-Cl-5-OMe U-4g 2-F-3-OCF_Three
cPr 3-Cl CF_Three   2-Cl-5-OCF_Three    U-4g 2-Cl-3-F
cPr 3-Br CF_Three   2-Br-5-F U-4g 2,3-di-Cl
cPr 3-Me CF_Three   2-Br-5-Cl U-4g 2-Cl-3-Br
cPr 3-CF_Three          CF_Three   2,5-di-Br U-4g 2-Cl-3-Me
cPr 3-OMe CF_Three   2-Br-5-Me U-4g 2-Cl-3-CF_Three
cPr 3-OCF_Three         CF_Three   2-Br-5-CF_Three     U-4g 2-Cl-3-OMe
cPr 4-F CF_Three   2-Br-5-OMe U-4g 2-Cl-3-OCF_Three
cPr 4-Cl CF_Three   2-Br-5-OCF_Three    U-4g 2-Br-3-F
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
cPr 4-Br CF_Three   2-Me-5-F U-4g 2-Br-3-Cl
cPr 4-Me CF_Three   2-Me-5-Cl U-4g 2,3-di-Br
cPr 4-CF_Three          CF_Three   2-Me-5-Br U-4g 2-Br-3-Me
cPr 4-OMe CF_Three   2,5-di-Me U-4g 2-Br-3-CF_Three
cPr 4-OCF_Three         CF_Three   2-Me-5-CF_Three     U-4g 2-Br-3-OMe
cPr 5-F CF_Three   2-Me-5-OMe U-4g 2-Br-3-OCF_Three
cPr 5-Cl CF_Three   2-Me-5-OCF_Three    U-4g 2-Me-3-F
cPr 5-Br CF_Three   2-CF_Three-5-F U-4g 2-Me-3-Cl
cPr 5-Me CF_Three   2-CF_Three-5-Cl U-4g 2-Me-3-Br
cPr 5-CF_Three          CF_Three   2-CF_Three-5-Br U-4g 2,3-di-Me
cPr 5-OMe CF_Three   2-CF_Three-5-Me U-4g 2-Me-3-CF_Three
cPr 5-OCF_Three         CF_Three   2,5-di-CF_Three     U-4g 2-Me-3-OMe
U-4b 2-F CF_Three   2-CF_Three-5-OMe U-4g 2-Me-3-OCF_Three
U-4b 2-Cl CF_Three   2-CF_Three-5-OCF_Three   U-4g 2-CF_Three-3-F
U-4b 2-Br CF_Three   2-OMe-5-F U-4g 2-CF_Three-3-Cl
U-4b 2-Me CF_Three   2-OMe-5-Cl U-4g 2-CF_Three-3-Br
U-4b 2-CF_Three          CF_Three   2-OMe-5-Br U-4g 2-CF_Three-3-Me
U-4b 2-OMe CF_Three   2-OMe-5-Me U-4g 2,3-di-CF_Three
U-4b 2-OCF_Three         CF_Three   2-OMe-5-CF_Three    U-4g 2-CF_Three-3-OMe
U-4b 3-F CF_Three   2,5-di-OMe U-4g 2-CF_Three-3-OCF_Three
U-4b 3-Cl CF_Three   2-OMe-5-OCF_Three   U-4g 2-OMe-3-F
U-4b 3-Br CF_Three   2-OCF_Three-5-F U-4g 2-OMe-3-Cl
U-4b 3-Me CF_Three   2-OCF_Three-5-Cl U-4g 2-OMe-3-Br
U-4b 3-CF_Three          CF_Three   2-OCF_Three-5-Br U-4g 2-OMe-3-Me
U-4b 3-OMe CF_Three   2-OCF_Three-5-Me U-4g 2-OMe-3-CF_Three
U-4b 3-OCF_Three         CF_Three   2-OCF_Three-5-CF_Three   U-4g 2,3-di-OMe
U-4b 4-F CF_Three   2-OCF_Three-5-OMe U-4g 2-OMe-3-OCF_Three
U-4b 4-Cl CF_Three   2,5-di-OCF_Three    U-4g 2-OCF_Three-3-F
U-4b 4-Br CF_Three   3,4-di-F U-4g 2-OCF_Three-3-Cl
U-4b 4-Me CF_Three   3-F-4-Cl U-4g 2-OCF_Three-3-Br
U-4b 4-CF_Three          CF_Three   3-F-4-Br U-4g 2-OCF_Three-3-Me
U-4b 4-OMe CF_Three   3-F-4-Me U-4g 2-OCF_Three-3-CF_Three
U-4b 4-OCF_Three         CF_Three   3-F-4-CF_Three      U-4g 2-OCF_Three-3-OMe
U-4b 5-F CF_Three   3-F-4-OMe U-4g 2,3-di-OCF_Three
U-4b 5-Cl CF_Three   3-F-4-OCF_Three     U-4g 2,4-di-F
U-4b 5-Br CF_Three   3-Cl-4-F U-4g 2-F-4-Cl
U-4b 5-Me CF_Three   3,4-di-Cl U-4g 2-F-4-Br
U-4b 5-CF_Three          CF_Three   3-Cl-4-Br U-4g 2-F-4-Me
U-4b 5-OMe CF_Three   3-Cl-4-Me U-4g 2-F-4-CF_Three
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
U-4b 5-OCF_Three         CF_Three   3-Cl-4-CF_Three     U-4g 2-F-4-OMe
U-4c 2-F CF_Three   3-Cl-4-OMe U-4g 2-F-4-OCF_Three
U-4c 2-Cl CF_Three   3-Cl-4-OCF_Three    U-4g 2-Cl-4-F
U-4c 2-Br CF_Three   3-Br-4-F U-4g 2,4-di-Cl
U-4c 2-Me CF_Three   3-Br-4-Cl U-4g 2-Cl-4-Br
U-4c 2-CF_Three          CF_Three   3,4-di-Br U-4g 2-Cl-4-Me
U-4c 2-OMe CF_Three   3-Br-4-Me U-4g 2-Cl-4-CF_Three
U-4c 2-OCF_Three         CF_Three   3-Br-4-CF_Three     U-4g 2-Cl-4-OMe
U-4c 3-F CF_Three   3-Br-4-OMe U-4g 2-Cl-4-OCF_Three
U-4c 3-Cl CF_Three   3-Br-4-OCF_Three    U-4g 2-Br-4-F
U-4c 3-Br CF_Three   3-Me-4-F U-4g 2-Br-4-Cl
U-4c 3-Me CF_Three   3-Me-4-Cl U-4g 2,4-di-Br
U-4c 3-CF_Three          CF_Three   3-Me-4-Br U-4g 2-Br-4-Me
U-4c 3-OMe CF_Three   3,4-di-Me U-4g 2-Br-4-CF_Three
U-4c 3-OCF_Three         CF_Three   3-Me-4-CF_Three     U-4g 2-Br-4-OMe
U-4c 4-F CF_Three   3-Me-4-OMe U-4g 2-Br-4-OCF_Three
U-4c 4-Cl CF_Three   3-Me-4-OCF_Three    U-4g 2-Me-4-F
U-4c 4-Br CF_Three   3-CF_Three-4-F U-4g 2-Me-4-Cl
U-4c 4-Me CF_Three   3-CF_Three-4-Cl U-4g 2-Me-4-Br
U-4c 4-CF_Three          CF_Three   3-CF_Three-4-Br U-4g 2,4-di-Me
U-4c 4-OMe CF_Three   3-CF_Three-4-Me U-4g 2-Me-4-CF_Three
U-4c 4-OCF_Three         CF_Three   3,4-di-CF_Three     U-4g 2-Me-4-OMe
U-4c 5-F CF_Three   3-CF_Three-4-OMe U-4g 2-Me-4-OCF_Three
U-4c 5-Cl CF_Three   3-CF_Three-4-OCF_Three   U-4g 2-CF_Three-4-F
U-4c 5-Br CF_Three   3-OMe-4-F U-4g 2-CF_Three-4-Cl
U-4c 5-Me CF_Three   3-OMe-4-Cl U-4g 2-CF_Three-4-Br
U-4c 5-CF_Three          CF_Three   3-OMe-4-Br U-4g 2-CF_Three-4-Me
U-4c 5-OMe CF_Three   3-OMe-4-Me U-4g 2,4-di-CF_Three
U-4c 5-OCF_Three         CF_Three   3-OMe-4-CF_Three    U-4g 2-CF_Three-4-OMe
U-4d 2-F CF_Three   3,4-di-OMe U-4g 2-CF_Three-4-OCF_Three
U-4d 2-Cl CF_Three   3-OMe-4-OCF_Three   U-4g 2-OMe-4-F
U-4d 2-Br CF_Three   3-OCF_Three-4-F U-4g 2-OMe-4-Cl
U-4d 2-Me CF_Three   3-OCF_Three-4-Cl U-4g 2-OMe-4-Br
U-4d 2-CF_Three          CF_Three   3-OCF_Three-4-Br U-4g 2-OMe-4-Me
U-4d 2-OMe CF_Three   3-OCF_Three-4-Me U-4g 2-OMe-4-CF_Three
U-4d 2-OCF_Three         CF_Three   3-OCF_Three-4-CF_Three   U-4g 2,4-di-OMe
U-4d 3-F CF_Three   3-OCF_Three-4-OMe U-4g 2-OMe-4-OCF_Three
U-4d 3-Cl CF_Three   3,4-di-OCF_Three    U-4g 2-OCF_Three-4-F
U-4d 3-Br CF_Three   3,5-di-F U-4g 2-OCF_Three-4-Cl
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
U-4d 3-Me CF_Three   3-F-5-Cl U-4g 2-OCF_Three-4-Br
U-4d 3-CF_Three          CF_Three   3-F-5-Br U-4g 2-OCF_Three-4-Me
U-4d 3-OMe CF_Three   3-F-5-Me U-4g 2-OCF_Three-4-CF_Three
U-4d 3-OCF_Three         CF_Three   3-F-5-CF_Three      U-4g 2-OCF_Three-4-OMe
U-4d 4-F CF_Three   3-F-5-OMe U-4g 2,4-di-OCF_Three
U-4d 4-Cl CF_Three   3-F-5-OCF_Three     U-4g 2,5-di-F
U-4d 4-Br CF_Three   3-Cl-5-F U-4g 2-F-5-Cl
U-4d 4-Me CF_Three   3,5-di-Cl U-4g 2-F-5-Br
U-4d 4-CF_Three          CF_Three   3-Cl-5-Br U-4g 2-F-5-Me
U-4d 4-OMe CF_Three   3-Cl-5-Me U-4g 2-F-5-CF_Three
U-4d 4-OCF_Three         CF_Three   3-Cl-5-CF_Three     U-4g 2-F-5-OMe
U-4d 5-F CF_Three   3-Cl-5-OMe U-4g 2-F-5-OCF_Three
U-4d 5-Cl CF_Three   3-Cl-5-OCF_Three    U-4g 2-Cl-5-F
U-4d 5-Br CF_Three   3-Br-5-F U-4g 2,5-di-Cl
U-4d 5-Me CF_Three   3-Br-5-Cl U-4g 2-Cl-5-Br
U-4d 5-CF_Three          CF_Three   3,5-di-Br U-4g 2-Cl-5-Me
U-4d 5-OMe CF_Three   3-Br-5-Me U-4g 2-Cl-5-CF_Three
U-4d 5-OCF_Three         CF_Three   3-Br-5-CF_Three     U-4g 2-Cl-5-OMe
U-4e 2-F CF_Three   3-Br-5-OMe U-4g 2-Cl-5-OCF_Three
U-4e 2-Cl CF_Three   3-Br-5-OCF_Three    U-4g 2-Br-5-F
U-4e 2-Br CF_Three   3-Me-5-F U-4g 2-Br-5-Cl
U-4e 2-Me CF_Three   3-Me-5-Cl U-4g 2,5-di-Br
U-4e 2-CF_Three          CF_Three   3-Me-5-Br U-4g 2-Br-5-Me
U-4e 2-OMe CF_Three   3,5-di-Me U-4g 2-Br-5-CF_Three
U-4e 2-OCF_Three         CF_Three   3-Me-5-CF_Three     U-4g 2-Br-5-OMe
U-4e 3-F CF_Three   3-Me-5-OMe U-4g 2-Br-5-OCF_Three
U-4e 3-Cl CF_Three   3-Me-5-OCF_Three    U-4g 2-Me-5-F
U-4e 3-Br CF_Three   3-CF_Three-5-F U-4g 2-Me-5-Cl
U-4e 3-Me CF_Three   3-CF_Three-5-Cl U-4g 2-Me-5-Br
U-4e 3-CF_Three          CF_Three   3-CF_Three-5-Br U-4g 2,5-di-Me
U-4e 3-OMe CF_Three   3-CF_Three-5-Me U-4g 2-Me-5-CF_Three
U-4e 3-OCF_Three         CF_Three   3,5-di-CF_Three     U-4g 2-Me-5-OMe
U-4e 4-F CF_Three   3-CF_Three-5-OMe U-4g 2-Me-5-OCF_Three
U-4e 4-Cl CF_Three   3-CF_Three-5-OCF_Three   U-4g 2-CF_Three-5-F
U-4e 4-Br CF_Three   3-OMe-5-F U-4g 2-CF_Three-5-Cl
U-4e 4-Me CF_Three   3-OMe-5-Cl U-4g 2-CF_Three-5-Br
U-4e 4-CF_Three          CF_Three   3-OMe-5-Br U-4g 2-CF_Three-5-Me
U-4e 4-OMe CF_Three   3-OMe-5-Me U-4g 2,5-di-CF_Three
U-4e 4-OCF_Three         CF_Three   3-OMe-5-CF_Three    U-4g 2-CF_Three-5-OMe
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
U-4e 5-F CF_Three   3,5-di-OMe U-4g 2-CF_Three-5-OCF_Three
U-4e 5-Cl CF_Three   3-OMe-5-OCF_Three   U-4g 2-OMe-5-F
U-4e 5-Br CF_Three   3-OCF_Three-5-F U-4g 2-OMe-5-Cl
U-4e 5-Me CF_Three   3-OCF_Three-5-Cl U-4g 2-OMe-5-Br
U-4e 5-CF_Three          CF_Three   3-OCF_Three-5-Br U-4g 2-OMe-5-Me
U-4e 5-OMe CF_Three   3-OCF_Three-5-Me U-4g 2-OMe-5-CF_Three
U-4e 5-OCF_Three         CF_Three   3-OCF_Three-5-CF_Three   U-4g 2,5-di-OMe
U-4f 2-F CF_Three   3-OCF_Three-5-OMe U-4g 2-OMe-5-OCF_Three
U-4f 2-Cl CF_Three   3,5-di-OCF_Three    U-4g 2-OCF_Three-5-F
U-4f 2-Br cPr 2,3-di-F U-4g 2-OCF_Three-5-Cl
U-4f 2-Me cPr 2-F-3-Cl U-4g 2-OCF_Three-5-Br
U-4f 2-CF_Three          cPr 2-F-3-Br U-4g 2-OCF_Three-5-Me
U-4f 2-OMe cPr 2-F-3-Me U-4g 2-OCF_Three-5-CF_Three
U-4f 2-OCF_Three         cPr 2-F-3-CF_Three      U-4g 2-OCF_Three-5-OMe
U-4f 3-F cPr 2-F-3-OMe U-4g 2,5-di-OCF_Three
U-4f 3-Cl cPr 2-F-3-OCF_Three     U-4g 3,4-di-F
U-4f 3-Br cPr 2-Cl-3-F U-4g 3-F-4-Cl
U-4f 3-Me cPr 2,3-di-Cl U-4g 3-F-4-Br
U-4f 3-CF_Three          cPr 2-Cl-3-Br U-4g 3-F-4-Me
U-4f 3-OMe cPr 2-Cl-3-Me U-4g 3-F-4-CF_Three
U-4f 3-OCF_Three         cPr 2-Cl-3-CF_Three     U-4g 3-F-4-OMe
U-4f 4-F cPr 2-Cl-3-OMe U-4g 3-F-4-OCF_Three
U-4f 4-Cl cPr 2-Cl-3-OCF_Three    U-4g 3-Cl-4-F
U-4f 4-Br cPr 2-Br-3-F U-4g 3,4-di-Cl
U-4f 4-Me cPr 2-Br-3-Cl U-4g 3-Cl-4-Br
U-4f 4-CF_Three          cPr 2,3-di-Br U-4g 3-Cl-4-Me
U-4f 4-OMe cPr 2-Br-3-Me U-4g 3-Cl-4-CF_Three
U-4f 4-OCF_Three         cPr 2-Br-3-CF_Three     U-4g 3-Cl-4-OMe
U-4f 5-F cPr 2-Br-3-OMe U-4g 3-Cl-4-OCF_Three
U-4f 5-Cl cPr 2-Br-3-OCF_Three    U-4g 3-Br-4-F
U-4f 5-Br cPr 2-Me-3-F U-4g 3-Br-4-Cl
U-4f 5-Me cPr 2-Me-3-Cl U-4g 3,4-di-Br
U-4f 5-CF_Three          cPr 2-Me-3-Br U-4g 3-Br-4-Me
U-4f 5-OMe cPr 2,3-di-Me U-4g 3-Br-4-CF_Three
U-4f 5-OCF_Three         cPr 2-Me-3-CF_Three     U-4g 3-Br-4-OMe
U-4g 2-F cPr 2-Me-3-OMe U-4g 3-Br-4-OCF_Three
U-4g 2-Cl cPr 2-Me-3-OCF_Three    U-4g 3-Me-4-F
U-4g 2-Br cPr 2-CF_Three-3-F U-4g 3-Me-4-Cl
U-4g 2-Me cPr 2-CF_Three-3-Cl U-4g 3-Me-4-Br
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
U-4g 2-CF_Three          cPr 2-CF_Three-3-Br U-4g 3,4-di-Me
U-4g 2-OMe cPr 2-CF_Three-3-Me U-4g 3-Me-4-CF_Three
U-4g 2-OCF_Three         cPr 2,3-di-CF_Three     U-4g 3-Me-4-OMe
U-4g 3-F cPr 2-CF_Three-3-OMe U-4g 3-Me-4-OCF_Three
U-4g 3-Cl cPr 2-CF_Three-3-OCF_Three   U-4g 3-CF_Three-4-F
U-4g 3-Br cPr 2-OMe-3-F U-4g 3-CF_Three-4-Cl
U-4g 3-Me cPr 2-OMe-3-Cl U-4g 3-CF_Three-4-Br
U-4g 3-CF_Three          cPr 2-OMe-3-Br U-4g 3-CF_Three-4-Me
U-4g 3-OMe cPr 2-OMe-3-Me U-4g 3,4-di-CF_Three
U-4g 3-OCF_Three         cPr 2-OMe-3-CF_Three    U-4g 3-CF_Three-4-OMe
U-4g 4-F cPr 2,3-di-OMe U-4g 3-CF_Three-4-OCF_Three
U-4g 4-Cl cPr 2-OMe-3-OCF_Three   U-4g 3-OMe-4-F
U-4g 4-Br cPr 2-OCF_Three-3-F U-4g 3-OMe-4-Cl
U-4g 4-Me cPr 2-OCF_Three-3-Cl U-4g 3-OMe-4-Br
U-4g 4-CF_Three          cPr 2-OCF_Three-3-Br U-4g 3-OMe-4-Me
U-4g 4-OMe cPr 2-OCF_Three-3-Me U-4g 3-OMe-4-CF_Three
U-4g 4-OCF_Three         cPr 2-OCF_Three-3-CF_Three   U-4g 3,4-di-OMe
U-4g 5-F cPr 2-OCF_Three-3-OMe U-4g 3-OMe-4-OCF_Three
U-4g 5-Cl cPr 2,3-di-OCF_Three    U-4g 3-OCF_Three-4-F
U-4g 5-Br cPr 2,4-di-F U-4g 3-OCF_Three-4-Cl
U-4g 5-Me cPr 2-F-4-Cl U-4g 3-OCF_Three-4-Br
U-4g 5-CF_Three          cPr 2-F-4-Br U-4g 3-OCF_Three-4-Me
U-4g 5-OMe cPr 2-F-4-Me U-4g 3-OCF_Three-4-CF_Three
U-4g 5-OCF_Three         cPr 2-F-4-CF_Three      U-4g 3-OCF_Three-4-OMe
OMe 2-F cPr 2-F-4-OMe U-4g 3,4-di-OCF_Three
OMe 2-Cl cPr 2-F-4-OCF_Three     U-4g 3,5-di-F
OMe 2-Br cPr 2-Cl-4-F U-4g 3-F-5-Cl
OMe 2-Me cPr 2,4-di-Cl U-4g 3-F-5-Br
OMe 2-CF_Three          cPr 2-Cl-4-Br U-4g 3-F-5-Me
OMe 2-OMe cPr 2-Cl-4-Me U-4g 3-F-5-CF_Three
OMe 2-OCF_Three         cPr 2-Cl-4-CF_Three     U-4g 3-F-5-OMe
OMe 3-F cPr 2-Cl-4-OMe U-4g 3-F-5-OCF_Three
OMe 3-Cl cPr 2-Cl-4-OCF_Three    U-4g 3-Cl-5-F
OMe 3-Br cPr 2-Br-4-F U-4g 3,5-di-Cl
OMe 3-Me cPr 2-Br-4-Cl U-4g 3-Cl-5-Br
OMe 3-CF_Three          cPr 2,4-di-Br U-4g 3-Cl-5-Me
OMe 3-OMe cPr 2-Br-4-Me U-4g 3-Cl-5-CF_Three
OMe 3-OCF_Three         cPr 2-Br-4-CF_Three     U-4g 3-Cl-5-OMe
OMe 4-F cPr 2-Br-4-OMe U-4g 3-Cl-5-OCF_Three
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
OMe 4-Cl cPr 2-Br-4-OCF_Three    U-4g 3-Br-5-F
OMe 4-Br cPr 2-Me-4-F U-4g 3-Br-5-Cl
OMe 4-Me cPr 2-Me-4-Cl U-4g 3,5-di-Br
OMe 4-CF_Three          cPr 2-Me-4-Br U-4g 3-Br-5-Me
OMe 4-OMe cPr 2,4-di-Me U-4g 3-Br-5-CF_Three
OMe 4-OCF_Three         cPr 2-Me-4-CF_Three     U-4g 3-Br-5-OMe
OMe 5-F cPr 2-Me-4-OMe U-4g 3-Br-5-OCF_Three
OMe 5-Cl cPr 2-Me-4-OCF_Three    U-4g 3-Me-5-F
OMe 5-Br cPr 2-CF_Three-4-F U-4g 3-Me-5-Cl
OMe 5-Me cPr 2-CF_Three-4-Cl U-4g 3-Me-5-Br
OMe 5-CF_Three          cPr 2-CF_Three-4-Br U-4g 3,5-di-Me
OMe 5-OMe cPr 2-CF_Three-4-Me U-4g 3-Me-5-CF_Three
OMe 5-OCF_Three         cPr 2,4-di-CF_Three     U-4g 3-Me-5-OMe
SMe 2-F cPr 2-CF_Three-4-OMe U-4g 3-Me-5-OCF_Three
SMe 2-Cl cPr 2-CF_Three-4-OCF_Three   U-4g 3-CF_Three-5-F
SMe 2-Br cPr 2-OMe-4-F U-4g 3-CF_Three-5-Cl
SMe 2-Me cPr 2-OMe-4-Cl U-4g 3-CF_Three-5-Br
SMe 2-CF_Three          cPr 2-OMe-4-Br U-4g 3-CF_Three-5-Me
SMe 2-OMe cPr 2-OMe-4-Me U-4g 3,5-di-CF_Three
SMe 2-OCF_Three         cPr 2-OMe-4-CF_Three    U-4g 3-CF_Three-5-OMe
SMe 3-F cPr 2,4-di-OMe U-4g 3-CF_Three-5-OCF_Three
SMe 3-Cl cPr 2-OMe-4-OCF_Three   U-4g 3-OMe-5-F
SMe 3-Br cPr 2-OCF_Three-4-F U-4g 3-OMe-5-Cl
SMe 3-Me cPr 2-OCF_Three-4-Cl U-4g 3-OMe-5-Br
SMe 3-CF_Three          cPr 2-OCF_Three-4-Br U-4g 3-OMe-5-Me
SMe 3-OMe cPr 2-OCF_Three-4-Me U-4g 3-OMe-5-CF_Three
SMe 3-OCF_Three         cPr 2-OCF_Three-4-CF_Three   U-4g 3,5-di-OMe
SMe 4-F cPr 2-OCF_Three-4-OMe U-4g 3-OMe-5-OCF_Three
SMe 4-Cl cPr 2,4-di-OCF_Three    U-4g 3-OCF_Three-5-F
SMe 4-Br cPr 2,5-di-F U-4g 3-OCF_Three-5-Cl
SMe 4-Me cPr 2-F-5-Cl U-4g 3-OCF_Three-5-Br
SMe 4-CF_Three          cPr 2-F-5-Br U-4g 3-OCF_Three-5-Me
SMe 4-OMe cPr 2-F-5-Me U-4g 3-OCF_Three-5-CF_Three
SMe 4-OCF_Three         cPr 2-F-5-CF_Three      U-4g 3-OCF_Three-5-OMe
SMe 5-F cPr 2-F-5-OMe U-4g 3,5-di-OCF_Three
SMe 5-Cl cPr 2-F-5-OCF_Three     OMe 2,3-di-F
SMe 5-Br cPr 2-Cl-5-F OMe 2-F-3-Cl
SMe 5-Me cPr 2,5-di-Cl OMe 2-F-3-Br
SMe 5-CF_Three          cPr 2-Cl-5-Br OMe 2-F-3-Me
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
SMe 5-OMe cPr 2-Cl-5-Me OMe 2-F-3-CF_Three
SMe 5-OCF_Three         cPr 2-Cl-5-CF_Three     OMe 2-F-3-OMe
Ac 2-F cPr 2-Cl-5-OMe OMe 2-F-3-OCF_Three
Ac 2-Cl cPr 2-Cl-5-OCF_Three    OMe 2-Cl-3-F
Ac 2-Br cPr 2-Br-5-F OMe 2,3-di-Cl
Ac 2-Me cPr 2-Br-5-Cl OMe 2-Cl-3-Br
Ac 2-CF_Three          cPr 2,5-di-Br OMe 2-Cl-3-Me
Ac 2-OMe cPr 2-Br-5-Me OMe 2-Cl-3-CF_Three
Ac 2-OCF_Three         cPr 2-Br-5-CF_Three     OMe 2-Cl-3-OMe
Ac 3-F cPr 2-Br-5-OMe OMe 2-Cl-3-OCF_Three
Ac 3-Cl cPr 2-Br-5-OCF_Three    OMe 2-Br-3-F
Ac 3-Br cPr 2-Me-5-F OMe 2-Br-3-Cl
Ac 3-Me cPr 2-Me-5-Cl OMe 2,3-di-Br
Ac 3-CF_Three          cPr 2-Me-5-Br OMe 2-Br-3-Me
Ac 3-OMe cPr 2,5-di-Me OMe 2-Br-3-CF_Three
Ac 3-OCF_Three         cPr 2-Me-5-CF_Three     OMe 2-Br-3-OMe
Ac 4-F cPr 2-Me-5-OMe OMe 2-Br-3-OCF_Three
Ac 4-Cl cPr 2-Me-5-OCF_Three    OMe 2-Me-3-F
Ac 4-Br cPr 2-CF_Three-5-F OMe 2-Me-3-Cl
Ac 4-Me cPr 2-CF_Three-5-Cl OMe 2-Me-3-Br
Ac 4-CF_Three          cPr 2-CF_Three-5-Br OMe 2,3-di-Me
Ac 4-OMe cPr 2-CF_Three-5-Me OMe 2-Me-3-CF_Three
Ac 4-OCF_Three         cPr 2,5-di-CF_Three     OMe 2-Me-3-OMe
Ac 5-F cPr 2-CF_Three-5-OMe OMe 2-Me-3-OCF_Three
Ac 5-Cl cPr 2-CF_Three-5-OCF_Three   OMe 2-CF_Three-3-F
Ac 5-Br cPr 2-OMe-5-F OMe 2-CF_Three-3-Cl
Ac 5-Me cPr 2-OMe-5-Cl OMe 2-CF_Three-3-Br
Ac 5-CF_Three          cPr 2-OMe-5-Br OMe 2-CF_Three-3-Me
Ac 5-OMe cPr 2-OMe-5-Me OMe 2,3-di-CF_Three
Ac 5-OCF_Three         cPr 2-OMe-5-CF_Three    OMe 2-CF_Three-3-OMe
cPen 2-F cPr 2,5-di-OMe OMe 2-CF_Three-3-OCF_Three
cPen 2-Cl cPr 2-OMe-5-OCF_Three   OMe 2-OMe-3-F
cPen 2-Br cPr 2-OCF_Three-5-F OMe 2-OMe-3-Cl
cPen 2-Me cPr 2-OCF_Three-5-Cl OMe 2-OMe-3-Br
cPen 2-CF_Three          cPr 2-OCF_Three-5-Br OMe 2-OMe-3-Me
cPen 2-OMe cPr 2-OCF_Three-5-Me OMe 2-OMe-3-CF_Three
cPen 2-OCF_Three         cPr 2-OCF_Three-5-CF_Three   OMe 2,3-di-OMe
cPen 3-F cPr 2-OCF_Three-5-OMe OMe 2-OMe-3-OCF_Three
cPen 3-Cl cPr 2,5-di-OCF_Three    OMe 2-OCF_Three-3-F
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
cPen 3-Br cPr 3,4-di-F OMe 2-OCF_Three-3-Cl
cPen 3-Me cPr 3-F-4-Cl OMe 2-OCF_Three-3-Br
cPen 3-CF_Three          cPr 3-F-4-Br OMe 2-OCF_Three-3-Me
cPen 3-OMe cPr 3-F-4-Me OMe 2-OCF_Three-3-CF_Three
cPen 3-OCF_Three         cPr 3-F-4-CF_Three      OMe 2-OCF_Three-3-OMe
cPen 4-F cPr 3-F-4-OMe OMe 2,3-di-OCF_Three
cPen 4-Cl cPr 3-F-4-OCF_Three     OMe 2,4-di-F
cPen 4-Br cPr 3-Cl-4-F OMe 2-F-4-Cl
cPen 4-Me cPr 3,4-di-Cl OMe 2-F-4-Br
cPen 4-CF_Three          cPr 3-Cl-4-Br OMe 2-F-4-Me
cPen 4-OMe cPr 3-Cl-4-Me OMe 2-F-4-CF_Three
cPen 4-OCF_Three         cPr 3-Cl-4-CF_Three     OMe 2-F-4-OMe
cPen 5-F cPr 3-Cl-4-OMe OMe 2-F-4-OCF_Three
cPen 5-Cl cPr 3-Cl-4-OCF_Three    OMe 2-Cl-4-F
cPen 5-Br cPr 3-Br-4-F OMe 2,4-di-Cl
cPen 5-Me cPr 3-Br-4-Cl OMe 2-Cl-4-Br
cPen 5-CF_Three          cPr 3,4-di-Br OMe 2-Cl-4-Me
cPen 5-OMe cPr 3-Br-4-Me OMe 2-Cl-4-CF_Three
cPen 5-OCF_Three         cPr 3-Br-4-CF_Three     OMe 2-Cl-4-OMe
U-1e 2-F cPr 3-Br-4-OMe OMe 2-Cl-4-OCF_Three
U-1e 2-Cl cPr 3-Br-4-OCF_Three    OMe 2-Br-4-F
U-1e 2-Br cPr 3-Me-4-F OMe 2-Br-4-Cl
U-1e 2-Me cPr 3-Me-4-Cl OMe 2,4-di-Br
U-1e 2-CF_Three          cPr 3-Me-4-Br OMe 2-Br-4-Me
U-1e 2-OMe cPr 3,4-di-Me OMe 2-Br-4-CF_Three
U-1e 2-OCF_Three         cPr 3-Me-4-CF_Three     OMe 2-Br-4-OMe
U-1e 3-F cPr 3-Me-4-OMe OMe 2-Br-4-OCF_Three
U-1e 3-Cl cPr 3-Me-4-OCF_Three    OMe 2-Me-4-F
U-1e 3-Br cPr 3-CF_Three-4-F OMe 2-Me-4-Cl
U-1e 3-Me cPr 3-CF_Three-4-Cl OMe 2-Me-4-Br
U-1e 3-CF_Three          cPr 3-CF_Three-4-Br OMe 2,4-di-Me
U-1e 3-OMe cPr 3-CF_Three-4-Me OMe 2-Me-4-CF_Three
U-1e 3-OCF_Three         cPr 3,4-di-CF_Three     OMe 2-Me-4-OMe
U-1e 4-F cPr 3-CF_Three-4-OMe OMe 2-Me-4-OCF_Three
U-1e 4-Cl cPr 3-CF_Three-4-OCF_Three   OMe 2-CF_Three-4-F
U-1e 4-Br cPr 3-OMe-4-F OMe 2-CF_Three-4-Cl
U-1e 4-Me cPr 3-OMe-4-Cl OMe 2-CF_Three-4-Br
U-1e 4-CF_Three          cPr 3-OMe-4-Br OMe 2-CF_Three-4-Me
U-1e 4-OMe cPr 3-OMe-4-Me OMe 2,4-di-CF_Three
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
U-1e 4-OCF_Three         cPr 3-OMe-4-CF_Three    OMe 2-CF_Three-4-OMe
U-1e 5-F cPr 3,4-di-OMe OMe 2-CF_Three-4-OCF_Three
U-1e 5-Cl cPr 3-OMe-4-OCF_Three   OMe 2-OMe-4-F
U-1e 5-Br cPr 3-OCF_Three-4-F OMe 2-OMe-4-Cl
U-1e 5-Me cPr 3-OCF_Three-4-Cl OMe 2-OMe-4-Br
U-1e 5-CF_Three          cPr 3-OCF_Three-4-Br OMe 2-OMe-4-Me
U-1e 5-OMe cPr 3-OCF_Three-4-Me OMe 2-OMe-4-CF_Three
U-1e 5-OCF_Three         cPr 3-OCF_Three-4-CF_Three   OMe 2,4-di-OMe
Me 2-Ac cPr 3-OCF_Three-4-OMe OMe 2-OMe-4-OCF_Three
Me 2- (U-3b) cPr 3,4-di-OCF_Three    OMe 2-OCF_Three-4-F
Me 2-CF₂H cPr 3,5-di-F OMe 2-OCF_Three-4-Cl
Me 2-CN cPr 3-F-5-Cl OMe 2-OCF_Three-4-Br
Me 2-Et cPr 3-F-5-Br OMe 2-OCF_Three-4-Me
Me 2-OCF₂H cPr 3-F-5-Me OMe 2-OCF_Three-4-CF_Three
Me 2-OEt cPr 3-F-5-CF_Three      OMe 2-OCF_Three-4-OMe
Me 2-C (O) CF_Three      cPr 3-F-5-OMe OMe 2,4-di-OCF_Three
Me 3-Ac cPr 3-F-5-OCF_Three     OMe 2,5-di-F
Me 3- (U-3b) cPr 3-Cl-5-F OMe 2-F-5-Cl
Me 3-CF₂H cPr 3,5-di-Cl OMe 2-F-5-Br
Me 3-CN cPr 3-Cl-5-Br OMe 2-F-5-Me
Me 3-Et cPr 3-Cl-5-Me OMe 2-F-5-CF_Three
Me 3-OCF₂H cPr 3-Cl-5-CF_Three     OMe 2-F-5-OMe
Me 3-OEt cPr 3-Cl-5-OMe OMe 2-F-5-OCF_Three
Me 3-C (O) CF_Three      cPr 3-Cl-5-OCF_Three    OMe 2-Cl-5-F
Me 4-Ac cPr 3-Br-5-F OMe 2,5-di-Cl
Me 4- (U-3b) cPr 3-Br-5-Cl OMe 2-Cl-5-Br
Me 4-CF₂H cPr 3,5-di-Br OMe 2-Cl-5-Me
Me 4-CN cPr 3-Br-5-Me OMe 2-Cl-5-CF_Three
Me 4-Et cPr 3-Br-5-CF_Three     OMe 2-Cl-5-OMe
Me 4-OCF₂H cPr 3-Br-5-OMe OMe 2-Cl-5-OCF_Three
Me 4-OEt cPr 3-Br-5-OCF_Three    OMe 2-Br-5-F
Me 4-C (O) CF_Three      cPr 3-Me-5-F OMe 2-Br-5-Cl
Me 5-Ac cPr 3-Me-5-Cl OMe 2,5-di-Br
Me 5- (U-3b) cPr 3-Me-5-Br OMe 2-Br-5-Me
Me 5-CF₂H cPr 3,5-di-Me OMe 2-Br-5-CF_Three
Me 5-CN cPr 3-Me-5-CF_Three     OMe 2-Br-5-OMe
Me 5-Et cPr 3-Me-5-OMe OMe 2-Br-5-OCF_Three
Me 5-OCF₂H cPr 3-Me-5-OCF_Three    OMe 2-Me-5-F
Me 5-OEt cPr 3-CF_Three-5-F OMe 2-Me-5-Cl
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
Me 5-C (O) CF_Three      cPr 3-CF_Three-5-Cl OMe 2-Me-5-Br
Et 2-Ac cPr 3-CF_Three-5-Br OMe 2,5-di-Me
Et 2- (U-3b) cPr 3-CF_Three-5-Me OMe 2-Me-5-CF_Three
Et 2-CF₂H cPr 3,5-di-CF_Three     OMe 2-Me-5-OMe
Et 2-CN cPr 3-CF_Three-5-OMe OMe 2-Me-5-OCF_Three
Et 2-Et cPr 3-CF_Three-5-OCF_Three   OMe 2-CF_Three-5-F
Et 2-OCF₂H cPr 3-OMe-5-F OMe 2-CF_Three-5-Cl
Et 2-OEt cPr 3-OMe-5-Cl OMe 2-CF_Three-5-Br
Et 2-C (O) CF_Three      cPr 3-OMe-5-Br OMe 2-CF_Three-5-Me
Et 3-Ac cPr 3-OMe-5-Me OMe 2,5-di-CF_Three
Et 3- (U-3b) cPr 3-OMe-5-CF_Three    OMe 2-CF_Three-5-OMe
Et 3-CF₂H cPr 3,5-di-OMe OMe 2-CF_Three-5-OCF_Three
Et 3-CN cPr 3-OMe-5-OCF_Three   OMe 2-OMe-5-F
Et 3-Et cPr 3-OCF_Three-5-F OMe 2-OMe-5-Cl
Et 3-OCF₂H cPr 3-OCF_Three-5-Cl OMe 2-OMe-5-Br
Et 3-OEt cPr 3-OCF_Three-5-Br OMe 2-OMe-5-Me
Et 3-C (O) CF_Three      cPr 3-OCF_Three-5-Me OMe 2-OMe-5-CF_Three
Et 4-Ac cPr 3-OCF_Three-5-CF_Three   OMe 2,5-di-OMe
Et 4- (U-3b) cPr 3-OCF_Three-5-OMe OMe 2-OMe-5-OCF_Three
Et 4-CF₂H cPr 3,5-di-OCF_Three    OMe 2-OCF_Three-5-F
Et 4-CN U-4b 2,3-di-F OMe 2-OCF_Three-5-Cl
Et 4-Et U-4b 2-F-3-Cl OMe 2-OCF_Three-5-Br
Et 4-OCF₂H U-4b 2-F-3-Br OMe 2-OCF_Three-5-Me
Et 4-OEt U-4b 2-F-3-Me OMe 2-OCF_Three-5-CF_Three
Et 4-C (O) CF_Three      U-4b 2-F-3-CF_Three      OMe 2-OCF_Three-5-OMe
Et 5-Ac U-4b 2-F-3-OMe OMe 2,5-di-OCF_Three
Et 5- (U-3b) U-4b 2-F-3-OCF_Three     OMe 3,4-di-F
Et 5-CF₂H U-4b 2-Cl-3-F OMe 3-F-4-Cl
Et 5-CN U-4b 2,3-di-Cl OMe 3-F-4-Br
Et 5-Et U-4b 2-Cl-3-Br OMe 3-F-4-Me
Et 5-OCF₂H U-4b 2-Cl-3-Me OMe 3-F-4-CF_Three
Et 5-OEt U-4b 2-Cl-3-CF_Three     OMe 3-F-4-OMe
Et 5-C (O) CF_Three      U-4b 2-Cl-3-OMe OMe 3-F-4-OCF_Three
iPr 2-Ac U-4b 2-Cl-3-OCF_Three    OMe 3-Cl-4-F
iPr 2- (U-3b) U-4b 2-Br-3-F OMe 3,4-di-Cl
iPr 2-CF₂H U-4b 2-Br-3-Cl OMe 3-Cl-4-Br
iPr 2-CN U-4b 2,3-di-Br OMe 3-Cl-4-Me
iPr 2-Et U-4b 2-Br-3-Me OMe 3-Cl-4-CF_Three
iPr 2-OCF₂H U-4b 2-Br-3-CF_Three     OMe 3-Cl-4-OMe
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
iPr 2-OEt U-4b 2-Br-3-OMe OMe 3-Cl-4-OCF_Three
iPr 2-C (O) CF_Three      U-4b 2-Br-3-OCF_Three    OMe 3-Br-4-F
iPr 3-Ac U-4b 2-Me-3-F OMe 3-Br-4-Cl
iPr 3- (U-3b) U-4b 2-Me-3-Cl OMe 3,4-di-Br
iPr 3-CF₂H U-4b 2-Me-3-Br OMe 3-Br-4-Me
iPr 3-CN U-4b 2,3-di-Me OMe 3-Br-4-CF_Three
iPr 3-Et U-4b 2-Me-3-CF_Three     OMe 3-Br-4-OMe
iPr 3-OCF₂H U-4b 2-Me-3-OMe OMe 3-Br-4-OCF_Three
iPr 3-OEt U-4b 2-Me-3-OCF_Three    OMe 3-Me-4-F
iPr 3-C (O) CF_Three      U-4b 2-CF_Three-3-F OMe 3-Me-4-Cl
iPr 4-Ac U-4b 2-CF_Three-3-Cl OMe 3-Me-4-Br
iPr 4- (U-3b) U-4b 2-CF_Three-3-Br OMe 3,4-di-Me
iPr 4-CF₂H U-4b 2-CF_Three-3-Me OMe 3-Me-4-CF_Three
iPr 4-CN U-4b 2,3-di-CF_Three     OMe 3-Me-4-OMe
iPr 4-Et U-4b 2-CF_Three-3-OMe OMe 3-Me-4-OCF_Three
iPr 4-OCF₂H U-4b 2-CF_Three-3-OCF_Three   OMe 3-CF_Three-4-F
iPr 4-OEt U-4b 2-OMe-3-F OMe 3-CF_Three-4-Cl
iPr 4-C (O) CF_Three      U-4b 2-OMe-3-Cl OMe 3-CF_Three-4-Br
iPr 5-Ac U-4b 2-OMe-3-Br OMe 3-CF_Three-4-Me
iPr 5- (U-3b) U-4b 2-OMe-3-Me OMe 3,4-di-CF_Three
iPr 5-CF₂H U-4b 2-OMe-3-CF_Three    OMe 3-CF_Three-4-OMe
iPr 5-CN U-4b 2,3-di-OMe OMe 3-CF_Three-4-OCF_Three
iPr 5-Et U-4b 2-OMe-3-OCF_Three   OMe 3-OMe-4-F
iPr 5-OCF₂H U-4b 2-OCF_Three-3-F OMe 3-OMe-4-Cl
iPr 5-OEt U-4b 2-OCF_Three-3-Cl OMe 3-OMe-4-Br
iPr 5-C (O) CF_Three      U-4b 2-OCF_Three-3-Br OMe 3-OMe-4-Me
U-4a 2-Ac U-4b 2-OCF_Three-3-Me OMe 3-OMe-4-CF_Three
U-4a 2- (U-3b) U-4b 2-OCF_Three-3-CF_Three   OMe 3,4-di-OMe
U-4a 2-CF₂H U-4b 2-OCF_Three-3-OMe OMe 3-OMe-4-OCF_Three
U-4a 2-CN U-4b 2,3-di-OCF_Three    OMe 3-OCF_Three-4-F
U-4a 2-Et U-4b 2,4-di-F OMe 3-OCF_Three-4-Cl
U-4a 2-OCF₂H U-4b 2-F-4-Cl OMe 3-OCF_Three-4-Br
U-4a 2-OEt U-4b 2-F-4-Br OMe 3-OCF_Three-4-Me
U-4a 2-C (O) CF_Three      U-4b 2-F-4-Me OMe 3-OCF_Three-4-CF_Three
U-4a 3-Ac U-4b 2-F-4-CF_Three      OMe 3-OCF_Three-4-OMe
U-4a 3- (U-3b) U-4b 2-F-4-OMe OMe 3,4-di-OCF_Three
U-4a 3-CF₂H U-4b 2-F-4-OCF_Three     OMe 3,5-di-F
U-4a 3-CN U-4b 2-Cl-4-F OMe 3-F-5-Cl
U-4a 3-Et U-4b 2,4-di-Cl OMe 3-F-5-Br
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
U-4a 3-OCF₂H U-4b 2-Cl-4-Br OMe 3-F-5-Me
U-4a 3-OEt U-4b 2-Cl-4-Me OMe 3-F-5-CF_Three
U-4a 3-C (O) CF_Three      U-4b 2-Cl-4-CF_Three     OMe 3-F-5-OMe
U-4a 4-Ac U-4b 2-Cl-4-OMe OMe 3-F-5-OCF_Three
U-4a 4- (U-3b) U-4b 2-Cl-4-OCF_Three    OMe 3-Cl-5-F
U-4a 4-CF₂H U-4b 2-Br-4-F OMe 3,5-di-Cl
U-4a 4-CN U-4b 2-Br-4-Cl OMe 3-Cl-5-Br
U-4a 4-Et U-4b 2,4-di-Br OMe 3-Cl-5-Me
U-4a 4-OCF₂H U-4b 2-Br-4-Me OMe 3-Cl-5-CF_Three
U-4a 4-OEt U-4b 2-Br-4-CF_Three     OMe 3-Cl-5-OMe
U-4a 4-C (O) CF_Three      U-4b 2-Br-4-OMe OMe 3-Cl-5-OCF_Three
U-4a 5-Ac U-4b 2-Br-4-OCF_Three    OMe 3-Br-5-F
U-4a 5- (U-3b) U-4b 2-Me-4-F OMe 3-Br-5-Cl
U-4a 5-CF₂H U-4b 2-Me-4-Cl OMe 3,5-di-Br
U-4a 5-CN U-4b 2-Me-4-Br OMe 3-Br-5-Me
U-4a 5-Et U-4b 2,4-di-Me OMe 3-Br-5-CF_Three
U-4a 5-OCF₂H U-4b 2-Me-4-CF_Three     OMe 3-Br-5-OMe
U-4a 5-OEt U-4b 2-Me-4-OMe OMe 3-Br-5-OCF_Three
U-4a 5-C (O) CF_Three      U-4b 2-Me-4-OCF_Three    OMe 3-Me-5-F
CF_Three   2-Ac U-4b 2-CF_Three-4-F OMe 3-Me-5-Cl
CF_Three   2- (U-3b) U-4b 2-CF_Three-4-Cl OMe 3-Me-5-Br
CF_Three   2-CF₂H U-4b 2-CF_Three-4-Br OMe 3,5-di-Me
CF_Three   2-CN U-4b 2-CF_Three-4-Me OMe 3-Me-5-CF_Three
CF_Three   2-Et U-4b 2,4-di-CF_Three     OMe 3-Me-5-OMe
CF_Three   2-OCF₂H U-4b 2-CF_Three-4-OMe OMe 3-Me-5-OCF_Three
CF_Three   2-OEt U-4b 2-CF_Three-4-OCF_Three   OMe 3-CF_Three-5-F
CF_Three   2-C (O) CF_Three      U-4b 2-OMe-4-F OMe 3-CF_Three-5-Cl
CF_Three   3-Ac U-4b 2-OMe-4-Cl OMe 3-CF_Three-5-Br
CF_Three   3- (U-3b) U-4b 2-OMe-4-Br OMe 3-CF_Three-5-Me
CF_Three   3-CF₂H U-4b 2-OMe-4-Me OMe 3,5-di-CF_Three
CF_Three   3-CN U-4b 2-OMe-4-CF_Three    OMe 3-CF_Three-5-OMe
CF_Three   3-Et U-4b 2,4-di-OMe OMe 3-CF_Three-5-OCF_Three
CF_Three   3-OCF₂H U-4b 2-OMe-4-OCF_Three   OMe 3-OMe-5-F
CF_Three   3-OEt U-4b 2-OCF_Three-4-F OMe 3-OMe-5-Cl
CF_Three   3-C (O) CF_Three      U-4b 2-OCF_Three-4-Cl OMe 3-OMe-5-Br
CF_Three   4-Ac U-4b 2-OCF_Three-4-Br OMe 3-OMe-5-Me
CF_Three   4- (U-3b) U-4b 2-OCF_Three-4-Me OMe 3-OMe-5-CF_Three
CF_Three   4-CF₂H U-4b 2-OCF_Three-4-CF_Three   OMe 3,5-di-OMe
CF_Three   4-CN U-4b 2-OCF_Three-4-OMe OMe 3-OMe-5-OCF_Three
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
CF_Three   4-Et U-4b 2,4-di-OCF_Three    OMe 3-OCF_Three-5-F
CF_Three   4-OCF₂H U-4b 2,5-di-F OMe 3-OCF_Three-5-Cl
CF_Three   4-OEt U-4b 2-F-5-Cl OMe 3-OCF_Three-5-Br
CF_Three   4-C (O) CF_Three      U-4b 2-F-5-Br OMe 3-OCF_Three-5-Me
CF_Three   5-Ac U-4b 2-F-5-Me OMe 3-OCF_Three-5-CF_Three
CF_Three   5- (U-3b) U-4b 2-F-5-CF_Three      OMe 3-OCF_Three-5-OMe
CF_Three   5-CF₂H U-4b 2-F-5-OMe OMe 3,5-di-OCF_Three
CF_Three   5-CN U-4b 2-F-5-OCF_Three     SMe 2,3-di-F
CF_Three   5-Et U-4b 2-Cl-5-F SMe 2-F-3-Cl
CF_Three   5-OCF₂H U-4b 2,5-di-Cl SMe 2-F-3-Br
CF_Three   5-OEt U-4b 2-Cl-5-Br SMe 2-F-3-Me
CF_Three   5-C (O) CF_Three      U-4b 2-Cl-5-Me SMe 2-F-3-CF_Three
cPr 2-Ac U-4b 2-Cl-5-CF_Three     SMe 2-F-3-OMe
cPr 2- (U-3b) U-4b 2-Cl-5-OMe SMe 2-F-3-OCF_Three
cPr 2-CF₂H U-4b 2-Cl-5-OCF_Three    SMe 2-Cl-3-F
cPr 2-CN U-4b 2-Br-5-F SMe 2,3-di-Cl
cPr 2-Et U-4b 2-Br-5-Cl SMe 2-Cl-3-Br
cPr 2-OCF₂H U-4b 2,5-di-Br SMe 2-Cl-3-Me
cPr 2-OEt U-4b 2-Br-5-Me SMe 2-Cl-3-CF_Three
cPr 2-C (O) CF_Three      U-4b 2-Br-5-CF_Three     SMe 2-Cl-3-OMe
cPr 3-Ac U-4b 2-Br-5-OMe SMe 2-Cl-3-OCF_Three
cPr 3- (U-3b) U-4b 2-Br-5-OCF_Three    SMe 2-Br-3-F
cPr 3-CF₂H U-4b 2-Me-5-F SMe 2-Br-3-Cl
cPr 3-CN U-4b 2-Me-5-Cl SMe 2,3-di-Br
cPr 3-Et U-4b 2-Me-5-Br SMe 2-Br-3-Me
cPr 3-OCF₂H U-4b 2,5-di-Me SMe 2-Br-3-CF_Three
cPr 3-OEt U-4b 2-Me-5-CF_Three     SMe 2-Br-3-OMe
cPr 3-C (O) CF_Three      U-4b 2-Me-5-OMe SMe 2-Br-3-OCF_Three
cPr 4-Ac U-4b 2-Me-5-OCF_Three    SMe 2-Me-3-F
cPr 4- (U-3b) U-4b 2-CF_Three-5-F SMe 2-Me-3-Cl
cPr 4-CF₂H U-4b 2-CF_Three-5-Cl SMe 2-Me-3-Br
cPr 4-CN U-4b 2-CF_Three-5-Br SMe 2,3-di-Me
cPr 4-Et U-4b 2-CF_Three-5-Me SMe 2-Me-3-CF_Three
cPr 4-OCF₂H U-4b 2,5-di-CF_Three     SMe 2-Me-3-OMe
cPr 4-OEt U-4b 2-CF_Three-5-OMe SMe 2-Me-3-OCF_Three
cPr 4-C (O) CF_Three      U-4b 2-CF_Three-5-OCF_Three   SMe 2-CF_Three-3-F
cPr 5-Ac U-4b 2-OMe-5-F SMe 2-CF_Three-3-Cl
cPr 5- (U-3b) U-4b 2-OMe-5-Cl SMe 2-CF_Three-3-Br
cPr 5-CF₂H U-4b 2-OMe-5-Br SMe 2-CF_Three-3-Me
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
cPr 5-CN U-4b 2-OMe-5-Me SMe 2,3-di-CF_Three
cPr 5-Et U-4b 2-OMe-5-CF_Three    SMe 2-CF_Three-3-OMe
cPr 5-OCF₂H U-4b 2,5-di-OMe SMe 2-CF_Three-3-OCF_Three
cPr 5-OEt U-4b 2-OMe-5-OCF_Three   SMe 2-OMe-3-F
cPr 5-C (O) CF_Three      U-4b 2-OCF_Three-5-F SMe 2-OMe-3-Cl
Me 2,3-di-F U-4b 2-OCF_Three-5-Cl SMe 2-OMe-3-Br
Me 2-F-3-Cl U-4b 2-OCF_Three-5-Br SMe 2-OMe-3-Me
Me 2-F-3-Br U-4b 2-OCF_Three-5-Me SMe 2-OMe-3-CF_Three
Me 2-F-3-Me U-4b 2-OCF_Three-5-CF_Three   SMe 2,3-di-OMe
Me 2-F-3-CF_Three      U-4b 2-OCF_Three-5-OMe SMe 2-OMe-3-OCF_Three
Me 2-F-3-OMe U-4b 2,5-di-OCF_Three    SMe 2-OCF_Three-3-F
Me 2-F-3-OCF_Three     U-4b 3,4-di-F SMe 2-OCF_Three-3-Cl
Me 2-Cl-3-F U-4b 3-F-4-Cl SMe 2-OCF_Three-3-Br
Me 2,3-di-Cl U-4b 3-F-4-Br SMe 2-OCF_Three-3-Me
Me 2-Cl-3-Br U-4b 3-F-4-Me SMe 2-OCF_Three-3-CF_Three
Me 2-Cl-3-Me U-4b 3-F-4-CF_Three      SMe 2-OCF_Three-3-OMe
Me 2-Cl-3-CF_Three     U-4b 3-F-4-OMe SMe 2,3-di-OCF_Three
Me 2-Cl-3-OMe U-4b 3-F-4-OCF_Three     SMe 2,4-di-F
Me 2-Cl-3-OCF_Three    U-4b 3-Cl-4-F SMe 2-F-4-Cl
Me 2-Br-3-F U-4b 3,4-di-Cl SMe 2-F-4-Br
Me 2-Br-3-Cl U-4b 3-Cl-4-Br SMe 2-F-4-Me
Me 2,3-di-Br U-4b 3-Cl-4-Me SMe 2-F-4-CF_Three
Me 2-Br-3-Me U-4b 3-Cl-4-CF_Three     SMe 2-F-4-OMe
Me 2-Br-3-CF_Three     U-4b 3-Cl-4-OMe SMe 2-F-4-OCF_Three
Me 2-Br-3-OMe U-4b 3-Cl-4-OCF_Three    SMe 2-Cl-4-F
Me 2-Br-3-OCF_Three    U-4b 3-Br-4-F SMe 2,4-di-Cl
Me 2-Me-3-F U-4b 3-Br-4-Cl SMe 2-Cl-4-Br
Me 2-Me-3-Cl U-4b 3,4-di-Br SMe 2-Cl-4-Me
Me 2-Me-3-Br U-4b 3-Br-4-Me SMe 2-Cl-4-CF_Three
Me 2,3-di-Me U-4b 3-Br-4-CF_Three     SMe 2-Cl-4-OMe
Me 2-Me-3-CF_Three     U-4b 3-Br-4-OMe SMe 2-Cl-4-OCF_Three
Me 2-Me-3-OMe U-4b 3-Br-4-OCF_Three    SMe 2-Br-4-F
Me 2-Me-3-OCF_Three    U-4b 3-Me-4-F SMe 2-Br-4-Cl
Me 2-CF_Three-3-F U-4b 3-Me-4-Cl SMe 2,4-di-Br
Me 2-CF_Three-3-Cl U-4b 3-Me-4-Br SMe 2-Br-4-Me
Me 2-CF_Three-3-Br U-4b 3,4-di-Me SMe 2-Br-4-CF_Three
Me 2-CF_Three-3-Me U-4b 3-Me-4-CF_Three     SMe 2-Br-4-OMe
Me 2,3-di-CF_Three     U-4b 3-Me-4-OMe SMe 2-Br-4-OCF_Three
Me 2-CF_Three-3-OMe U-4b 3-Me-4-OCF_Three    SMe 2-Me-4-F
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
Me 2-CF_Three-3-OCF_Three   U-4b 3-CF_Three-4-F SMe 2-Me-4-Cl
Me 2-OMe-3-F U-4b 3-CF_Three-4-Cl SMe 2-Me-4-Br
Me 2-OMe-3-Cl U-4b 3-CF_Three-4-Br SMe 2,4-di-Me
Me 2-OMe-3-Br U-4b 3-CF_Three-4-Me SMe 2-Me-4-CF_Three
Me 2-OMe-3-Me U-4b 3,4-di-CF_Three     SMe 2-Me-4-OMe
Me 2-OMe-3-CF_Three    U-4b 3-CF_Three-4-OMe SMe 2-Me-4-OCF_Three
Me 2,3-di-OMe U-4b 3-CF_Three-4-OCF_Three   SMe 2-CF_Three-4-F
Me 2-OMe-3-OCF_Three   U-4b 3-OMe-4-F SMe 2-CF_Three-4-Cl
Me 2-OCF_Three-3-F U-4b 3-OMe-4-Cl SMe 2-CF_Three-4-Br
Me 2-OCF_Three-3-Cl U-4b 3-OMe-4-Br SMe 2-CF_Three-4-Me
Me 2-OCF_Three-3-Br U-4b 3-OMe-4-Me SMe 2,4-di-CF_Three
Me 2-OCF_Three-3-Me U-4b 3-OMe-4-CF_Three    SMe 2-CF_Three-4-OMe
Me 2-OCF_Three-3-CF_Three   U-4b 3,4-di-OMe SMe 2-CF_Three-4-OCF_Three
Me 2-OCF_Three-3-OMe U-4b 3-OMe-4-OCF_Three   SMe 2-OMe-4-F
Me 2,3-di-OCF_Three    U-4b 3-OCF_Three-4-F SMe 2-OMe-4-Cl
Me 2,4-di-F U-4b 3-OCF_Three-4-Cl SMe 2-OMe-4-Br
Me 2-F-4-Cl U-4b 3-OCF_Three-4-Br SMe 2-OMe-4-Me
Me 2-F-4-Br U-4b 3-OCF_Three-4-Me SMe 2-OMe-4-CF_Three
Me 2-F-4-Me U-4b 3-OCF_Three-4-CF_Three   SMe 2,4-di-OMe
Me 2-F-4-CF_Three      U-4b 3-OCF_Three-4-OMe SMe 2-OMe-4-OCF_Three
Me 2-F-4-OMe U-4b 3,4-di-OCF_Three    SMe 2-OCF_Three-4-F
Me 2-F-4-OCF_Three     U-4b 3,5-di-F SMe 2-OCF_Three-4-Cl
Me 2-Cl-4-F U-4b 3-F-5-Cl SMe 2-OCF_Three-4-Br
Me 2,4-di-Cl U-4b 3-F-5-Br SMe 2-OCF_Three-4-Me
Me 2-Cl-4-Br U-4b 3-F-5-Me SMe 2-OCF_Three-4-CF_Three
Me 2-Cl-4-Me U-4b 3-F-5-CF_Three      SMe 2-OCF_Three-4-OMe
Me 2-Cl-4-CF_Three     U-4b 3-F-5-OMe SMe 2,4-di-OCF_Three
Me 2-Cl-4-OMe U-4b 3-F-5-OCF_Three     SMe 2,5-di-F
Me 2-Cl-4-OCF_Three    U-4b 3-Cl-5-F SMe 2-F-5-Cl
Me 2-Br-4-F U-4b 3,5-di-Cl SMe 2-F-5-Br
Me 2-Br-4-Cl U-4b 3-Cl-5-Br SMe 2-F-5-Me
Me 2,4-di-Br U-4b 3-Cl-5-Me SMe 2-F-5-CF_Three
Me 2-Br-4-Me U-4b 3-Cl-5-CF_Three     SMe 2-F-5-OMe
Me 2-Br-4-CF_Three     U-4b 3-Cl-5-OMe SMe 2-F-5-OCF_Three
Me 2-Br-4-OMe U-4b 3-Cl-5-OCF_Three    SMe 2-Cl-5-F
Me 2-Br-4-OCF_Three    U-4b 3-Br-5-F SMe 2,5-di-Cl
Me 2-Me-4-F U-4b 3-Br-5-Cl SMe 2-Cl-5-Br
Me 2-Me-4-Cl U-4b 3,5-di-Br SMe 2-Cl-5-Me
Me 2-Me-4-Br U-4b 3-Br-5-Me SMe 2-Cl-5-CF_Three
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
Me 2,4-di-Me U-4b 3-Br-5-CF_Three     SMe 2-Cl-5-OMe
Me 2-Me-4-CF_Three     U-4b 3-Br-5-OMe SMe 2-Cl-5-OCF_Three
Me 2-Me-4-OMe U-4b 3-Br-5-OCF_Three    SMe 2-Br-5-F
Me 2-Me-4-OCF_Three    U-4b 3-Me-5-F SMe 2-Br-5-Cl
Me 2-CF_Three-4-F U-4b 3-Me-5-Cl SMe 2,5-di-Br
Me 2-CF_Three-4-Cl U-4b 3-Me-5-Br SMe 2-Br-5-Me
Me 2-CF_Three-4-Br U-4b 3,5-di-Me SMe 2-Br-5-CF_Three
Me 2-CF_Three-4-Me U-4b 3-Me-5-CF_Three     SMe 2-Br-5-OMe
Me 2,4-di-CF_Three     U-4b 3-Me-5-OMe SMe 2-Br-5-OCF_Three
Me 2-CF_Three-4-OMe U-4b 3-Me-5-OCF_Three    SMe 2-Me-5-F
Me 2-CF_Three-4-OCF_Three   U-4b 3-CF_Three-5-F SMe 2-Me-5-Cl
Me 2-OMe-4-F U-4b 3-CF_Three-5-Cl SMe 2-Me-5-Br
Me 2-OMe-4-Cl U-4b 3-CF_Three-5-Br SMe 2,5-di-Me
Me 2-OMe-4-Br U-4b 3-CF_Three-5-Me SMe 2-Me-5-CF_Three
Me 2-OMe-4-Me U-4b 3,5-di-CF_Three     SMe 2-Me-5-OMe
Me 2-OMe-4-CF_Three    U-4b 3-CF_Three-5-OMe SMe 2-Me-5-OCF_Three
Me 2,4-di-OMe U-4b 3-CF_Three-5-OCF_Three   SMe 2-CF_Three-5-F
Me 2-OMe-4-OCF_Three   U-4b 3-OMe-5-F SMe 2-CF_Three-5-Cl
Me 2-OCF_Three-4-F U-4b 3-OMe-5-Cl SMe 2-CF_Three-5-Br
Me 2-OCF_Three-4-Cl U-4b 3-OMe-5-Br SMe 2-CF_Three-5-Me
Me 2-OCF_Three-4-Br U-4b 3-OMe-5-Me SMe 2,5-di-CF_Three
Me 2-OCF_Three-4-Me U-4b 3-OMe-5-CF_Three    SMe 2-CF_Three-5-OMe
Me 2-OCF_Three-4-CF_Three   U-4b 3,5-di-OMe SMe 2-CF_Three-5-OCF_Three
Me 2-OCF_Three-4-OMe U-4b 3-OMe-5-OCF_Three   SMe 2-OMe-5-F
Me 2,4-di-OCF_Three    U-4b 3-OCF_Three-5-F SMe 2-OMe-5-Cl
Me 2,5-di-F U-4b 3-OCF_Three-5-Cl SMe 2-OMe-5-Br
Me 2-F-5-Cl U-4b 3-OCF_Three-5-Br SMe 2-OMe-5-Me
Me 2-F-5-Br U-4b 3-OCF_Three-5-Me SMe 2-OMe-5-CF_Three
Me 2-F-5-Me U-4b 3-OCF_Three-5-CF_Three   SMe 2,5-di-OMe
Me 2-F-5-CF_Three      U-4b 3-OCF_Three-5-OMe SMe 2-OMe-5-OCF_Three
Me 2-F-5-OMe U-4b 3,5-di-OCF_Three    SMe 2-OCF_Three-5-F
Me 2-F-5-OCF_Three     U-4c 2,3-di-F SMe 2-OCF_Three-5-Cl
Me 2-Cl-5-F U-4c 2-F-3-Cl SMe 2-OCF_Three-5-Br
Me 2,5-di-Cl U-4c 2-F-3-Br SMe 2-OCF_Three-5-Me
Me 2-Cl-5-Br U-4c 2-F-3-Me SMe 2-OCF_Three-5-CF_Three
Me 2-Cl-5-Me U-4c 2-F-3-CF_Three      SMe 2-OCF_Three-5-OMe
Me 2-Cl-5-CF_Three     U-4c 2-F-3-OMe SMe 2,5-di-OCF_Three
Me 2-Cl-5-OMe U-4c 2-F-3-OCF_Three     SMe 3,4-di-F
Me 2-Cl-5-OCF_Three    U-4c 2-Cl-3-F SMe 3-F-4-Cl
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
Me 2-Br-5-F U-4c 2,3-di-Cl SMe 3-F-4-Br
Me 2-Br-5-Cl U-4c 2-Cl-3-Br SMe 3-F-4-Me
Me 2,5-di-Br U-4c 2-Cl-3-Me SMe 3-F-4-CF_Three
Me 2-Br-5-Me U-4c 2-Cl-3-CF_Three     SMe 3-F-4-OMe
Me 2-Br-5-CF_Three     U-4c 2-Cl-3-OMe SMe 3-F-4-OCF_Three
Me 2-Br-5-OMe U-4c 2-Cl-3-OCF_Three    SMe 3-Cl-4-F
Me 2-Br-5-OCF_Three    U-4c 2-Br-3-F SMe 3,4-di-Cl
Me 2-Me-5-F U-4c 2-Br-3-Cl SMe 3-Cl-4-Br
Me 2-Me-5-Cl U-4c 2,3-di-Br SMe 3-Cl-4-Me
Me 2-Me-5-Br U-4c 2-Br-3-Me SMe 3-Cl-4-CF_Three
Me 2,5-di-Me U-4c 2-Br-3-CF_Three     SMe 3-Cl-4-OMe
Me 2-Me-5-CF_Three     U-4c 2-Br-3-OMe SMe 3-Cl-4-OCF_Three
Me 2-Me-5-OMe U-4c 2-Br-3-OCF_Three    SMe 3-Br-4-F
Me 2-Me-5-OCF_Three    U-4c 2-Me-3-F SMe 3-Br-4-Cl
Me 2-CF_Three-5-F U-4c 2-Me-3-Cl SMe 3,4-di-Br
Me 2-CF_Three-5-Cl U-4c 2-Me-3-Br SMe 3-Br-4-Me
Me 2-CF_Three-5-Br U-4c 2,3-di-Me SMe 3-Br-4-CF_Three
Me 2-CF_Three-5-Me U-4c 2-Me-3-CF_Three     SMe 3-Br-4-OMe
Me 2,5-di-CF_Three     U-4c 2-Me-3-OMe SMe 3-Br-4-OCF_Three
Me 2-CF_Three-5-OMe U-4c 2-Me-3-OCF_Three    SMe 3-Me-4-F
Me 2-CF_Three-5-OCF_Three   U-4c 2-CF_Three-3-F SMe 3-Me-4-Cl
Me 2-OMe-5-F U-4c 2-CF_Three-3-Cl SMe 3-Me-4-Br
Me 2-OMe-5-Cl U-4c 2-CF_Three-3-Br SMe 3,4-di-Me
Me 2-OMe-5-Br U-4c 2-CF_Three-3-Me SMe 3-Me-4-CF_Three
Me 2-OMe-5-Me U-4c 2,3-di-CF_Three     SMe 3-Me-4-OMe
Me 2-OMe-5-CF_Three    U-4c 2-CF_Three-3-OMe SMe 3-Me-4-OCF_Three
Me 2,5-di-OMe U-4c 2-CF_Three-3-OCF_Three   SMe 3-CF_Three-4-F
Me 2-OMe-5-OCF_Three   U-4c 2-OMe-3-F SMe 3-CF_Three-4-Cl
Me 2-OCF_Three-5-F U-4c 2-OMe-3-Cl SMe 3-CF_Three-4-Br
Me 2-OCF_Three-5-Cl U-4c 2-OMe-3-Br SMe 3-CF_Three-4-Me
Me 2-OCF_Three-5-Br U-4c 2-OMe-3-Me SMe 3,4-di-CF_Three
Me 2-OCF_Three-5-Me U-4c 2-OMe-3-CF_Three    SMe 3-CF_Three-4-OMe
Me 2-OCF_Three-5-CF_Three   U-4c 2,3-di-OMe SMe 3-CF_Three-4-OCF_Three
Me 2-OCF_Three-5-OMe U-4c 2-OMe-3-OCF_Three   SMe 3-OMe-4-F
Me 2,5-di-OCF_Three    U-4c 2-OCF_Three-3-F SMe 3-OMe-4-Cl
Me 3,4-di-F U-4c 2-OCF_Three-3-Cl SMe 3-OMe-4-Br
Me 3-F-4-Cl U-4c 2-OCF_Three-3-Br SMe 3-OMe-4-Me
Me 3-F-4-Br U-4c 2-OCF_Three-3-Me SMe 3-OMe-4-CF_Three
Me 3-F-4-Me U-4c 2-OCF_Three-3-CF_Three   SMe 3,4-di-OMe
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
Me 3-F-4-CF_Three      U-4c 2-OCF_Three-3-OMe SMe 3-OMe-4-OCF_Three
Me 3-F-4-OMe U-4c 2,3-di-OCF_Three    SMe 3-OCF_Three-4-F
Me 3-F-4-OCF_Three     U-4c 2,4-di-F SMe 3-OCF_Three-4-Cl
Me 3-Cl-4-F U-4c 2-F-4-Cl SMe 3-OCF_Three-4-Br
Me 3,4-di-Cl U-4c 2-F-4-Br SMe 3-OCF_Three-4-Me
Me 3-Cl-4-Br U-4c 2-F-4-Me SMe 3-OCF_Three-4-CF_Three
Me 3-Cl-4-Me U-4c 2-F-4-CF_Three      SMe 3-OCF_Three-4-OMe
Me 3-Cl-4-CF_Three     U-4c 2-F-4-OMe SMe 3,4-di-OCF_Three
Me 3-Cl-4-OMe U-4c 2-F-4-OCF_Three     SMe 3,5-di-F
Me 3-Cl-4-OCF_Three    U-4c 2-Cl-4-F SMe 3-F-5-Cl
Me 3-Br-4-F U-4c 2,4-di-Cl SMe 3-F-5-Br
Me 3-Br-4-Cl U-4c 2-Cl-4-Br SMe 3-F-5-Me
Me 3,4-di-Br U-4c 2-Cl-4-Me SMe 3-F-5-CF_Three
Me 3-Br-4-Me U-4c 2-Cl-4-CF_Three     SMe 3-F-5-OMe
Me 3-Br-4-CF_Three     U-4c 2-Cl-4-OMe SMe 3-F-5-OCF_Three
Me 3-Br-4-OMe U-4c 2-Cl-4-OCF_Three    SMe 3-Cl-5-F
Me 3-Br-4-OCF_Three    U-4c 2-Br-4-F SMe 3,5-di-Cl
Me 3-Me-4-F U-4c 2-Br-4-Cl SMe 3-Cl-5-Br
Me 3-Me-4-Cl U-4c 2,4-di-Br SMe 3-Cl-5-Me
Me 3-Me-4-Br U-4c 2-Br-4-Me SMe 3-Cl-5-CF_Three
Me 3,4-di-Me U-4c 2-Br-4-CF_Three     SMe 3-Cl-5-OMe
Me 3-Me-4-CF_Three     U-4c 2-Br-4-OMe SMe 3-Cl-5-OCF_Three
Me 3-Me-4-OMe U-4c 2-Br-4-OCF_Three    SMe 3-Br-5-F
Me 3-Me-4-OCF_Three    U-4c 2-Me-4-F SMe 3-Br-5-Cl
Me 3-CF_Three-4-F U-4c 2-Me-4-Cl SMe 3,5-di-Br
Me 3-CF_Three-4-Cl U-4c 2-Me-4-Br SMe 3-Br-5-Me
Me 3-CF_Three-4-Br U-4c 2,4-di-Me SMe 3-Br-5-CF_Three
Me 3-CF_Three-4-Me U-4c 2-Me-4-CF_Three     SMe 3-Br-5-OMe
Me 3,4-di-CF_Three     U-4c 2-Me-4-OMe SMe 3-Br-5-OCF_Three
Me 3-CF_Three-4-OMe U-4c 2-Me-4-OCF_Three    SMe 3-Me-5-F
Me 3-CF_Three-4-OCF_Three   U-4c 2-CF_Three-4-F SMe 3-Me-5-Cl
Me 3-OMe-4-F U-4c 2-CF_Three-4-Cl SMe 3-Me-5-Br
Me 3-OMe-4-Cl U-4c 2-CF_Three-4-Br SMe 3,5-di-Me
Me 3-OMe-4-Br U-4c 2-CF_Three-4-Me SMe 3-Me-5-CF_Three
Me 3-OMe-4-Me U-4c 2,4-di-CF_Three     SMe 3-Me-5-OMe
Me 3-OMe-4-CF_Three    U-4c 2-CF_Three-4-OMe SMe 3-Me-5-OCF_Three
Me 3,4-di-OMe U-4c 2-CF_Three-4-OCF_Three   SMe 3-CF_Three-5-F
Me 3-OMe-4-OCF_Three   U-4c 2-OMe-4-F SMe 3-CF_Three-5-Cl
Me 3-OCF_Three-4-F U-4c 2-OMe-4-Cl SMe 3-CF_Three-5-Br
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
Me 3-OCF_Three-4-Cl U-4c 2-OMe-4-Br SMe 3-CF_Three-5-Me
Me 3-OCF_Three-4-Br U-4c 2-OMe-4-Me SMe 3,5-di-CF_Three
Me 3-OCF_Three-4-Me U-4c 2-OMe-4-CF_Three    SMe 3-CF_Three-5-OMe
Me 3-OCF_Three-4-CF_Three   U-4c 2,4-di-OMe SMe 3-CF_Three-5-OCF_Three
Me 3-OCF_Three-4-OMe U-4c 2-OMe-4-OCF_Three   SMe 3-OMe-5-F
Me 3,4-di-OCF_Three    U-4c 2-OCF_Three-4-F SMe 3-OMe-5-Cl
Me 3,5-di-F U-4c 2-OCF_Three-4-Cl SMe 3-OMe-5-Br
Me 3-F-5-Cl U-4c 2-OCF_Three-4-Br SMe 3-OMe-5-Me
Me 3-F-5-Br U-4c 2-OCF_Three-4-Me SMe 3-OMe-5-CF_Three
Me 3-F-5-Me U-4c 2-OCF_Three-4-CF_Three   SMe 3,5-di-OMe
Me 3-F-5-CF_Three      U-4c 2-OCF_Three-4-OMe SMe 3-OMe-5-OCF_Three
Me 3-F-5-OMe U-4c 2,4-di-OCF_Three    SMe 3-OCF_Three-5-F
Me 3-F-5-OCF_Three     U-4c 2,5-di-F SMe 3-OCF_Three-5-Cl
Me 3-Cl-5-F U-4c 2-F-5-Cl SMe 3-OCF_Three-5-Br
Me 3,5-di-Cl U-4c 2-F-5-Br SMe 3-OCF_Three-5-Me
Me 3-Cl-5-Br U-4c 2-F-5-Me SMe 3-OCF_Three-5-CF_Three
Me 3-Cl-5-Me U-4c 2-F-5-CF_Three      SMe 3-OCF_Three-5-OMe
Me 3-Cl-5-CF_Three     U-4c 2-F-5-OMe SMe 3,5-di-OCF_Three
Me 3-Cl-5-OMe U-4c 2-F-5-OCF_Three     Ac 2,3-di-F
Me 3-Cl-5-OCF_Three    U-4c 2-Cl-5-F Ac 2-F-3-Cl
Me 3-Br-5-F U-4c 2,5-di-Cl Ac 2-F-3-Br
Me 3-Br-5-Cl U-4c 2-Cl-5-Br Ac 2-F-3-Me
Me 3,5-di-Br U-4c 2-Cl-5-Me Ac 2-F-3-CF_Three
Me 3-Br-5-Me U-4c 2-Cl-5-CF_Three     Ac 2-F-3-OMe
Me 3-Br-5-CF_Three     U-4c 2-Cl-5-OMe Ac 2-F-3-OCF_Three
Me 3-Br-5-OMe U-4c 2-Cl-5-OCF_Three    Ac 2-Cl-3-F
Me 3-Br-5-OCF_Three    U-4c 2-Br-5-F Ac 2,3-di-Cl
Me 3-Me-5-F U-4c 2-Br-5-Cl Ac 2-Cl-3-Br
Me 3-Me-5-Cl U-4c 2,5-di-Br Ac 2-Cl-3-Me
Me 3-Me-5-Br U-4c 2-Br-5-Me Ac 2-Cl-3-CF_Three
Me 3,5-di-Me U-4c 2-Br-5-CF_Three     Ac 2-Cl-3-OMe
Me 3-Me-5-CF_Three     U-4c 2-Br-5-OMe Ac 2-Cl-3-OCF_Three
Me 3-Me-5-OMe U-4c 2-Br-5-OCF_Three    Ac 2-Br-3-F
Me 3-Me-5-OCF_Three    U-4c 2-Me-5-F Ac 2-Br-3-Cl
Me 3-CF_Three-5-F U-4c 2-Me-5-Cl Ac 2,3-di-Br
Me 3-CF_Three-5-Cl U-4c 2-Me-5-Br Ac 2-Br-3-Me
Me 3-CF_Three-5-Br U-4c 2,5-di-Me Ac 2-Br-3-CF_Three
Me 3-CF_Three-5-Me U-4c 2-Me-5-CF_Three     Ac 2-Br-3-OMe
Me 3,5-di-CF_Three     U-4c 2-Me-5-OMe Ac 2-Br-3-OCF_Three
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
Me 3-CF_Three-5-OMe U-4c 2-Me-5-OCF_Three    Ac 2-Me-3-F
Me 3-CF_Three-5-OCF_Three   U-4c 2-CF_Three-5-F Ac 2-Me-3-Cl
Me 3-OMe-5-F U-4c 2-CF_Three-5-Cl Ac 2-Me-3-Br
Me 3-OMe-5-Cl U-4c 2-CF_Three-5-Br Ac 2,3-di-Me
Me 3-OMe-5-Br U-4c 2-CF_Three-5-Me Ac 2-Me-3-CF_Three
Me 3-OMe-5-Me U-4c 2,5-di-CF_Three     Ac 2-Me-3-OMe
Me 3-OMe-5-CF_Three    U-4c 2-CF_Three-5-OMe Ac 2-Me-3-OCF_Three
Me 3,5-di-OMe U-4c 2-CF_Three-5-OCF_Three   Ac 2-CF_Three-3-F
Me 3-OMe-5-OCF_Three   U-4c 2-OMe-5-F Ac 2-CF_Three-3-Cl
Me 3-OCF_Three-5-F U-4c 2-OMe-5-Cl Ac 2-CF_Three-3-Br
Me 3-OCF_Three-5-Cl U-4c 2-OMe-5-Br Ac 2-CF_Three-3-Me
Me 3-OCF_Three-5-Br U-4c 2-OMe-5-Me Ac 2,3-di-CF_Three
Me 3-OCF_Three-5-Me U-4c 2-OMe-5-CF_Three    Ac 2-CF_Three-3-OMe
Me 3-OCF_Three-5-CF_Three   U-4c 2,5-di-OMe Ac 2-CF_Three-3-OCF_Three
Me 3-OCF_Three-5-OMe U-4c 2-OMe-5-OCF_Three   Ac 2-OMe-3-F
Me 3,5-di-OCF_Three    U-4c 2-OCF_Three-5-F Ac 2-OMe-3-Cl
Et 2,3-di-F U-4c 2-OCF_Three-5-Cl Ac 2-OMe-3-Br
Et 2-F-3-Cl U-4c 2-OCF_Three-5-Br Ac 2-OMe-3-Me
Et 2-F-3-Br U-4c 2-OCF_Three-5-Me Ac 2-OMe-3-CF_Three
Et 2-F-3-Me U-4c 2-OCF_Three-5-CF_Three   Ac 2,3-di-OMe
Et 2-F-3-CF_Three      U-4c 2-OCF_Three-5-OMe Ac 2-OMe-3-OCF_Three
Et 2-F-3-OMe U-4c 2,5-di-OCF_Three    Ac 2-OCF_Three-3-F
Et 2-F-3-OCF_Three     U-4c 3,4-di-F Ac 2-OCF_Three-3-Cl
Et 2-Cl-3-F U-4c 3-F-4-Cl Ac 2-OCF_Three-3-Br
Et 2,3-di-Cl U-4c 3-F-4-Br Ac 2-OCF_Three-3-Me
Et 2-Cl-3-Br U-4c 3-F-4-Me Ac 2-OCF_Three-3-CF_Three
Et 2-Cl-3-Me U-4c 3-F-4-CF_Three      Ac 2-OCF_Three-3-OMe
Et 2-Cl-3-CF_Three     U-4c 3-F-4-OMe Ac 2,3-di-OCF_Three
Et 2-Cl-3-OMe U-4c 3-F-4-OCF_Three     Ac 2,4-di-F
Et 2-Cl-3-OCF_Three    U-4c 3-Cl-4-F Ac 2-F-4-Cl
Et 2-Br-3-F U-4c 3,4-di-Cl Ac 2-F-4-Br
Et 2-Br-3-Cl U-4c 3-Cl-4-Br Ac 2-F-4-Me
Et 2,3-di-Br U-4c 3-Cl-4-Me Ac 2-F-4-CF_Three
Et 2-Br-3-Me U-4c 3-Cl-4-CF_Three     Ac 2-F-4-OMe
Et 2-Br-3-CF_Three     U-4c 3-Cl-4-OMe Ac 2-F-4-OCF_Three
Et 2-Br-3-OMe U-4c 3-Cl-4-OCF_Three    Ac 2-Cl-4-F
Et 2-Br-3-OCF_Three    U-4c 3-Br-4-F Ac 2,4-di-Cl
Et 2-Me-3-F U-4c 3-Br-4-Cl Ac 2-Cl-4-Br
Et 2-Me-3-Cl U-4c 3,4-di-Br Ac 2-Cl-4-Me
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
Et 2-Me-3-Br U-4c 3-Br-4-Me Ac 2-Cl-4-CF_Three
Et 2,3-di-Me U-4c 3-Br-4-CF_Three     Ac 2-Cl-4-OMe
Et 2-Me-3-CF_Three     U-4c 3-Br-4-OMe Ac 2-Cl-4-OCF_Three
Et 2-Me-3-OMe U-4c 3-Br-4-OCF_Three    Ac 2-Br-4-F
Et 2-Me-3-OCF_Three    U-4c 3-Me-4-F Ac 2-Br-4-Cl
Et 2-CF_Three-3-F U-4c 3-Me-4-Cl Ac 2,4-di-Br
Et 2-CF_Three-3-Cl U-4c 3-Me-4-Br Ac 2-Br-4-Me
Et 2-CF_Three-3-Br U-4c 3,4-di-Me Ac 2-Br-4-CF_Three
Et 2-CF_Three-3-Me U-4c 3-Me-4-CF_Three     Ac 2-Br-4-OMe
Et 2,3-di-CF_Three     U-4c 3-Me-4-OMe Ac 2-Br-4-OCF_Three
Et 2-CF_Three-3-OMe U-4c 3-Me-4-OCF_Three    Ac 2-Me-4-F
Et 2-CF_Three-3-OCF_Three   U-4c 3-CF_Three-4-F Ac 2-Me-4-Cl
Et 2-OMe-3-F U-4c 3-CF_Three-4-Cl Ac 2-Me-4-Br
Et 2-OMe-3-Cl U-4c 3-CF_Three-4-Br Ac 2,4-di-Me
Et 2-OMe-3-Br U-4c 3-CF_Three-4-Me Ac 2-Me-4-CF_Three
Et 2-OMe-3-Me U-4c 3,4-di-CF_Three     Ac 2-Me-4-OMe
Et 2-OMe-3-CF_Three    U-4c 3-CF_Three-4-OMe Ac 2-Me-4-OCF_Three
Et 2,3-di-OMe U-4c 3-CF_Three-4-OCF_Three   Ac 2-CF_Three-4-F
Et 2-OMe-3-OCF_Three   U-4c 3-OMe-4-F Ac 2-CF_Three-4-Cl
Et 2-OCF_Three-3-F U-4c 3-OMe-4-Cl Ac 2-CF_Three-4-Br
Et 2-OCF_Three-3-Cl U-4c 3-OMe-4-Br Ac 2-CF_Three-4-Me
Et 2-OCF_Three-3-Br U-4c 3-OMe-4-Me Ac 2,4-di-CF_Three
Et 2-OCF_Three-3-Me U-4c 3-OMe-4-CF_Three    Ac 2-CF_Three-4-OMe
Et 2-OCF_Three-3-CF_Three   U-4c 3,4-di-OMe Ac 2-CF_Three-4-OCF_Three
Et 2-OCF_Three-3-OMe U-4c 3-OMe-4-OCF_Three   Ac 2-OMe-4-F
Et 2,3-di-OCF_Three    U-4c 3-OCF_Three-4-F Ac 2-OMe-4-Cl
Et 2,4-di-F U-4c 3-OCF_Three-4-Cl Ac 2-OMe-4-Br
Et 2-F-4-Cl U-4c 3-OCF_Three-4-Br Ac 2-OMe-4-Me
Et 2-F-4-Br U-4c 3-OCF_Three-4-Me Ac 2-OMe-4-CF_Three
Et 2-F-4-Me U-4c 3-OCF_Three-4-CF_Three   Ac 2,4-di-OMe
Et 2-F-4-CF_Three      U-4c 3-OCF_Three-4-OMe Ac 2-OMe-4-OCF_Three
Et 2-F-4-OMe U-4c 3,4-di-OCF_Three    Ac 2-OCF_Three-4-F
Et 2-F-4-OCF_Three     U-4c 3,5-di-F Ac 2-OCF_Three-4-Cl
Et 2-Cl-4-F U-4c 3-F-5-Cl Ac 2-OCF_Three-4-Br
Et 2,4-di-Cl U-4c 3-F-5-Br Ac 2-OCF_Three-4-Me
Et 2-Cl-4-Br U-4c 3-F-5-Me Ac 2-OCF_Three-4-CF_Three
Et 2-Cl-4-Me U-4c 3-F-5-CF_Three      Ac 2-OCF_Three-4-OMe
Et 2-Cl-4-CF_Three     U-4c 3-F-5-OMe Ac 2,4-di-OCF_Three
Et 2-Cl-4-OMe U-4c 3-F-5-OCF_Three     Ac 2,5-di-F
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
Et 2-Cl-4-OCF_Three    U-4c 3-Cl-5-F Ac 2-F-5-Cl
Et 2-Br-4-F U-4c 3,5-di-Cl Ac 2-F-5-Br
Et 2-Br-4-Cl U-4c 3-Cl-5-Br Ac 2-F-5-Me
Et 2,4-di-Br U-4c 3-Cl-5-Me Ac 2-F-5-CF_Three
Et 2-Br-4-Me U-4c 3-Cl-5-CF_Three     Ac 2-F-5-OMe
Et 2-Br-4-CF_Three     U-4c 3-Cl-5-OMe Ac 2-F-5-OCF_Three
Et 2-Br-4-OMe U-4c 3-Cl-5-OCF_Three    Ac 2-Cl-5-F
Et 2-Br-4-OCF_Three    U-4c 3-Br-5-F Ac 2,5-di-Cl
Et 2-Me-4-F U-4c 3-Br-5-Cl Ac 2-Cl-5-Br
Et 2-Me-4-Cl U-4c 3,5-di-Br Ac 2-Cl-5-Me
Et 2-Me-4-Br U-4c 3-Br-5-Me Ac 2-Cl-5-CF_Three
Et 2,4-di-Me U-4c 3-Br-5-CF_Three     Ac 2-Cl-5-OMe
Et 2-Me-4-CF_Three     U-4c 3-Br-5-OMe Ac 2-Cl-5-OCF_Three
Et 2-Me-4-OMe U-4c 3-Br-5-OCF_Three    Ac 2-Br-5-F
Et 2-Me-4-OCF_Three    U-4c 3-Me-5-F Ac 2-Br-5-Cl
Et 2-CF_Three-4-F U-4c 3-Me-5-Cl Ac 2,5-di-Br
Et 2-CF_Three-4-Cl U-4c 3-Me-5-Br Ac 2-Br-5-Me
Et 2-CF_Three-4-Br U-4c 3,5-di-Me Ac 2-Br-5-CF_Three
Et 2-CF_Three-4-Me U-4c 3-Me-5-CF_Three     Ac 2-Br-5-OMe
Et 2,4-di-CF_Three     U-4c 3-Me-5-OMe Ac 2-Br-5-OCF_Three
Et 2-CF_Three-4-OMe U-4c 3-Me-5-OCF_Three    Ac 2-Me-5-F
Et 2-CF_Three-4-OCF_Three   U-4c 3-CF_Three-5-F Ac 2-Me-5-Cl
Et 2-OMe-4-F U-4c 3-CF_Three-5-Cl Ac 2-Me-5-Br
Et 2-OMe-4-Cl U-4c 3-CF_Three-5-Br Ac 2,5-di-Me
Et 2-OMe-4-Br U-4c 3-CF_Three-5-Me Ac 2-Me-5-CF_Three
Et 2-OMe-4-Me U-4c 3,5-di-CF_Three     Ac 2-Me-5-OMe
Et 2-OMe-4-CF_Three    U-4c 3-CF_Three-5-OMe Ac 2-Me-5-OCF_Three
Et 2,4-di-OMe U-4c 3-CF_Three-5-OCF_Three   Ac 2-CF_Three-5-F
Et 2-OMe-4-OCF_Three   U-4c 3-OMe-5-F Ac 2-CF_Three-5-Cl
Et 2-OCF_Three-4-F U-4c 3-OMe-5-Cl Ac 2-CF_Three-5-Br
Et 2-OCF_Three-4-Cl U-4c 3-OMe-5-Br Ac 2-CF_Three-5-Me
Et 2-OCF_Three-4-Br U-4c 3-OMe-5-Me Ac 2,5-di-CF_Three
Et 2-OCF_Three-4-Me U-4c 3-OMe-5-CF_Three    Ac 2-CF_Three-5-OMe
Et 2-OCF_Three-4-CF_Three   U-4c 3,5-di-OMe Ac 2-CF_Three-5-OCF_Three
Et 2-OCF_Three-4-OMe U-4c 3-OMe-5-OCF_Three   Ac 2-OMe-5-F
Et 2,4-di-OCF_Three    U-4c 3-OCF_Three-5-F Ac 2-OMe-5-Cl
Et 2,5-di-F U-4c 3-OCF_Three-5-Cl Ac 2-OMe-5-Br
Et 2-F-5-Cl U-4c 3-OCF_Three-5-Br Ac 2-OMe-5-Me
Et 2-F-5-Br U-4c 3-OCF_Three-5-Me Ac 2-OMe-5-CF_Three
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
Et 2-F-5-Me U-4c 3-OCF_Three-5-CF_Three   Ac 2,5-di-OMe
Et 2-F-5-CF_Three      U-4c 3-OCF_Three-5-OMe Ac 2-OMe-5-OCF_Three
Et 2-F-5-OMe U-4c 3,5-di-OCF_Three    Ac 2-OCF_Three-5-F
Et 2-F-5-OCF_Three     U-4d 2,3-di-F Ac 2-OCF_Three-5-Cl
Et 2-Cl-5-F U-4d 2-F-3-Cl Ac 2-OCF_Three-5-Br
Et 2,5-di-Cl U-4d 2-F-3-Br Ac 2-OCF_Three-5-Me
Et 2-Cl-5-Br U-4d 2-F-3-Me Ac 2-OCF_Three-5-CF_Three
Et 2-Cl-5-Me U-4d 2-F-3-CF_Three      Ac 2-OCF_Three-5-OMe
Et 2-Cl-5-CF_Three     U-4d 2-F-3-OMe Ac 2,5-di-OCF_Three
Et 2-Cl-5-OMe U-4d 2-F-3-OCF_Three     Ac 3,4-di-F
Et 2-Cl-5-OCF_Three    U-4d 2-Cl-3-F Ac 3-F-4-Cl
Et 2-Br-5-F U-4d 2,3-di-Cl Ac 3-F-4-Br
Et 2-Br-5-Cl U-4d 2-Cl-3-Br Ac 3-F-4-Me
Et 2,5-di-Br U-4d 2-Cl-3-Me Ac 3-F-4-CF_Three
Et 2-Br-5-Me U-4d 2-Cl-3-CF_Three     Ac 3-F-4-OMe
Et 2-Br-5-CF_Three     U-4d 2-Cl-3-OMe Ac 3-F-4-OCF_Three
Et 2-Br-5-OMe U-4d 2-Cl-3-OCF_Three    Ac 3-Cl-4-F
Et 2-Br-5-OCF_Three    U-4d 2-Br-3-F Ac 3,4-di-Cl
Et 2-Me-5-F U-4d 2-Br-3-Cl Ac 3-Cl-4-Br
Et 2-Me-5-Cl U-4d 2,3-di-Br Ac 3-Cl-4-Me
Et 2-Me-5-Br U-4d 2-Br-3-Me Ac 3-Cl-4-CF_Three
Et 2,5-di-Me U-4d 2-Br-3-CF_Three     Ac 3-Cl-4-OMe
Et 2-Me-5-CF_Three     U-4d 2-Br-3-OMe Ac 3-Cl-4-OCF_Three
Et 2-Me-5-OMe U-4d 2-Br-3-OCF_Three    Ac 3-Br-4-F
Et 2-Me-5-OCF_Three    U-4d 2-Me-3-F Ac 3-Br-4-Cl
Et 2-CF_Three-5-F U-4d 2-Me-3-Cl Ac 3,4-di-Br
Et 2-CF_Three-5-Cl U-4d 2-Me-3-Br Ac 3-Br-4-Me
Et 2-CF_Three-5-Br U-4d 2,3-di-Me Ac 3-Br-4-CF_Three
Et 2-CF_Three-5-Me U-4d 2-Me-3-CF_Three     Ac 3-Br-4-OMe
Et 2,5-di-CF_Three     U-4d 2-Me-3-OMe Ac 3-Br-4-OCF_Three
Et 2-CF_Three-5-OMe U-4d 2-Me-3-OCF_Three    Ac 3-Me-4-F
Et 2-CF_Three-5-OCF_Three   U-4d 2-CF_Three-3-F Ac 3-Me-4-Cl
Et 2-OMe-5-F U-4d 2-CF_Three-3-Cl Ac 3-Me-4-Br
Et 2-OMe-5-Cl U-4d 2-CF_Three-3-Br Ac 3,4-di-Me
Et 2-OMe-5-Br U-4d 2-CF_Three-3-Me Ac 3-Me-4-CF_Three
Et 2-OMe-5-Me U-4d 2,3-di-CF_Three     Ac 3-Me-4-OMe
Et 2-OMe-5-CF_Three    U-4d 2-CF_Three-3-OMe Ac 3-Me-4-OCF_Three
Et 2,5-di-OMe U-4d 2-CF_Three-3-OCF_Three   Ac 3-CF_Three-4-F
Et 2-OMe-5-OCF_Three   U-4d 2-OMe-3-F Ac 3-CF_Three-4-Cl
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
Et 2-OCF_Three-5-F U-4d 2-OMe-3-Cl Ac 3-CF_Three-4-Br
Et 2-OCF_Three-5-Cl U-4d 2-OMe-3-Br Ac 3-CF_Three-4-Me
Et 2-OCF_Three-5-Br U-4d 2-OMe-3-Me Ac 3,4-di-CF_Three
Et 2-OCF_Three-5-Me U-4d 2-OMe-3-CF_Three    Ac 3-CF_Three-4-OMe
Et 2-OCF_Three-5-CF_Three   U-4d 2,3-di-OMe Ac 3-CF_Three-4-OCF_Three
Et 2-OCF_Three-5-OMe U-4d 2-OMe-3-OCF_Three   Ac 3-OMe-4-F
Et 2,5-di-OCF_Three    U-4d 2-OCF_Three-3-F Ac 3-OMe-4-Cl
Et 3,4-di-F U-4d 2-OCF_Three-3-Cl Ac 3-OMe-4-Br
Et 3-F-4-Cl U-4d 2-OCF_Three-3-Br Ac 3-OMe-4-Me
Et 3-F-4-Br U-4d 2-OCF_Three-3-Me Ac 3-OMe-4-CF_Three
Et 3-F-4-Me U-4d 2-OCF_Three-3-CF_Three   Ac 3,4-di-OMe
Et 3-F-4-CF_Three      U-4d 2-OCF_Three-3-OMe Ac 3-OMe-4-OCF_Three
Et 3-F-4-OMe U-4d 2,3-di-OCF_Three    Ac 3-OCF_Three-4-F
Et 3-F-4-OCF_Three     U-4d 2,4-di-F Ac 3-OCF_Three-4-Cl
Et 3-Cl-4-F U-4d 2-F-4-Cl Ac 3-OCF_Three-4-Br
Et 3,4-di-Cl U-4d 2-F-4-Br Ac 3-OCF_Three-4-Me
Et 3-Cl-4-Br U-4d 2-F-4-Me Ac 3-OCF_Three-4-CF_Three
Et 3-Cl-4-Me U-4d 2-F-4-CF_Three      Ac 3-OCF_Three-4-OMe
Et 3-Cl-4-CF_Three     U-4d 2-F-4-OMe Ac 3,4-di-OCF_Three
Et 3-Cl-4-OMe U-4d 2-F-4-OCF_Three     Ac 3,5-di-F
Et 3-Cl-4-OCF_Three    U-4d 2-Cl-4-F Ac 3-F-5-Cl
Et 3-Br-4-F U-4d 2,4-di-Cl Ac 3-F-5-Br
Et 3-Br-4-Cl U-4d 2-Cl-4-Br Ac 3-F-5-Me
Et 3,4-di-Br U-4d 2-Cl-4-Me Ac 3-F-5-CF_Three
Et 3-Br-4-Me U-4d 2-Cl-4-CF_Three     Ac 3-F-5-OMe
Et 3-Br-4-CF_Three     U-4d 2-Cl-4-OMe Ac 3-F-5-OCF_Three
Et 3-Br-4-OMe U-4d 2-Cl-4-OCF_Three    Ac 3-Cl-5-F
Et 3-Br-4-OCF_Three    U-4d 2-Br-4-F Ac 3,5-di-Cl
Et 3-Me-4-F U-4d 2-Br-4-Cl Ac 3-Cl-5-Br
Et 3-Me-4-Cl U-4d 2,4-di-Br Ac 3-Cl-5-Me
Et 3-Me-4-Br U-4d 2-Br-4-Me Ac 3-Cl-5-CF_Three
Et 3,4-di-Me U-4d 2-Br-4-CF_Three     Ac 3-Cl-5-OMe
Et 3-Me-4-CF_Three     U-4d 2-Br-4-OMe Ac 3-Cl-5-OCF_Three
Et 3-Me-4-OMe U-4d 2-Br-4-OCF_Three    Ac 3-Br-5-F
Et 3-Me-4-OCF_Three    U-4d 2-Me-4-F Ac 3-Br-5-Cl
Et 3-CF_Three-4-F U-4d 2-Me-4-Cl Ac 3,5-di-Br
Et 3-CF_Three-4-Cl U-4d 2-Me-4-Br Ac 3-Br-5-Me
Et 3-CF_Three-4-Br U-4d 2,4-di-Me Ac 3-Br-5-CF_Three
Et 3-CF_Three-4-Me U-4d 2-Me-4-CF_Three     Ac 3-Br-5-OMe
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
Et 3,4-di-CF_Three     U-4d 2-Me-4-OMe Ac 3-Br-5-OCF_Three
Et 3-CF_Three-4-OMe U-4d 2-Me-4-OCF_Three    Ac 3-Me-5-F
Et 3-CF_Three-4-OCF_Three   U-4d 2-CF_Three-4-F Ac 3-Me-5-Cl
Et 3-OMe-4-F U-4d 2-CF_Three-4-Cl Ac 3-Me-5-Br
Et 3-OMe-4-Cl U-4d 2-CF_Three-4-Br Ac 3,5-di-Me
Et 3-OMe-4-Br U-4d 2-CF_Three-4-Me Ac 3-Me-5-CF_Three
Et 3-OMe-4-Me U-4d 2,4-di-CF_Three     Ac 3-Me-5-OMe
Et 3-OMe-4-CF_Three    U-4d 2-CF_Three-4-OMe Ac 3-Me-5-OCF_Three
Et 3,4-di-OMe U-4d 2-CF_Three-4-OCF_Three   Ac 3-CF_Three-5-F
Et 3-OMe-4-OCF_Three   U-4d 2-OMe-4-F Ac 3-CF_Three-5-Cl
Et 3-OCF_Three-4-F U-4d 2-OMe-4-Cl Ac 3-CF_Three-5-Br
Et 3-OCF_Three-4-Cl U-4d 2-OMe-4-Br Ac 3-CF_Three-5-Me
Et 3-OCF_Three-4-Br U-4d 2-OMe-4-Me Ac 3,5-di-CF_Three
Et 3-OCF_Three-4-Me U-4d 2-OMe-4-CF_Three    Ac 3-CF_Three-5-OMe
Et 3-OCF_Three-4-CF_Three   U-4d 2,4-di-OMe Ac 3-CF_Three-5-OCF_Three
Et 3-OCF_Three-4-OMe U-4d 2-OMe-4-OCF_Three   Ac 3-OMe-5-F
Et 3,4-di-OCF_Three    U-4d 2-OCF_Three-4-F Ac 3-OMe-5-Cl
Et 3,5-di-F U-4d 2-OCF_Three-4-Cl Ac 3-OMe-5-Br
Et 3-F-5-Cl U-4d 2-OCF_Three-4-Br Ac 3-OMe-5-Me
Et 3-F-5-Br U-4d 2-OCF_Three-4-Me Ac 3-OMe-5-CF_Three
Et 3-F-5-Me U-4d 2-OCF_Three-4-CF_Three   Ac 3,5-di-OMe
Et 3-F-5-CF_Three      U-4d 2-OCF_Three-4-OMe Ac 3-OMe-5-OCF_Three
Et 3-F-5-OMe U-4d 2,4-di-OCF_Three    Ac 3-OCF_Three-5-F
Et 3-F-5-OCF_Three     U-4d 2,5-di-F Ac 3-OCF_Three-5-Cl
Et 3-Cl-5-F U-4d 2-F-5-Cl Ac 3-OCF_Three-5-Br
Et 3,5-di-Cl U-4d 2-F-5-Br Ac 3-OCF_Three-5-Me
Et 3-Cl-5-Br U-4d 2-F-5-Me Ac 3-OCF_Three-5-CF_Three
Et 3-Cl-5-Me U-4d 2-F-5-CF_Three      Ac 3-OCF_Three-5-OMe
Et 3-Cl-5-CF_Three     U-4d 2-F-5-OMe Ac 3,5-di-OCF_Three
Et 3-Cl-5-OMe U-4d 2-F-5-OCF_Three     cPen 2,3-di-F
Et 3-Cl-5-OCF_Three    U-4d 2-Cl-5-F cPen 2-F-3-Cl
Et 3-Br-5-F U-4d 2,5-di-Cl cPen 2-F-3-Br
Et 3-Br-5-Cl U-4d 2-Cl-5-Br cPen 2-F-3-Me
Et 3,5-di-Br U-4d 2-Cl-5-Me cPen 2-F-3-CF_Three
Et 3-Br-5-Me U-4d 2-Cl-5-CF_Three     cPen 2-F-3-OMe
Et 3-Br-5-CF_Three     U-4d 2-Cl-5-OMe cPen 2-F-3-OCF_Three
Et 3-Br-5-OMe U-4d 2-Cl-5-OCF_Three    cPen 2-Cl-3-F
Et 3-Br-5-OCF_Three    U-4d 2-Br-5-F cPen 2,3-di-Cl
Et 3-Me-5-F U-4d 2-Br-5-Cl cPen 2-Cl-3-Br
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
Et 3-Me-5-Cl U-4d 2,5-di-Br cPen 2-Cl-3-Me
Et 3-Me-5-Br U-4d 2-Br-5-Me cPen 2-Cl-3-CF_Three
Et 3,5-di-Me U-4d 2-Br-5-CF_Three     cPen 2-Cl-3-OMe
Et 3-Me-5-CF_Three     U-4d 2-Br-5-OMe cPen 2-Cl-3-OCF_Three
Et 3-Me-5-OMe U-4d 2-Br-5-OCF_Three    cPen 2-Br-3-F
Et 3-Me-5-OCF_Three    U-4d 2-Me-5-F cPen 2-Br-3-Cl
Et 3-CF_Three-5-F U-4d 2-Me-5-Cl cPen 2,3-di-Br
Et 3-CF_Three-5-Cl U-4d 2-Me-5-Br cPen 2-Br-3-Me
Et 3-CF_Three-5-Br U-4d 2,5-di-Me cPen 2-Br-3-CF_Three
Et 3-CF_Three-5-Me U-4d 2-Me-5-CF_Three     cPen 2-Br-3-OMe
Et 3,5-di-CF_Three     U-4d 2-Me-5-OMe cPen 2-Br-3-OCF_Three
Et 3-CF_Three-5-OMe U-4d 2-Me-5-OCF_Three    cPen 2-Me-3-F
Et 3-CF_Three-5-OCF_Three   U-4d 2-CF_Three-5-F cPen 2-Me-3-Cl
Et 3-OMe-5-F U-4d 2-CF_Three-5-Cl cPen 2-Me-3-Br
Et 3-OMe-5-Cl U-4d 2-CF_Three-5-Br cPen 2,3-di-Me
Et 3-OMe-5-Br U-4d 2-CF_Three-5-Me cPen 2-Me-3-CF_Three
Et 3-OMe-5-Me U-4d 2,5-di-CF_Three     cPen 2-Me-3-OMe
Et 3-OMe-5-CF_Three    U-4d 2-CF_Three-5-OMe cPen 2-Me-3-OCF_Three
Et 3,5-di-OMe U-4d 2-CF_Three-5-OCF_Three   cPen 2-CF_Three-3-F
Et 3-OMe-5-OCF_Three   U-4d 2-OMe-5-F cPen 2-CF_Three-3-Cl
Et 3-OCF_Three-5-F U-4d 2-OMe-5-Cl cPen 2-CF_Three-3-Br
Et 3-OCF_Three-5-Cl U-4d 2-OMe-5-Br cPen 2-CF_Three-3-Me
Et 3-OCF_Three-5-Br U-4d 2-OMe-5-Me cPen 2,3-di-CF_Three
Et 3-OCF_Three-5-Me U-4d 2-OMe-5-CF_Three    cPen 2-CF_Three-3-OMe
Et 3-OCF_Three-5-CF_Three   U-4d 2,5-di-OMe cPen 2-CF_Three-3-OCF_Three
Et 3-OCF_Three-5-OMe U-4d 2-OMe-5-OCF_Three   cPen 2-OMe-3-F
Et 3,5-di-OCF_Three    U-4d 2-OCF_Three-5-F cPen 2-OMe-3-Cl
iPr 2,3-di-F U-4d 2-OCF_Three-5-Cl cPen 2-OMe-3-Br
iPr 2-F-3-Cl U-4d 2-OCF_Three-5-Br cPen 2-OMe-3-Me
iPr 2-F-3-Br U-4d 2-OCF_Three-5-Me cPen 2-OMe-3-CF_Three
iPr 2-F-3-Me U-4d 2-OCF_Three-5-CF_Three   cPen 2,3-di-OMe
iPr 2-F-3-CF_Three      U-4d 2-OCF_Three-5-OMe cPen 2-OMe-3-OCF_Three
iPr 2-F-3-OMe U-4d 2,5-di-OCF_Three    cPen 2-OCF_Three-3-F
iPr 2-F-3-OCF_Three     U-4d 3,4-di-F cPen 2-OCF_Three-3-Cl
iPr 2-Cl-3-F U-4d 3-F-4-Cl cPen 2-OCF_Three-3-Br
iPr 2,3-di-Cl U-4d 3-F-4-Br cPen 2-OCF_Three-3-Me
iPr 2-Cl-3-Br U-4d 3-F-4-Me cPen 2-OCF_Three-3-CF_Three
iPr 2-Cl-3-Me U-4d 3-F-4-CF_Three      cPen 2-OCF_Three-3-OMe
iPr 2-Cl-3-CF_Three     U-4d 3-F-4-OMe cPen 2,3-di-OCF_Three
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
iPr 2-Cl-3-OMe U-4d 3-F-4-OCF_Three     cPen 2,4-di-F
iPr 2-Cl-3-OCF_Three    U-4d 3-Cl-4-F cPen 2-F-4-Cl
iPr 2-Br-3-F U-4d 3,4-di-Cl cPen 2-F-4-Br
iPr 2-Br-3-Cl U-4d 3-Cl-4-Br cPen 2-F-4-Me
iPr 2,3-di-Br U-4d 3-Cl-4-Me cPen 2-F-4-CF_Three
iPr 2-Br-3-Me U-4d 3-Cl-4-CF_Three     cPen 2-F-4-OMe
iPr 2-Br-3-CF_Three     U-4d 3-Cl-4-OMe cPen 2-F-4-OCF_Three
iPr 2-Br-3-OMe U-4d 3-Cl-4-OCF_Three    cPen 2-Cl-4-F
iPr 2-Br-3-OCF_Three    U-4d 3-Br-4-F cPen 2,4-di-Cl
iPr 2-Me-3-F U-4d 3-Br-4-Cl cPen 2-Cl-4-Br
iPr 2-Me-3-Cl U-4d 3,4-di-Br cPen 2-Cl-4-Me
iPr 2-Me-3-Br U-4d 3-Br-4-Me cPen 2-Cl-4-CF_Three
iPr 2,3-di-Me U-4d 3-Br-4-CF_Three     cPen 2-Cl-4-OMe
iPr 2-Me-3-CF_Three     U-4d 3-Br-4-OMe cPen 2-Cl-4-OCF_Three
iPr 2-Me-3-OMe U-4d 3-Br-4-OCF_Three    cPen 2-Br-4-F
iPr 2-Me-3-OCF_Three    U-4d 3-Me-4-F cPen 2-Br-4-Cl
iPr 2-CF_Three-3-F U-4d 3-Me-4-Cl cPen 2,4-di-Br
iPr 2-CF_Three-3-Cl U-4d 3-Me-4-Br cPen 2-Br-4-Me
iPr 2-CF_Three-3-Br U-4d 3,4-di-Me cPen 2-Br-4-CF_Three
iPr 2-CF_Three-3-Me U-4d 3-Me-4-CF_Three     cPen 2-Br-4-OMe
iPr 2,3-di-CF_Three     U-4d 3-Me-4-OMe cPen 2-Br-4-OCF_Three
iPr 2-CF_Three-3-OMe U-4d 3-Me-4-OCF_Three    cPen 2-Me-4-F
iPr 2-CF_Three-3-OCF_Three   U-4d 3-CF_Three-4-F cPen 2-Me-4-Cl
iPr 2-OMe-3-F U-4d 3-CF_Three-4-Cl cPen 2-Me-4-Br
iPr 2-OMe-3-Cl U-4d 3-CF_Three-4-Br cPen 2,4-di-Me
iPr 2-OMe-3-Br U-4d 3-CF_Three-4-Me cPen 2-Me-4-CF_Three
iPr 2-OMe-3-Me U-4d 3,4-di-CF_Three     cPen 2-Me-4-OMe
iPr 2-OMe-3-CF_Three    U-4d 3-CF_Three-4-OMe cPen 2-Me-4-OCF_Three
iPr 2,3-di-OMe U-4d 3-CF_Three-4-OCF_Three   cPen 2-CF_Three-4-F
iPr 2-OMe-3-OCF_Three   U-4d 3-OMe-4-F cPen 2-CF_Three-4-Cl
iPr 2-OCF_Three-3-F U-4d 3-OMe-4-Cl cPen 2-CF_Three-4-Br
iPr 2-OCF_Three-3-Cl U-4d 3-OMe-4-Br cPen 2-CF_Three-4-Me
iPr 2-OCF_Three-3-Br U-4d 3-OMe-4-Me cPen 2,4-di-CF_Three
iPr 2-OCF_Three-3-Me U-4d 3-OMe-4-CF_Three    cPen 2-CF_Three-4-OMe
iPr 2-OCF_Three-3-CF_Three   U-4d 3,4-di-OMe cPen 2-CF_Three-4-OCF_Three
iPr 2-OCF_Three-3-OMe U-4d 3-OMe-4-OCF_Three   cPen 2-OMe-4-F
iPr 2,3-di-OCF_Three    U-4d 3-OCF_Three-4-F cPen 2-OMe-4-Cl
iPr 2,4-di-F U-4d 3-OCF_Three-4-Cl cPen 2-OMe-4-Br
iPr 2-F-4-Cl U-4d 3-OCF_Three-4-Br cPen 2-OMe-4-Me
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
iPr 2-F-4-Br U-4d 3-OCF_Three-4-Me cPen 2-OMe-4-CF_Three
iPr 2-F-4-Me U-4d 3-OCF_Three-4-CF_Three   cPen 2,4-di-OMe
iPr 2-F-4-CF_Three      U-4d 3-OCF_Three-4-OMe cPen 2-OMe-4-OCF_Three
iPr 2-F-4-OMe U-4d 3,4-di-OCF_Three    cPen 2-OCF_Three-4-F
iPr 2-F-4-OCF_Three     U-4d 3,5-di-F cPen 2-OCF_Three-4-Cl
iPr 2-Cl-4-F U-4d 3-F-5-Cl cPen 2-OCF_Three-4-Br
iPr 2,4-di-Cl U-4d 3-F-5-Br cPen 2-OCF_Three-4-Me
iPr 2-Cl-4-Br U-4d 3-F-5-Me cPen 2-OCF_Three-4-CF_Three
iPr 2-Cl-4-Me U-4d 3-F-5-CF_Three      cPen 2-OCF_Three-4-OMe
iPr 2-Cl-4-CF_Three     U-4d 3-F-5-OMe cPen 2,4-di-OCF_Three
iPr 2-Cl-4-OMe U-4d 3-F-5-OCF_Three     cPen 2,5-di-F
iPr 2-Cl-4-OCF_Three    U-4d 3-Cl-5-F cPen 2-F-5-Cl
iPr 2-Br-4-F U-4d 3,5-di-Cl cPen 2-F-5-Br
iPr 2-Br-4-Cl U-4d 3-Cl-5-Br cPen 2-F-5-Me
iPr 2,4-di-Br U-4d 3-Cl-5-Me cPen 2-F-5-CF_Three
iPr 2-Br-4-Me U-4d 3-Cl-5-CF_Three     cPen 2-F-5-OMe
iPr 2-Br-4-CF_Three     U-4d 3-Cl-5-OMe cPen 2-F-5-OCF_Three
iPr 2-Br-4-OMe U-4d 3-Cl-5-OCF_Three    cPen 2-Cl-5-F
iPr 2-Br-4-OCF_Three    U-4d 3-Br-5-F cPen 2,5-di-Cl
iPr 2-Me-4-F U-4d 3-Br-5-Cl cPen 2-Cl-5-Br
iPr 2-Me-4-Cl U-4d 3,5-di-Br cPen 2-Cl-5-Me
iPr 2-Me-4-Br U-4d 3-Br-5-Me cPen 2-Cl-5-CF_Three
iPr 2,4-di-Me U-4d 3-Br-5-CF_Three     cPen 2-Cl-5-OMe
iPr 2-Me-4-CF_Three     U-4d 3-Br-5-OMe cPen 2-Cl-5-OCF_Three
iPr 2-Me-4-OMe U-4d 3-Br-5-OCF_Three    cPen 2-Br-5-F
iPr 2-Me-4-OCF_Three    U-4d 3-Me-5-F cPen 2-Br-5-Cl
iPr 2-CF_Three-4-F U-4d 3-Me-5-Cl cPen 2,5-di-Br
iPr 2-CF_Three-4-Cl U-4d 3-Me-5-Br cPen 2-Br-5-Me
iPr 2-CF_Three-4-Br U-4d 3,5-di-Me cPen 2-Br-5-CF_Three
iPr 2-CF_Three-4-Me U-4d 3-Me-5-CF_Three     cPen 2-Br-5-OMe
iPr 2,4-di-CF_Three     U-4d 3-Me-5-OMe cPen 2-Br-5-OCF_Three
iPr 2-CF_Three-4-OMe U-4d 3-Me-5-OCF_Three    cPen 2-Me-5-F
iPr 2-CF_Three-4-OCF_Three   U-4d 3-CF_Three-5-F cPen 2-Me-5-Cl
iPr 2-OMe-4-F U-4d 3-CF_Three-5-Cl cPen 2-Me-5-Br
iPr 2-OMe-4-Cl U-4d 3-CF_Three-5-Br cPen 2,5-di-Me
iPr 2-OMe-4-Br U-4d 3-CF_Three-5-Me cPen 2-Me-5-CF_Three
iPr 2-OMe-4-Me U-4d 3,5-di-CF_Three     cPen 2-Me-5-OMe
iPr 2-OMe-4-CF_Three    U-4d 3-CF_Three-5-OMe cPen 2-Me-5-OCF_Three
iPr 2,4-di-OMe U-4d 3-CF_Three-5-OCF_Three   cPen 2-CF_Three-5-F
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
iPr 2-OMe-4-OCF_Three   U-4d 3-OMe-5-F cPen 2-CF_Three-5-Cl
iPr 2-OCF_Three-4-F U-4d 3-OMe-5-Cl cPen 2-CF_Three-5-Br
iPr 2-OCF_Three-4-Cl U-4d 3-OMe-5-Br cPen 2-CF_Three-5-Me
iPr 2-OCF_Three-4-Br U-4d 3-OMe-5-Me cPen 2,5-di-CF_Three
iPr 2-OCF_Three-4-Me U-4d 3-OMe-5-CF_Three    cPen 2-CF_Three-5-OMe
iPr 2-OCF_Three-4-CF_Three   U-4d 3,5-di-OMe cPen 2-CF_Three-5-OCF_Three
iPr 2-OCF_Three-4-OMe U-4d 3-OMe-5-OCF_Three   cPen 2-OMe-5-F
iPr 2,4-di-OCF_Three    U-4d 3-OCF_Three-5-F cPen 2-OMe-5-Cl
iPr 2,5-di-F U-4d 3-OCF_Three-5-Cl cPen 2-OMe-5-Br
iPr 2-F-5-Cl U-4d 3-OCF_Three-5-Br cPen 2-OMe-5-Me
iPr 2-F-5-Br U-4d 3-OCF_Three-5-Me cPen 2-OMe-5-CF_Three
iPr 2-F-5-Me U-4d 3-OCF_Three-5-CF_Three   cPen 2,5-di-OMe
iPr 2-F-5-CF_Three      U-4d 3-OCF_Three-5-OMe cPen 2-OMe-5-OCF_Three
iPr 2-F-5-OMe U-4d 3,5-di-OCF_Three    cPen 2-OCF_Three-5-F
iPr 2-F-5-OCF_Three     U-4e 2,3-di-F cPen 2-OCF_Three-5-Cl
iPr 2-Cl-5-F U-4e 2-F-3-Cl cPen 2-OCF_Three-5-Br
iPr 2,5-di-Cl U-4e 2-F-3-Br cPen 2-OCF_Three-5-Me
iPr 2-Cl-5-Br U-4e 2-F-3-Me cPen 2-OCF_Three-5-CF_Three
iPr 2-Cl-5-Me U-4e 2-F-3-CF_Three      cPen 2-OCF_Three-5-OMe
iPr 2-Cl-5-CF_Three     U-4e 2-F-3-OMe cPen 2,5-di-OCF_Three
iPr 2-Cl-5-OMe U-4e 2-F-3-OCF_Three     cPen 3,4-di-F
iPr 2-Cl-5-OCF_Three    U-4e 2-Cl-3-F cPen 3-F-4-Cl
iPr 2-Br-5-F U-4e 2,3-di-Cl cPen 3-F-4-Br
iPr 2-Br-5-Cl U-4e 2-Cl-3-Br cPen 3-F-4-Me
iPr 2,5-di-Br U-4e 2-Cl-3-Me cPen 3-F-4-CF_Three
iPr 2-Br-5-Me U-4e 2-Cl-3-CF_Three     cPen 3-F-4-OMe
iPr 2-Br-5-CF_Three     U-4e 2-Cl-3-OMe cPen 3-F-4-OCF_Three
iPr 2-Br-5-OMe U-4e 2-Cl-3-OCF_Three    cPen 3-Cl-4-F
iPr 2-Br-5-OCF_Three    U-4e 2-Br-3-F cPen 3,4-di-Cl
iPr 2-Me-5-F U-4e 2-Br-3-Cl cPen 3-Cl-4-Br
iPr 2-Me-5-Cl U-4e 2,3-di-Br cPen 3-Cl-4-Me
iPr 2-Me-5-Br U-4e 2-Br-3-Me cPen 3-Cl-4-CF_Three
iPr 2,5-di-Me U-4e 2-Br-3-CF_Three     cPen 3-Cl-4-OMe
iPr 2-Me-5-CF_Three     U-4e 2-Br-3-OMe cPen 3-Cl-4-OCF_Three
iPr 2-Me-5-OMe U-4e 2-Br-3-OCF_Three    cPen 3-Br-4-F
iPr 2-Me-5-OCF_Three    U-4e 2-Me-3-F cPen 3-Br-4-Cl
iPr 2-CF_Three-5-F U-4e 2-Me-3-Cl cPen 3,4-di-Br
iPr 2-CF_Three-5-Cl U-4e 2-Me-3-Br cPen 3-Br-4-Me
iPr 2-CF_Three-5-Br U-4e 2,3-di-Me cPen 3-Br-4-CF_Three
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
iPr 2-CF_Three-5-Me U-4e 2-Me-3-CF_Three     cPen 3-Br-4-OMe
iPr 2,5-di-CF_Three     U-4e 2-Me-3-OMe cPen 3-Br-4-OCF_Three
iPr 2-CF_Three-5-OMe U-4e 2-Me-3-OCF_Three    cPen 3-Me-4-F
iPr 2-CF_Three-5-OCF_Three   U-4e 2-CF_Three-3-F cPen 3-Me-4-Cl
iPr 2-OMe-5-F U-4e 2-CF_Three-3-Cl cPen 3-Me-4-Br
iPr 2-OMe-5-Cl U-4e 2-CF_Three-3-Br cPen 3,4-di-Me
iPr 2-OMe-5-Br U-4e 2-CF_Three-3-Me cPen 3-Me-4-CF_Three
iPr 2-OMe-5-Me U-4e 2,3-di-CF_Three     cPen 3-Me-4-OMe
iPr 2-OMe-5-CF_Three    U-4e 2-CF_Three-3-OMe cPen 3-Me-4-OCF_Three
iPr 2,5-di-OMe U-4e 2-CF_Three-3-OCF_Three   cPen 3-CF_Three-4-F
iPr 2-OMe-5-OCF_Three   U-4e 2-OMe-3-F cPen 3-CF_Three-4-Cl
iPr 2-OCF_Three-5-F U-4e 2-OMe-3-Cl cPen 3-CF_Three-4-Br
iPr 2-OCF_Three-5-Cl U-4e 2-OMe-3-Br cPen 3-CF_Three-4-Me
iPr 2-OCF_Three-5-Br U-4e 2-OMe-3-Me cPen 3,4-di-CF_Three
iPr 2-OCF_Three-5-Me U-4e 2-OMe-3-CF_Three    cPen 3-CF_Three-4-OMe
iPr 2-OCF_Three-5-CF_Three   U-4e 2,3-di-OMe cPen 3-CF_Three-4-OCF_Three
iPr 2-OCF_Three-5-OMe U-4e 2-OMe-3-OCF_Three   cPen 3-OMe-4-F
iPr 2,5-di-OCF_Three    U-4e 2-OCF_Three-3-F cPen 3-OMe-4-Cl
iPr 3,4-di-F U-4e 2-OCF_Three-3-Cl cPen 3-OMe-4-Br
iPr 3-F-4-Cl U-4e 2-OCF_Three-3-Br cPen 3-OMe-4-Me
iPr 3-F-4-Br U-4e 2-OCF_Three-3-Me cPen 3-OMe-4-CF_Three
iPr 3-F-4-Me U-4e 2-OCF_Three-3-CF_Three   cPen 3,4-di-OMe
iPr 3-F-4-CF_Three      U-4e 2-OCF_Three-3-OMe cPen 3-OMe-4-OCF_Three
iPr 3-F-4-OMe U-4e 2,3-di-OCF_Three    cPen 3-OCF_Three-4-F
iPr 3-F-4-OCF_Three     U-4e 2,4-di-F cPen 3-OCF_Three-4-Cl
iPr 3-Cl-4-F U-4e 2-F-4-Cl cPen 3-OCF_Three-4-Br
iPr 3,4-di-Cl U-4e 2-F-4-Br cPen 3-OCF_Three-4-Me
iPr 3-Cl-4-Br U-4e 2-F-4-Me cPen 3-OCF_Three-4-CF_Three
iPr 3-Cl-4-Me U-4e 2-F-4-CF_Three      cPen 3-OCF_Three-4-OMe
iPr 3-Cl-4-CF_Three     U-4e 2-F-4-OMe cPen 3,4-di-OCF_Three
iPr 3-Cl-4-OMe U-4e 2-F-4-OCF_Three     cPen 3,5-di-F
iPr 3-Cl-4-OCF_Three    U-4e 2-Cl-4-F cPen 3-F-5-Cl
iPr 3-Br-4-F U-4e 2,4-di-Cl cPen 3-F-5-Br
iPr 3-Br-4-Cl U-4e 2-Cl-4-Br cPen 3-F-5-Me
iPr 3,4-di-Br U-4e 2-Cl-4-Me cPen 3-F-5-CF_Three
iPr 3-Br-4-Me U-4e 2-Cl-4-CF_Three     cPen 3-F-5-OMe
iPr 3-Br-4-CF_Three     U-4e 2-Cl-4-OMe cPen 3-F-5-OCF_Three
iPr 3-Br-4-OMe U-4e 2-Cl-4-OCF_Three    cPen 3-Cl-5-F
iPr 3-Br-4-OCF_Three    U-4e 2-Br-4-F cPen 3,5-di-Cl
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
iPr 3-Me-4-F U-4e 2-Br-4-Cl cPen 3-Cl-5-Br
iPr 3-Me-4-Cl U-4e 2,4-di-Br cPen 3-Cl-5-Me
iPr 3-Me-4-Br U-4e 2-Br-4-Me cPen 3-Cl-5-CF_Three
iPr 3,4-di-Me U-4e 2-Br-4-CF_Three     cPen 3-Cl-5-OMe
iPr 3-Me-4-CF_Three     U-4e 2-Br-4-OMe cPen 3-Cl-5-OCF_Three
iPr 3-Me-4-OMe U-4e 2-Br-4-OCF_Three    cPen 3-Br-5-F
iPr 3-Me-4-OCF_Three    U-4e 2-Me-4-F cPen 3-Br-5-Cl
iPr 3-CF_Three-4-F U-4e 2-Me-4-Cl cPen 3,5-di-Br
iPr 3-CF_Three-4-Cl U-4e 2-Me-4-Br cPen 3-Br-5-Me
iPr 3-CF_Three-4-Br U-4e 2,4-di-Me cPen 3-Br-5-CF_Three
iPr 3-CF_Three-4-Me U-4e 2-Me-4-CF_Three     cPen 3-Br-5-OMe
iPr 3,4-di-CF_Three     U-4e 2-Me-4-OMe cPen 3-Br-5-OCF_Three
iPr 3-CF_Three-4-OMe U-4e 2-Me-4-OCF_Three    cPen 3-Me-5-F
iPr 3-CF_Three-4-OCF_Three   U-4e 2-CF_Three-4-F cPen 3-Me-5-Cl
iPr 3-OMe-4-F U-4e 2-CF_Three-4-Cl cPen 3-Me-5-Br
iPr 3-OMe-4-Cl U-4e 2-CF_Three-4-Br cPen 3,5-di-Me
iPr 3-OMe-4-Br U-4e 2-CF_Three-4-Me cPen 3-Me-5-CF_Three
iPr 3-OMe-4-Me U-4e 2,4-di-CF_Three     cPen 3-Me-5-OMe
iPr 3-OMe-4-CF_Three    U-4e 2-CF_Three-4-OMe cPen 3-Me-5-OCF_Three
iPr 3,4-di-OMe U-4e 2-CF_Three-4-OCF_Three   cPen 3-CF_Three-5-F
iPr 3-OMe-4-OCF_Three   U-4e 2-OMe-4-F cPen 3-CF_Three-5-Cl
iPr 3-OCF_Three-4-F U-4e 2-OMe-4-Cl cPen 3-CF_Three-5-Br
iPr 3-OCF_Three-4-Cl U-4e 2-OMe-4-Br cPen 3-CF_Three-5-Me
iPr 3-OCF_Three-4-Br U-4e 2-OMe-4-Me cPen 3,5-di-CF_Three
iPr 3-OCF_Three-4-Me U-4e 2-OMe-4-CF_Three    cPen 3-CF_Three-5-OMe
iPr 3-OCF_Three-4-CF_Three   U-4e 2,4-di-OMe cPen 3-CF_Three-5-OCF_Three
iPr 3-OCF_Three-4-OMe U-4e 2-OMe-4-OCF_Three   cPen 3-OMe-5-F
iPr 3,4-di-OCF_Three    U-4e 2-OCF_Three-4-F cPen 3-OMe-5-Cl
iPr 3,5-di-F U-4e 2-OCF_Three-4-Cl cPen 3-OMe-5-Br
iPr 3-F-5-Cl U-4e 2-OCF_Three-4-Br cPen 3-OMe-5-Me
iPr 3-F-5-Br U-4e 2-OCF_Three-4-Me cPen 3-OMe-5-CF_Three
iPr 3-F-5-Me U-4e 2-OCF_Three-4-CF_Three   cPen 3,5-di-OMe
iPr 3-F-5-CF_Three      U-4e 2-OCF_Three-4-OMe cPen 3-OMe-5-OCF_Three
iPr 3-F-5-OMe U-4e 2,4-di-OCF_Three    cPen 3-OCF_Three-5-F
iPr 3-F-5-OCF_Three     U-4e 2,5-di-F cPen 3-OCF_Three-5-Cl
iPr 3-Cl-5-F U-4e 2-F-5-Cl cPen 3-OCF_Three-5-Br
iPr 3,5-di-Cl U-4e 2-F-5-Br cPen 3-OCF_Three-5-Me
iPr 3-Cl-5-Br U-4e 2-F-5-Me cPen 3-OCF_Three-5-CF_Three
iPr 3-Cl-5-Me U-4e 2-F-5-CF_Three      cPen 3-OCF_Three-5-OMe
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
iPr 3-Cl-5-CF_Three     U-4e 2-F-5-OMe cPen 3,5-di-OCF_Three
iPr 3-Cl-5-OMe U-4e 2-F-5-OCF_Three     U-1e 2,3-di-F
iPr 3-Cl-5-OCF_Three    U-4e 2-Cl-5-F U-1e 2-F-3-Cl
iPr 3-Br-5-F U-4e 2,5-di-Cl U-1e 2-F-3-Br
iPr 3-Br-5-Cl U-4e 2-Cl-5-Br U-1e 2-F-3-Me
iPr 3,5-di-Br U-4e 2-Cl-5-Me U-1e 2-F-3-CF_Three
iPr 3-Br-5-Me U-4e 2-Cl-5-CF_Three     U-1e 2-F-3-OMe
iPr 3-Br-5-CF_Three     U-4e 2-Cl-5-OMe U-1e 2-F-3-OCF_Three
iPr 3-Br-5-OMe U-4e 2-Cl-5-OCF_Three    U-1e 2-Cl-3-F
iPr 3-Br-5-OCF_Three    U-4e 2-Br-5-F U-1e 2,3-di-Cl
iPr 3-Me-5-F U-4e 2-Br-5-Cl U-1e 2-Cl-3-Br
iPr 3-Me-5-Cl U-4e 2,5-di-Br U-1e 2-Cl-3-Me
iPr 3-Me-5-Br U-4e 2-Br-5-Me U-1e 2-Cl-3-CF_Three
iPr 3,5-di-Me U-4e 2-Br-5-CF_Three     U-1e 2-Cl-3-OMe
iPr 3-Me-5-CF_Three     U-4e 2-Br-5-OMe U-1e 2-Cl-3-OCF_Three
iPr 3-Me-5-OMe U-4e 2-Br-5-OCF_Three    U-1e 2-Br-3-F
iPr 3-Me-5-OCF_Three    U-4e 2-Me-5-F U-1e 2-Br-3-Cl
iPr 3-CF_Three-5-F U-4e 2-Me-5-Cl U-1e 2,3-di-Br
iPr 3-CF_Three-5-Cl U-4e 2-Me-5-Br U-1e 2-Br-3-Me
iPr 3-CF_Three-5-Br U-4e 2,5-di-Me U-1e 2-Br-3-CF_Three
iPr 3-CF_Three-5-Me U-4e 2-Me-5-CF_Three     U-1e 2-Br-3-OMe
iPr 3,5-di-CF_Three     U-4e 2-Me-5-OMe U-1e 2-Br-3-OCF_Three
iPr 3-CF_Three-5-OMe U-4e 2-Me-5-OCF_Three    U-1e 2-Me-3-F
iPr 3-CF_Three-5-OCF_Three   U-4e 2-CF_Three-5-F U-1e 2-Me-3-Cl
iPr 3-OMe-5-F U-4e 2-CF_Three-5-Cl U-1e 2-Me-3-Br
iPr 3-OMe-5-Cl U-4e 2-CF_Three-5-Br U-1e 2,3-di-Me
iPr 3-OMe-5-Br U-4e 2-CF_Three-5-Me U-1e 2-Me-3-CF_Three
iPr 3-OMe-5-Me U-4e 2,5-di-CF_Three     U-1e 2-Me-3-OMe
iPr 3-OMe-5-CF_Three    U-4e 2-CF_Three-5-OMe U-1e 2-Me-3-OCF_Three
iPr 3,5-di-OMe U-4e 2-CF_Three-5-OCF_Three  U-1e 2-CF_Three-3-F
iPr 3-OMe-5-OCF_Three   U-4e 2-OMe-5-F U-1e 2-CF_Three-3-Cl
iPr 3-OCF_Three-5-F U-4e 2-OMe-5-Cl U-1e 2-CF_Three-3-Br
iPr 3-OCF_Three-5-Cl U-4e 2-OMe-5-Br U-1e 2-CF_Three-3-Me
iPr 3-OCF_Three-5-Br U-4e 2-OMe-5-Me U-1e 2,3-di-CF_Three
iPr 3-OCF_Three-5-Me U-4e 2-OMe-5-CF_Three    U-1e 2-CF_Three-3-OMe
iPr 3-OCF_Three-5-CF_Three   U-4e 2,5-di-OMe U-1e 2-CF_Three-3-OCF_Three
iPr 3-OCF_Three-5-OMe U-4e 2-OMe-5-OCF_Three   U-1e 2-OMe-3-F
iPr 3,5-di-OCF_Three    U-4e 2-OCF_Three-5-F U-1e 2-OMe-3-Cl
U-4a 2,3-di-F U-4e 2-OCF_Three-5-Cl U-1e 2-OMe-3-Br
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
U-4a 2-F-3-Cl U-4e 2-OCF_Three-5-Br U-1e 2-OMe-3-Me
U-4a 2-F-3-Br U-4e 2-OCF_Three-5-Me U-1e 2-OMe-3-CF_Three
U-4a 2-F-3-Me U-4e 2-OCF_Three-5-CF_Three   U-1e 2,3-di-OMe
U-4a 2-F-3-CF_Three      U-4e 2-OCF_Three-5-OMe U-1e 2-OMe-3-OCF_Three
U-4a 2-F-3-OMe U-4e 2,5-di-OCF_Three    U-1e 2-OCF_Three-3-F
U-4a 2-F-3-OCF_Three     U-4e 3,4-di-F U-1e 2-OCF_Three-3-Cl
U-4a 2-Cl-3-F U-4e 3-F-4-Cl U-1e 2-OCF_Three-3-Br
U-4a 2,3-di-Cl U-4e 3-F-4-Br U-1e 2-OCF_Three-3-Me
U-4a 2-Cl-3-Br U-4e 3-F-4-Me U-1e 2-OCF_Three-3-CF_Three
U-4a 2-Cl-3-Me U-4e 3-F-4-CF_Three      U-1e 2-OCF_Three-3-OMe
U-4a 2-Cl-3-CF_Three     U-4e 3-F-4-OMe U-1e 2,3-di-OCF_Three
U-4a 2-Cl-3-OMe U-4e 3-F-4-OCF_Three     U-1e 2,4-di-F
U-4a 2-Cl-3-OCF_Three    U-4e 3-Cl-4-F U-1e 2-F-4-Cl
U-4a 2-Br-3-F U-4e 3,4-di-Cl U-1e 2-F-4-Br
U-4a 2-Br-3-Cl U-4e 3-Cl-4-Br U-1e 2-F-4-Me
U-4a 2,3-di-Br U-4e 3-Cl-4-Me U-1e 2-F-4-CF_Three
U-4a 2-Br-3-Me U-4e 3-Cl-4-CF_Three     U-1e 2-F-4-OMe
U-4a 2-Br-3-CF_Three     U-4e 3-Cl-4-OMe U-1e 2-F-4-OCF_Three
U-4a 2-Br-3-OMe U-4e 3-Cl-4-OCF_Three    U-1e 2-Cl-4-F
U-4a 2-Br-3-OCF_Three    U-4e 3-Br-4-F U-1e 2,4-di-Cl
U-4a 2-Me-3-F U-4e 3-Br-4-Cl U-1e 2-Cl-4-Br
U-4a 2-Me-3-Cl U-4e 3,4-di-Br U-1e 2-Cl-4-Me
U-4a 2-Me-3-Br U-4e 3-Br-4-Me U-1e 2-Cl-4-CF_Three
U-4a 2,3-di-Me U-4e 3-Br-4-CF_Three     U-1e 2-Cl-4-OMe
U-4a 2-Me-3-CF_Three     U-4e 3-Br-4-OMe U-1e 2-Cl-4-OCF_Three
U-4a 2-Me-3-OMe U-4e 3-Br-4-OCF_Three    U-1e 2-Br-4-F
U-4a 2-Me-3-OCF_Three    U-4e 3-Me-4-F U-1e 2-Br-4-Cl
U-4a 2-CF_Three-3-F U-4e 3-Me-4-Cl U-1e 2,4-di-Br
U-4a 2-CF_Three-3-Cl U-4e 3-Me-4-Br U-1e 2-Br-4-Me
U-4a 2-CF_Three-3-Br U-4e 3,4-di-Me U-1e 2-Br-4-CF_Three
U-4a 2-CF_Three-3-Me U-4e 3-Me-4-CF_Three     U-1e 2-Br-4-OMe
U-4a 2,3-di-CF_Three     U-4e 3-Me-4-OMe U-1e 2-Br-4-OCF_Three
U-4a 2-CF_Three-3-OMe U-4e 3-Me-4-OCF_Three    U-1e 2-Me-4-F
U-4a 2-CF_Three-3-OCF_Three   U-4e 3-CF_Three-4-F U-1e 2-Me-4-Cl
U-4a 2-OMe-3-F U-4e 3-CF_Three-4-Cl U-1e 2-Me-4-Br
U-4a 2-OMe-3-Cl U-4e 3-CF_Three-4-Br U-1e 2,4-di-Me
U-4a 2-OMe-3-Br U-4e 3-CF_Three-4-Me U-1e 2-Me-4-CF_Three
U-4a 2-OMe-3-Me U-4e 3,4-di-CF_Three     U-1e 2-Me-4-OMe
U-4a 2-OMe-3-CF_Three    U-4e 3-CF_Three-4-OMe U-1e 2-Me-4-OCF_Three
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
U-4a 2,3-di-OMe U-4e 3-CF_Three-4-OCF_Three   U-1e 2-CF_Three-4-F
U-4a 2-OMe-3-OCF_Three   U-4e 3-OMe-4-F U-1e 2-CF_Three-4-Cl
U-4a 2-OCF_Three-3-F U-4e 3-OMe-4-Cl U-1e 2-CF_Three-4-Br
U-4a 2-OCF_Three-3-Cl U-4e 3-OMe-4-Br U-1e 2-CF_Three-4-Me
U-4a 2-OCF_Three-3-Br U-4e 3-OMe-4-Me U-1e 2,4-di-CF_Three
U-4a 2-OCF_Three-3-Me U-4e 3-OMe-4-CF_Three    U-1e 2-CF_Three-4-OMe
U-4a 2-OCF_Three-3-CF_Three   U-4e 3,4-di-OMe U-1e 2-CF_Three-4-OCF_Three
U-4a 2-OCF_Three-3-OMe U-4e 3-OMe-4-OCF_Three   U-1e 2-OMe-4-F
U-4a 2,3-di-OCF_Three    U-4e 3-OCF_Three-4-F U-1e 2-OMe-4-Cl
U-4a 2,4-di-F U-4e 3-OCF_Three-4-Cl U-1e 2-OMe-4-Br
U-4a 2-F-4-Cl U-4e 3-OCF_Three-4-Br U-1e 2-OMe-4-Me
U-4a 2-F-4-Br U-4e 3-OCF_Three-4-Me U-1e 2-OMe-4-CF_Three
U-4a 2-F-4-Me U-4e 3-OCF_Three-4-CF_Three   U-1e 2,4-di-OMe
U-4a 2-F-4-CF_Three      U-4e 3-OCF_Three-4-OMe U-1e 2-OMe-4-OCF_Three
U-4a 2-F-4-OMe U-4e 3,4-di-OCF_Three    U-1e 2-OCF_Three-4-F
U-4a 2-F-4-OCF_Three     U-4e 3,5-di-F U-1e 2-OCF_Three-4-Cl
U-4a 2-Cl-4-F U-4e 3-F-5-Cl U-1e 2-OCF_Three-4-Br
U-4a 2,4-di-Cl U-4e 3-F-5-Br U-1e 2-OCF_Three-4-Me
U-4a 2-Cl-4-Br U-4e 3-F-5-Me U-1e 2-OCF_Three-4-CF_Three
U-4a 2-Cl-4-Me U-4e 3-F-5-CF_Three      U-1e 2-OCF_Three-4-OMe
U-4a 2-Cl-4-CF_Three     U-4e 3-F-5-OMe U-1e 2,4-di-OCF_Three
U-4a 2-Cl-4-OMe U-4e 3-F-5-OCF_Three     U-1e 2,5-di-F
U-4a 2-Cl-4-OCF_Three    U-4e 3-Cl-5-F U-1e 2-F-5-Cl
U-4a 2-Br-4-F U-4e 3,5-di-Cl U-1e 2-F-5-Br
U-4a 2-Br-4-Cl U-4e 3-Cl-5-Br U-1e 2-F-5-Me
U-4a 2,4-di-Br U-4e 3-Cl-5-Me U-1e 2-F-5-CF_Three
U-4a 2-Br-4-Me U-4e 3-Cl-5-CF_Three     U-1e 2-F-5-OMe
U-4a 2-Br-4-CF_Three     U-4e 3-Cl-5-OMe U-1e 2-F-5-OCF_Three
U-4a 2-Br-4-OMe U-4e 3-Cl-5-OCF_Three    U-1e 2-Cl-5-F
U-4a 2-Br-4-OCF_Three    U-4e 3-Br-5-F U-1e 2,5-di-Cl
U-4a 2-Me-4-F U-4e 3-Br-5-Cl U-1e 2-Cl-5-Br
U-4a 2-Me-4-Cl U-4e 3,5-di-Br U-1e 2-Cl-5-Me
U-4a 2-Me-4-Br U-4e 3-Br-5-Me U-1e 2-Cl-5-CF_Three
U-4a 2,4-di-Me U-4e 3-Br-5-CF_Three     U-1e 2-Cl-5-OMe
U-4a 2-Me-4-CF_Three     U-4e 3-Br-5-OMe U-1e 2-Cl-5-OCF_Three
U-4a 2-Me-4-OMe U-4e 3-Br-5-OCF_Three    U-1e 2-Br-5-F
U-4a 2-Me-4-OCF_Three    U-4e 3-Me-5-F U-1e 2-Br-5-Cl
U-4a 2-CF_Three-4-F U-4e 3-Me-5-Cl U-1e 2,5-di-Br
U-4a 2-CF_Three-4-Cl U-4e 3-Me-5-Br U-1e 2-Br-5-Me
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
U-4a 2-CF_Three-4-Br U-4e 3,5-di-Me U-1e 2-Br-5-CF_Three
U-4a 2-CF_Three-4-Me U-4e 3-Me-5-CF_Three     U-1e 2-Br-5-OMe
U-4a 2,4-di-CF_Three     U-4e 3-Me-5-OMe U-1e 2-Br-5-OCF_Three
U-4a 2-CF_Three-4-OMe U-4e 3-Me-5-OCF_Three    U-1e 2-Me-5-F
U-4a 2-CF_Three-4-OCF_Three   U-4e 3-CF_Three-5-F U-1e 2-Me-5-Cl
U-4a 2-OMe-4-F U-4e 3-CF_Three-5-Cl U-1e 2-Me-5-Br
U-4a 2-OMe-4-Cl U-4e 3-CF_Three-5-Br U-1e 2,5-di-Me
U-4a 2-OMe-4-Br U-4e 3-CF_Three-5-Me U-1e 2-Me-5-CF_Three
U-4a 2-OMe-4-Me U-4e 3,5-di-CF_Three     U-1e 2-Me-5-OMe
U-4a 2-OMe-4-CF_Three    U-4e 3-CF_Three-5-OMe U-1e 2-Me-5-OCF_Three
U-4a 2,4-di-OMe U-4e 3-CF_Three-5-OCF_Three   U-1e 2-CF_Three-5-F
U-4a 2-OMe-4-OCF_Three   U-4e 3-OMe-5-F U-1e 2-CF_Three-5-Cl
U-4a 2-OCF_Three-4-F U-4e 3-OMe-5-Cl U-1e 2-CF_Three-5-Br
U-4a 2-OCF_Three-4-Cl U-4e 3-OMe-5-Br U-1e 2-CF_Three-5-Me
U-4a 2-OCF_Three-4-Br U-4e 3-OMe-5-Me U-1e 2,5-di-CF_Three
U-4a 2-OCF_Three-4-Me U-4e 3-OMe-5-CF_Three    U-1e 2-CF_Three-5-OMe
U-4a 2-OCF_Three-4-CF_Three   U-4e 3,5-di-OMe U-1e 2-CF_Three-5-OCF_Three
U-4a 2-OCF_Three-4-OMe U-4e 3-OMe-5-OCF_Three   U-1e 2-OMe-5-F
U-4a 2,4-di-OCF_Three    U-4e 3-OCF_Three-5-F U-1e 2-OMe-5-Cl
U-4a 2,5-di-F U-4e 3-OCF_Three-5-Cl U-1e 2-OMe-5-Br
U-4a 2-F-5-Cl U-4e 3-OCF_Three-5-Br U-1e 2-OMe-5-Me
U-4a 2-F-5-Br U-4e 3-OCF_Three-5-Me U-1e 2-OMe-5-CF_Three
U-4a 2-F-5-Me U-4e 3-OCF_Three-5-CF_Three   U-1e 2,5-di-OMe
U-4a 2-F-5-CF_Three      U-4e 3-OCF_Three-5-OMe U-1e 2-OMe-5-OCF_Three
U-4a 2-F-5-OMe U-4e 3,5-di-OCF_Three    U-1e 2-OCF_Three-5-F
U-4a 2-F-5-OCF_Three     U-4f 2,3-di-F U-1e 2-OCF_Three-5-Cl
U-4a 2-Cl-5-F U-4f 2-F-3-Cl U-1e 2-OCF_Three-5-Br
U-4a 2,5-di-Cl U-4f 2-F-3-Br U-1e 2-OCF_Three-5-Me
U-4a 2-Cl-5-Br U-4f 2-F-3-Me U-1e 2-OCF_Three-5-CF_Three
U-4a 2-Cl-5-Me U-4f 2-F-3-CF_Three      U-1e 2-OCF_Three-5-OMe
U-4a 2-Cl-5-CF_Three     U-4f 2-F-3-OMe U-1e 2,5-di-OCF_Three
U-4a 2-Cl-5-OMe U-4f 2-F-3-OCF_Three     U-1e 3,4-di-F
U-4a 2-Cl-5-OCF_Three    U-4f 2-Cl-3-F U-1e 3-F-4-Cl
U-4a 2-Br-5-F U-4f 2,3-di-Cl U-1e 3-F-4-Br
U-4a 2-Br-5-Cl U-4f 2-Cl-3-Br U-1e 3-F-4-Me
U-4a 2,5-di-Br U-4f 2-Cl-3-Me U-1e 3-F-4-CF_Three
U-4a 2-Br-5-Me U-4f 2-Cl-3-CF_Three     U-1e 3-F-4-OMe
U-4a 2-Br-5-CF_Three     U-4f 2-Cl-3-OMe U-1e 3-F-4-OCF_Three
U-4a 2-Br-5-OMe U-4f 2-Cl-3-OCF_Three    U-1e 3-Cl-4-F
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
U-4a 2-Br-5-OCF_Three    U-4f 2-Br-3-F U-1e 3,4-di-Cl
U-4a 2-Me-5-F U-4f 2-Br-3-Cl U-1e 3-Cl-4-Br
U-4a 2-Me-5-Cl U-4f 2,3-di-Br U-1e 3-Cl-4-Me
U-4a 2-Me-5-Br U-4f 2-Br-3-Me U-1e 3-Cl-4-CF_Three
U-4a 2,5-di-Me U-4f 2-Br-3-CF_Three     U-1e 3-Cl-4-OMe
U-4a 2-Me-5-CF_Three     U-4f 2-Br-3-OMe U-1e 3-Cl-4-OCF_Three
U-4a 2-Me-5-OMe U-4f 2-Br-3-OCF_Three    U-1e 3-Br-4-F
U-4a 2-Me-5-OCF_Three    U-4f 2-Me-3-F U-1e 3-Br-4-Cl
U-4a 2-CF_Three-5-F U-4f 2-Me-3-Cl U-1e 3,4-di-Br
U-4a 2-CF_Three-5-Cl U-4f 2-Me-3-Br U-1e 3-Br-4-Me
U-4a 2-CF_Three-5-Br U-4f 2,3-di-Me U-1e 3-Br-4-CF_Three
U-4a 2-CF_Three-5-Me U-4f 2-Me-3-CF_Three     U-1e 3-Br-4-OMe
U-4a 2,5-di-CF_Three     U-4f 2-Me-3-OMe U-1e 3-Br-4-OCF_Three
U-4a 2-CF_Three-5-OMe U-4f 2-Me-3-OCF_Three    U-1e 3-Me-4-F
U-4a 2-CF_Three-5-OCF_Three   U-4f 2-CF_Three-3-F U-1e 3-Me-4-Cl
U-4a 2-OMe-5-F U-4f 2-CF_Three-3-Cl U-1e 3-Me-4-Br
U-4a 2-OMe-5-Cl U-4f 2-CF_Three-3-Br U-1e 3,4-di-Me
U-4a 2-OMe-5-Br U-4f 2-CF_Three-3-Me U-1e 3-Me-4-CF_Three
U-4a 2-OMe-5-Me U-4f 2,3-di-CF_Three     U-1e 3-Me-4-OMe
U-4a 2-OMe-5-CF_Three    U-4f 2-CF_Three-3-OMe U-1e 3-Me-4-OCF_Three
U-4a 2,5-di-OMe U-4f 2-CF_Three-3-OCF_Three   U-1e 3-CF_Three-4-F
U-4a 2-OMe-5-OCF_Three   U-4f 2-OMe-3-F U-1e 3-CF_Three-4-Cl
U-4a 2-OCF_Three-5-F U-4f 2-OMe-3-Cl U-1e 3-CF_Three-4-Br
U-4a 2-OCF_Three-5-Cl U-4f 2-OMe-3-Br U-1e 3-CF_Three-4-Me
U-4a 2-OCF_Three-5-Br U-4f 2-OMe-3-Me U-1e 3,4-di-CF_Three
U-4a 2-OCF_Three-5-Me U-4f 2-OMe-3-CF_Three    U-1e 3-CF_Three-4-OMe
U-4a 2-OCF_Three-5-CF_Three  U-4f 2,3-di-OMe U-1e 3-CF_Three-4-OCF_Three
U-4a 2-OCF_Three-5-OMe U-4f 2-OMe-3-OCF_Three   U-1e 3-OMe-4-F
U-4a 2,5-di-OCF_Three    U-4f 2-OCF_Three-3-F U-1e 3-OMe-4-Cl
U-4a 3,4-di-F U-4f 2-OCF_Three-3-Cl U-1e 3-OMe-4-Br
U-4a 3-F-4-Cl U-4f 2-OCF_Three-3-Br U-1e 3-OMe-4-Me
U-4a 3-F-4-Br U-4f 2-OCF_Three-3-Me U-1e 3-OMe-4-CF_Three
U-4a 3-F-4-Me U-4f 2-OCF_Three-3-CF_Three   U-1e 3,4-di-OMe
U-4a 3-F-4-CF_Three      U-4f 2-OCF_Three-3-OMe U-1e 3-OMe-4-OCF_Three
U-4a 3-F-4-OMe U-4f 2,3-di-OCF_Three    U-1e 3-OCF_Three-4-F
U-4a 3-F-4-OCF_Three     U-4f 2,4-di-F U-1e 3-OCF_Three-4-Cl
U-4a 3-Cl-4-F U-4f 2-F-4-Cl U-1e 3-OCF_Three-4-Br
U-4a 3,4-di-Cl U-4f 2-F-4-Br U-1e 3-OCF_Three-4-Me
U-4a 3-Cl-4-Br U-4f 2-F-4-Me U-1e 3-OCF_Three-4-CF_Three
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
U-4a 3-Cl-4-Me U-4f 2-F-4-CF_Three      U-1e 3-OCF_Three-4-OMe
U-4a 3-Cl-4-CF_Three     U-4f 2-F-4-OMe U-1e 3,4-di-OCF_Three
U-4a 3-Cl-4-OMe U-4f 2-F-4-OCF_Three     U-1e 3,5-di-F
U-4a 3-Cl-4-OCF_Three    U-4f 2-Cl-4-F U-1e 3-F-5-Cl
U-4a 3-Br-4-F U-4f 2,4-di-Cl U-1e 3-F-5-Br
U-4a 3-Br-4-Cl U-4f 2-Cl-4-Br U-1e 3-F-5-Me
U-4a 3,4-di-Br U-4f 2-Cl-4-Me U-1e 3-F-5-CF_Three
U-4a 3-Br-4-Me U-4f 2-Cl-4-CF_Three     U-1e 3-F-5-OMe
U-4a 3-Br-4-CF_Three     U-4f 2-Cl-4-OMe U-1e 3-F-5-OCF_Three
U-4a 3-Br-4-OMe U-4f 2-Cl-4-OCF_Three    U-1e 3-Cl-5-F
U-4a 3-Br-4-OCF_Three    U-4f 2-Br-4-F U-1e 3,5-di-Cl
U-4a 3-Me-4-F U-4f 2-Br-4-Cl U-1e 3-Cl-5-Br
U-4a 3-Me-4-Cl U-4f 2,4-di-Br U-1e 3-Cl-5-Me
U-4a 3-Me-4-Br U-4f 2-Br-4-Me U-1e 3-Cl-5-CF_Three
U-4a 3,4-di-Me U-4f 2-Br-4-CF_Three     U-1e 3-Cl-5-OMe
U-4a 3-Me-4-CF_Three     U-4f 2-Br-4-OMe U-1e 3-Cl-5-OCF_Three
U-4a 3-Me-4-OMe U-4f 2-Br-4-OCF_Three    U-1e 3-Br-5-F
U-4a 3-Me-4-OCF_Three    U-4f 2-Me-4-F U-1e 3-Br-5-Cl
U-4a 3-CF_Three-4-F U-4f 2-Me-4-Cl U-1e 3,5-di-Br
U-4a 3-CF_Three-4-Cl U-4f 2-Me-4-Br U-1e 3-Br-5-Me
U-4a 3-CF_Three-4-Br U-4f 2,4-di-Me U-1e 3-Br-5-CF_Three
U-4a 3-CF_Three-4-Me U-4f 2-Me-4-CF_Three     U-1e 3-Br-5-OMe
U-4a 3,4-di-CF_Three     U-4f 2-Me-4-OMe U-1e 3-Br-5-OCF_Three
U-4a 3-CF_Three-4-OMe U-4f 2-Me-4-OCF_Three    U-1e 3-Me-5-F
U-4a 3-CF_Three-4-OCF_Three   U-4f 2-CF_Three-4-F U-1e 3-Me-5-Cl
U-4a 3-OMe-4-F U-4f 2-CF_Three-4-Cl U-1e 3-Me-5-Br
U-4a 3-OMe-4-Cl U-4f 2-CF_Three-4-Br U-1e 3,5-di-Me
U-4a 3-OMe-4-Br U-4f 2-CF_Three-4-Me U-1e 3-Me-5-CF_Three
U-4a 3-OMe-4-Me U-4f 2,4-di-CF_Three     U-1e 3-Me-5-OMe
U-4a 3-OMe-4-CF_Three    U-4f 2-CF_Three-4-OMe U-1e 3-Me-5-OCF_Three
U-4a 3,4-di-OMe U-4f 2-CF_Three-4-OCF_Three   U-1e 3-CF_Three-5-F
U-4a 3-OMe-4-OCF_Three   U-4f 2-OMe-4-F U-1e 3-CF_Three-5-Cl
U-4a 3-OCF_Three-4-F U-4f 2-OMe-4-Cl U-1e 3-CF_Three-5-Br
U-4a 3-OCF_Three-4-Cl U-4f 2-OMe-4-Br U-1e 3-CF_Three-5-Me
U-4a 3-OCF_Three-4-Br U-4f 2-OMe-4-Me U-1e 3,5-di-CF_Three
U-4a 3-OCF_Three-4-Me U-4f 2-OMe-4-CF_Three    U-1e 3-CF_Three-5-OMe
U-4a 3-OCF_Three-4-CF_Three   U-4f 2,4-di-OMe U-1e 3-CF_Three-5-OCF_Three
U-4a 3-OCF_Three-4-OMe U-4f 2-OMe-4-OCF_Three   U-1e 3-OMe-5-F
U-4a 3,4-di-OCF_Three    U-4f 2-OCF_Three-4-F U-1e 3-OMe-5-Cl
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued) [Table 1] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
U-4a 3,5-di-F U-4f 2-OCF_Three-4-Cl U-1e 3-OMe-5-Br
U-4a 3-F-5-Cl U-4f 2-OCF_Three-4-Br U-1e 3-OMe-5-Me
U-4a 3-F-5-Br U-4f 2-OCF_Three-4-Me U-1e 3-OMe-5-CF_Three
U-4a 3-F-5-Me U-4f 2-OCF_Three-4-CF_Three   U-1e 3,5-di-OMe
U-4a 3-F-5-CF_Three      U-4f 2-OCF_Three-4-OMe U-1e 3-OMe-5-OCF_Three
U-4a 3-F-5-OMe U-4f 2,4-di-OCF_Three    U-1e 3-OCF_Three-5-F
U-4a 3-F-5-OCF_Three     U-4f 2,5-di-F U-1e 3-OCF_Three-5-Cl
U-4a 3-Cl-5-F U-4f 2-F-5-Cl U-1e 3-OCF_Three-5-Br
U-4a 3,5-di-Cl U-4f 2-F-5-Br U-1e 3-OCF_Three-5-Me
U-4a 3-Cl-5-Br U-4f 2-F-5-Me U-1e 3-OCF_Three-5-CF_Three
U-4a 3-Cl-5-Me U-4f 2-F-5-CF_Three      U-1e 3-OCF_Three-5-OMe
U-4a 3-Cl-5-CF_Three     U-4f 2-F-5-OMe U-1e 3,5-di-OCF_Three
--------- --------- ------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Me 2-F-3-Ac cPr 3-Cl-4-Ac
Me 2-F-3- (U-3b) cPr 3-Cl-4- (U-3b)
Me 2-F-3-CF₂H cPr 3-Cl-4-CF₂H
Me 2-F-3-CN cPr 3-Cl-4-CN
Me 2-F-3-Et cPr 3-Cl-4-Et
Me 2-F-3-OCF₂H cPr 3-Cl-4-OCF₂H
Me 2-F-3-OEt cPr 3-Cl-4-OEt
Me 2-F-3-C (O) CF_Three       cPr 3-Cl-4-C (O) CF_Three
Me 2-Cl-3-Ac cPr 3-Br-4-Ac
Me 2-Cl-3- (U-3b) cPr 3-Br-4- (U-3b)
Me 2-Cl-3-CF₂H cPr 3-Br-4-CF₂H
Me 2-Cl-3-CN cPr 3-Br-4-CN
Me 2-Cl-3-Et cPr 3-Br-4-Et
Me 2-Cl-3-OCF₂H cPr 3-Br-4-OCF₂H
Me 2-Cl-3-OEt cPr 3-Br-4-OEt
Me 2-Cl-3-C (O) CF_Three      cPr 3-Br-4-C (O) CF_Three
Me 2-Br-3-Ac cPr 3-Me-4-Ac
Me 2-Br-3- (U-3b) cPr 3-Me-4- (U-3b)
Me 2-Br-3-CF₂H cPr 3-Me-4-CF₂H
Me 2-Br-3-CN cPr 3-Me-4-CN
Me 2-Br-3-Et cPr 3-Me-4-Et
Me 2-Br-3-OCF₂H cPr 3-Me-4-OCF₂H
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Me 2-Br-3-OEt cPr 3-Me-4-OEt
Me 2-Br-3-C (O) CF_Three      cPr 3-Me-4-C (O) CF_Three
Me 2-Me-3-Ac cPr 3-CF_Three-4-Ac
Me 2-Me-3- (U-3b) cPr 3-CF_Three-4- (U-3b)
Me 2-Me-3-CF₂H cPr 3-CF_Three-4-CF₂H
Me 2-Me-3-CN cPr 3-CF_Three-4-CN
Me 2-Me-3-Et cPr 3-CF_Three-4-Et
Me 2-Me-3-OCF₂H cPr 3-CF_Three-4-OCF₂H
Me 2-Me-3-OEt cPr 3-CF_Three-4-OEt
Me 2-Me-3-C (O) CF_Three      cPr 3-CF_Three-4-C (O) CF_Three
Me 2-CF_Three-3-Ac cPr 3-OMe-4-Ac
Me 2-CF_Three-3- (U-3b) cPr 3-OMe-4- (U-3b)
Me 2-CF_Three-3-CF₂H cPr 3-OMe-4-CF₂H
Me 2-CF_Three-3-CN cPr 3-OMe-4-CN
Me 2-CF_Three-3-Et cPr 3-OMe-4-Et
Me 2-CF_Three-3-OCF₂H cPr 3-OMe-4-OCF₂H
Me 2-CF_Three-3-OEt cPr 3-OMe-4-OEt
Me 2-CF_Three-3-C (O) CF_Three     cPr 3-OMe-4-C (O) CF_Three
Me 2-OMe-3-Ac cPr 3-OCF_Three-4-Ac
Me 2-OMe-3- (U-3b) cPr 3-OCF_Three-4- (U-3b)
Me 2-OMe-3-CF₂H cPr 3-OCF_Three-4-CF₂H
Me 2-OMe-3-CN cPr 3-OCF_Three-4-CN
Me 2-OMe-3-Et cPr 3-OCF_Three-4-Et
Me 2-OMe-3-OCF₂H cPr 3-OCF_Three-4-OCF₂H
Me 2-OMe-3-OEt cPr 3-OCF_Three-4-OEt
Me 2-OMe-3-C (O) CF_Three     cPr 3-OCF_Three-4-C (O) CF_Three
Me 2-OCF_Three-3-Ac cPr 3-F-5-Ac
Me 2-OCF_Three-3- (U-3b) cPr 3-F-5- (U-3b)
Me 2-OCF_Three-3-CF₂H cPr 3-F-5-CF₂H
Me 2-OCF_Three-3-CN cPr 3-F-5-CN
Me 2-OCF_Three-3-Et cPr 3-F-5-Et
Me 2-OCF_Three-3-OCF₂H cPr 3-F-5-OCF₂H
Me 2-OCF_Three-3-OEt cPr 3-F-5-OEt
Me 2-OCF_Three-3-C (O) CF_Three    cPr 3-F-5-C (O) CF_Three
Me 2-F-4-Ac cPr 3-Cl-5-Ac
Me 2-F-4- (U-3b) cPr 3-Cl-5- (U-3b)
Me 2-F-4-CF₂H cPr 3-Cl-5-CF₂H
Me 2-F-4-CN cPr 3-Cl-5-CN
Me 2-F-4-Et cPr 3-Cl-5-Et
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Me 2-F-4-OCF₂H cPr 3-Cl-5-OCF₂H
Me 2-F-4-OEt cPr 3-Cl-5-OEt
Me 2-F-4-C (O) CF_Three       cPr 3-Cl-5-C (O) CF_Three
Me 2-Cl-4-Ac cPr 3-Br-5-Ac
Me 2-Cl-4- (U-3b) cPr 3-Br-5- (U-3b)
Me 2-Cl-4-CF₂H cPr 3-Br-5-CF₂H
Me 2-Cl-4-CN cPr 3-Br-5-CN
Me 2-Cl-4-Et cPr 3-Br-5-Et
Me 2-Cl-4-OCF₂H cPr 3-Br-5-OCF₂H
Me 2-Cl-4-OEt cPr 3-Br-5-OEt
Me 2-Cl-4-C (O) CF_Three      cPr 3-Br-5-C (O) CF_Three
Me 2-Br-4-Ac cPr 3-Me-5-Ac
Me 2-Br-4- (U-3b) cPr 3-Me-5- (U-3b)
Me 2-Br-4-CF₂H cPr 3-Me-5-CF₂H
Me 2-Br-4-CN cPr 3-Me-5-CN
Me 2-Br-4-Et cPr 3-Me-5-Et
Me 2-Br-4-OCF₂H cPr 3-Me-5-OCF₂H
Me 2-Br-4-OEt cPr 3-Me-5-OEt
Me 2-Br-4-C (O) CF_Three      cPr 3-Me-5-C (O) CF_Three
Me 2-Me-4-Ac cPr 3-CF_Three-5-Ac
Me 2-Me-4- (U-3b) cPr 3-CF_Three-5- (U-3b)
Me 2-Me-4-CF₂H cPr 3-CF_Three-5-CF₂H
Me 2-Me-4-CN cPr 3-CF_Three-5-CN
Me 2-Me-4-Et cPr 3-CF_Three-5-Et
Me 2-Me-4-OCF₂H cPr 3-CF_Three-5-OCF₂H
Me 2-Me-4-OEt cPr 3-CF_Three-5-OEt
Me 2-Me-4-C (O) CF_Three      cPr 3-CF_Three-5-C (O) CF_Three
Me 2-CF_Three-4-Ac cPr 3-OMe-5-Ac
Me 2-CF_Three-4- (U-3b) cPr 3-OMe-5- (U-3b)
Me 2-CF_Three-4-CF₂H cPr 3-OMe-5-CF₂H
Me 2-CF_Three-4-CN cPr 3-OMe-5-CN
Me 2-CF_Three-4-Et cPr 3-OMe-5-Et
Me 2-CF_Three-4-OCF₂H cPr 3-OMe-5-OCF₂H
Me 2-CF_Three-4-OEt cPr 3-OMe-5-OEt
Me 2-CF_Three-4-C (O) CF_Three     cPr 3-OMe-5-C (O) CF_Three
Me 2-OMe-4-Ac cPr 3-OCF_Three-5-Ac
Me 2-OMe-4- (U-3b) cPr 3-OCF_Three-5- (U-3b)
Me 2-OMe-4-CF₂H cPr 3-OCF_Three-5-CF₂H
Me 2-OMe-4-CN cPr 3-OCF_Three-5-CN
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Me 2-OMe-4-Et cPr 3-OCF_Three-5-Et
Me 2-OMe-4-OCF₂H cPr 3-OCF_Three-5-OCF₂H
Me 2-OMe-4-OEt cPr 3-OCF_Three-5-OEt
Me 2-OMe-4-C (O) CF_Three     cPr 3-OCF_Three-5-C (O) CF_Three
Me 2-OCF_Three-4-Ac cPr 2-Ac-3-F
Me 2-OCF_Three-4- (U-3b) cPr 2-Ac-3-Cl
Me 2-OCF_Three-4-CF₂H cPr 2-Ac-3-Br
Me 2-OCF_Three-4-CN cPr 2-Ac-3-Me
Me 2-OCF_Three-4-Et cPr 2-Ac-3-CF_Three
Me 2-OCF_Three-4-OCF₂H cPr 2-Ac-3-OMe
Me 2-OCF_Three-4-OEt cPr 2-Ac-3-OCF_Three
Me 2-OCF_Three-4-C (O) CF_Three    cPr 2- (U-3b) -3-F
Me 2-F-5-Ac cPr 2- (U-3b) -3-Cl
Me 2-F-5- (U-3b) cPr 2- (U-3b) -3-Br
Me 2-F-5-CF₂H cPr 2- (U-3b) -3-Me
Me 2-F-5-CN cPr 2- (U-3b) -3-CF_Three
Me 2-F-5-Et cPr 2- (U-3b) -3-OMe
Me 2-F-5-OCF₂H cPr 2- (U-3b) -3-OCF_Three
Me 2-F-5-OEt cPr 2-CF₂H-3-F
Me 2-F-5-C (O) CF_Three       cPr 2-CF₂H-3-Cl
Me 2-Cl-5-Ac cPr 2-CF₂H-3-Br
Me 2-Cl-5- (U-3b) cPr 2-CF₂H-3-Me
Me 2-Cl-5-CF₂H cPr 2-CF₂H-3-CF_Three
Me 2-Cl-5-CN cPr 2-CF₂H-3-OMe
Me 2-Cl-5-Et cPr 2-CF₂H-3-OCF_Three
Me 2-Cl-5-OCF₂H cPr 2-CN-3-F
Me 2-Cl-5-OEt cPr 2-CN-3-Cl
Me 2-Cl-5-C (O) CF_Three      cPr 2-CN-3-Br
Me 2-Br-5-Ac cPr 2-CN-3-Me
Me 2-Br-5- (U-3b) cPr 2-CN-3-CF_Three
Me 2-Br-5-CF₂H cPr 2-CN-3-OMe
Me 2-Br-5-CN cPr 2-CN-3-OCF_Three
Me 2-Br-5-Et cPr 2-Et-3-F
Me 2-Br-5-OCF₂H cPr 2-Et-3-Cl
Me 2-Br-5-OEt cPr 2-Et-3-Br
Me 2-Br-5-C (O) CF_Three      cPr 2-Et-3-Me
Me 2-Me-5-Ac cPr 2-Et-3-CF_Three
Me 2-Me-5- (U-3b) cPr 2-Et-3-OMe
Me 2-Me-5-CF₂H cPr 2-Et-3-OCF_Three
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Me 2-Me-5-CN cPr 2-OCF₂H-3-F
Me 2-Me-5-Et cPr 2-OCF₂H-3-Cl
Me 2-Me-5-OCF₂H cPr 2-OCF₂H-3-Br
Me 2-Me-5-OEt cPr 2-OCF₂H-3-Me
Me 2-Me-5-C (O) CF_Three      cPr 2-OCF₂H-3-CF_Three
Me 2-CF_Three-5-Ac cPr 2-OCF₂H-3-OMe
Me 2-CF_Three-5- (U-3b) cPr 2-OCF₂H-3-OCF_Three
Me 2-CF_Three-5-CF₂H cPr 2-OEt-3-F
Me 2-CF_Three-5-CN cPr 2-OEt-3-Cl
Me 2-CF_Three-5-Et cPr 2-OEt-3-Br
Me 2-CF_Three-5-OCF₂H cPr 2-OEt-3-Me
Me 2-CF_Three-5-OEt cPr 2-OEt-3-CF_Three
Me 2-CF_Three-5-C (O) CF_Three     cPr 2-OEt-3-OMe
Me 2-OMe-5-Ac cPr 2-OEt-3-OCF_Three
Me 2-OMe-5- (U-3b) cPr 2-C (O) CF_Three-3-F
Me 2-OMe-5-CF₂H cPr 2-C (O) CF_Three-3-Cl
Me 2-OMe-5-CN cPr 2-C (O) CF_Three-3-Br
Me 2-OMe-5-Et cPr 2-C (O) CF_Three-3-Me
Me 2-OMe-5-OCF₂H cPr 2-C (O) CF_Three-3-CF_Three
Me 2-OMe-5-OEt cPr 2-C (O) CF_Three-3-OMe
Me 2-OMe-5-C (O) CF_Three     cPr 2-C (O) CF_Three-3-OCF_Three
Me 2-OCF_Three-5-Ac cPr 2-Ac-4-F
Me 2-OCF_Three-5- (U-3b) cPr 2-Ac-4-Cl
Me 2-OCF_Three-5-CF₂H cPr 2-Ac-4-Br
Me 2-OCF_Three-5-CN cPr 2-Ac-4-Me
Me 2-OCF_Three-5-Et cPr 2-Ac-4-CF_Three
Me 2-OCF_Three-5-OCF₂H cPr 2-Ac-4-OMe
Me 2-OCF_Three-5-OEt cPr 2-Ac-4-OCF_Three
Me 2-OCF_Three-5-C (O) CF_Three    cPr 2- (U-3b) -4-F
Me 3-F-4-Ac cPr 2- (U-3b) -4-Cl
Me 3-F-4- (U-3b) cPr 2- (U-3b) -4-Br
Me 3-F-4-CF₂H cPr 2- (U-3b) -4-Me
Me 3-F-4-CN cPr 2- (U-3b) -4-CF_Three
Me 3-F-4-Et cPr 2- (U-3b) -4-OMe
Me 3-F-4-OCF₂H cPr 2- (U-3b) -4-OCF_Three
Me 3-F-4-OEt cPr 2-CF₂H-4-F
Me 3-F-4-C (O) CF_Three       cPr 2-CF₂H-4-Cl
Me 3-Cl-4-Ac cPr 2-CF₂H-4-Br
Me 3-Cl-4- (U-3b) cPr 2-CF₂H-4-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Me 3-Cl-4-CF₂H cPr 2-CF₂H-4-CF_Three
Me 3-Cl-4-CN cPr 2-CF₂H-4-OMe
Me 3-Cl-4-Et cPr 2-CF₂H-4-OCF_Three
Me 3-Cl-4-OCF₂H cPr 2-CN-4-F
Me 3-Cl-4-OEt cPr 2-CN-4-Cl
Me 3-Cl-4-C (O) CF_Three      cPr 2-CN-4-Br
Me 3-Br-4-Ac cPr 2-CN-4-Me
Me 3-Br-4- (U-3b) cPr 2-CN-4-CF_Three
Me 3-Br-4-CF₂H cPr 2-CN-4-OMe
Me 3-Br-4-CN cPr 2-CN-4-OCF_Three
Me 3-Br-4-Et cPr 2-Et-4-F
Me 3-Br-4-OCF₂H cPr 2-Et-4-Cl
Me 3-Br-4-OEt cPr 2-Et-4-Br
Me 3-Br-4-C (O) CF_Three      cPr 2-Et-4-Me
Me 3-Me-4-Ac cPr 2-Et-4-CF_Three
Me 3-Me-4- (U-3b) cPr 2-Et-4-OMe
Me 3-Me-4-CF₂H cPr 2-Et-4-OCF_Three
Me 3-Me-4-CN cPr 2-OCF₂H-4-F
Me 3-Me-4-Et cPr 2-OCF₂H-4-Cl
Me 3-Me-4-OCF₂H cPr 2-OCF₂H-4-Br
Me 3-Me-4-OEt cPr 2-OCF₂H-4-Me
Me 3-Me-4-C (O) CF_Three      cPr 2-OCF₂H-4-CF_Three
Me 3-CF_Three-4-Ac cPr 2-OCF₂H-4-OMe
Me 3-CF_Three-4- (U-3b) cPr 2-OCF₂H-4-OCF_Three
Me 3-CF_Three-4-CF₂H cPr 2-OEt-4-F
Me 3-CF_Three-4-CN cPr 2-OEt-4-Cl
Me 3-CF_Three-4-Et cPr 2-OEt-4-Br
Me 3-CF_Three-4-OCF₂H cPr 2-OEt-4-Me
Me 3-CF_Three-4-OEt cPr 2-OEt-4-CF_Three
Me 3-CF_Three-4-C (O) CF_Three     cPr 2-OEt-4-OMe
Me 3-OMe-4-Ac cPr 2-OEt-4-OCF_Three
Me 3-OMe-4- (U-3b) cPr 2-C (O) CF_Three-4-F
Me 3-OMe-4-CF₂H cPr 2-C (O) CF_Three-4-Cl
Me 3-OMe-4-CN cPr 2-C (O) CF_Three-4-Br
Me 3-OMe-4-Et cPr 2-C (O) CF_Three-4-Me
Me 3-OMe-4-OCF₂H cPr 2-C (O) CF_Three-4-CF_Three
Me 3-OMe-4-OEt cPr 2-C (O) CF_Three-4-OMe
Me 3-OMe-4-C (O) CF_Three     cPr 2-C (O) CF_Three-4-OCF_Three
Me 3-OCF_Three-4-Ac cPr 2-Ac-5-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Me 3-OCF_Three-4- (U-3b) cPr 2-Ac-5-Cl
Me 3-OCF_Three-4-CF₂H cPr 2-Ac-5-Br
Me 3-OCF_Three-4-CN cPr 2-Ac-5-Me
Me 3-OCF_Three-4-Et cPr 2-Ac-5-CF_Three
Me 3-OCF_Three-4-OCF₂H cPr 2-Ac-5-OMe
Me 3-OCF_Three-4-OEt cPr 2-Ac-5-OCF_Three
Me 3-OCF_Three-4-C (O) CF_Three    cPr 2- (U-3b) -5-F
Me 3-F-5-Ac cPr 2- (U-3b) -5-Cl
Me 3-F-5- (U-3b) cPr 2- (U-3b) -5-Br
Me 3-F-5-CF₂H cPr 2- (U-3b) -5-Me
Me 3-F-5-CN cPr 2- (U-3b) -5-CF_Three
Me 3-F-5-Et cPr 2- (U-3b) -5-OMe
Me 3-F-5-OCF₂H cPr 2- (U-3b) -5-OCF_Three
Me 3-F-5-OEt cPr 2-CF₂H-5-F
Me 3-F-5-C (O) CF_Three       cPr 2-CF₂H-5-Cl
Me 3-Cl-5-Ac cPr 2-CF₂H-5-Br
Me 3-Cl-5- (U-3b) cPr 2-CF₂H-5-Me
Me 3-Cl-5-CF₂H cPr 2-CF₂H-5-CF_Three
Me 3-Cl-5-CN cPr 2-CF₂H-5-OMe
Me 3-Cl-5-Et cPr 2-CF₂H-5-OCF_Three
Me 3-Cl-5-OCF₂H cPr 2-CN-5-F
Me 3-Cl-5-OEt cPr 2-CN-5-Cl
Me 3-Cl-5-C (O) CF_Three      cPr 2-CN-5-Br
Me 3-Br-5-Ac cPr 2-CN-5-Me
Me 3-Br-5- (U-3b) cPr 2-CN-5-CF_Three
Me 3-Br-5-CF₂H cPr 2-CN-5-OMe
Me 3-Br-5-CN cPr 2-CN-5-OCF_Three
Me 3-Br-5-Et cPr 2-Et-5-F
Me 3-Br-5-OCF₂H cPr 2-Et-5-Cl
Me 3-Br-5-OEt cPr 2-Et-5-Br
Me 3-Br-5-C (O) CF_Three      cPr 2-Et-5-Me
Me 3-Me-5-Ac cPr 2-Et-5-CF_Three
Me 3-Me-5- (U-3b) cPr 2-Et-5-OMe
Me 3-Me-5-CF₂H cPr 2-Et-5-OCF_Three
Me 3-Me-5-CN cPr 2-OCF₂H-5-F
Me 3-Me-5-Et cPr 2-OCF₂H-5-Cl
Me 3-Me-5-OCF₂H cPr 2-OCF₂H-5-Br
Me 3-Me-5-OEt cPr 2-OCF₂H-5-Me
Me 3-Me-5-C (O) CF_Three      cPr 2-OCF₂H-5-CF_Three
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Me 3-CF_Three-5-Ac cPr 2-OCF₂H-5-OMe
Me 3-CF_Three-5- (U-3b) cPr 2-OCF₂H-5-OCF_Three
Me 3-CF_Three-5-CF₂H cPr 2-OEt-5-F
Me 3-CF_Three-5-CN cPr 2-OEt-5-Cl
Me 3-CF_Three-5-Et cPr 2-OEt-5-Br
Me 3-CF_Three-5-OCF₂H cPr 2-OEt-5-Me
Me 3-CF_Three-5-OEt cPr 2-OEt-5-CF_Three
Me 3-CF_Three-5-C (O) CF_Three     cPr 2-OEt-5-OMe
Me 3-OMe-5-Ac cPr 2-OEt-5-OCF_Three
Me 3-OMe-5- (U-3b) cPr 2-C (O) CF_Three-5-F
Me 3-OMe-5-CF₂H cPr 2-C (O) CF_Three-5-Cl
Me 3-OMe-5-CN cPr 2-C (O) CF_Three-5-Br
Me 3-OMe-5-Et cPr 2-C (O) CF_Three-5-Me
Me 3-OMe-5-OCF₂H cPr 2-C (O) CF_Three-5-CF_Three
Me 3-OMe-5-OEt cPr 2-C (O) CF_Three-5-OMe
Me 3-OMe-5-C (O) CF_Three     cPr 2-C (O) CF_Three-5-OCF_Three
Me 3-OCF_Three-5-Ac cPr 3-Ac-4-F
Me 3-OCF_Three-5- (U-3b) cPr 3-Ac-4-Cl
Me 3-OCF_Three-5-CF₂H cPr 3-Ac-4-Br
Me 3-OCF_Three-5-CN cPr 3-Ac-4-Me
Me 3-OCF_Three-5-Et cPr 3-Ac-4-CF_Three
Me 3-OCF_Three-5-OCF₂H cPr 3-Ac-4-OMe
Me 3-OCF_Three-5-OEt cPr 3-Ac-4-OCF_Three
Me 3-OCF_Three-5-C (O) CF_Three    cPr 3- (U-3b) -4-F
Me 2-Ac-3-F cPr 3- (U-3b) -4-Cl
Me 2-Ac-3-Cl cPr 3- (U-3b) -4-Br
Me 2-Ac-3-Br cPr 3- (U-3b) -4-Me
Me 2-Ac-3-Me cPr 3- (U-3b) -4-CF_Three
Me 2-Ac-3-CF_Three          cPr 3- (U-3b) -4-OMe
Me 2-Ac-3-OMe cPr 3- (U-3b) -4-OCF_Three
Me 2-Ac-3-OCF_Three         cPr 3-CF₂H-4-F
Me 2- (U-3b) -3-F cPr 3-CF₂H-4-Cl
Me 2- (U-3b) -3-Cl cPr 3-CF₂H-4-Br
Me 2- (U-3b) -3-Br cPr 3-CF₂H-4-Me
Me 2- (U-3b) -3-Me cPr 3-CF₂H-4-CF_Three
Me 2- (U-3b) -3-CF_Three      cPr 3-CF₂H-4-OMe
Me 2- (U-3b) -3-OMe cPr 3-CF₂H-4-OCF_Three
Me 2- (U-3b) -3-OCF_Three     cPr 3-CN-4-F
Me 2-CF₂H-3-F cPr 3-CN-4-Cl
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Me 2-CF₂H-3-Cl cPr 3-CN-4-Br
Me 2-CF₂H-3-Br cPr 3-CN-4-Me
Me 2-CF₂H-3-Me cPr 3-CN-4-CF_Three
Me 2-CF₂H-3-CF_Three        cPr 3-CN-4-OMe
Me 2-CF₂H-3-OMe cPr 3-CN-4-OCF_Three
Me 2-CF₂H-3-OCF_Three       cPr 3-Et-4-F
Me 2-CN-3-F cPr 3-Et-4-Cl
Me 2-CN-3-Cl cPr 3-Et-4-Br
Me 2-CN-3-Br cPr 3-Et-4-Me
Me 2-CN-3-Me cPr 3-Et-4-CF_Three
Me 2-CN-3-CF_Three          cPr 3-Et-4-OMe
Me 2-CN-3-OMe cPr 3-Et-4-OCF_Three
Me 2-CN-3-OCF_Three         cPr 3-OCF₂H-4-F
Me 2-Et-3-F cPr 3-OCF₂H-4-Cl
Me 2-Et-3-Cl cPr 3-OCF₂H-4-Br
Me 2-Et-3-Br cPr 3-OCF₂H-4-Me
Me 2-Et-3-Me cPr 3-OCF₂H-4-CF_Three
Me 2-Et-3-CF_Three          cPr 3-OCF₂H-4-OMe
Me 2-Et-3-OMe cPr 3-OCF₂H-4-OCF_Three
Me 2-Et-3-OCF_Three         cPr 3-OEt-4-F
Me 2-OCF₂H-3-F cPr 3-OEt-4-Cl
Me 2-OCF₂H-3-Cl cPr 3-OEt-4-Br
Me 2-OCF₂H-3-Br cPr 3-OEt-4-Me
Me 2-OCF₂H-3-Me cPr 3-OEt-4-CF_Three
Me 2-OCF₂H-3-CF_Three       cPr 3-OEt-4-OMe
Me 2-OCF₂H-3-OMe cPr 3-OEt-4-OCF_Three
Me 2-OCF₂H-3-OCF_Three      cPr 3-C (O) CF_Three-4-F
Me 2-OEt-3-F cPr 3-C (O) CF_Three-4-Cl
Me 2-OEt-3-Cl cPr 3-C (O) CF_Three-4-Br
Me 2-OEt-3-Br cPr 3-C (O) CF_Three-4-Me
Me 2-OEt-3-Me cPr 3-C (O) CF_Three-4-CF_Three
Me 2-OEt-3-CF_Three         cPr 3-C (O) CF_Three-4-OMe
Me 2-OEt-3-OMe cPr 3-C (O) CF_Three-4-OCF_Three
Me 2-OEt-3-OCF_Three        cPr 3-Ac-5-F
Me 2-C (O) CF_Three-3-F cPr 3-Ac-5-Cl
Me 2-C (O) CF_Three-3-Cl cPr 3-Ac-5-Br
Me 2-C (O) CF_Three-3-Br cPr 3-Ac-5-Me
Me 2-C (O) CF_Three-3-Me cPr 3-Ac-5-CF_Three
Me 2-C (O) CF_Three-3-CF_Three     cPr 3-Ac-5-OMe
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Me 2-C (O) CF_Three-3-OMe cPr 3-Ac-5-OCF_Three
Me 2-C (O) CF_Three-3-OCF_Three    cPr 3- (U-3b) -5-F
Me 2-Ac-4-F cPr 3- (U-3b) -5-Cl
Me 2-Ac-4-Cl cPr 3- (U-3b) -5-Br
Me 2-Ac-4-Br cPr 3- (U-3b) -5-Me
Me 2-Ac-4-Me cPr 3- (U-3b) -5-CF_Three
Me 2-Ac-4-CF_Three          cPr 3- (U-3b) -5-OMe
Me 2-Ac-4-OMe cPr 3- (U-3b) -5-OCF_Three
Me 2-Ac-4-OCF_Three         cPr 3-CF₂H-5-F
Me 2- (U-3b) -4-F cPr 3-CF₂H-5-Cl
Me 2- (U-3b) -4-Cl cPr 3-CF₂H-5-Br
Me 2- (U-3b) -4-Br cPr 3-CF₂H-5-Me
Me 2- (U-3b) -4-Me cPr 3-CF₂H-5-CF_Three
Me 2- (U-3b) -4-CF_Three      cPr 3-CF₂H-5-OMe
Me 2- (U-3b) -4-OMe cPr 3-CF₂H-5-OCF_Three
Me 2- (U-3b) -4-OCF_Three     cPr 3-CN-5-F
Me 2-CF₂H-4-F cPr 3-CN-5-Cl
Me 2-CF₂H-4-Cl cPr 3-CN-5-Br
Me 2-CF₂H-4-Br cPr 3-CN-5-Me
Me 2-CF₂H-4-Me cPr 3-CN-5-CF_Three
Me 2-CF₂H-4-CF_Three        cPr 3-CN-5-OMe
Me 2-CF₂H-4-OMe cPr 3-CN-5-OCF_Three
Me 2-CF₂H-4-OCF_Three       cPr 3-Et-5-F
Me 2-CN-4-F cPr 3-Et-5-Cl
Me 2-CN-4-Cl cPr 3-Et-5-Br
Me 2-CN-4-Br cPr 3-Et-5-Me
Me 2-CN-4-Me cPr 3-Et-5-CF_Three
Me 2-CN-4-CF_Three          cPr 3-Et-5-OMe
Me 2-CN-4-OMe cPr 3-Et-5-OCF_Three
Me 2-CN-4-OCF_Three         cPr 3-OCF₂H-5-F
Me 2-Et-4-F cPr 3-OCF₂H-5-Cl
Me 2-Et-4-Cl cPr 3-OCF₂H-5-Br
Me 2-Et-4-Br cPr 3-OCF₂H-5-Me
Me 2-Et-4-Me cPr 3-OCF₂H-5-CF_Three
Me 2-Et-4-CF_Three          cPr 3-OCF₂H-5-OMe
Me 2-Et-4-OMe cPr 3-OCF₂H-5-OCF_Three
Me 2-Et-4-OCF_Three         cPr 3-OEt-5-F
Me 2-OCF₂H-4-F cPr 3-OEt-5-Cl
Me 2-OCF₂H-4-Cl cPr 3-OEt-5-Br
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Me 2-OCF₂H-4-Br cPr 3-OEt-5-Me
Me 2-OCF₂H-4-Me cPr 3-OEt-5-CF_Three
Me 2-OCF₂H-4-CF_Three       cPr 3-OEt-5-OMe
Me 2-OCF₂H-4-OMe cPr 3-OEt-5-OCF_Three
Me 2-OCF₂H-4-OCF_Three      cPr 3-C (O) CF_Three-5-F
Me 2-OEt-4-F cPr 3-C (O) CF_Three-5-Cl
Me 2-OEt-4-Cl cPr 3-C (O) CF_Three-5-Br
Me 2-OEt-4-Br cPr 3-C (O) CF_Three-5-Me
Me 2-OEt-4-Me cPr 3-C (O) CF_Three-5-CF_Three
Me 2-OEt-4-CF_Three         cPr 3-C (O) CF_Three-5-OMe
Me 2-OEt-4-OMe cPr 3-C (O) CF_Three-5-OCF_Three
Me 2-OEt-4-OCF_Three        Me 2,3,4-tri-F
Me 2-C (O) CF_Three-4-F Me 2,3-di-F-4-Cl
Me 2-C (O) CF_Three-4-Cl Me 2,3-di-F-4-Br
Me 2-C (O) CF_Three-4-Br Me 2,3-di-F-4-Me
Me 2-C (O) CF_Three-4-Me Me 2,3-di-F-4-CF_Three
Me 2-C (O) CF_Three-4-CF_Three     Me 2,3-di-F-4-OMe
Me 2-C (O) CF_Three-4-OMe Me 2,4-di-F-3-Cl
Me 2-C (O) CF_Three-4-OCF_Three    Me 2-F-3,4-di-Cl
Me 2-Ac-5-F Me 2-F-3-Cl-4-Br
Me 2-Ac-5-Cl Me 2-F-3-Cl-4-Me
Me 2-Ac-5-Br Me 2-F-3-Cl-4-CF_Three
Me 2-Ac-5-Me Me 2-F-3-Cl-4-OMe
Me 2-Ac-5-CF_Three          Me 2,4-di-F-3-Br
Me 2-Ac-5-OMe Me 2-F-3-Br-4-Cl
Me 2-Ac-5-OCF_Three         Me 2-F-3,4-di-Br
Me 2- (U-3b) -5-F Me 2-F-3-Br-4-Me
Me 2- (U-3b) -5-Cl Me 2-F-3-Br-4-CF_Three
Me 2- (U-3b) -5-Br Me 2-F-3-Br-4-OMe
Me 2- (U-3b) -5-Me Me 2,4-di-F-3-Me
Me 2- (U-3b) -5-CF_Three      Me 2-F-3-Me-4-Cl
Me 2- (U-3b) -5-OMe Me 2-F-3-Me-4-Br
Me 2- (U-3b) -5-OCF_Three     Me 2-F-3,4-di-Me
Me 2-CF₂H-5-F Me 2-F-3-Me-4-CF_Three
Me 2-CF₂H-5-Cl Me 2-F-3-Me-4-OMe
Me 2-CF₂H-5-Br Me 2,4-di-F-3-CF_Three
Me 2-CF₂H-5-Me Me 2-F-3-CF_Three-4-Cl
Me 2-CF₂H-5-CF_Three        Me 2-F-3-CF_Three-4-Br
Me 2-CF₂H-5-OMe Me 2-F-3-CF_Three-4-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Me 2-CF₂H-5-OCF_Three       Me 2-F-3,4-di-CF_Three
Me 2-CN-5-F Me 2-F-3-CF_Three-4-OMe
Me 2-CN-5-Cl Me 2,4-di-F-3-OMe
Me 2-CN-5-Br Me 2-F-3-OMe-4-Cl
Me 2-CN-5-Me Me 2-F-3-OMe-4-Br
Me 2-CN-5-CF_Three          Me 2-F-3-OMe-4-Me
Me 2-CN-5-OMe Me 2-F-3-OMe-4-CF_Three
Me 2-CN-5-OCF_Three         Me 2-F-3,4-di-OMe
Me 2-Et-5-F Me 2,3,5-tri-F
Me 2-Et-5-Cl Me 2,3-di-F-5-Cl
Me 2-Et-5-Br Me 2,3-di-F-5-Br
Me 2-Et-5-Me Me 2,3-di-F-5-Me
Me 2-Et-5-CF_Three          Me 2,3-di-F-5-CF_Three
Me 2-Et-5-OMe Me 2,3-di-F-5-OMe
Me 2-Et-5-OCF_Three         Me 2,5-di-F-3-Cl
Me 2-OCF₂H-5-F Me 2-F-3,5-di-Cl
Me 2-OCF₂H-5-Cl Me 2-F-3-Cl-5-Br
Me 2-OCF₂H-5-Br Me 2-F-3-Cl-5-Me
Me 2-OCF₂H-5-Me Me 2-F-3-Cl-5-CF_Three
Me 2-OCF₂H-5-CF_Three       Me 2-F-3-Cl-5-OMe
Me 2-OCF₂H-5-OMe Me 2,5-di-F-3-Br
Me 2-OCF₂H-5-OCF_Three      Me 2-F-3-Br-5-Cl
Me 2-OEt-5-F Me 2-F-3,5-di-Br
Me 2-OEt-5-Cl Me 2-F-3-Br-5-Me
Me 2-OEt-5-Br Me 2-F-3-Br-5-CF_Three
Me 2-OEt-5-Me Me 2-F-3-Br-5-OMe
Me 2-OEt-5-CF_Three         Me 2,5-di-F-3-Me
Me 2-OEt-5-OMe Me 2-F-3-Me-5-Cl
Me 2-OEt-5-OCF_Three        Me 2-F-3-Me-5-Br
Me 2-C (O) CF_Three-5-F Me 2-F-3,5-di-Me
Me 2-C (O) CF_Three-5-Cl Me 2-F-3-Me-5-CF_Three
Me 2-C (O) CF_Three-5-Br Me 2-F-3-Me-5-OMe
Me 2-C (O) CF_Three-5-Me Me 2,5-di-F-3-CF_Three
Me 2-C (O) CF_Three-5-CF_Three     Me 2-F-3-CF_Three-5-Cl
Me 2-C (O) CF_Three-5-OMe Me 2-F-3-CF_Three-5-Br
Me 2-C (O) CF_Three-5-OCF_Three    Me 2-F-3-CF_Three-5-Me
Me 3-Ac-4-F Me 2-F-3,5-di-CF_Three
Me 3-Ac-4-Cl Me 2-F-3-CF_Three-5-OMe
Me 3-Ac-4-Br Me 2,5-di-F-3-OMe
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Me 3-Ac-4-Me Me 2-F-3-OMe-5-Cl
Me 3-Ac-4-CF_Three          Me 2-F-3-OMe-5-Br
Me 3-Ac-4-OMe Me 2-F-3-OMe-5-Me
Me 3-Ac-4-OCF_Three         Me 2-F-3-OMe-5-CF_Three
Me 3- (U-3b) -4-F Me 2-F-3,5-di-OMe
Me 3- (U-3b) -4-Cl Me 2,4,5-tri-F
Me 3- (U-3b) -4-Br Me 2,4-di-F-5-Cl
Me 3- (U-3b) -4-Me Me 2,4-di-F-5-Br
Me 3- (U-3b) -4-CF_Three      Me 2,4-di-F-5-Me
Me 3- (U-3b) -4-OMe Me 2,4-di-F-5-CF_Three
Me 3- (U-3b) -4-OCF_Three     Me 2,4-di-F-5-OMe
Me 3-CF₂H-4-F Me 2,5-di-F-4-Cl
Me 3-CF₂H-4-Cl Me 2-F-4,5-di-Cl
Me 3-CF₂H-4-Br Me 2-F-4-Cl-5-Br
Me 3-CF₂H-4-Me Me 2-F-4-Cl-5-Me
Me 3-CF₂H-4-CF_Three        Me 2-F-4-Cl-5-CF_Three
Me 3-CF₂H-4-OMe Me 2-F-4-Cl-5-OMe
Me 3-CF₂H-4-OCF_Three       Me 2,5-di-F-4-Br
Me 3-CN-4-F Me 2-F-4-Br-5-Cl
Me 3-CN-4-Cl Me 2-F-4,5-di-Br
Me 3-CN-4-Br Me 2-F-4-Br-5-Me
Me 3-CN-4-Me Me 2-F-4-Br-5-CF_Three
Me 3-CN-4-CF_Three          Me 2-F-4-Br-5-OMe
Me 3-CN-4-OMe Me 2,5-di-F-4-Me
Me 3-CN-4-OCF_Three         Me 2-F-4-Me-5-Cl
Me 3-Et-4-F Me 2-F-4-Me-5-Br
Me 3-Et-4-Cl Me 2-F-4,5-di-Me
Me 3-Et-4-Br Me 2-F-4-Me-5-CF_Three
Me 3-Et-4-Me Me 2-F-4-Me-5-OMe
Me 3-Et-4-CF_Three          Me 2,5-di-F-4-CF_Three
Me 3-Et-4-OMe Me 2-F-4-CF_Three-5-Cl
Me 3-Et-4-OCF_Three         Me 2-F-4-CF_Three-5-Br
Me 3-OCF₂H-4-F Me 2-F-4-CF_Three-5-Me
Me 3-OCF₂H-4-Cl Me 2-F-4,5-di-CF_Three
Me 3-OCF₂H-4-Br Me 2-F-4-CF_Three-5-OMe
Me 3-OCF₂H-4-Me Me 2,5-di-F-4-OMe
Me 3-OCF₂H-4-CF_Three       Me 2-F-4-OMe-5-Cl
Me 3-OCF₂H-4-OMe Me 2-F-4-OMe-5-Br
Me 3-OCF₂H-4-OCF_Three      Me 2-F-4-OMe-5-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Me 3-OEt-4-F Me 2-F-4-OMe-5-CF_Three
Me 3-OEt-4-Cl Me 2-F-4,5-di-OMe
Me 3-OEt-4-Br Me 3,4,5-tri-F
Me 3-OEt-4-Me Me 3,4-di-F-5-Cl
Me 3-OEt-4-CF_Three         Me 3,4-di-F-5-Br
Me 3-OEt-4-OMe Me 3,4-di-F-5-Me
Me 3-OEt-4-OCF_Three        Me 3,4-di-F-5-CF_Three
Me 3-C (O) CF_Three-4-F Me 3,4-di-F-5-OMe
Me 3-C (O) CF_Three-4-Cl Me 3,5-di-F-4-Cl
Me 3-C (O) CF_Three-4-Br Me 3-F-4,5-di-Cl
Me 3-C (O) CF_Three-4-Me Me 3-F-4-Cl-5-Br
Me 3-C (O) CF_Three-4-CF_Three     Me 3-F-4-Cl-5-Me
Me 3-C (O) CF_Three-4-OMe Me 3-F-4-Cl-5-CF_Three
Me 3-C (O) CF_Three-4-OCF_Three    Me 3-F-4-Cl-5-OMe
Me 3-Ac-5-F Me 3,5-di-F-4-Br
Me 3-Ac-5-Cl Me 3-F-4-Br-5-Cl
Me 3-Ac-5-Br Me 3-F-4,5-di-Br
Me 3-Ac-5-Me Me 3-F-4-Br-5-Me
Me 3-Ac-5-CF_Three          Me 3-F-4-Br-5-CF_Three
Me 3-Ac-5-OMe Me 3-F-4-Br-5-OMe
Me 3-Ac-5-OCF_Three         Me 3,5-di-F-4-Me
Me 3- (U-3b) -5-F Me 3-F-4-Me-5-Cl
Me 3- (U-3b) -5-Cl Me 3-F-4-Me-5-Br
Me 3- (U-3b) -5-Br Me 3-F-4,5-di-Me
Me 3- (U-3b) -5-Me Me 3-F-4-Me-5-CF_Three
Me 3- (U-3b) -5-CF_Three      Me 3-F-4-Me-5-OMe
Me 3- (U-3b) -5-OMe Me 3,5-di-F-4-CF_Three
Me 3- (U-3b) -5-OCF_Three     Me 3-F-4-CF_Three-5-Cl
Me 3-CF₂H-5-F Me 3-F-4-CF_Three-5-Br
Me 3-CF₂H-5-Cl Me 3-F-4-CF_Three-5-Me
Me 3-CF₂H-5-Br Me 3-F-4,5-di-CF_Three
Me 3-CF₂H-5-Me Me 3-F-4-CF_Three-5-OMe
Me 3-CF₂H-5-CF_Three        Me 3,5-di-F-4-OMe
Me 3-CF₂H-5-OMe Me 3-F-4-OMe-5-Cl
Me 3-CF₂H-5-OCF_Three       Me 3-F-4-OMe-5-Br
Me 3-CN-5-F Me 3-F-4-OMe-5-Me
Me 3-CN-5-Cl Me 3-F-4-OMe-5-CF_Three
Me 3-CN-5-Br Me 3-F-4,5-di-OMe
Me 3-CN-5-Me Me 2-Cl-3,4-di-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Me 3-CN-5-CF_Three          Me 2,4-di-Cl-3-F
Me 3-CN-5-OMe Me 2-Cl-3-F-4-Br
Me 3-CN-5-OCF_Three         Me 2-Cl-3-F-4-Me
Me 3-Et-5-F Me 2-Cl-3-F-4-CF_Three
Me 3-Et-5-Cl Me 2-Cl-3-F-4-OMe
Me 3-Et-5-Br Me 2,3-di-Cl-4-F
Me 3-Et-5-Me Me 2,3,4-tri-Cl
Me 3-Et-5-CF_Three          Me 2,3-di-Cl-4-Br
Me 3-Et-5-OMe Me 2,3-di-Cl-4-Me
Me 3-Et-5-OCF_Three         Me 2,3-di-Cl-4-CF_Three
Me 3-OCF₂H-5-F Me 2,3-di-Cl-4-OMe
Me 3-OCF₂H-5-Cl Me 2-Cl-3-Br-4-F
Me 3-OCF₂H-5-Br Me 2,4-di-Cl-3-Br
Me 3-OCF₂H-5-Me Me 2-Cl-3,4-di-Br
Me 3-OCF₂H-5-CF_Three       Me 2-Cl-3-Br-4-Me
Me 3-OCF₂H-5-OMe Me 2-Cl-3-Br-4-CF_Three
Me 3-OCF₂H-5-OCF_Three      Me 2-Cl-3-Br-4-OMe
Me 3-OEt-5-F Me 2-Cl-3-Me-4-F
Me 3-OEt-5-Cl Me 2,4-di-Cl-3-Me
Me 3-OEt-5-Br Me 2-Cl-3-Me-4-Br
Me 3-OEt-5-Me Me 2-Cl-3,4-di-Me
Me 3-OEt-5-CF_Three         Me 2-Cl-3-Me-4-CF_Three
Me 3-OEt-5-OMe Me 2-Cl-3-Me-4-OMe
Me 3-OEt-5-OCF_Three        Me 2-Cl-3-CF_Three-4-F
Me 3-C (O) CF_Three-5-F Me 2,4-di-Cl-3-CF_Three
Me 3-C (O) CF_Three-5-Cl Me 2-Cl-3-CF_Three-4-Br
Me 3-C (O) CF_Three-5-Br Me 2-Cl-3-CF_Three-4-Me
Me 3-C (O) CF_Three-5-Me Me 2-Cl-3,4-di-CF_Three
Me 3-C (O) CF_Three-5-CF_Three     Me 2-Cl-3-CF_Three-4-OMe
Me 3-C (O) CF_Three-5-OMe Me 2-Cl-3-OMe-4-F
Me 3-C (O) CF_Three-5-OCF_Three    Me 2,4-di-Cl-3-OMe
Et 2-F-3-Ac Me 2-Cl-3-OMe-4-Br
Et 2-F-3- (U-3b) Me 2-Cl-3-OMe-4-Me
Et 2-F-3-CF₂H Me 2-Cl-3-OMe-4-CF_Three
Et 2-F-3-CN Me 2-Cl-3,4-di-OMe
Et 2-F-3-Et Me 2-Cl-3,5-di-F
Et 2-F-3-OCF₂H Me 2,5-di-Cl-3-F
Et 2-F-3-OEt Me 2-Cl-3-F-5-Br
Et 2-F-3-C (O) CF_Three       Me 2-Cl-3-F-5-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Et 2-Cl-3-Ac Me 2-Cl-3-F-5-CF_Three
Et 2-Cl-3- (U-3b) Me 2-Cl-3-F-5-OMe
Et 2-Cl-3-CF₂H Me 2,3-di-Cl-5-F
Et 2-Cl-3-CN Me 2,3,5-tri-Cl
Et 2-Cl-3-Et Me 2,3-di-Cl-5-Br
Et 2-Cl-3-OCF₂H Me 2,3-di-Cl-5-Me
Et 2-Cl-3-OEt Me 2,3-di-Cl-5-CF_Three
Et 2-Cl-3-C (O) CF_Three      Me 2,3-di-Cl-5-OMe
Et 2-Br-3-Ac Me 2-Cl-3-Br-5-F
Et 2-Br-3- (U-3b) Me 2,5-di-Cl-3-Br
Et 2-Br-3-CF₂H Me 2-Cl-3,5-di-Br
Et 2-Br-3-CN Me 2-Cl-3-Br-5-Me
Et 2-Br-3-Et Me 2-Cl-3-Br-5-CF_Three
Et 2-Br-3-OCF₂H Me 2-Cl-3-Br-5-OMe
Et 2-Br-3-OEt Me 2-Cl-3-Me-5-F
Et 2-Br-3-C (O) CF_Three      Me 2,5-di-Cl-3-Me
Et 2-Me-3-Ac Me 2-Cl-3-Me-5-Br
Et 2-Me-3- (U-3b) Me 2-Cl-3,5-di-Me
Et 2-Me-3-CF₂H Me 2-Cl-3-Me-5-CF_Three
Et 2-Me-3-CN Me 2-Cl-3-Me-5-OMe
Et 2-Me-3-Et Me 2-Cl-3-CF_Three-5-F
Et 2-Me-3-OCF₂H Me 2,5-di-Cl-3-CF_Three
Et 2-Me-3-OEt Me 2-Cl-3-CF_Three-5-Br
Et 2-Me-3-C (O) CF_Three      Me 2-Cl-3-CF_Three-5-Me
Et 2-CF_Three-3-Ac Me 2-Cl-3,5-di-CF_Three
Et 2-CF_Three-3- (U-3b) Me 2-Cl-3-CF_Three-5-OMe
Et 2-CF_Three-3-CF₂H Me 2-Cl-3-OMe-5-F
Et 2-CF_Three-3-CN Me 2,5-di-Cl-3-OMe
Et 2-CF_Three-3-Et Me 2-Cl-3-OMe-5-Br
Et 2-CF_Three-3-OCF₂H Me 2-Cl-3-OMe-5-Me
Et 2-CF_Three-3-OEt Me 2-Cl-3-OMe-5-CF_Three
Et 2-CF_Three-3-C (O) CF_Three     Me 2-Cl-3,5-di-OMe
Et 2-OMe-3-Ac Me 2-Cl-4,5-di-F
Et 2-OMe-3- (U-3b) Me 2,5-di-Cl-4-F
Et 2-OMe-3-CF₂H Me 2-Cl-4-F-5-Br
Et 2-OMe-3-CN Me 2-Cl-4-F-5-Me
Et 2-OMe-3-Et Me 2-Cl-4-F-5-CF_Three
Et 2-OMe-3-OCF₂H Me 2-Cl-4-F-5-OMe
Et 2-OMe-3-OEt Me 2,4-di-Cl-5-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Et 2-OMe-3-C (O) CF_Three     Me 2,4,5-tri-Cl
Et 2-OCF_Three-3-Ac Me 2,4-di-Cl-5-Br
Et 2-OCF_Three-3- (U-3b) Me 2,4-di-Cl-5-Me
Et 2-OCF_Three-3-CF₂H Me 2,4-di-Cl-5-CF_Three
Et 2-OCF_Three-3-CN Me 2,4-di-Cl-5-OMe
Et 2-OCF_Three-3-Et Me 2-Cl-4-Br-5-F
Et 2-OCF_Three-3-OCF₂H Me 2,5-di-Cl-4-Br
Et 2-OCF_Three-3-OEt Me 2-Cl-4,5-di-Br
Et 2-OCF_Three-3-C (O) CF_Three    Me 2-Cl-4-Br-5-Me
Et 2-F-4-Ac Me 2-Cl-4-Br-5-CF_Three
Et 2-F-4- (U-3b) Me 2-Cl-4-Br-5-OMe
Et 2-F-4-CF₂H Me 2-Cl-4-Me-5-F
Et 2-F-4-CN Me 2,5-di-Cl-4-Me
Et 2-F-4-Et Me 2-Cl-4-Me-5-Br
Et 2-F-4-OCF₂H Me 2-Cl-4,5-di-Me
Et 2-F-4-OEt Me 2-Cl-4-Me-5-CF_Three
Et 2-F-4-C (O) CF_Three       Me 2-Cl-4-Me-5-OMe
Et 2-Cl-4-Ac Me 2-Cl-4-CF_Three-5-F
Et 2-Cl-4- (U-3b) Me 2,5-di-Cl-4-CF_Three
Et 2-Cl-4-CF₂H Me 2-Cl-4-CF_Three-5-Br
Et 2-Cl-4-CN Me 2-Cl-4-CF_Three-5-Me
Et 2-Cl-4-Et Me 2-Cl-4,5-di-CF_Three
Et 2-Cl-4-OCF₂H Me 2-Cl-4-CF_Three-5-OMe
Et 2-Cl-4-OEt Me 2-Cl-4-OMe-5-F
Et 2-Cl-4-C (O) CF_Three      Me 2,5-di-Cl-4-OMe
Et 2-Br-4-Ac Me 2-Cl-4-OMe-5-Br
Et 2-Br-4- (U-3b) Me 2-Cl-4-OMe-5-Me
Et 2-Br-4-CF₂H Me 2-Cl-4-OMe-5-CF_Three
Et 2-Br-4-CN Me 2-Cl-4,5-di-OMe
Et 2-Br-4-Et Me 3-Cl-4,5-di-F
Et 2-Br-4-OCF₂H Me 3,5-di-Cl-4-F
Et 2-Br-4-OEt Me 3-Cl-4-F-5-Br
Et 2-Br-4-C (O) CF_Three      Me 3-Cl-4-F-5-Me
Et 2-Me-4-Ac Me 3-Cl-4-F-5-CF_Three
Et 2-Me-4- (U-3b) Me 3-Cl-4-F-5-OMe
Et 2-Me-4-CF₂H Me 3,4-di-Cl-5-F
Et 2-Me-4-CN Me 3,4,5-tri-Cl
Et 2-Me-4-Et Me 3,4-di-Cl-5-Br
Et 2-Me-4-OCF₂H Me 3,4-di-Cl-5-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Et 2-Me-4-OEt Me 3,4-di-Cl-5-CF_Three
Et 2-Me-4-C (O) CF_Three      Me 3,4-di-Cl-5-OMe
Et 2-CF_Three-4-Ac Me 3-Cl-4-Br-5-F
Et 2-CF_Three-4- (U-3b) Me 3,5-di-Cl-4-Br
Et 2-CF_Three-4-CF₂H Me 3-Cl-4,5-di-Br
Et 2-CF_Three-4-CN Me 3-Cl-4-Br-5-Me
Et 2-CF_Three-4-Et Me 3-Cl-4-Br-5-CF_Three
Et 2-CF_Three-4-OCF₂H Me 3-Cl-4-Br-5-OMe
Et 2-CF_Three-4-OEt Me 3-Cl-4-Me-5-F
Et 2-CF_Three-4-C (O) CF_Three     Me 3,5-di-Cl-4-Me
Et 2-OMe-4-Ac Me 3-Cl-4-Me-5-Br
Et 2-OMe-4- (U-3b) Me 3-Cl-4,5-di-Me
Et 2-OMe-4-CF₂H Me 3-Cl-4-Me-5-CF_Three
Et 2-OMe-4-CN Me 3-Cl-4-Me-5-OMe
Et 2-OMe-4-Et Me 3-Cl-4-CF_Three-5-F
Et 2-OMe-4-OCF₂H Me 3,5-di-Cl-4-CF_Three
Et 2-OMe-4-OEt Me 3-Cl-4-CF_Three-5-Br
Et 2-OMe-4-C (O) CF_Three     Me 3-Cl-4-CF_Three-5-Me
Et 2-OCF_Three-4-Ac Me 3-Cl-4,5-di-CF_Three
Et 2-OCF_Three-4- (U-3b) Me 3-Cl-4-CF_Three-5-OMe
Et 2-OCF_Three-4-CF₂H Me 3-Cl-4-OMe-5-F
Et 2-OCF_Three-4-CN Me 3,5-di-Cl-4-OMe
Et 2-OCF_Three-4-Et Me 3-Cl-4-OMe-5-Br
Et 2-OCF_Three-4-OCF₂H Me 3-Cl-4-OMe-5-Me
Et 2-OCF_Three-4-OEt Me 3-Cl-4-OMe-5-CF_Three
Et 2-OCF_Three-4-C (O) CF_Three    Me 3-Cl-4,5-di-OMe
Et 2-F-5-Ac Me 2-Br-3,4-di-F
Et 2-F-5- (U-3b) Me 2-Br-3-F-4-Cl
Et 2-F-5-CF₂H Me 2,4-di-Br-3-F
Et 2-F-5-CN Me 2-Br-3-F-4-Me
Et 2-F-5-Et Me 2-Br-3-F-4-CF_Three
Et 2-F-5-OCF₂H Me 2-Br-3-F-4-OMe
Et 2-F-5-OEt Me 2-Br-3-Cl-4-F
Et 2-F-5-C (O) CF_Three       Me 2-Br-3,4-di-Cl
Et 2-Cl-5-Ac Me 2,4-di-Br-3-Cl
Et 2-Cl-5- (U-3b) Me 2-Br-3-Cl-4-Me
Et 2-Cl-5-CF₂H Me 2-Br-3-Cl-4-CF_Three
Et 2-Cl-5-CN Me 2-Br-3-Cl-4-OMe
Et 2-Cl-5-Et Me 2,3-di-Br-4-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Et 2-Cl-5-OCF₂H Me 2,3-di-Br-4-Cl
Et 2-Cl-5-OEt Me 2,3,4-tri-Br
Et 2-Cl-5-C (O) CF_Three      Me 2,3-di-Br-4-Me
Et 2-Br-5-Ac Me 2,3-di-Br-4-CF_Three
Et 2-Br-5- (U-3b) Me 2,3-di-Br-4-OMe
Et 2-Br-5-CF₂H Me 2-Br-3-Me-4-F
Et 2-Br-5-CN Me 2-Br-3-Me-4-Cl
Et 2-Br-5-Et Me 2,4-di-Br-3-Me
Et 2-Br-5-OCF₂H Me 2-Br-3,4-di-Me
Et 2-Br-5-OEt Me 2-Br-3-Me-4-CF_Three
Et 2-Br-5-C (O) CF_Three      Me 2-Br-3-Me-4-OMe
Et 2-Me-5-Ac Me 2-Br-3-CF_Three-4-F
Et 2-Me-5- (U-3b) Me 2-Br-3-CF_Three-4-Cl
Et 2-Me-5-CF₂H Me 2,4-di-Br-3-CF_Three
Et 2-Me-5-CN Me 2-Br-3-CF_Three-4-Me
Et 2-Me-5-Et Me 2-Br-3,4-di-CF_Three
Et 2-Me-5-OCF₂H Me 2-Br-3-CF_Three-4-OMe
Et 2-Me-5-OEt Me 2-Br-3-OMe-4-F
Et 2-Me-5-C (O) CF_Three      Me 2-Br-3-OMe-4-Cl
Et 2-CF_Three-5-Ac Me 2,4-di-Br-3-OMe
Et 2-CF_Three-5- (U-3b) Me 2-Br-3-OMe-4-Me
Et 2-CF_Three-5-CF₂H Me 2-Br-3-OMe-4-CF_Three
Et 2-CF_Three-5-CN Me 2-Br-3,4-di-OMe
Et 2-CF_Three-5-Et Me 2-Br-3,5-di-F
Et 2-CF_Three-5-OCF₂H Me 2-Br-3-F-5-Cl
Et 2-CF_Three-5-OEt Me 2,5-di-Br-3-F
Et 2-CF_Three-5-C (O) CF_Three     Me 2-Br-3-F-5-Me
Et 2-OMe-5-Ac Me 2-Br-3-F-5-CF_Three
Et 2-OMe-5- (U-3b) Me 2-Br-3-F-5-OMe
Et 2-OMe-5-CF₂H Me 2-Br-3-Cl-5-F
Et 2-OMe-5-CN Me 2-Br-3,5-di-Cl
Et 2-OMe-5-Et Me 2,5-di-Br-3-Cl
Et 2-OMe-5-OCF₂H Me 2-Br-3-Cl-5-Me
Et 2-OMe-5-OEt Me 2-Br-3-Cl-5-CF_Three
Et 2-OMe-5-C (O) CF_Three     Me 2-Br-3-Cl-5-OMe
Et 2-OCF_Three-5-Ac Me 2,3-di-Br-5-F
Et 2-OCF_Three-5- (U-3b) Me 2,3-di-Br-5-Cl
Et 2-OCF_Three-5-CF₂H Me 2,3,5-tri-Br
Et 2-OCF_Three-5-CN Me 2,3-di-Br-5-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Et 2-OCF_Three-5-Et Me 2,3-di-Br-5-CF_Three
Et 2-OCF_Three-5-OCF₂H Me 2,3-di-Br-5-OMe
Et 2-OCF_Three-5-OEt Me 2-Br-3-Me-5-F
Et 2-OCF_Three-5-C (O) CF_Three    Me 2-Br-3-Me-5-Cl
Et 3-F-4-Ac Me 2,5-di-Br-3-Me
Et 3-F-4- (U-3b) Me 2-Br-3,5-di-Me
Et 3-F-4-CF₂H Me 2-Br-3-Me-5-CF_Three
Et 3-F-4-CN Me 2-Br-3-Me-5-OMe
Et 3-F-4-Et Me 2-Br-3-CF_Three-5-F
Et 3-F-4-OCF₂H Me 2-Br-3-CF_Three-5-Cl
Et 3-F-4-OEt Me 2,5-di-Br-3-CF_Three
Et 3-F-4-C (O) CF_Three       Me 2-Br-3-CF_Three-5-Me
Et 3-Cl-4-Ac Me 2-Br-3,5-di-CF_Three
Et 3-Cl-4- (U-3b) Me 2-Br-3-CF_Three-5-OMe
Et 3-Cl-4-CF₂H Me 2-Br-3-OMe-5-F
Et 3-Cl-4-CN Me 2-Br-3-OMe-5-Cl
Et 3-Cl-4-Et Me 2,5-di-Br-3-OMe
Et 3-Cl-4-OCF₂H Me 2-Br-3-OMe-5-Me
Et 3-Cl-4-OEt Me 2-Br-3-OMe-5-CF_Three
Et 3-Cl-4-C (O) CF_Three      Me 2-Br-3,5-di-OMe
Et 3-Br-4-Ac Me 2-Br-4,5-di-F
Et 3-Br-4- (U-3b) Me 2-Br-4-F-5-Cl
Et 3-Br-4-CF₂H Me 2,5-di-Br-4-F
Et 3-Br-4-CN Me 2-Br-4-F-5-Me
Et 3-Br-4-Et Me 2-Br-4-F-5-CF_Three
Et 3-Br-4-OCF₂H Me 2-Br-4-F-5-OMe
Et 3-Br-4-OEt Me 2-Br-4-Cl-5-F
Et 3-Br-4-C (O) CF_Three      Me 2-Br-4,5-di-Cl
Et 3-Me-4-Ac Me 2,5-di-Br-4-Cl
Et 3-Me-4- (U-3b) Me 2-Br-4-Cl-5-Me
Et 3-Me-4-CF₂H Me 2-Br-4-Cl-5-CF_Three
Et 3-Me-4-CN Me 2-Br-4-Cl-5-OMe
Et 3-Me-4-Et Me 2,4-di-Br-5-F
Et 3-Me-4-OCF₂H Me 2,4-di-Br-5-Cl
Et 3-Me-4-OEt Me 2,4,5-tri-Br
Et 3-Me-4-C (O) CF_Three      Me 2,4-di-Br-5-Me
Et 3-CF_Three-4-Ac Me 2,4-di-Br-5-CF_Three
Et 3-CF_Three-4- (U-3b) Me 2,4-di-Br-5-OMe
Et 3-CF_Three-4-CF₂H Me 2-Br-4-Me-5-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Et 3-CF_Three-4-CN Me 2-Br-4-Me-5-Cl
Et 3-CF_Three-4-Et Me 2,5-di-Br-4-Me
Et 3-CF_Three-4-OCF₂H Me 2-Br-4,5-di-Me
Et 3-CF_Three-4-OEt Me 2-Br-4-Me-5-CF_Three
Et 3-CF_Three-4-C (O) CF_Three     Me 2-Br-4-Me-5-OMe
Et 3-OMe-4-Ac Me 2-Br-4-CF_Three-5-F
Et 3-OMe-4- (U-3b) Me 2-Br-4-CF_Three-5-Cl
Et 3-OMe-4-CF₂H Me 2,5-di-Br-4-CF_Three
Et 3-OMe-4-CN Me 2-Br-4-CF_Three-5-Me
Et 3-OMe-4-Et Me 2-Br-4,5-di-CF_Three
Et 3-OMe-4-OCF₂H Me 2-Br-4-CF_Three-5-OMe
Et 3-OMe-4-OEt Me 2-Br-4-OMe-5-F
Et 3-OMe-4-C (O) CF_Three     Me 2-Br-4-OMe-5-Cl
Et 3-OCF_Three-4-Ac Me 2,5-di-Br-4-OMe
Et 3-OCF_Three-4- (U-3b) Me 2-Br-4-OMe-5-Me
Et 3-OCF_Three-4-CF₂H Me 2-Br-4-OMe-5-CF_Three
Et 3-OCF_Three-4-CN Me 2-Br-4,5-di-OMe
Et 3-OCF_Three-4-Et Me 3-Br-4,5-di-F
Et 3-OCF_Three-4-OCF₂H Me 3-Br-4-F-5-Cl
Et 3-OCF_Three-4-OEt Me 3,5-di-Br-4-F
Et 3-OCF_Three-4-C (O) CF_Three    Me 3-Br-4-F-5-Me
Et 3-F-5-Ac Me 3-Br-4-F-5-CF_Three
Et 3-F-5- (U-3b) Me 3-Br-4-F-5-OMe
Et 3-F-5-CF₂H Me 3-Br-4-Cl-5-F
Et 3-F-5-CN Me 3-Br-4,5-di-Cl
Et 3-F-5-Et Me 3,5-di-Br-4-Cl
Et 3-F-5-OCF₂H Me 3-Br-4-Cl-5-Me
Et 3-F-5-OEt Me 3-Br-4-Cl-5-CF_Three
Et 3-F-5-C (O) CF_Three       Me 3-Br-4-Cl-5-OMe
Et 3-Cl-5-Ac Me 3,4-di-Br-5-F
Et 3-Cl-5- (U-3b) Me 3,4-di-Br-5-Cl
Et 3-Cl-5-CF₂H Me 3,4,5-tri-Br
Et 3-Cl-5-CN Me 3,4-di-Br-5-Me
Et 3-Cl-5-Et Me 3,4-di-Br-5-CF_Three
Et 3-Cl-5-OCF₂H Me 3,4-di-Br-5-OMe
Et 3-Cl-5-OEt Me 3-Br-4-Me-5-F
Et 3-Cl-5-C (O) CF_Three      Me 3-Br-4-Me-5-Cl
Et 3-Br-5-Ac Me 3,5-di-Br-4-Me
Et 3-Br-5- (U-3b) Me 3-Br-4,5-di-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Et 3-Br-5-CF₂H Me 3-Br-4-Me-5-CF_Three
Et 3-Br-5-CN Me 3-Br-4-Me-5-OMe
Et 3-Br-5-Et Me 3-Br-4-CF_Three-5-F
Et 3-Br-5-OCF₂H Me 3-Br-4-CF_Three-5-Cl
Et 3-Br-5-OEt Me 3,5-di-Br-4-CF_Three
Et 3-Br-5-C (O) CF_Three      Me 3-Br-4-CF_Three-5-Me
Et 3-Me-5-Ac Me 3-Br-4,5-di-CF_Three
Et 3-Me-5- (U-3b) Me 3-Br-4-CF_Three-5-OMe
Et 3-Me-5-CF₂H Me 3-Br-4-OMe-5-F
Et 3-Me-5-CN Me 3-Br-4-OMe-5-Cl
Et 3-Me-5-Et Me 3,5-di-Br-4-OMe
Et 3-Me-5-OCF₂H Me 3-Br-4-OMe-5-Me
Et 3-Me-5-OEt Me 3-Br-4-OMe-5-CF_Three
Et 3-Me-5-C (O) CF_Three      Me 3-Br-4,5-di-OMe
Et 3-CF_Three-5-Ac Me 2-Me-3,4-di-F
Et 3-CF_Three-5- (U-3b) Me 2-Me-3-F-4-Cl
Et 3-CF_Three-5-CF₂H Me 2-Me-3-F-4-Br
Et 3-CF_Three-5-CN Me 2,4-di-Me-3-F
Et 3-CF_Three-5-Et Me 2-Me-3-F-4-CF_Three
Et 3-CF_Three-5-OCF₂H Me 2-Me-3-F-4-OMe
Et 3-CF_Three-5-OEt Me 2-Me-3-Cl-4-F
Et 3-CF_Three-5-C (O) CF_Three     Me 2-Me-3,4-di-Cl
Et 3-OMe-5-Ac Me 2-Me-3-Cl-4-Br
Et 3-OMe-5- (U-3b) Me 2,4-di-Me-3-Cl
Et 3-OMe-5-CF₂H Me 2-Me-3-Cl-4-CF_Three
Et 3-OMe-5-CN Me 2-Me-3-Cl-4-OMe
Et 3-OMe-5-Et Me 2-Me-3-Br-4-F
Et 3-OMe-5-OCF₂H Me 2-Me-3-Br-4-Cl
Et 3-OMe-5-OEt Me 2-Me-3,4-di-Br
Et 3-OMe-5-C (O) CF_Three     Me 2,4-di-Me-3-Br
Et 3-OCF_Three-5-Ac Me 2-Me-3-Br-4-CF_Three
Et 3-OCF_Three-5- (U-3b) Me 2-Me-3-Br-4-OMe
Et 3-OCF_Three-5-CF₂H Me 2,3-di-Me-4-F
Et 3-OCF_Three-5-CN Me 2,3-di-Me-4-Cl
Et 3-OCF_Three-5-Et Me 2,3-di-Me-4-Br
Et 3-OCF_Three-5-OCF₂H Me 2,3,4-tri-Me
Et 3-OCF_Three-5-OEt Me 2,3-di-Me-4-CF_Three
Et 3-OCF_Three-5-C (O) CF_Three    Me 2,3-di-Me-4-OMe
Et 2-Ac-3-F Me 2-Me-3-CF_Three-4-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Et 2-Ac-3-Cl Me 2-Me-3-CF_Three-4-Cl
Et 2-Ac-3-Br Me 2-Me-3-CF_Three-4-Br
Et 2-Ac-3-Me Me 2,4-di-Me-3-CF_Three
Et 2-Ac-3-CF_Three          Me 2-Me-3,4-di-CF_Three
Et 2-Ac-3-OMe Me 2-Me-3-CF_Three-4-OMe
Et 2-Ac-3-OCF_Three         Me 2-Me-3-OMe-4-F
Et 2- (U-3b) -3-F Me 2-Me-3-OMe-4-Cl
Et 2- (U-3b) -3-Cl Me 2-Me-3-OMe-4-Br
Et 2- (U-3b) -3-Br Me 2,4-di-Me-3-OMe
Et 2- (U-3b) -3-Me Me 2-Me-3-OMe-4-CF_Three
Et 2- (U-3b) -3-CF_Three      Me 2-Me-3,4-di-OMe
Et 2- (U-3b) -3-OMe Me 2-Me-3,5-di-F
Et 2- (U-3b) -3-OCF_Three     Me 2-Me-3-F-5-Cl
Et 2-CF₂H-3-F Me 2-Me-3-F-5-Br
Et 2-CF₂H-3-Cl Me 2,5-di-Me-3-F
Et 2-CF₂H-3-Br Me 2-Me-3-F-5-CF_Three
Et 2-CF₂H-3-Me Me 2-Me-3-F-5-OMe
Et 2-CF₂H-3-CF_Three        Me 2-Me-3-Cl-5-F
Et 2-CF₂H-3-OMe Me 2-Me-3,5-di-Cl
Et 2-CF₂H-3-OCF_Three       Me 2-Me-3-Cl-5-Br
Et 2-CN-3-F Me 2,5-di-Me-3-Cl
Et 2-CN-3-Cl Me 2-Me-3-Cl-5-CF_Three
Et 2-CN-3-Br Me 2-Me-3-Cl-5-OMe
Et 2-CN-3-Me Me 2-Me-3-Br-5-F
Et 2-CN-3-CF_Three          Me 2-Me-3-Br-5-Cl
Et 2-CN-3-OMe Me 2-Me-3,5-di-Br
Et 2-CN-3-OCF_Three         Me 2,5-di-Me-3-Br
Et 2-Et-3-F Me 2-Me-3-Br-5-CF_Three
Et 2-Et-3-Cl Me 2-Me-3-Br-5-OMe
Et 2-Et-3-Br Me 2,3-di-Me-5-F
Et 2-Et-3-Me Me 2,3-di-Me-5-Cl
Et 2-Et-3-CF_Three          Me 2,3-di-Me-5-Br
Et 2-Et-3-OMe Me 2,3,5-tri-Me
Et 2-Et-3-OCF_Three         Me 2,3-di-Me-5-CF_Three
Et 2-OCF₂H-3-F Me 2,3-di-Me-5-OMe
Et 2-OCF₂H-3-Cl Me 2-Me-3-CF_Three-5-F
Et 2-OCF₂H-3-Br Me 2-Me-3-CF_Three-5-Cl
Et 2-OCF₂H-3-Me Me 2-Me-3-CF_Three-5-Br
Et 2-OCF₂H-3-CF_Three       Me 2,5-di-Me-3-CF_Three
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Et 2-OCF₂H-3-OMe Me 2-Me-3,5-di-CF_Three
Et 2-OCF₂H-3-OCF_Three      Me 2-Me-3-CF_Three-5-OMe
Et 2-OEt-3-F Me 2-Me-3-OMe-5-F
Et 2-OEt-3-Cl Me 2-Me-3-OMe-5-Cl
Et 2-OEt-3-Br Me 2-Me-3-OMe-5-Br
Et 2-OEt-3-Me Me 2,5-di-Me-3-OMe
Et 2-OEt-3-CF_Three         Me 2-Me-3-OMe-5-CF_Three
Et 2-OEt-3-OMe Me 2-Me-3,5-di-OMe
Et 2-OEt-3-OCF_Three        Me 2-Me-4,5-di-F
Et 2-C (O) CF_Three-3-F Me 2-Me-4-F-5-Cl
Et 2-C (O) CF_Three-3-Cl Me 2-Me-4-F-5-Br
Et 2-C (O) CF_Three-3-Br Me 2,5-di-Me-4-F
Et 2-C (O) CF_Three-3-Me Me 2-Me-4-F-5-CF_Three
Et 2-C (O) CF_Three-3-CF_Three     Me 2-Me-4-F-5-OMe
Et 2-C (O) CF_Three-3-OMe Me 2-Me-4-Cl-5-F
Et 2-C (O) CF_Three-3-OCF_Three    Me 2-Me-4,5-di-Cl
Et 2-Ac-4-F Me 2-Me-4-Cl-5-Br
Et 2-Ac-4-Cl Me 2,5-di-Me-4-Cl
Et 2-Ac-4-Br Me 2-Me-4-Cl-5-CF_Three
Et 2-Ac-4-Me Me 2-Me-4-Cl-5-OMe
Et 2-Ac-4-CF_Three          Me 2-Me-4-Br-5-F
Et 2-Ac-4-OMe Me 2-Me-4-Br-5-Cl
Et 2-Ac-4-OCF_Three         Me 2-Me-4,5-di-Br
Et 2- (U-3b) -4-F Me 2,5-di-Me-4-Br
Et 2- (U-3b) -4-Cl Me 2-Me-4-Br-5-CF_Three
Et 2- (U-3b) -4-Br Me 2-Me-4-Br-5-OMe
Et 2- (U-3b) -4-Me Me 2,4-di-Me-5-F
Et 2- (U-3b) -4-CF_Three      Me 2,4-di-Me-5-Cl
Et 2- (U-3b) -4-OMe Me 2,4-di-Me-5-Br
Et 2- (U-3b) -4-OCF_Three     Me 2,4,5-tri-Me
Et 2-CF₂H-4-F Me 2,4-di-Me-5-CF_Three
Et 2-CF₂H-4-Cl Me 2,4-di-Me-5-OMe
Et 2-CF₂H-4-Br Me 2-Me-4-CF_Three-5-F
Et 2-CF₂H-4-Me Me 2-Me-4-CF_Three-5-Cl
Et 2-CF₂H-4-CF_Three        Me 2-Me-4-CF_Three-5-Br
Et 2-CF₂H-4-OMe Me 2,5-di-Me-4-CF_Three
Et 2-CF₂H-4-OCF_Three       Me 2-Me-4,5-di-CF_Three
Et 2-CN-4-F Me 2-Me-4-CF_Three-5-OMe
Et 2-CN-4-Cl Me 2-Me-4-OMe-5-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Et 2-CN-4-Br Me 2-Me-4-OMe-5-Cl
Et 2-CN-4-Me Me 2-Me-4-OMe-5-Br
Et 2-CN-4-CF_Three          Me 2,5-di-Me-4-OMe
Et 2-CN-4-OMe Me 2-Me-4-OMe-5-CF_Three
Et 2-CN-4-OCF_Three         Me 2-Me-4,5-di-OMe
Et 2-Et-4-F Me 3-Me-4,5-di-F
Et 2-Et-4-Cl Me 3-Me-4-F-5-Cl
Et 2-Et-4-Br Me 3-Me-4-F-5-Br
Et 2-Et-4-Me Me 3,5-di-Me-4-F
Et 2-Et-4-CF_Three          Me 3-Me-4-F-5-CF_Three
Et 2-Et-4-OMe Me 3-Me-4-F-5-OMe
Et 2-Et-4-OCF_Three         Me 3-Me-4-Cl-5-F
Et 2-OCF₂H-4-F Me 3-Me-4,5-di-Cl
Et 2-OCF₂H-4-Cl Me 3-Me-4-Cl-5-Br
Et 2-OCF₂H-4-Br Me 3,5-di-Me-4-Cl
Et 2-OCF₂H-4-Me Me 3-Me-4-Cl-5-CF_Three
Et 2-OCF₂H-4-CF_Three       Me 3-Me-4-Cl-5-OMe
Et 2-OCF₂H-4-OMe Me 3-Me-4-Br-5-F
Et 2-OCF₂H-4-OCF_Three      Me 3-Me-4-Br-5-Cl
Et 2-OEt-4-F Me 3-Me-4,5-di-Br
Et 2-OEt-4-Cl Me 3,5-di-Me-4-Br
Et 2-OEt-4-Br Me 3-Me-4-Br-5-CF_Three
Et 2-OEt-4-Me Me 3-Me-4-Br-5-OMe
Et 2-OEt-4-CF_Three         Me 3,4-di-Me-5-F
Et 2-OEt-4-OMe Me 3,4-di-Me-5-Cl
Et 2-OEt-4-OCF_Three        Me 3,4-di-Me-5-Br
Et 2-C (O) CF_Three-4-F Me 3,4,5-tri-Me
Et 2-C (O) CF_Three-4-Cl Me 3,4-di-Me-5-CF_Three
Et 2-C (O) CF_Three-4-Br Me 3,4-di-Me-5-OMe
Et 2-C (O) CF_Three-4-Me Me 3-Me-4-CF_Three-5-F
Et 2-C (O) CF_Three-4-CF_Three     Me 3-Me-4-CF_Three-5-Cl
Et 2-C (O) CF_Three-4-OMe Me 3-Me-4-CF_Three-5-Br
Et 2-C (O) CF_Three-4-OCF_Three    Me 3,5-di-Me-4-CF_Three
Et 2-Ac-5-F Me 3-Me-4,5-di-CF_Three
Et 2-Ac-5-Cl Me 3-Me-4-CF_Three-5-OMe
Et 2-Ac-5-Br Me 3-Me-4-OMe-5-F
Et 2-Ac-5-Me Me 3-Me-4-OMe-5-Cl
Et 2-Ac-5-CF_Three          Me 3-Me-4-OMe-5-Br
Et 2-Ac-5-OMe Me 3,5-di-Me-4-OMe
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Et 2-Ac-5-OCF_Three         Me 3-Me-4-OMe-5-CF_Three
Et 2- (U-3b) -5-F Me 3-Me-4,5-di-OMe
Et 2- (U-3b) -5-Cl Me 2-CF_Three-3,4-di-F
Et 2- (U-3b) -5-Br Me 2-CF_Three-3-F-4-Cl
Et 2- (U-3b) -5-Me Me 2-CF_Three-3-F-4-Br
Et 2- (U-3b) -5-CF_Three      Me 2-CF_Three-3-F-4-Me
Et 2- (U-3b) -5-OMe Me 2,4-di-CF_Three-3-F
Et 2- (U-3b) -5-OCF_Three     Me 2-CF_Three-3-F-4-OMe
Et 2-CF₂H-5-F Me 2-CF_Three-3-Cl-4-F
Et 2-CF₂H-5-Cl Me 2-CF_Three-3,4-di-Cl
Et 2-CF₂H-5-Br Me 2-CF_Three-3-Cl-4-Br
Et 2-CF₂H-5-Me Me 2-CF_Three-3-Cl-4-Me
Et 2-CF₂H-5-CF_Three        Me 2,4-di-CF_Three-3-Cl
Et 2-CF₂H-5-OMe Me 2-CF_Three-3-Cl-4-OMe
Et 2-CF₂H-5-OCF_Three       Me 2-CF_Three-3-Br-4-F
Et 2-CN-5-F Me 2-CF_Three-3-Br-4-Cl
Et 2-CN-5-Cl Me 2-CF_Three-3,4-di-Br
Et 2-CN-5-Br Me 2-CF_Three-3-Br-4-Me
Et 2-CN-5-Me Me 2,4-di-CF_Three-3-Br
Et 2-CN-5-CF_Three          Me 2-CF_Three-3-Br-4-OMe
Et 2-CN-5-OMe Me 2-CF_Three-3-Me-4-F
Et 2-CN-5-OCF_Three         Me 2-CF_Three-3-Me-4-Cl
Et 2-Et-5-F Me 2-CF_Three-3-Me-4-Br
Et 2-Et-5-Cl Me 2-CF_Three-3,4-di-Me
Et 2-Et-5-Br Me 2,4-di-CF_Three-3-Me
Et 2-Et-5-Me Me 2-CF_Three-3-Me-4-OMe
Et 2-Et-5-CF_Three          Me 2,3-di-CF_Three-4-F
Et 2-Et-5-OMe Me 2,3-di-CF_Three-4-Cl
Et 2-Et-5-OCF_Three         Me 2,3-di-CF_Three-4-Br
Et 2-OCF₂H-5-F Me 2,3-di-CF_Three-4-Me
Et 2-OCF₂H-5-Cl Me 2,3,4-tri-CF_Three
Et 2-OCF₂H-5-Br Me 2,3-di-CF_Three-4-OMe
Et 2-OCF₂H-5-Me Me 2-CF_Three-3-OMe-4-F
Et 2-OCF₂H-5-CF_Three       Me 2-CF_Three-3-OMe-4-Cl
Et 2-OCF₂H-5-OMe Me 2-CF_Three-3-OMe-4-Br
Et 2-OCF₂H-5-OCF_Three      Me 2-CF_Three-3-OMe-4-Me
Et 2-OEt-5-F Me 2,4-di-CF_Three-3-OMe
Et 2-OEt-5-Cl Me 2-CF_Three-3,4-di-OMe
Et 2-OEt-5-Br Me 2-CF_Three-3,5-di-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Et 2-OEt-5-Me Me 2-CF_Three-3-F-5-Cl
Et 2-OEt-5-CF_Three         Me 2-CF_Three-3-F-5-Br
Et 2-OEt-5-OMe Me 2-CF_Three-3-F-5-Me
Et 2-OEt-5-OCF_Three        Me 2,5-di-CF_Three-3-F
Et 2-C (O) CF_Three-5-F Me 2-CF_Three-3-F-5-OMe
Et 2-C (O) CF_Three-5-Cl Me 2-CF_Three-3-Cl-5-F
Et 2-C (O) CF_Three-5-Br Me 2-CF_Three-3,5-di-Cl
Et 2-C (O) CF_Three-5-Me Me 2-CF_Three-3-Cl-5-Br
Et 2-C (O) CF_Three-5-CF_Three     Me 2-CF_Three-3-Cl-5-Me
Et 2-C (O) CF_Three-5-OMe Me 2,5-di-CF_Three-3-Cl
Et 2-C (O) CF_Three-5-OCF_Three    Me 2-CF_Three-3-Cl-5-OMe
Et 3-Ac-4-F Me 2-CF_Three-3-Br-5-F
Et 3-Ac-4-Cl Me 2-CF_Three-3-Br-5-Cl
Et 3-Ac-4-Br Me 2-CF_Three-3,5-di-Br
Et 3-Ac-4-Me Me 2-CF_Three-3-Br-5-Me
Et 3-Ac-4-CF_Three          Me 2,5-di-CF_Three-3-Br
Et 3-Ac-4-OMe Me 2-CF_Three-3-Br-5-OMe
Et 3-Ac-4-OCF_Three         Me 2-CF_Three-3-Me-5-F
Et 3- (U-3b) -4-F Me 2-CF_Three-3-Me-5-Cl
Et 3- (U-3b) -4-Cl Me 2-CF_Three-3-Me-5-Br
Et 3- (U-3b) -4-Br Me 2-CF_Three-3,5-di-Me
Et 3- (U-3b) -4-Me Me 2,5-di-CF_Three-3-Me
Et 3- (U-3b) -4-CF_Three      Me 2-CF_Three-3-Me-5-OMe
Et 3- (U-3b) -4-OMe Me 2,3-di-CF_Three-5-F
Et 3- (U-3b) -4-OCF_Three     Me 2,3-di-CF_Three-5-Cl
Et 3-CF₂H-4-F Me 2,3-di-CF_Three-5-Br
Et 3-CF₂H-4-Cl Me 2,3-di-CF_Three-5-Me
Et 3-CF₂H-4-Br Me 2,3,5-tri-CF_Three
Et 3-CF₂H-4-Me Me 2,3-di-CF_Three-5-OMe
Et 3-CF₂H-4-CF_Three        Me 2-CF_Three-3-OMe-5-F
Et 3-CF₂H-4-OMe Me 2-CF_Three-3-OMe-5-Cl
Et 3-CF₂H-4-OCF_Three       Me 2-CF_Three-3-OMe-5-Br
Et 3-CN-4-F Me 2-CF_Three-3-OMe-5-Me
Et 3-CN-4-Cl Me 2,5-di-CF_Three-3-OMe
Et 3-CN-4-Br Me 2-CF_Three-3,5-di-OMe
Et 3-CN-4-Me Me 2-CF_Three-4,5-di-F
Et 3-CN-4-CF_Three          Me 2-CF_Three-4-F-5-Cl
Et 3-CN-4-OMe Me 2-CF_Three-4-F-5-Br
Et 3-CN-4-OCF_Three         Me 2-CF_Three-4-F-5-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Et 3-Et-4-F Me 2,5-di-CF_Three-4-F
Et 3-Et-4-Cl Me 2-CF_Three-4-F-5-OMe
Et 3-Et-4-Br Me 2-CF_Three-4-Cl-5-F
Et 3-Et-4-Me Me 2-CF_Three-4,5-di-Cl
Et 3-Et-4-CF_Three          Me 2-CF_Three-4-Cl-5-Br
Et 3-Et-4-OMe Me 2-CF_Three-4-Cl-5-Me
Et 3-Et-4-OCF_Three         Me 2,5-di-CF_Three-4-Cl
Et 3-OCF₂H-4-F Me 2-CF_Three-4-Cl-5-OMe
Et 3-OCF₂H-4-Cl Me 2-CF_Three-4-Br-5-F
Et 3-OCF₂H-4-Br Me 2-CF_Three-4-Br-5-Cl
Et 3-OCF₂H-4-Me Me 2-CF_Three-4,5-di-Br
Et 3-OCF₂H-4-CF_Three       Me 2-CF_Three-4-Br-5-Me
Et 3-OCF₂H-4-OMe Me 2,5-di-CF_Three-4-Br
Et 3-OCF₂H-4-OCF_Three      Me 2-CF_Three-4-Br-5-OMe
Et 3-OEt-4-F Me 2-CF_Three-4-Me-5-F
Et 3-OEt-4-Cl Me 2-CF_Three-4-Me-5-Cl
Et 3-OEt-4-Br Me 2-CF_Three-4-Me-5-Br
Et 3-OEt-4-Me Me 2-CF_Three-4,5-di-Me
Et 3-OEt-4-CF_Three         Me 2,5-di-CF_Three-4-Me
Et 3-OEt-4-OMe Me 2-CF_Three-4-Me-5-OMe
Et 3-OEt-4-OCF_Three        Me 2,4-di-CF_Three-5-F
Et 3-C (O) CF_Three-4-F Me 2,4-di-CF_Three-5-Cl
Et 3-C (O) CF_Three-4-Cl Me 2,4-di-CF_Three-5-Br
Et 3-C (O) CF_Three-4-Br Me 2,4-di-CF_Three-5-Me
Et 3-C (O) CF_Three-4-Me Me 2,4,5-tri-CF_Three
Et 3-C (O) CF_Three-4-CF_Three     Me 2,4-di-CF_Three-5-OMe
Et 3-C (O) CF_Three-4-OMe Me 2-CF_Three-4-OMe-5-F
Et 3-C (O) CF_Three-4-OCF_Three    Me 2-CF_Three-4-OMe-5-Cl
Et 3-Ac-5-F Me 2-CF_Three-4-OMe-5-Br
Et 3-Ac-5-Cl Me 2-CF_Three-4-OMe-5-Me
Et 3-Ac-5-Br Me 2,5-di-CF_Three-4-OMe
Et 3-Ac-5-Me Me 2-CF_Three-4,5-di-OMe
Et 3-Ac-5-CF_Three          Me 3-CF_Three-4,5-di-F
Et 3-Ac-5-OMe Me 3-CF_Three-4-F-5-Cl
Et 3-Ac-5-OCF_Three         Me 3-CF_Three-4-F-5-Br
Et 3- (U-3b) -5-F Me 3-CF_Three-4-F-5-Me
Et 3- (U-3b) -5-Cl Me 3,5-di-CF_Three-4-F
Et 3- (U-3b) -5-Br Me 3-CF_Three-4-F-5-OMe
Et 3- (U-3b) -5-Me Me 3-CF_Three-4-Cl-5-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Et 3- (U-3b) -5-CF_Three      Me 3-CF_Three-4,5-di-Cl
Et 3- (U-3b) -5-OMe Me 3-CF_Three-4-Cl-5-Br
Et 3- (U-3b) -5-OCF_Three     Me 3-CF_Three-4-Cl-5-Me
Et 3-CF₂H-5-F Me 3,5-di-CF_Three-4-Cl
Et 3-CF₂H-5-Cl Me 3-CF_Three-4-Cl-5-OMe
Et 3-CF₂H-5-Br Me 3-CF_Three-4-Br-5-F
Et 3-CF₂H-5-Me Me 3-CF_Three-4-Br-5-Cl
Et 3-CF₂H-5-CF_Three        Me 3-CF_Three-4,5-di-Br
Et 3-CF₂H-5-OMe Me 3-CF_Three-4-Br-5-Me
Et 3-CF₂H-5-OCF_Three       Me 3,5-di-CF_Three-4-Br
Et 3-CN-5-F Me 3-CF_Three-4-Br-5-OMe
Et 3-CN-5-Cl Me 3-CF_Three-4-Me-5-F
Et 3-CN-5-Br Me 3-CF_Three-4-Me-5-Cl
Et 3-CN-5-Me Me 3-CF_Three-4-Me-5-Br
Et 3-CN-5-CF_Three          Me 3-CF_Three-4,5-di-Me
Et 3-CN-5-OMe Me 3,5-di-CF_Three-4-Me
Et 3-CN-5-OCF_Three         Me 3-CF_Three-4-Me-5-OMe
Et 3-Et-5-F Me 3,4-di-CF_Three-5-F
Et 3-Et-5-Cl Me 3,4-di-CF_Three-5-Cl
Et 3-Et-5-Br Me 3,4-di-CF_Three-5-Br
Et 3-Et-5-Me Me 3,4-di-CF_Three-5-Me
Et 3-Et-5-CF_Three          Me 3,4,5-tri-CF_Three
Et 3-Et-5-OMe Me 3,4-di-CF_Three-5-OMe
Et 3-Et-5-OCF_Three         Me 3-CF_Three-4-OMe-5-F
Et 3-OCF₂H-5-F Me 3-CF_Three-4-OMe-5-Cl
Et 3-OCF₂H-5-Cl Me 3-CF_Three-4-OMe-5-Br
Et 3-OCF₂H-5-Br Me 3-CF_Three-4-OMe-5-Me
Et 3-OCF₂H-5-Me Me 3,5-di-CF_Three-4-OMe
Et 3-OCF₂H-5-CF_Three       Me 3-CF_Three-4,5-di-OMe
Et 3-OCF₂H-5-OMe Me 2-OMe-3,4-di-F
Et 3-OCF₂H-5-OCF_Three      Me 2-OMe-3-F-4-Cl
Et 3-OEt-5-F Me 2-OMe-3-F-4-Br
Et 3-OEt-5-Cl Me 2-OMe-3-F-4-Me
Et 3-OEt-5-Br Me 2-OMe-3-F-4-CF_Three
Et 3-OEt-5-Me Me 2,4-di-OMe-3-F
Et 3-OEt-5-CF_Three         Me 2-OMe-3-Cl-4-F
Et 3-OEt-5-OMe Me 2-OMe-3,4-di-Cl
Et 3-OEt-5-OCF_Three        Me 2-OMe-3-Cl-4-Br
Et 3-C (O) CF_Three-5-F Me 2-OMe-3-Cl-4-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
Et 3-C (O) CF_Three-5-Cl Me 2-OMe-3-Cl-4-CF_Three
Et 3-C (O) CF_Three-5-Br Me 2,4-di-OMe-3-Cl
Et 3-C (O) CF_Three-5-Me Me 2-OMe-3-Br-4-F
Et 3-C (O) CF_Three-5-CF_Three     Me 2-OMe-3-Br-4-Cl
Et 3-C (O) CF_Three-5-OMe Me 2-OMe-3,4-di-Br
Et 3-C (O) CF_Three-5-OCF_Three    Me 2-OMe-3-Br-4-Me
iPr 2-F-3-Ac Me 2-OMe-3-Br-4-CF_Three
iPr 2-F-3- (U-3b) Me 2,4-di-OMe-3-Br
iPr 2-F-3-CF₂H Me 2-OMe-3-Me-4-F
iPr 2-F-3-CN Me 2-OMe-3-Me-4-Cl
iPr 2-F-3-Et Me 2-OMe-3-Me-4-Br
iPr 2-F-3-OCF₂H Me 2-OMe-3,4-di-Me
iPr 2-F-3-OEt Me 2-OMe-3-Me-4-CF_Three
iPr 2-F-3-C (O) CF_Three       Me 2,4-di-OMe-3-Me
iPr 2-Cl-3-Ac Me 2-OMe-3-CF_Three-4-F
iPr 2-Cl-3- (U-3b) Me 2-OMe-3-CF_Three-4-Cl
iPr 2-Cl-3-CF₂H Me 2-OMe-3-CF_Three-4-Br
iPr 2-Cl-3-CN Me 2-OMe-3-CF_Three-4-Me
iPr 2-Cl-3-Et Me 2-OMe-3,4-di-CF_Three
iPr 2-Cl-3-OCF₂H Me 2,4-di-OMe-3-CF_Three
iPr 2-Cl-3-OEt Me 2,3-di-OMe-4-F
iPr 2-Cl-3-C (O) CF_Three      Me 2,3-di-OMe-4-Cl
iPr 2-Br-3-Ac Me 2,3-di-OMe-4-Br
iPr 2-Br-3- (U-3b) Me 2,3-di-OMe-4-Me
iPr 2-Br-3-CF₂H Me 2,3-di-OMe-4-CF_Three
iPr 2-Br-3-CN Me 2,3,4-tri-OMe
iPr 2-Br-3-Et Me 2-OMe-3,5-di-F
iPr 2-Br-3-OCF₂H Me 2-OMe-3-F-5-Cl
iPr 2-Br-3-OEt Me 2-OMe-3-F-5-Br
iPr 2-Br-3-C (O) CF_Three      Me 2-OMe-3-F-5-Me
iPr 2-Me-3-Ac Me 2-OMe-3-F-5-CF_Three
iPr 2-Me-3- (U-3b) Me 2,5-di-OMe-3-F
iPr 2-Me-3-CF₂H Me 2-OMe-3-Cl-5-F
iPr 2-Me-3-CN Me 2-OMe-3,5-di-Cl
iPr 2-Me-3-Et Me 2-OMe-3-Cl-5-Br
iPr 2-Me-3-OCF₂H Me 2-OMe-3-Cl-5-Me
iPr 2-Me-3-OEt Me 2-OMe-3-Cl-5-CF_Three
iPr 2-Me-3-C (O) CF_Three      Me 2,5-di-OMe-3-Cl
iPr 2-CF_Three-3-Ac Me 2-OMe-3-Br-5-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
iPr 2-CF_Three-3- (U-3b) Me 2-OMe-3-Br-5-Cl
iPr 2-CF_Three-3-CF₂H Me 2-OMe-3,5-di-Br
iPr 2-CF_Three-3-CN Me 2-OMe-3-Br-5-Me
iPr 2-CF_Three-3-Et Me 2-OMe-3-Br-5-CF_Three
iPr 2-CF_Three-3-OCF₂H Me 2,5-di-OMe-3-Br
iPr 2-CF_Three-3-OEt Me 2-OMe-3-Me-5-F
iPr 2-CF_Three-3-C (O) CF_Three     Me 2-OMe-3-Me-5-Cl
iPr 2-OMe-3-Ac Me 2-OMe-3-Me-5-Br
iPr 2-OMe-3- (U-3b) Me 2-OMe-3,5-di-Me
iPr 2-OMe-3-CF₂H Me 2-OMe-3-Me-5-CF_Three
iPr 2-OMe-3-CN Me 2,5-di-OMe-3-Me
iPr 2-OMe-3-Et Me 2-OMe-3-CF_Three-5-F
iPr 2-OMe-3-OCF₂H Me 2-OMe-3-CF_Three-5-Cl
iPr 2-OMe-3-OEt Me 2-OMe-3-CF_Three-5-Br
iPr 2-OMe-3-C (O) CF_Three     Me 2-OMe-3-CF_Three-5-Me
iPr 2-OCF_Three-3-Ac Me 2-OMe-3,5-di-CF_Three
iPr 2-OCF_Three-3- (U-3b) Me 2,5-di-OMe-3-CF_Three
iPr 2-OCF_Three-3-CF₂H Me 2,3-di-OMe-5-F
iPr 2-OCF_Three-3-CN Me 2,3-di-OMe-5-Cl
iPr 2-OCF_Three-3-Et Me 2,3-di-OMe-5-Br
iPr 2-OCF_Three-3-OCF₂H Me 2,3-di-OMe-5-Me
iPr 2-OCF_Three-3-OEt Me 2,3-di-OMe-5-CF_Three
iPr 2-OCF_Three-3-C (O) CF_Three    Me 2,3,5-tri-OMe
iPr 2-F-4-Ac Me 2-OMe-4,5-di-F
iPr 2-F-4- (U-3b) Me 2-OMe-4-F-5-Cl
iPr 2-F-4-CF₂H Me 2-OMe-4-F-5-Br
iPr 2-F-4-CN Me 2-OMe-4-F-5-Me
iPr 2-F-4-Et Me 2-OMe-4-F-5-CF_Three
iPr 2-F-4-OCF₂H Me 2,5-di-OMe-4-F
iPr 2-F-4-OEt Me 2-OMe-4-Cl-5-F
iPr 2-F-4-C (O) CF_Three       Me 2-OMe-4,5-di-Cl
iPr 2-Cl-4-Ac Me 2-OMe-4-Cl-5-Br
iPr 2-Cl-4- (U-3b) Me 2-OMe-4-Cl-5-Me
iPr 2-Cl-4-CF₂H Me 2-OMe-4-Cl-5-CF_Three
iPr 2-Cl-4-CN Me 2,5-di-OMe-4-Cl
iPr 2-Cl-4-Et Me 2-OMe-4-Br-5-F
iPr 2-Cl-4-OCF₂H Me 2-OMe-4-Br-5-Cl
iPr 2-Cl-4-OEt Me 2-OMe-4,5-di-Br
iPr 2-Cl-4-C (O) CF_Three      Me 2-OMe-4-Br-5-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
iPr 2-Br-4-Ac Me 2-OMe-4-Br-5-CF_Three
iPr 2-Br-4- (U-3b) Me 2,5-di-OMe-4-Br
iPr 2-Br-4-CF₂H Me 2-OMe-4-Me-5-F
iPr 2-Br-4-CN Me 2-OMe-4-Me-5-Cl
iPr 2-Br-4-Et Me 2-OMe-4-Me-5-Br
iPr 2-Br-4-OCF₂H Me 2-OMe-4,5-di-Me
iPr 2-Br-4-OEt Me 2-OMe-4-Me-5-CF_Three
iPr 2-Br-4-C (O) CF_Three      Me 2,5-di-OMe-4-Me
iPr 2-Me-4-Ac Me 2-OMe-4-CF_Three-5-F
iPr 2-Me-4- (U-3b) Me 2-OMe-4-CF_Three-5-Cl
iPr 2-Me-4-CF₂H Me 2-OMe-4-CF_Three-5-Br
iPr 2-Me-4-CN Me 2-OMe-4-CF_Three-5-Me
iPr 2-Me-4-Et Me 2-OMe-4,5-di-CF_Three
iPr 2-Me-4-OCF₂H Me 2,5-di-OMe-4-CF_Three
iPr 2-Me-4-OEt Me 2,4-di-OMe-5-F
iPr 2-Me-4-C (O) CF_Three      Me 2,4-di-OMe-5-Cl
iPr 2-CF_Three-4-Ac Me 2,4-di-OMe-5-Br
iPr 2-CF_Three-4- (U-3b) Me 2,4-di-OMe-5-Me
iPr 2-CF_Three-4-CF₂H Me 2,4-di-OMe-5-CF_Three
iPr 2-CF_Three-4-CN Me 2,4,5-tri-OMe
iPr 2-CF_Three-4-Et Me 3-OMe-4,5-di-F
iPr 2-CF_Three-4-OCF₂H Me 3-OMe-4-F-5-Cl
iPr 2-CF_Three-4-OEt Me 3-OMe-4-F-5-Br
iPr 2-CF_Three-4-C (O) CF_Three     Me 3-OMe-4-F-5-Me
iPr 2-OMe-4-Ac Me 3-OMe-4-F-5-CF_Three
iPr 2-OMe-4- (U-3b) Me 3,5-di-OMe-4-F
iPr 2-OMe-4-CF₂H Me 3-OMe-4-Cl-5-F
iPr 2-OMe-4-CN Me 3-OMe-4,5-di-Cl
iPr 2-OMe-4-Et Me 3-OMe-4-Cl-5-Br
iPr 2-OMe-4-OCF₂H Me 3-OMe-4-Cl-5-Me
iPr 2-OMe-4-OEt Me 3-OMe-4-Cl-5-CF_Three
iPr 2-OMe-4-C (O) CF_Three     Me 3,5-di-OMe-4-Cl
iPr 2-OCF_Three-4-Ac Me 3-OMe-4-Br-5-F
iPr 2-OCF_Three-4- (U-3b) Me 3-OMe-4-Br-5-Cl
iPr 2-OCF_Three-4-CF₂H Me 3-OMe-4,5-di-Br
iPr 2-OCF_Three-4-CN Me 3-OMe-4-Br-5-Me
iPr 2-OCF_Three-4-Et Me 3-OMe-4-Br-5-CF_Three
iPr 2-OCF_Three-4-OCF₂H Me 3,5-di-OMe-4-Br
iPr 2-OCF_Three-4-OEt Me 3-OMe-4-Me-5-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
iPr 2-OCF_Three-4-C (O) CF_Three    Me 3-OMe-4-Me-5-Cl
iPr 2-F-5-Ac Me 3-OMe-4-Me-5-Br
iPr 2-F-5- (U-3b) Me 3-OMe-4,5-di-Me
iPr 2-F-5-CF₂H Me 3-OMe-4-Me-5-CF_Three
iPr 2-F-5-CN Me 3,5-di-OMe-4-Me
iPr 2-F-5-Et Me 3-OMe-4-CF_Three-5-F
iPr 2-F-5-OCF₂H Me 3-OMe-4-CF_Three-5-Cl
iPr 2-F-5-OEt Me 3-OMe-4-CF_Three-5-Br
iPr 2-F-5-C (O) CF_Three       Me 3-OMe-4-CF_Three-5-Me
iPr 2-Cl-5-Ac Me 3-OMe-4,5-di-CF_Three
iPr 2-Cl-5- (U-3b) Me 3,5-di-OMe-4-CF_Three
iPr 2-Cl-5-CF₂H Me 3,4-di-OMe-5-F
iPr 2-Cl-5-CN Me 3,4-di-OMe-5-Cl
iPr 2-Cl-5-Et Me 3,4-di-OMe-5-Br
iPr 2-Cl-5-OCF₂H Me 3,4-di-OMe-5-Me
iPr 2-Cl-5-OEt Me 3,4-di-OMe-5-CF_Three
iPr 2-Cl-5-C (O) CF_Three      Me 3,4,5-tri-OMe
iPr 2-Br-5-Ac Et 2,3,4-tri-F
iPr 2-Br-5- (U-3b) Et 2,3-di-F-4-Cl
iPr 2-Br-5-CF₂H Et 2,3-di-F-4-Br
iPr 2-Br-5-CN Et 2,3-di-F-4-Me
iPr 2-Br-5-Et Et 2,3-di-F-4-CF_Three
iPr 2-Br-5-OCF₂H Et 2,3-di-F-4-OMe
iPr 2-Br-5-OEt Et 2,4-di-F-3-Cl
iPr 2-Br-5-C (O) CF_Three      Et 2-F-3,4-di-Cl
iPr 2-Me-5-Ac Et 2-F-3-Cl-4-Br
iPr 2-Me-5- (U-3b) Et 2-F-3-Cl-4-Me
iPr 2-Me-5-CF₂H Et 2-F-3-Cl-4-CF_Three
iPr 2-Me-5-CN Et 2-F-3-Cl-4-OMe
iPr 2-Me-5-Et Et 2,4-di-F-3-Br
iPr 2-Me-5-OCF₂H Et 2-F-3-Br-4-Cl
iPr 2-Me-5-OEt Et 2-F-3,4-di-Br
iPr 2-Me-5-C (O) CF_Three      Et 2-F-3-Br-4-Me
iPr 2-CF_Three-5-Ac Et 2-F-3-Br-4-CF_Three
iPr 2-CF_Three-5- (U-3b) Et 2-F-3-Br-4-OMe
iPr 2-CF_Three-5-CF₂H Et 2,4-di-F-3-Me
iPr 2-CF_Three-5-CN Et 2-F-3-Me-4-Cl
iPr 2-CF_Three-5-Et Et 2-F-3-Me-4-Br
iPr 2-CF_Three-5-OCF₂H Et 2-F-3,4-di-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
iPr 2-CF_Three-5-OEt Et 2-F-3-Me-4-CF_Three
iPr 2-CF_Three-5-C (O) CF_Three     Et 2-F-3-Me-4-OMe
iPr 2-OMe-5-Ac Et 2,4-di-F-3-CF_Three
iPr 2-OMe-5- (U-3b) Et 2-F-3-CF_Three-4-Cl
iPr 2-OMe-5-CF₂H Et 2-F-3-CF_Three-4-Br
iPr 2-OMe-5-CN Et 2-F-3-CF_Three-4-Me
iPr 2-OMe-5-Et Et 2-F-3,4-di-CF_Three
iPr 2-OMe-5-OCF₂H Et 2-F-3-CF_Three-4-OMe
iPr 2-OMe-5-OEt Et 2,4-di-F-3-OMe
iPr 2-OMe-5-C (O) CF_Three     Et 2-F-3-OMe-4-Cl
iPr 2-OCF_Three-5-Ac Et 2-F-3-OMe-4-Br
iPr 2-OCF_Three-5- (U-3b) Et 2-F-3-OMe-4-Me
iPr 2-OCF_Three-5-CF₂H Et 2-F-3-OMe-4-CF_Three
iPr 2-OCF_Three-5-CN Et 2-F-3,4-di-OMe
iPr 2-OCF_Three-5-Et Et 2,3,5-tri-F
iPr 2-OCF_Three-5-OCF₂H Et 2,3-di-F-5-Cl
iPr 2-OCF_Three-5-OEt Et 2,3-di-F-5-Br
iPr 2-OCF_Three-5-C (O) CF_Three    Et 2,3-di-F-5-Me
iPr 3-F-4-Ac Et 2,3-di-F-5-CF_Three
iPr 3-F-4- (U-3b) Et 2,3-di-F-5-OMe
iPr 3-F-4-CF₂H Et 2,5-di-F-3-Cl
iPr 3-F-4-CN Et 2-F-3,5-di-Cl
iPr 3-F-4-Et Et 2-F-3-Cl-5-Br
iPr 3-F-4-OCF₂H Et 2-F-3-Cl-5-Me
iPr 3-F-4-OEt Et 2-F-3-Cl-5-CF_Three
iPr 3-F-4-C (O) CF_Three       Et 2-F-3-Cl-5-OMe
iPr 3-Cl-4-Ac Et 2,5-di-F-3-Br
iPr 3-Cl-4- (U-3b) Et 2-F-3-Br-5-Cl
iPr 3-Cl-4-CF₂H Et 2-F-3,5-di-Br
iPr 3-Cl-4-CN Et 2-F-3-Br-5-Me
iPr 3-Cl-4-Et Et 2-F-3-Br-5-CF_Three
iPr 3-Cl-4-OCF₂H Et 2-F-3-Br-5-OMe
iPr 3-Cl-4-OEt Et 2,5-di-F-3-Me
iPr 3-Cl-4-C (O) CF_Three      Et 2-F-3-Me-5-Cl
iPr 3-Br-4-Ac Et 2-F-3-Me-5-Br
iPr 3-Br-4- (U-3b) Et 2-F-3,5-di-Me
iPr 3-Br-4-CF₂H Et 2-F-3-Me-5-CF_Three
iPr 3-Br-4-CN Et 2-F-3-Me-5-OMe
iPr 3-Br-4-Et Et 2,5-di-F-3-CF_Three
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
iPr 3-Br-4-OCF₂H Et 2-F-3-CF_Three-5-Cl
iPr 3-Br-4-OEt Et 2-F-3-CF_Three-5-Br
iPr 3-Br-4-C (O) CF_Three      Et 2-F-3-CF_Three-5-Me
iPr 3-Me-4-Ac Et 2-F-3,5-di-CF_Three
iPr 3-Me-4- (U-3b) Et 2-F-3-CF_Three-5-OMe
iPr 3-Me-4-CF₂H Et 2,5-di-F-3-OMe
iPr 3-Me-4-CN Et 2-F-3-OMe-5-Cl
iPr 3-Me-4-Et Et 2-F-3-OMe-5-Br
iPr 3-Me-4-OCF₂H Et 2-F-3-OMe-5-Me
iPr 3-Me-4-OEt Et 2-F-3-OMe-5-CF_Three
iPr 3-Me-4-C (O) CF_Three      Et 2-F-3,5-di-OMe
iPr 3-CF_Three-4-Ac Et 2,4,5-tri-F
iPr 3-CF_Three-4- (U-3b) Et 2,4-di-F-5-Cl
iPr 3-CF_Three-4-CF₂H Et 2,4-di-F-5-Br
iPr 3-CF_Three-4-CN Et 2,4-di-F-5-Me
iPr 3-CF_Three-4-Et Et 2,4-di-F-5-CF_Three
iPr 3-CF_Three-4-OCF₂H Et 2,4-di-F-5-OMe
iPr 3-CF_Three-4-OEt Et 2,5-di-F-4-Cl
iPr 3-CF_Three-4-C (O) CF_Three     Et 2-F-4,5-di-Cl
iPr 3-OMe-4-Ac Et 2-F-4-Cl-5-Br
iPr 3-OMe-4- (U-3b) Et 2-F-4-Cl-5-Me
iPr 3-OMe-4-CF₂H Et 2-F-4-Cl-5-CF_Three
iPr 3-OMe-4-CN Et 2-F-4-Cl-5-OMe
iPr 3-OMe-4-Et Et 2,5-di-F-4-Br
iPr 3-OMe-4-OCF₂H Et 2-F-4-Br-5-Cl
iPr 3-OMe-4-OEt Et 2-F-4,5-di-Br
iPr 3-OMe-4-C (O) CF_Three     Et 2-F-4-Br-5-Me
iPr 3-OCF_Three-4-Ac Et 2-F-4-Br-5-CF_Three
iPr 3-OCF_Three-4- (U-3b) Et 2-F-4-Br-5-OMe
iPr 3-OCF_Three-4-CF₂H Et 2,5-di-F-4-Me
iPr 3-OCF_Three-4-CN Et 2-F-4-Me-5-Cl
iPr 3-OCF_Three-4-Et Et 2-F-4-Me-5-Br
iPr 3-OCF_Three-4-OCF₂H Et 2-F-4,5-di-Me
iPr 3-OCF_Three-4-OEt Et 2-F-4-Me-5-CF_Three
iPr 3-OCF_Three-4-C (O) CF_Three    Et 2-F-4-Me-5-OMe
iPr 3-F-5-Ac Et 2,5-di-F-4-CF_Three
iPr 3-F-5- (U-3b) Et 2-F-4-CF_Three-5-Cl
iPr 3-F-5-CF₂H Et 2-F-4-CF_Three-5-Br
iPr 3-F-5-CN Et 2-F-4-CF_Three-5-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
iPr 3-F-5-Et Et 2-F-4,5-di-CF_Three
iPr 3-F-5-OCF₂H Et 2-F-4-CF_Three-5-OMe
iPr 3-F-5-OEt Et 2,5-di-F-4-OMe
iPr 3-F-5-C (O) CF_Three       Et 2-F-4-OMe-5-Cl
iPr 3-Cl-5-Ac Et 2-F-4-OMe-5-Br
iPr 3-Cl-5- (U-3b) Et 2-F-4-OMe-5-Me
iPr 3-Cl-5-CF₂H Et 2-F-4-OMe-5-CF_Three
iPr 3-Cl-5-CN Et 2-F-4,5-di-OMe
iPr 3-Cl-5-Et Et 3,4,5-tri-F
iPr 3-Cl-5-OCF₂H Et 3,4-di-F-5-Cl
iPr 3-Cl-5-OEt Et 3,4-di-F-5-Br
iPr 3-Cl-5-C (O) CF_Three      Et 3,4-di-F-5-Me
iPr 3-Br-5-Ac Et 3,4-di-F-5-CF_Three
iPr 3-Br-5- (U-3b) Et 3,4-di-F-5-OMe
iPr 3-Br-5-CF₂H Et 3,5-di-F-4-Cl
iPr 3-Br-5-CN Et 3-F-4,5-di-Cl
iPr 3-Br-5-Et Et 3-F-4-Cl-5-Br
iPr 3-Br-5-OCF₂H Et 3-F-4-Cl-5-Me
iPr 3-Br-5-OEt Et 3-F-4-Cl-5-CF_Three
iPr 3-Br-5-C (O) CF_Three      Et 3-F-4-Cl-5-OMe
iPr 3-Me-5-Ac Et 3,5-di-F-4-Br
iPr 3-Me-5- (U-3b) Et 3-F-4-Br-5-Cl
iPr 3-Me-5-CF₂H Et 3-F-4,5-di-Br
iPr 3-Me-5-CN Et 3-F-4-Br-5-Me
iPr 3-Me-5-Et Et 3-F-4-Br-5-CF_Three
iPr 3-Me-5-OCF₂H Et 3-F-4-Br-5-OMe
iPr 3-Me-5-OEt Et 3,5-di-F-4-Me
iPr 3-Me-5-C (O) CF_Three      Et 3-F-4-Me-5-Cl
iPr 3-CF_Three-5-Ac Et 3-F-4-Me-5-Br
iPr 3-CF_Three-5- (U-3b) Et 3-F-4,5-di-Me
iPr 3-CF_Three-5-CF₂H Et 3-F-4-Me-5-CF_Three
iPr 3-CF_Three-5-CN Et 3-F-4-Me-5-OMe
iPr 3-CF_Three-5-Et Et 3,5-di-F-4-CF_Three
iPr 3-CF_Three-5-OCF₂H Et 3-F-4-CF_Three-5-Cl
iPr 3-CF_Three-5-OEt Et 3-F-4-CF_Three-5-Br
iPr 3-CF_Three-5-C (O) CF_Three     Et 3-F-4-CF_Three-5-Me
iPr 3-OMe-5-Ac Et 3-F-4,5-di-CF_Three
iPr 3-OMe-5- (U-3b) Et 3-F-4-CF_Three-5-OMe
iPr 3-OMe-5-CF₂H Et 3,5-di-F-4-OMe
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
iPr 3-OMe-5-CN Et 3-F-4-OMe-5-Cl
iPr 3-OMe-5-Et Et 3-F-4-OMe-5-Br
iPr 3-OMe-5-OCF₂H Et 3-F-4-OMe-5-Me
iPr 3-OMe-5-OEt Et 3-F-4-OMe-5-CF_Three
iPr 3-OMe-5-C (O) CF_Three     Et 3-F-4,5-di-OMe
iPr 3-OCF_Three-5-Ac Et 2-Cl-3,4-di-F
iPr 3-OCF_Three-5- (U-3b) Et 2,4-di-Cl-3-F
iPr 3-OCF_Three-5-CF₂H Et 2-Cl-3-F-4-Br
iPr 3-OCF_Three-5-CN Et 2-Cl-3-F-4-Me
iPr 3-OCF_Three-5-Et Et 2-Cl-3-F-4-CF_Three
iPr 3-OCF_Three-5-OCF₂H Et 2-Cl-3-F-4-OMe
iPr 3-OCF_Three-5-OEt Et 2,3-di-Cl-4-F
iPr 3-OCF_Three-5-C (O) CF_Three    Et 2,3,4-tri-Cl
iPr 2-Ac-3-F Et 2,3-di-Cl-4-Br
iPr 2-Ac-3-Cl Et 2,3-di-Cl-4-Me
iPr 2-Ac-3-Br Et 2,3-di-Cl-4-CF_Three
iPr 2-Ac-3-Me Et 2,3-di-Cl-4-OMe
iPr 2-Ac-3-CF_Three          Et 2-Cl-3-Br-4-F
iPr 2-Ac-3-OMe Et 2,4-di-Cl-3-Br
iPr 2-Ac-3-OCF_Three         Et 2-Cl-3,4-di-Br
iPr 2- (U-3b) -3-F Et 2-Cl-3-Br-4-Me
iPr 2- (U-3b) -3-Cl Et 2-Cl-3-Br-4-CF_Three
iPr 2- (U-3b) -3-Br Et 2-Cl-3-Br-4-OMe
iPr 2- (U-3b) -3-Me Et 2-Cl-3-Me-4-F
iPr 2- (U-3b) -3-CF_Three      Et 2,4-di-Cl-3-Me
iPr 2- (U-3b) -3-OMe Et 2-Cl-3-Me-4-Br
iPr 2- (U-3b) -3-OCF_Three     Et 2-Cl-3,4-di-Me
iPr 2-CF₂H-3-F Et 2-Cl-3-Me-4-CF_Three
iPr 2-CF₂H-3-Cl Et 2-Cl-3-Me-4-OMe
iPr 2-CF₂H-3-Br Et 2-Cl-3-CF_Three-4-F
iPr 2-CF₂H-3-Me Et 2,4-di-Cl-3-CF_Three
iPr 2-CF₂H-3-CF_Three        Et 2-Cl-3-CF_Three-4-Br
iPr 2-CF₂H-3-OMe Et 2-Cl-3-CF_Three-4-Me
iPr 2-CF₂H-3-OCF_Three       Et 2-Cl-3,4-di-CF_Three
iPr 2-CN-3-F Et 2-Cl-3-CF_Three-4-OMe
iPr 2-CN-3-Cl Et 2-Cl-3-OMe-4-F
iPr 2-CN-3-Br Et 2,4-di-Cl-3-OMe
iPr 2-CN-3-Me Et 2-Cl-3-OMe-4-Br
iPr 2-CN-3-CF_Three          Et 2-Cl-3-OMe-4-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
iPr 2-CN-3-OMe Et 2-Cl-3-OMe-4-CF_Three
iPr 2-CN-3-OCF_Three         Et 2-Cl-3,4-di-OMe
iPr 2-Et-3-F Et 2-Cl-3,5-di-F
iPr 2-Et-3-Cl Et 2,5-di-Cl-3-F
iPr 2-Et-3-Br Et 2-Cl-3-F-5-Br
iPr 2-Et-3-Me Et 2-Cl-3-F-5-Me
iPr 2-Et-3-CF_Three          Et 2-Cl-3-F-5-CF_Three
iPr 2-Et-3-OMe Et 2-Cl-3-F-5-OMe
iPr 2-Et-3-OCF_Three         Et 2,3-di-Cl-5-F
iPr 2-OCF₂H-3-F Et 2,3,5-tri-Cl
iPr 2-OCF₂H-3-Cl Et 2,3-di-Cl-5-Br
iPr 2-OCF₂H-3-Br Et 2,3-di-Cl-5-Me
iPr 2-OCF₂H-3-Me Et 2,3-di-Cl-5-CF_Three
iPr 2-OCF₂H-3-CF_Three       Et 2,3-di-Cl-5-OMe
iPr 2-OCF₂H-3-OMe Et 2-Cl-3-Br-5-F
iPr 2-OCF₂H-3-OCF_Three      Et 2,5-di-Cl-3-Br
iPr 2-OEt-3-F Et 2-Cl-3,5-di-Br
iPr 2-OEt-3-Cl Et 2-Cl-3-Br-5-Me
iPr 2-OEt-3-Br Et 2-Cl-3-Br-5-CF_Three
iPr 2-OEt-3-Me Et 2-Cl-3-Br-5-OMe
iPr 2-OEt-3-CF_Three         Et 2-Cl-3-Me-5-F
iPr 2-OEt-3-OMe Et 2,5-di-Cl-3-Me
iPr 2-OEt-3-OCF_Three        Et 2-Cl-3-Me-5-Br
iPr 2-C (O) CF_Three-3-F Et 2-Cl-3,5-di-Me
iPr 2-C (O) CF_Three-3-Cl Et 2-Cl-3-Me-5-CF_Three
iPr 2-C (O) CF_Three-3-Br Et 2-Cl-3-Me-5-OMe
iPr 2-C (O) CF_Three-3-Me Et 2-Cl-3-CF_Three-5-F
iPr 2-C (O) CF_Three-3-CF_Three     Et 2,5-di-Cl-3-CF_Three
iPr 2-C (O) CF_Three-3-OMe Et 2-Cl-3-CF_Three-5-Br
iPr 2-C (O) CF_Three-3-OCF_Three    Et 2-Cl-3-CF_Three-5-Me
iPr 2-Ac-4-F Et 2-Cl-3,5-di-CF_Three
iPr 2-Ac-4-Cl Et 2-Cl-3-CF_Three-5-OMe
iPr 2-Ac-4-Br Et 2-Cl-3-OMe-5-F
iPr 2-Ac-4-Me Et 2,5-di-Cl-3-OMe
iPr 2-Ac-4-CF_Three          Et 2-Cl-3-OMe-5-Br
iPr 2-Ac-4-OMe Et 2-Cl-3-OMe-5-Me
iPr 2-Ac-4-OCF_Three         Et 2-Cl-3-OMe-5-CF_Three
iPr 2- (U-3b) -4-F Et 2-Cl-3,5-di-OMe
iPr 2- (U-3b) -4-Cl Et 2-Cl-4,5-di-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
iPr 2- (U-3b) -4-Br Et 2,5-di-Cl-4-F
iPr 2- (U-3b) -4-Me Et 2-Cl-4-F-5-Br
iPr 2- (U-3b) -4-CF_Three      Et 2-Cl-4-F-5-Me
iPr 2- (U-3b) -4-OMe Et 2-Cl-4-F-5-CF_Three
iPr 2- (U-3b) -4-OCF_Three     Et 2-Cl-4-F-5-OMe
iPr 2-CF₂H-4-F Et 2,4-di-Cl-5-F
iPr 2-CF₂H-4-Cl Et 2,4,5-tri-Cl
iPr 2-CF₂H-4-Br Et 2,4-di-Cl-5-Br
iPr 2-CF₂H-4-Me Et 2,4-di-Cl-5-Me
iPr 2-CF₂H-4-CF_Three        Et 2,4-di-Cl-5-CF_Three
iPr 2-CF₂H-4-OMe Et 2,4-di-Cl-5-OMe
iPr 2-CF₂H-4-OCF_Three       Et 2-Cl-4-Br-5-F
iPr 2-CN-4-F Et 2,5-di-Cl-4-Br
iPr 2-CN-4-Cl Et 2-Cl-4,5-di-Br
iPr 2-CN-4-Br Et 2-Cl-4-Br-5-Me
iPr 2-CN-4-Me Et 2-Cl-4-Br-5-CF_Three
iPr 2-CN-4-CF_Three          Et 2-Cl-4-Br-5-OMe
iPr 2-CN-4-OMe Et 2-Cl-4-Me-5-F
iPr 2-CN-4-OCF_Three         Et 2,5-di-Cl-4-Me
iPr 2-Et-4-F Et 2-Cl-4-Me-5-Br
iPr 2-Et-4-Cl Et 2-Cl-4,5-di-Me
iPr 2-Et-4-Br Et 2-Cl-4-Me-5-CF_Three
iPr 2-Et-4-Me Et 2-Cl-4-Me-5-OMe
iPr 2-Et-4-CF_Three          Et 2-Cl-4-CF_Three-5-F
iPr 2-Et-4-OMe Et 2,5-di-Cl-4-CF_Three
iPr 2-Et-4-OCF_Three         Et 2-Cl-4-CF_Three-5-Br
iPr 2-OCF₂H-4-F Et 2-Cl-4-CF_Three-5-Me
iPr 2-OCF₂H-4-Cl Et 2-Cl-4,5-di-CF_Three
iPr 2-OCF₂H-4-Br Et 2-Cl-4-CF_Three-5-OMe
iPr 2-OCF₂H-4-Me Et 2-Cl-4-OMe-5-F
iPr 2-OCF₂H-4-CF_Three       Et 2,5-di-Cl-4-OMe
iPr 2-OCF₂H-4-OMe Et 2-Cl-4-OMe-5-Br
iPr 2-OCF₂H-4-OCF_Three      Et 2-Cl-4-OMe-5-Me
iPr 2-OEt-4-F Et 2-Cl-4-OMe-5-CF_Three
iPr 2-OEt-4-Cl Et 2-Cl-4,5-di-OMe
iPr 2-OEt-4-Br Et 3-Cl-4,5-di-F
iPr 2-OEt-4-Me Et 3,5-di-Cl-4-F
iPr 2-OEt-4-CF_Three         Et 3-Cl-4-F-5-Br
iPr 2-OEt-4-OMe Et 3-Cl-4-F-5-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
iPr 2-OEt-4-OCF_Three        Et 3-Cl-4-F-5-CF_Three
iPr 2-C (O) CF_Three-4-F Et 3-Cl-4-F-5-OMe
iPr 2-C (O) CF_Three-4-Cl Et 3,4-di-Cl-5-F
iPr 2-C (O) CF_Three-4-Br Et 3,4,5-tri-Cl
iPr 2-C (O) CF_Three-4-Me Et 3,4-di-Cl-5-Br
iPr 2-C (O) CF_Three-4-CF_Three     Et 3,4-di-Cl-5-Me
iPr 2-C (O) CF_Three-4-OMe Et 3,4-di-Cl-5-CF_Three
iPr 2-C (O) CF_Three-4-OCF_Three    Et 3,4-di-Cl-5-OMe
iPr 2-Ac-5-F Et 3-Cl-4-Br-5-F
iPr 2-Ac-5-Cl Et 3,5-di-Cl-4-Br
iPr 2-Ac-5-Br Et 3-Cl-4,5-di-Br
iPr 2-Ac-5-Me Et 3-Cl-4-Br-5-Me
iPr 2-Ac-5-CF_Three          Et 3-Cl-4-Br-5-CF_Three
iPr 2-Ac-5-OMe Et 3-Cl-4-Br-5-OMe
iPr 2-Ac-5-OCF_Three         Et 3-Cl-4-Me-5-F
iPr 2- (U-3b) -5-F Et 3,5-di-Cl-4-Me
iPr 2- (U-3b) -5-Cl Et 3-Cl-4-Me-5-Br
iPr 2- (U-3b) -5-Br Et 3-Cl-4,5-di-Me
iPr 2- (U-3b) -5-Me Et 3-Cl-4-Me-5-CF_Three
iPr 2- (U-3b) -5-CF_Three      Et 3-Cl-4-Me-5-OMe
iPr 2- (U-3b) -5-OMe Et 3-Cl-4-CF_Three-5-F
iPr 2- (U-3b) -5-OCF_Three     Et 3,5-di-Cl-4-CF_Three
iPr 2-CF₂H-5-F Et 3-Cl-4-CF_Three-5-Br
iPr 2-CF₂H-5-Cl Et 3-Cl-4-CF_Three-5-Me
iPr 2-CF₂H-5-Br Et 3-Cl-4,5-di-CF_Three
iPr 2-CF₂H-5-Me Et 3-Cl-4-CF_Three-5-OMe
iPr 2-CF₂H-5-CF_Three        Et 3-Cl-4-OMe-5-F
iPr 2-CF₂H-5-OMe Et 3,5-di-Cl-4-OMe
iPr 2-CF₂H-5-OCF_Three       Et 3-Cl-4-OMe-5-Br
iPr 2-CN-5-F Et 3-Cl-4-OMe-5-Me
iPr 2-CN-5-Cl Et 3-Cl-4-OMe-5-CF_Three
iPr 2-CN-5-Br Et 3-Cl-4,5-di-OMe
iPr 2-CN-5-Me Et 2-Br-3,4-di-F
iPr 2-CN-5-CF_Three          Et 2-Br-3-F-4-Cl
iPr 2-CN-5-OMe Et 2,4-di-Br-3-F
iPr 2-CN-5-OCF_Three         Et 2-Br-3-F-4-Me
iPr 2-Et-5-F Et 2-Br-3-F-4-CF_Three
iPr 2-Et-5-Cl Et 2-Br-3-F-4-OMe
iPr 2-Et-5-Br Et 2-Br-3-Cl-4-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
iPr 2-Et-5-Me Et 2-Br-3,4-di-Cl
iPr 2-Et-5-CF_Three          Et 2,4-di-Br-3-Cl
iPr 2-Et-5-OMe Et 2-Br-3-Cl-4-Me
iPr 2-Et-5-OCF_Three         Et 2-Br-3-Cl-4-CF_Three
iPr 2-OCF₂H-5-F Et 2-Br-3-Cl-4-OMe
iPr 2-OCF₂H-5-Cl Et 2,3-di-Br-4-F
iPr 2-OCF₂H-5-Br Et 2,3-di-Br-4-Cl
iPr 2-OCF₂H-5-Me Et 2,3,4-tri-Br
iPr 2-OCF₂H-5-CF_Three       Et 2,3-di-Br-4-Me
iPr 2-OCF₂H-5-OMe Et 2,3-di-Br-4-CF_Three
iPr 2-OCF₂H-5-OCF_Three      Et 2,3-di-Br-4-OMe
iPr 2-OEt-5-F Et 2-Br-3-Me-4-F
iPr 2-OEt-5-Cl Et 2-Br-3-Me-4-Cl
iPr 2-OEt-5-Br Et 2,4-di-Br-3-Me
iPr 2-OEt-5-Me Et 2-Br-3,4-di-Me
iPr 2-OEt-5-CF_Three         Et 2-Br-3-Me-4-CF_Three
iPr 2-OEt-5-OMe Et 2-Br-3-Me-4-OMe
iPr 2-OEt-5-OCF_Three        Et 2-Br-3-CF_Three-4-F
iPr 2-C (O) CF_Three-5-F Et 2-Br-3-CF_Three-4-Cl
iPr 2-C (O) CF_Three-5-Cl Et 2,4-di-Br-3-CF_Three
iPr 2-C (O) CF_Three-5-Br Et 2-Br-3-CF_Three-4-Me
iPr 2-C (O) CF_Three-5-Me Et 2-Br-3,4-di-CF_Three
iPr 2-C (O) CF_Three-5-CF_Three     Et 2-Br-3-CF_Three-4-OMe
iPr 2-C (O) CF_Three-5-OMe Et 2-Br-3-OMe-4-F
iPr 2-C (O) CF_Three-5-OCF_Three    Et 2-Br-3-OMe-4-Cl
iPr 3-Ac-4-F Et 2,4-di-Br-3-OMe
iPr 3-Ac-4-Cl Et 2-Br-3-OMe-4-Me
iPr 3-Ac-4-Br Et 2-Br-3-OMe-4-CF_Three
iPr 3-Ac-4-Me Et 2-Br-3,4-di-OMe
iPr 3-Ac-4-CF_Three          Et 2-Br-3,5-di-F
iPr 3-Ac-4-OMe Et 2-Br-3-F-5-Cl
iPr 3-Ac-4-OCF_Three         Et 2,5-di-Br-3-F
iPr 3- (U-3b) -4-F Et 2-Br-3-F-5-Me
iPr 3- (U-3b) -4-Cl Et 2-Br-3-F-5-CF_Three
iPr 3- (U-3b) -4-Br Et 2-Br-3-F-5-OMe
iPr 3- (U-3b) -4-Me Et 2-Br-3-Cl-5-F
iPr 3- (U-3b) -4-CF_Three      Et 2-Br-3,5-di-Cl
iPr 3- (U-3b) -4-OMe Et 2,5-di-Br-3-Cl
iPr 3- (U-3b) -4-OCF_Three     Et 2-Br-3-Cl-5-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
iPr 3-CF₂H-4-F Et 2-Br-3-Cl-5-CF_Three
iPr 3-CF₂H-4-Cl Et 2-Br-3-Cl-5-OMe
iPr 3-CF₂H-4-Br Et 2,3-di-Br-5-F
iPr 3-CF₂H-4-Me Et 2,3-di-Br-5-Cl
iPr 3-CF₂H-4-CF_Three        Et 2,3,5-tri-Br
iPr 3-CF₂H-4-OMe Et 2,3-di-Br-5-Me
iPr 3-CF₂H-4-OCF_Three       Et 2,3-di-Br-5-CF_Three
iPr 3-CN-4-F Et 2,3-di-Br-5-OMe
iPr 3-CN-4-Cl Et 2-Br-3-Me-5-F
iPr 3-CN-4-Br Et 2-Br-3-Me-5-Cl
iPr 3-CN-4-Me Et 2,5-di-Br-3-Me
iPr 3-CN-4-CF_Three          Et 2-Br-3,5-di-Me
iPr 3-CN-4-OMe Et 2-Br-3-Me-5-CF_Three
iPr 3-CN-4-OCF_Three         Et 2-Br-3-Me-5-OMe
iPr 3-Et-4-F Et 2-Br-3-CF_Three-5-F
iPr 3-Et-4-Cl Et 2-Br-3-CF_Three-5-Cl
iPr 3-Et-4-Br Et 2,5-di-Br-3-CF_Three
iPr 3-Et-4-Me Et 2-Br-3-CF_Three-5-Me
iPr 3-Et-4-CF_Three          Et 2-Br-3,5-di-CF_Three
iPr 3-Et-4-OMe Et 2-Br-3-CF_Three-5-OMe
iPr 3-Et-4-OCF_Three         Et 2-Br-3-OMe-5-F
iPr 3-OCF₂H-4-F Et 2-Br-3-OMe-5-Cl
iPr 3-OCF₂H-4-Cl Et 2,5-di-Br-3-OMe
iPr 3-OCF₂H-4-Br Et 2-Br-3-OMe-5-Me
iPr 3-OCF₂H-4-Me Et 2-Br-3-OMe-5-CF_Three
iPr 3-OCF₂H-4-CF_Three       Et 2-Br-3,5-di-OMe
iPr 3-OCF₂H-4-OMe Et 2-Br-4,5-di-F
iPr 3-OCF₂H-4-OCF_Three      Et 2-Br-4-F-5-Cl
iPr 3-OEt-4-F Et 2,5-di-Br-4-F
iPr 3-OEt-4-Cl Et 2-Br-4-F-5-Me
iPr 3-OEt-4-Br Et 2-Br-4-F-5-CF_Three
iPr 3-OEt-4-Me Et 2-Br-4-F-5-OMe
iPr 3-OEt-4-CF_Three         Et 2-Br-4-Cl-5-F
iPr 3-OEt-4-OMe Et 2-Br-4,5-di-Cl
iPr 3-OEt-4-OCF_Three        Et 2,5-di-Br-4-Cl
iPr 3-C (O) CF_Three-4-F Et 2-Br-4-Cl-5-Me
iPr 3-C (O) CF_Three-4-Cl Et 2-Br-4-Cl-5-CF_Three
iPr 3-C (O) CF_Three-4-Br Et 2-Br-4-Cl-5-OMe
iPr 3-C (O) CF_Three-4-Me Et 2,4-di-Br-5-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
iPr 3-C (O) CF_Three-4-CF_Three     Et 2,4-di-Br-5-Cl
iPr 3-C (O) CF_Three-4-OMe Et 2,4,5-tri-Br
iPr 3-C (O) CF_Three-4-OCF_Three    Et 2,4-di-Br-5-Me
iPr 3-Ac-5-F Et 2,4-di-Br-5-CF_Three
iPr 3-Ac-5-Cl Et 2,4-di-Br-5-OMe
iPr 3-Ac-5-Br Et 2-Br-4-Me-5-F
iPr 3-Ac-5-Me Et 2-Br-4-Me-5-Cl
iPr 3-Ac-5-CF_Three          Et 2,5-di-Br-4-Me
iPr 3-Ac-5-OMe Et 2-Br-4,5-di-Me
iPr 3-Ac-5-OCF_Three         Et 2-Br-4-Me-5-CF_Three
iPr 3- (U-3b) -5-F Et 2-Br-4-Me-5-OMe
iPr 3- (U-3b) -5-Cl Et 2-Br-4-CF_Three-5-F
iPr 3- (U-3b) -5-Br Et 2-Br-4-CF_Three-5-Cl
iPr 3- (U-3b) -5-Me Et 2,5-di-Br-4-CF_Three
iPr 3- (U-3b) -5-CF_Three      Et 2-Br-4-CF_Three-5-Me
iPr 3- (U-3b) -5-OMe Et 2-Br-4,5-di-CF_Three
iPr 3- (U-3b) -5-OCF_Three     Et 2-Br-4-CF_Three-5-OMe
iPr 3-CF₂H-5-F Et 2-Br-4-OMe-5-F
iPr 3-CF₂H-5-Cl Et 2-Br-4-OMe-5-Cl
iPr 3-CF₂H-5-Br Et 2,5-di-Br-4-OMe
iPr 3-CF₂H-5-Me Et 2-Br-4-OMe-5-Me
iPr 3-CF₂H-5-CF_Three        Et 2-Br-4-OMe-5-CF_Three
iPr 3-CF₂H-5-OMe Et 2-Br-4,5-di-OMe
iPr 3-CF₂H-5-OCF_Three       Et 3-Br-4,5-di-F
iPr 3-CN-5-F Et 3-Br-4-F-5-Cl
iPr 3-CN-5-Cl Et 3,5-di-Br-4-F
iPr 3-CN-5-Br Et 3-Br-4-F-5-Me
iPr 3-CN-5-Me Et 3-Br-4-F-5-CF_Three
iPr 3-CN-5-CF_Three          Et 3-Br-4-F-5-OMe
iPr 3-CN-5-OMe Et 3-Br-4-Cl-5-F
iPr 3-CN-5-OCF_Three         Et 3-Br-4,5-di-Cl
iPr 3-Et-5-F Et 3,5-di-Br-4-Cl
iPr 3-Et-5-Cl Et 3-Br-4-Cl-5-Me
iPr 3-Et-5-Br Et 3-Br-4-Cl-5-CF_Three
iPr 3-Et-5-Me Et 3-Br-4-Cl-5-OMe
iPr 3-Et-5-CF_Three          Et 3,4-di-Br-5-F
iPr 3-Et-5-OMe Et 3,4-di-Br-5-Cl
iPr 3-Et-5-OCF_Three         Et 3,4,5-tri-Br
iPr 3-OCF₂H-5-F Et 3,4-di-Br-5-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
iPr 3-OCF₂H-5-Cl Et 3,4-di-Br-5-CF_Three
iPr 3-OCF₂H-5-Br Et 3,4-di-Br-5-OMe
iPr 3-OCF₂H-5-Me Et 3-Br-4-Me-5-F
iPr 3-OCF₂H-5-CF_Three       Et 3-Br-4-Me-5-Cl
iPr 3-OCF₂H-5-OMe Et 3,5-di-Br-4-Me
iPr 3-OCF₂H-5-OCF_Three      Et 3-Br-4,5-di-Me
iPr 3-OEt-5-F Et 3-Br-4-Me-5-CF_Three
iPr 3-OEt-5-Cl Et 3-Br-4-Me-5-OMe
iPr 3-OEt-5-Br Et 3-Br-4-CF_Three-5-F
iPr 3-OEt-5-Me Et 3-Br-4-CF_Three-5-Cl
iPr 3-OEt-5-CF_Three         Et 3,5-di-Br-4-CF_Three
iPr 3-OEt-5-OMe Et 3-Br-4-CF_Three-5-Me
iPr 3-OEt-5-OCF_Three        Et 3-Br-4,5-di-CF_Three
iPr 3-C (O) CF_Three-5-F Et 3-Br-4-CF_Three-5-OMe
iPr 3-C (O) CF_Three-5-Cl Et 3-Br-4-OMe-5-F
iPr 3-C (O) CF_Three-5-Br Et 3-Br-4-OMe-5-Cl
iPr 3-C (O) CF_Three-5-Me Et 3,5-di-Br-4-OMe
iPr 3-C (O) CF_Three-5-CF_Three     Et 3-Br-4-OMe-5-Me
iPr 3-C (O) CF_Three-5-OMe Et 3-Br-4-OMe-5-CF_Three
iPr 3-C (O) CF_Three-5-OCF_Three    Et 3-Br-4,5-di-OMe
U-4a 2-F-3-Ac Et 2-Me-3,4-di-F
U-4a 2-F-3- (U-3b) Et 2-Me-3-F-4-Cl
U-4a 2-F-3-CF₂H Et 2-Me-3-F-4-Br
U-4a 2-F-3-CN Et 2,4-di-Me-3-F
U-4a 2-F-3-Et Et 2-Me-3-F-4-CF_Three
U-4a 2-F-3-OCF₂H Et 2-Me-3-F-4-OMe
U-4a 2-F-3-OEt Et 2-Me-3-Cl-4-F
U-4a 2-F-3-C (O) CF_Three       Et 2-Me-3,4-di-Cl
U-4a 2-Cl-3-Ac Et 2-Me-3-Cl-4-Br
U-4a 2-Cl-3- (U-3b) Et 2,4-di-Me-3-Cl
U-4a 2-Cl-3-CF₂H Et 2-Me-3-Cl-4-CF_Three
U-4a 2-Cl-3-CN Et 2-Me-3-Cl-4-OMe
U-4a 2-Cl-3-Et Et 2-Me-3-Br-4-F
U-4a 2-Cl-3-OCF₂H Et 2-Me-3-Br-4-Cl
U-4a 2-Cl-3-OEt Et 2-Me-3,4-di-Br
U-4a 2-Cl-3-C (O) CF_Three      Et 2,4-di-Me-3-Br
U-4a 2-Br-3-Ac Et 2-Me-3-Br-4-CF_Three
U-4a 2-Br-3- (U-3b) Et 2-Me-3-Br-4-OMe
U-4a 2-Br-3-CF₂H Et 2,3-di-Me-4-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
U-4a 2-Br-3-CN Et 2,3-di-Me-4-Cl
U-4a 2-Br-3-Et Et 2,3-di-Me-4-Br
U-4a 2-Br-3-OCF₂H Et 2,3,4-tri-Me
U-4a 2-Br-3-OEt Et 2,3-di-Me-4-CF_Three
U-4a 2-Br-3-C (O) CF_Three      Et 2,3-di-Me-4-OMe
U-4a 2-Me-3-Ac Et 2-Me-3-CF_Three-4-F
U-4a 2-Me-3- (U-3b) Et 2-Me-3-CF_Three-4-Cl
U-4a 2-Me-3-CF₂H Et 2-Me-3-CF_Three-4-Br
U-4a 2-Me-3-CN Et 2,4-di-Me-3-CF_Three
U-4a 2-Me-3-Et Et 2-Me-3,4-di-CF_Three
U-4a 2-Me-3-OCF₂H Et 2-Me-3-CF_Three-4-OMe
U-4a 2-Me-3-OEt Et 2-Me-3-OMe-4-F
U-4a 2-Me-3-C (O) CF_Three      Et 2-Me-3-OMe-4-Cl
U-4a 2-CF_Three-3-Ac Et 2-Me-3-OMe-4-Br
U-4a 2-CF_Three-3- (U-3b) Et 2,4-di-Me-3-OMe
U-4a 2-CF_Three-3-CF₂H Et 2-Me-3-OMe-4-CF_Three
U-4a 2-CF_Three-3-CN Et 2-Me-3,4-di-OMe
U-4a 2-CF_Three-3-Et Et 2-Me-3,5-di-F
U-4a 2-CF_Three-3-OCF₂H Et 2-Me-3-F-5-Cl
U-4a 2-CF_Three-3-OEt Et 2-Me-3-F-5-Br
U-4a 2-CF_Three-3-C (O) CF_Three     Et 2,5-di-Me-3-F
U-4a 2-OMe-3-Ac Et 2-Me-3-F-5-CF_Three
U-4a 2-OMe-3- (U-3b) Et 2-Me-3-F-5-OMe
U-4a 2-OMe-3-CF₂H Et 2-Me-3-Cl-5-F
U-4a 2-OMe-3-CN Et 2-Me-3,5-di-Cl
U-4a 2-OMe-3-Et Et 2-Me-3-Cl-5-Br
U-4a 2-OMe-3-OCF₂H Et 2,5-di-Me-3-Cl
U-4a 2-OMe-3-OEt Et 2-Me-3-Cl-5-CF_Three
U-4a 2-OMe-3-C (O) CF_Three     Et 2-Me-3-Cl-5-OMe
U-4a 2-OCF_Three-3-Ac Et 2-Me-3-Br-5-F
U-4a 2-OCF_Three-3- (U-3b) Et 2-Me-3-Br-5-Cl
U-4a 2-OCF_Three-3-CF₂H Et 2-Me-3,5-di-Br
U-4a 2-OCF_Three-3-CN Et 2,5-di-Me-3-Br
U-4a 2-OCF_Three-3-Et Et 2-Me-3-Br-5-CF_Three
U-4a 2-OCF_Three-3-OCF₂H Et 2-Me-3-Br-5-OMe
U-4a 2-OCF_Three-3-OEt Et 2,3-di-Me-5-F
U-4a 2-OCF_Three-3-C (O) CF_Three    Et 2,3-di-Me-5-Cl
U-4a 2-F-4-Ac Et 2,3-di-Me-5-Br
U-4a 2-F-4- (U-3b) Et 2,3,5-tri-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
U-4a 2-F-4-CF₂H Et 2,3-di-Me-5-CF_Three
U-4a 2-F-4-CN Et 2,3-di-Me-5-OMe
U-4a 2-F-4-Et Et 2-Me-3-CF_Three-5-F
U-4a 2-F-4-OCF₂H Et 2-Me-3-CF_Three-5-Cl
U-4a 2-F-4-OEt Et 2-Me-3-CF_Three-5-Br
U-4a 2-F-4-C (O) CF_Three       Et 2,5-di-Me-3-CF_Three
U-4a 2-Cl-4-Ac Et 2-Me-3,5-di-CF_Three
U-4a 2-Cl-4- (U-3b) Et 2-Me-3-CF_Three-5-OMe
U-4a 2-Cl-4-CF₂H Et 2-Me-3-OMe-5-F
U-4a 2-Cl-4-CN Et 2-Me-3-OMe-5-Cl
U-4a 2-Cl-4-Et Et 2-Me-3-OMe-5-Br
U-4a 2-Cl-4-OCF₂H Et 2,5-di-Me-3-OMe
U-4a 2-Cl-4-OEt Et 2-Me-3-OMe-5-CF_Three
U-4a 2-Cl-4-C (O) CF_Three      Et 2-Me-3,5-di-OMe
U-4a 2-Br-4-Ac Et 2-Me-4,5-di-F
U-4a 2-Br-4- (U-3b) Et 2-Me-4-F-5-Cl
U-4a 2-Br-4-CF₂H Et 2-Me-4-F-5-Br
U-4a 2-Br-4-CN Et 2,5-di-Me-4-F
U-4a 2-Br-4-Et Et 2-Me-4-F-5-CF_Three
U-4a 2-Br-4-OCF₂H Et 2-Me-4-F-5-OMe
U-4a 2-Br-4-OEt Et 2-Me-4-Cl-5-F
U-4a 2-Br-4-C (O) CF_Three      Et 2-Me-4,5-di-Cl
U-4a 2-Me-4-Ac Et 2-Me-4-Cl-5-Br
U-4a 2-Me-4- (U-3b) Et 2,5-di-Me-4-Cl
U-4a 2-Me-4-CF₂H Et 2-Me-4-Cl-5-CF_Three
U-4a 2-Me-4-CN Et 2-Me-4-Cl-5-OMe
U-4a 2-Me-4-Et Et 2-Me-4-Br-5-F
U-4a 2-Me-4-OCF₂H Et 2-Me-4-Br-5-Cl
U-4a 2-Me-4-OEt Et 2-Me-4,5-di-Br
U-4a 2-Me-4-C (O) CF_Three      Et 2,5-di-Me-4-Br
U-4a 2-CF_Three-4-Ac Et 2-Me-4-Br-5-CF_Three
U-4a 2-CF_Three-4- (U-3b) Et 2-Me-4-Br-5-OMe
U-4a 2-CF_Three-4-CF₂H Et 2,4-di-Me-5-F
U-4a 2-CF_Three-4-CN Et 2,4-di-Me-5-Cl
U-4a 2-CF_Three-4-Et Et 2,4-di-Me-5-Br
U-4a 2-CF_Three-4-OCF₂H Et 2,4,5-tri-Me
U-4a 2-CF_Three-4-OEt Et 2,4-di-Me-5-CF_Three
U-4a 2-CF_Three-4-C (O) CF_Three     Et 2,4-di-Me-5-OMe
U-4a 2-OMe-4-Ac Et 2-Me-4-CF_Three-5-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
U-4a 2-OMe-4- (U-3b) Et 2-Me-4-CF_Three-5-Cl
U-4a 2-OMe-4-CF₂H Et 2-Me-4-CF_Three-5-Br
U-4a 2-OMe-4-CN Et 2,5-di-Me-4-CF_Three
U-4a 2-OMe-4-Et Et 2-Me-4,5-di-CF_Three
U-4a 2-OMe-4-OCF₂H Et 2-Me-4-CF_Three-5-OMe
U-4a 2-OMe-4-OEt Et 2-Me-4-OMe-5-F
U-4a 2-OMe-4-C (O) CF_Three     Et 2-Me-4-OMe-5-Cl
U-4a 2-OCF_Three-4-Ac Et 2-Me-4-OMe-5-Br
U-4a 2-OCF_Three-4- (U-3b) Et 2,5-di-Me-4-OMe
U-4a 2-OCF_Three-4-CF₂H Et 2-Me-4-OMe-5-CF_Three
U-4a 2-OCF_Three-4-CN Et 2-Me-4,5-di-OMe
U-4a 2-OCF_Three-4-Et Et 3-Me-4,5-di-F
U-4a 2-OCF_Three-4-OCF₂H Et 3-Me-4-F-5-Cl
U-4a 2-OCF_Three-4-OEt Et 3-Me-4-F-5-Br
U-4a 2-OCF_Three-4-C (O) CF_Three    Et 3,5-di-Me-4-F
U-4a 2-F-5-Ac Et 3-Me-4-F-5-CF_Three
U-4a 2-F-5- (U-3b) Et 3-Me-4-F-5-OMe
U-4a 2-F-5-CF₂H Et 3-Me-4-Cl-5-F
U-4a 2-F-5-CN Et 3-Me-4,5-di-Cl
U-4a 2-F-5-Et Et 3-Me-4-Cl-5-Br
U-4a 2-F-5-OCF₂H Et 3,5-di-Me-4-Cl
U-4a 2-F-5-OEt Et 3-Me-4-Cl-5-CF_Three
U-4a 2-F-5-C (O) CF_Three       Et 3-Me-4-Cl-5-OMe
U-4a 2-Cl-5-Ac Et 3-Me-4-Br-5-F
U-4a 2-Cl-5- (U-3b) Et 3-Me-4-Br-5-Cl
U-4a 2-Cl-5-CF₂H Et 3-Me-4,5-di-Br
U-4a 2-Cl-5-CN Et 3,5-di-Me-4-Br
U-4a 2-Cl-5-Et Et 3-Me-4-Br-5-CF_Three
U-4a 2-Cl-5-OCF₂H Et 3-Me-4-Br-5-OMe
U-4a 2-Cl-5-OEt Et 3,4-di-Me-5-F
U-4a 2-Cl-5-C (O) CF_Three      Et 3,4-di-Me-5-Cl
U-4a 2-Br-5-Ac Et 3,4-di-Me-5-Br
U-4a 2-Br-5- (U-3b) Et 3,4,5-tri-Me
U-4a 2-Br-5-CF₂H Et 3,4-di-Me-5-CF_Three
U-4a 2-Br-5-CN Et 3,4-di-Me-5-OMe
U-4a 2-Br-5-Et Et 3-Me-4-CF_Three-5-F
U-4a 2-Br-5-OCF₂H Et 3-Me-4-CF_Three-5-Cl
U-4a 2-Br-5-OEt Et 3-Me-4-CF_Three-5-Br
U-4a 2-Br-5-C (O) CF_Three      Et 3,5-di-Me-4-CF_Three
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
U-4a 2-Me-5-Ac Et 3-Me-4,5-di-CF_Three
U-4a 2-Me-5- (U-3b) Et 3-Me-4-CF_Three-5-OMe
U-4a 2-Me-5-CF₂H Et 3-Me-4-OMe-5-F
U-4a 2-Me-5-CN Et 3-Me-4-OMe-5-Cl
U-4a 2-Me-5-Et Et 3-Me-4-OMe-5-Br
U-4a 2-Me-5-OCF₂H Et 3,5-di-Me-4-OMe
U-4a 2-Me-5-OEt Et 3-Me-4-OMe-5-CF_Three
U-4a 2-Me-5-C (O) CF_Three      Et 3-Me-4,5-di-OMe
U-4a 2-CF_Three-5-Ac Et 2-CF_Three-3,4-di-F
U-4a 2-CF_Three-5- (U-3b) Et 2-CF_Three-3-F-4-Cl
U-4a 2-CF_Three-5-CF₂H Et 2-CF_Three-3-F-4-Br
U-4a 2-CF_Three-5-CN Et 2-CF_Three-3-F-4-Me
U-4a 2-CF_Three-5-Et Et 2,4-di-CF_Three-3-F
U-4a 2-CF_Three-5-OCF₂H Et 2-CF_Three-3-F-4-OMe
U-4a 2-CF_Three-5-OEt Et 2-CF_Three-3-Cl-4-F
U-4a 2-CF_Three-5-C (O) CF_Three     Et 2-CF_Three-3,4-di-Cl
U-4a 2-OMe-5-Ac Et 2-CF_Three-3-Cl-4-Br
U-4a 2-OMe-5- (U-3b) Et 2-CF_Three-3-Cl-4-Me
U-4a 2-OMe-5-CF₂H Et 2,4-di-CF_Three-3-Cl
U-4a 2-OMe-5-CN Et 2-CF_Three-3-Cl-4-OMe
U-4a 2-OMe-5-Et Et 2-CF_Three-3-Br-4-F
U-4a 2-OMe-5-OCF₂H Et 2-CF_Three-3-Br-4-Cl
U-4a 2-OMe-5-OEt Et 2-CF_Three-3,4-di-Br
U-4a 2-OMe-5-C (O) CF_Three     Et 2-CF_Three-3-Br-4-Me
U-4a 2-OCF_Three-5-Ac Et 2,4-di-CF_Three-3-Br
U-4a 2-OCF_Three-5- (U-3b) Et 2-CF_Three-3-Br-4-OMe
U-4a 2-OCF_Three-5-CF₂H Et 2-CF_Three-3-Me-4-F
U-4a 2-OCF_Three-5-CN Et 2-CF_Three-3-Me-4-Cl
U-4a 2-OCF_Three-5-Et Et 2-CF_Three-3-Me-4-Br
U-4a 2-OCF_Three-5-OCF₂H Et 2-CF_Three-3,4-di-Me
U-4a 2-OCF_Three-5-OEt Et 2,4-di-CF_Three-3-Me
U-4a 2-OCF_Three-5-C (O) CF_Three    Et 2-CF_Three-3-Me-4-OMe
U-4a 3-F-4-Ac Et 2,3-di-CF_Three-4-F
U-4a 3-F-4- (U-3b) Et 2,3-di-CF_Three-4-Cl
U-4a 3-F-4-CF₂H Et 2,3-di-CF_Three-4-Br
U-4a 3-F-4-CN Et 2,3-di-CF_Three-4-Me
U-4a 3-F-4-Et Et 2,3,4-tri-CF_Three
U-4a 3-F-4-OCF₂H Et 2,3-di-CF_Three-4-OMe
U-4a 3-F-4-OEt Et 2-CF_Three-3-OMe-4-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
U-4a 3-F-4-C (O) CF_Three       Et 2-CF_Three-3-OMe-4-Cl
U-4a 3-Cl-4-Ac Et 2-CF_Three-3-OMe-4-Br
U-4a 3-Cl-4- (U-3b) Et 2-CF_Three-3-OMe-4-Me
U-4a 3-Cl-4-CF₂H Et 2,4-di-CF_Three-3-OMe
U-4a 3-Cl-4-CN Et 2-CF_Three-3,4-di-OMe
U-4a 3-Cl-4-Et Et 2-CF_Three-3,5-di-F
U-4a 3-Cl-4-OCF₂H Et 2-CF_Three-3-F-5-Cl
U-4a 3-Cl-4-OEt Et 2-CF_Three-3-F-5-Br
U-4a 3-Cl-4-C (O) CF_Three      Et 2-CF_Three-3-F-5-Me
U-4a 3-Br-4-Ac Et 2,5-di-CF_Three-3-F
U-4a 3-Br-4- (U-3b) Et 2-CF_Three-3-F-5-OMe
U-4a 3-Br-4-CF₂H Et 2-CF_Three-3-Cl-5-F
U-4a 3-Br-4-CN Et 2-CF_Three-3,5-di-Cl
U-4a 3-Br-4-Et Et 2-CF_Three-3-Cl-5-Br
U-4a 3-Br-4-OCF₂H Et 2-CF_Three-3-Cl-5-Me
U-4a 3-Br-4-OEt Et 2,5-di-CF_Three-3-Cl
U-4a 3-Br-4-C (O) CF_Three      Et 2-CF_Three-3-Cl-5-OMe
U-4a 3-Me-4-Ac Et 2-CF_Three-3-Br-5-F
U-4a 3-Me-4- (U-3b) Et 2-CF_Three-3-Br-5-Cl
U-4a 3-Me-4-CF₂H Et 2-CF_Three-3,5-di-Br
U-4a 3-Me-4-CN Et 2-CF_Three-3-Br-5-Me
U-4a 3-Me-4-Et Et 2,5-di-CF_Three-3-Br
U-4a 3-Me-4-OCF₂H Et 2-CF_Three-3-Br-5-OMe
U-4a 3-Me-4-OEt Et 2-CF_Three-3-Me-5-F
U-4a 3-Me-4-C (O) CF_Three      Et 2-CF_Three-3-Me-5-Cl
U-4a 3-CF_Three-4-Ac Et 2-CF_Three-3-Me-5-Br
U-4a 3-CF_Three-4- (U-3b) Et 2-CF_Three-3,5-di-Me
U-4a 3-CF_Three-4-CF₂H Et 2,5-di-CF_Three-3-Me
U-4a 3-CF_Three-4-CN Et 2-CF_Three-3-Me-5-OMe
U-4a 3-CF_Three-4-Et Et 2,3-di-CF_Three-5-F
U-4a 3-CF_Three-4-OCF₂H Et 2,3-di-CF_Three-5-Cl
U-4a 3-CF_Three-4-OEt Et 2,3-di-CF_Three-5-Br
U-4a 3-CF_Three-4-C (O) CF_Three     Et 2,3-di-CF_Three-5-Me
U-4a 3-OMe-4-Ac Et 2,3,5-tri-CF_Three
U-4a 3-OMe-4- (U-3b) Et 2,3-di-CF_Three-5-OMe
U-4a 3-OMe-4-CF₂H Et 2-CF_Three-3-OMe-5-F
U-4a 3-OMe-4-CN Et 2-CF_Three-3-OMe-5-Cl
U-4a 3-OMe-4-Et Et 2-CF_Three-3-OMe-5-Br
U-4a 3-OMe-4-OCF₂H Et 2-CF_Three-3-OMe-5-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
U-4a 3-OMe-4-OEt Et 2,5-di-CF_Three-3-OMe
U-4a 3-OMe-4-C (O) CF_Three     Et 2-CF_Three-3,5-di-OMe
U-4a 3-OCF_Three-4-Ac Et 2-CF_Three-4,5-di-F
U-4a 3-OCF_Three-4- (U-3b) Et 2-CF_Three-4-F-5-Cl
U-4a 3-OCF_Three-4-CF₂H Et 2-CF_Three-4-F-5-Br
U-4a 3-OCF_Three-4-CN Et 2-CF_Three-4-F-5-Me
U-4a 3-OCF_Three-4-Et Et 2,5-di-CF_Three-4-F
U-4a 3-OCF_Three-4-OCF₂H Et 2-CF_Three-4-F-5-OMe
U-4a 3-OCF_Three-4-OEt Et 2-CF_Three-4-Cl-5-F
U-4a 3-OCF_Three-4-C (O) CF_Three    Et 2-CF_Three-4,5-di-Cl
U-4a 3-F-5-Ac Et 2-CF_Three-4-Cl-5-Br
U-4a 3-F-5- (U-3b) Et 2-CF_Three-4-Cl-5-Me
U-4a 3-F-5-CF₂H Et 2,5-di-CF_Three-4-Cl
U-4a 3-F-5-CN Et 2-CF_Three-4-Cl-5-OMe
U-4a 3-F-5-Et Et 2-CF_Three-4-Br-5-F
U-4a 3-F-5-OCF₂H Et 2-CF_Three-4-Br-5-Cl
U-4a 3-F-5-OEt Et 2-CF_Three-4,5-di-Br
U-4a 3-F-5-C (O) CF_Three       Et 2-CF_Three-4-Br-5-Me
U-4a 3-Cl-5-Ac Et 2,5-di-CF_Three-4-Br
U-4a 3-Cl-5- (U-3b) Et 2-CF_Three-4-Br-5-OMe
U-4a 3-Cl-5-CF₂H Et 2-CF_Three-4-Me-5-F
U-4a 3-Cl-5-CN Et 2-CF_Three-4-Me-5-Cl
U-4a 3-Cl-5-Et Et 2-CF_Three-4-Me-5-Br
U-4a 3-Cl-5-OCF₂H Et 2-CF_Three-4,5-di-Me
U-4a 3-Cl-5-OEt Et 2,5-di-CF_Three-4-Me
U-4a 3-Cl-5-C (O) CF_Three      Et 2-CF_Three-4-Me-5-OMe
U-4a 3-Br-5-Ac Et 2,4-di-CF_Three-5-F
U-4a 3-Br-5- (U-3b) Et 2,4-di-CF_Three-5-Cl
U-4a 3-Br-5-CF₂H Et 2,4-di-CF_Three-5-Br
U-4a 3-Br-5-CN Et 2,4-di-CF_Three-5-Me
U-4a 3-Br-5-Et Et 2,4,5-tri-CF_Three
U-4a 3-Br-5-OCF₂H Et 2,4-di-CF_Three-5-OMe
U-4a 3-Br-5-OEt Et 2-CF_Three-4-OMe-5-F
U-4a 3-Br-5-C (O) CF_Three      Et 2-CF_Three-4-OMe-5-Cl
U-4a 3-Me-5-Ac Et 2-CF_Three-4-OMe-5-Br
U-4a 3-Me-5- (U-3b) Et 2-CF_Three-4-OMe-5-Me
U-4a 3-Me-5-CF₂H Et 2,5-di-CF_Three-4-OMe
U-4a 3-Me-5-CN Et 2-CF_Three-4,5-di-OMe
U-4a 3-Me-5-Et Et 3-CF_Three-4,5-di-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
U-4a 3-Me-5-OCF₂H Et 3-CF_Three-4-F-5-Cl
U-4a 3-Me-5-OEt Et 3-CF_Three-4-F-5-Br
U-4a 3-Me-5-C (O) CF_Three      Et 3-CF_Three-4-F-5-Me
U-4a 3-CF_Three-5-Ac Et 3,5-di-CF_Three-4-F
U-4a 3-CF_Three-5- (U-3b) Et 3-CF_Three-4-F-5-OMe
U-4a 3-CF_Three-5-CF₂H Et 3-CF_Three-4-Cl-5-F
U-4a 3-CF_Three-5-CN Et 3-CF_Three-4,5-di-Cl
U-4a 3-CF_Three-5-Et Et 3-CF_Three-4-Cl-5-Br
U-4a 3-CF_Three-5-OCF₂H Et 3-CF_Three-4-Cl-5-Me
U-4a 3-CF_Three-5-OEt Et 3,5-di-CF_Three-4-Cl
U-4a 3-CF_Three-5-C (O) CF_Three     Et 3-CF_Three-4-Cl-5-OMe
U-4a 3-OMe-5-Ac Et 3-CF_Three-4-Br-5-F
U-4a 3-OMe-5- (U-3b) Et 3-CF_Three-4-Br-5-Cl
U-4a 3-OMe-5-CF₂H Et 3-CF_Three-4,5-di-Br
U-4a 3-OMe-5-CN Et 3-CF_Three-4-Br-5-Me
U-4a 3-OMe-5-Et Et 3,5-di-CF_Three-4-Br
U-4a 3-OMe-5-OCF₂H Et 3-CF_Three-4-Br-5-OMe
U-4a 3-OMe-5-OEt Et 3-CF_Three-4-Me-5-F
U-4a 3-OMe-5-C (O) CF_Three     Et 3-CF_Three-4-Me-5-Cl
U-4a 3-OCF_Three-5-Ac Et 3-CF_Three-4-Me-5-Br
U-4a 3-OCF_Three-5- (U-3b) Et 3-CF_Three-4,5-di-Me
U-4a 3-OCF_Three-5-CF₂H Et 3,5-di-CF_Three-4-Me
U-4a 3-OCF_Three-5-CN Et 3-CF_Three-4-Me-5-OMe
U-4a 3-OCF_Three-5-Et Et 3,4-di-CF_Three-5-F
U-4a 3-OCF_Three-5-OCF₂H Et 3,4-di-CF_Three-5-Cl
U-4a 3-OCF_Three-5-OEt Et 3,4-di-CF_Three-5-Br
U-4a 3-OCF_Three-5-C (O) CF_Three    Et 3,4-di-CF_Three-5-Me
U-4a 2-Ac-3-F Et 3,4,5-tri-CF_Three
U-4a 2-Ac-3-Cl Et 3,4-di-CF_Three-5-OMe
U-4a 2-Ac-3-Br Et 3-CF_Three-4-OMe-5-F
U-4a 2-Ac-3-Me Et 3-CF_Three-4-OMe-5-Cl
U-4a 2-Ac-3-CF_Three          Et 3-CF_Three-4-OMe-5-Br
U-4a 2-Ac-3-OMe Et 3-CF_Three-4-OMe-5-Me
U-4a 2-Ac-3-OCF_Three         Et 3,5-di-CF_Three-4-OMe
U-4a 2- (U-3b) -3-F Et 3-CF_Three-4,5-di-OMe
U-4a 2- (U-3b) -3-Cl Et 2-OMe-3,4-di-F
U-4a 2- (U-3b) -3-Br Et 2-OMe-3-F-4-Cl
U-4a 2- (U-3b) -3-Me Et 2-OMe-3-F-4-Br
U-4a 2- (U-3b) -3-CF_Three      Et 2-OMe-3-F-4-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
U-4a 2- (U-3b) -3-OMe Et 2-OMe-3-F-4-CF_Three
U-4a 2- (U-3b) -3-OCF_Three     Et 2,4-di-OMe-3-F
U-4a 2-CF₂H-3-F Et 2-OMe-3-Cl-4-F
U-4a 2-CF₂H-3-Cl Et 2-OMe-3,4-di-Cl
U-4a 2-CF₂H-3-Br Et 2-OMe-3-Cl-4-Br
U-4a 2-CF₂H-3-Me Et 2-OMe-3-Cl-4-Me
U-4a 2-CF₂H-3-CF_Three        Et 2-OMe-3-Cl-4-CF_Three
U-4a 2-CF₂H-3-OMe Et 2,4-di-OMe-3-Cl
U-4a 2-CF₂H-3-OCF_Three       Et 2-OMe-3-Br-4-F
U-4a 2-CN-3-F Et 2-OMe-3-Br-4-Cl
U-4a 2-CN-3-Cl Et 2-OMe-3,4-di-Br
U-4a 2-CN-3-Br Et 2-OMe-3-Br-4-Me
U-4a 2-CN-3-Me Et 2-OMe-3-Br-4-CF_Three
U-4a 2-CN-3-CF_Three          Et 2,4-di-OMe-3-Br
U-4a 2-CN-3-OMe Et 2-OMe-3-Me-4-F
U-4a 2-CN-3-OCF_Three         Et 2-OMe-3-Me-4-Cl
U-4a 2-Et-3-F Et 2-OMe-3-Me-4-Br
U-4a 2-Et-3-Cl Et 2-OMe-3,4-di-Me
U-4a 2-Et-3-Br Et 2-OMe-3-Me-4-CF_Three
U-4a 2-Et-3-Me Et 2,4-di-OMe-3-Me
U-4a 2-Et-3-CF_Three          Et 2-OMe-3-CF_Three-4-F
U-4a 2-Et-3-OMe Et 2-OMe-3-CF_Three-4-Cl
U-4a 2-Et-3-OCF_Three         Et 2-OMe-3-CF_Three-4-Br
U-4a 2-OCF₂H-3-F Et 2-OMe-3-CF_Three-4-Me
U-4a 2-OCF₂H-3-Cl Et 2-OMe-3,4-di-CF_Three
U-4a 2-OCF₂H-3-Br Et 2,4-di-OMe-3-CF_Three
U-4a 2-OCF₂H-3-Me Et 2,3-di-OMe-4-F
U-4a 2-OCF₂H-3-CF_Three       Et 2,3-di-OMe-4-Cl
U-4a 2-OCF₂H-3-OMe Et 2,3-di-OMe-4-Br
U-4a 2-OCF₂H-3-OCF_Three      Et 2,3-di-OMe-4-Me
U-4a 2-OEt-3-F Et 2,3-di-OMe-4-CF_Three
U-4a 2-OEt-3-Cl Et 2,3,4-tri-OMe
U-4a 2-OEt-3-Br Et 2-OMe-3,5-di-F
U-4a 2-OEt-3-Me Et 2-OMe-3-F-5-Cl
U-4a 2-OEt-3-CF_Three         Et 2-OMe-3-F-5-Br
U-4a 2-OEt-3-OMe Et 2-OMe-3-F-5-Me
U-4a 2-OEt-3-OCF_Three        Et 2-OMe-3-F-5-CF_Three
U-4a 2-C (O) CF_Three-3-F Et 2,5-di-OMe-3-F
U-4a 2-C (O) CF_Three-3-Cl Et 2-OMe-3-Cl-5-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
U-4a 2-C (O) CF_Three-3-Br Et 2-OMe-3,5-di-Cl
U-4a 2-C (O) CF_Three-3-Me Et 2-OMe-3-Cl-5-Br
U-4a 2-C (O) CF_Three-3-CF_Three     Et 2-OMe-3-Cl-5-Me
U-4a 2-C (O) CF_Three-3-OMe Et 2-OMe-3-Cl-5-CF_Three
U-4a 2-C (O) CF_Three-3-OCF_Three    Et 2,5-di-OMe-3-Cl
U-4a 2-Ac-4-F Et 2-OMe-3-Br-5-F
U-4a 2-Ac-4-Cl Et 2-OMe-3-Br-5-Cl
U-4a 2-Ac-4-Br Et 2-OMe-3,5-di-Br
U-4a 2-Ac-4-Me Et 2-OMe-3-Br-5-Me
U-4a 2-Ac-4-CF_Three          Et 2-OMe-3-Br-5-CF_Three
U-4a 2-Ac-4-OMe Et 2,5-di-OMe-3-Br
U-4a 2-Ac-4-OCF_Three         Et 2-OMe-3-Me-5-F
U-4a 2- (U-3b) -4-F Et 2-OMe-3-Me-5-Cl
U-4a 2- (U-3b) -4-Cl Et 2-OMe-3-Me-5-Br
U-4a 2- (U-3b) -4-Br Et 2-OMe-3,5-di-Me
U-4a 2- (U-3b) -4-Me Et 2-OMe-3-Me-5-CF_Three
U-4a 2- (U-3b) -4-CF_Three      Et 2,5-di-OMe-3-Me
U-4a 2- (U-3b) -4-OMe Et 2-OMe-3-CF_Three-5-F
U-4a 2- (U-3b) -4-OCF_Three     Et 2-OMe-3-CF_Three-5-Cl
U-4a 2-CF₂H-4-F Et 2-OMe-3-CF_Three-5-Br
U-4a 2-CF₂H-4-Cl Et 2-OMe-3-CF_Three-5-Me
U-4a 2-CF₂H-4-Br Et 2-OMe-3,5-di-CF_Three
U-4a 2-CF₂H-4-Me Et 2,5-di-OMe-3-CF_Three
U-4a 2-CF₂H-4-CF_Three        Et 2,3-di-OMe-5-F
U-4a 2-CF₂H-4-OMe Et 2,3-di-OMe-5-Cl
U-4a 2-CF₂H-4-OCF_Three       Et 2,3-di-OMe-5-Br
U-4a 2-CN-4-F Et 2,3-di-OMe-5-Me
U-4a 2-CN-4-Cl Et 2,3-di-OMe-5-CF_Three
U-4a 2-CN-4-Br Et 2,3,5-tri-OMe
U-4a 2-CN-4-Me Et 2-OMe-4,5-di-F
U-4a 2-CN-4-CF_Three          Et 2-OMe-4-F-5-Cl
U-4a 2-CN-4-OMe Et 2-OMe-4-F-5-Br
U-4a 2-CN-4-OCF_Three         Et 2-OMe-4-F-5-Me
U-4a 2-Et-4-F Et 2-OMe-4-F-5-CF_Three
U-4a 2-Et-4-Cl Et 2,5-di-OMe-4-F
U-4a 2-Et-4-Br Et 2-OMe-4-Cl-5-F
U-4a 2-Et-4-Me Et 2-OMe-4,5-di-Cl
U-4a 2-Et-4-CF_Three          Et 2-OMe-4-Cl-5-Br
U-4a 2-Et-4-OMe Et 2-OMe-4-Cl-5-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
U-4a 2-Et-4-OCF_Three         Et 2-OMe-4-Cl-5-CF_Three
U-4a 2-OCF₂H-4-F Et 2,5-di-OMe-4-Cl
U-4a 2-OCF₂H-4-Cl Et 2-OMe-4-Br-5-F
U-4a 2-OCF₂H-4-Br Et 2-OMe-4-Br-5-Cl
U-4a 2-OCF₂H-4-Me Et 2-OMe-4,5-di-Br
U-4a 2-OCF₂H-4-CF_Three       Et 2-OMe-4-Br-5-Me
U-4a 2-OCF₂H-4-OMe Et 2-OMe-4-Br-5-CF_Three
U-4a 2-OCF₂H-4-OCF_Three      Et 2,5-di-OMe-4-Br
U-4a 2-OEt-4-F Et 2-OMe-4-Me-5-F
U-4a 2-OEt-4-Cl Et 2-OMe-4-Me-5-Cl
U-4a 2-OEt-4-Br Et 2-OMe-4-Me-5-Br
U-4a 2-OEt-4-Me Et 2-OMe-4,5-di-Me
U-4a 2-OEt-4-CF_Three         Et 2-OMe-4-Me-5-CF_Three
U-4a 2-OEt-4-OMe Et 2,5-di-OMe-4-Me
U-4a 2-OEt-4-OCF_Three        Et 2-OMe-4-CF_Three-5-F
U-4a 2-C (O) CF_Three-4-F Et 2-OMe-4-CF_Three-5-Cl
U-4a 2-C (O) CF_Three-4-Cl Et 2-OMe-4-CF_Three-5-Br
U-4a 2-C (O) CF_Three-4-Br Et 2-OMe-4-CF_Three-5-Me
U-4a 2-C (O) CF_Three-4-Me Et 2-OMe-4,5-di-CF_Three
U-4a 2-C (O) CF_Three-4-CF_Three     Et 2,5-di-OMe-4-CF_Three
U-4a 2-C (O) CF_Three-4-OMe Et 2,4-di-OMe-5-F
U-4a 2-C (O) CF_Three-4-OCF_Three    Et 2,4-di-OMe-5-Cl
U-4a 2-Ac-5-F Et 2,4-di-OMe-5-Br
U-4a 2-Ac-5-Cl Et 2,4-di-OMe-5-Me
U-4a 2-Ac-5-Br Et 2,4-di-OMe-5-CF_Three
U-4a 2-Ac-5-Me Et 2,4,5-tri-OMe
U-4a 2-Ac-5-CF_Three          Et 3-OMe-4,5-di-F
U-4a 2-Ac-5-OMe Et 3-OMe-4-F-5-Cl
U-4a 2-Ac-5-OCF_Three         Et 3-OMe-4-F-5-Br
U-4a 2- (U-3b) -5-F Et 3-OMe-4-F-5-Me
U-4a 2- (U-3b) -5-Cl Et 3-OMe-4-F-5-CF_Three
U-4a 2- (U-3b) -5-Br Et 3,5-di-OMe-4-F
U-4a 2- (U-3b) -5-Me Et 3-OMe-4-Cl-5-F
U-4a 2- (U-3b) -5-CF_Three      Et 3-OMe-4,5-di-Cl
U-4a 2- (U-3b) -5-OMe Et 3-OMe-4-Cl-5-Br
U-4a 2- (U-3b) -5-OCF_Three     Et 3-OMe-4-Cl-5-Me
U-4a 2-CF₂H-5-F Et 3-OMe-4-Cl-5-CF_Three
U-4a 2-CF₂H-5-Cl Et 3,5-di-OMe-4-Cl
U-4a 2-CF₂H-5-Br Et 3-OMe-4-Br-5-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
U-4a 2-CF₂H-5-Me Et 3-OMe-4-Br-5-Cl
U-4a 2-CF₂H-5-CF_Three        Et 3-OMe-4,5-di-Br
U-4a 2-CF₂H-5-OMe Et 3-OMe-4-Br-5-Me
U-4a 2-CF₂H-5-OCF_Three       Et 3-OMe-4-Br-5-CF_Three
U-4a 2-CN-5-F Et 3,5-di-OMe-4-Br
U-4a 2-CN-5-Cl Et 3-OMe-4-Me-5-F
U-4a 2-CN-5-Br Et 3-OMe-4-Me-5-Cl
U-4a 2-CN-5-Me Et 3-OMe-4-Me-5-Br
U-4a 2-CN-5-CF_Three          Et 3-OMe-4,5-di-Me
U-4a 2-CN-5-OMe Et 3-OMe-4-Me-5-CF_Three
U-4a 2-CN-5-OCF_Three         Et 3,5-di-OMe-4-Me
U-4a 2-Et-5-F Et 3-OMe-4-CF_Three-5-F
U-4a 2-Et-5-Cl Et 3-OMe-4-CF_Three-5-Cl
U-4a 2-Et-5-Br Et 3-OMe-4-CF_Three-5-Br
U-4a 2-Et-5-Me Et 3-OMe-4-CF_Three-5-Me
U-4a 2-Et-5-CF_Three          Et 3-OMe-4,5-di-CF_Three
U-4a 2-Et-5-OMe Et 3,5-di-OMe-4-CF_Three
U-4a 2-Et-5-OCF_Three         Et 3,4-di-OMe-5-F
U-4a 2-OCF₂H-5-F Et 3,4-di-OMe-5-Cl
U-4a 2-OCF₂H-5-Cl Et 3,4-di-OMe-5-Br
U-4a 2-OCF₂H-5-Br Et 3,4-di-OMe-5-Me
U-4a 2-OCF₂H-5-Me Et 3,4-di-OMe-5-CF_Three
U-4a 2-OCF₂H-5-CF_Three       Et 3,4,5-tri-OMe
U-4a 2-OCF₂H-5-OMe cPr 2,3,4-tri-F
U-4a 2-OCF₂H-5-OCF_Three      cPr 2,3-di-F-4-Cl
U-4a 2-OEt-5-F cPr 2,3-di-F-4-Br
U-4a 2-OEt-5-Cl cPr 2,3-di-F-4-Me
U-4a 2-OEt-5-Br cPr 2,3-di-F-4-CF_Three
U-4a 2-OEt-5-Me cPr 2,3-di-F-4-OMe
U-4a 2-OEt-5-CF_Three         cPr 2,4-di-F-3-Cl
U-4a 2-OEt-5-OMe cPr 2-F-3,4-di-Cl
U-4a 2-OEt-5-OCF_Three        cPr 2-F-3-Cl-4-Br
U-4a 2-C (O) CF_Three-5-F cPr 2-F-3-Cl-4-Me
U-4a 2-C (O) CF_Three-5-Cl cPr 2-F-3-Cl-4-CF_Three
U-4a 2-C (O) CF_Three-5-Br cPr 2-F-3-Cl-4-OMe
U-4a 2-C (O) CF_Three-5-Me cPr 2,4-di-F-3-Br
U-4a 2-C (O) CF_Three-5-CF_Three     cPr 2-F-3-Br-4-Cl
U-4a 2-C (O) CF_Three-5-OMe cPr 2-F-3,4-di-Br
U-4a 2-C (O) CF_Three-5-OCF_Three    cPr 2-F-3-Br-4-Me
U-4a 3-Ac-4-F cPr 2-F-3-Br-4-CF_Three
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
U-4a 3-Ac-4-Cl cPr 2-F-3-Br-4-OMe
U-4a 3-Ac-4-Br cPr 2,4-di-F-3-Me
U-4a 3-Ac-4-Me cPr 2-F-3-Me-4-Cl
U-4a 3-Ac-4-CF_Three          cPr 2-F-3-Me-4-Br
U-4a 3-Ac-4-OMe cPr 2-F-3,4-di-Me
U-4a 3-Ac-4-OCF_Three         cPr 2-F-3-Me-4-CF_Three
U-4a 3- (U-3b) -4-F cPr 2-F-3-Me-4-OMe
U-4a 3- (U-3b) -4-Cl cPr 2,4-di-F-3-CF_Three
U-4a 3- (U-3b) -4-Br cPr 2-F-3-CF_Three-4-Cl
U-4a 3- (U-3b) -4-Me cPr 2-F-3-CF_Three-4-Br
U-4a 3- (U-3b) -4-CF_Three      cPr 2-F-3-CF_Three-4-Me
U-4a 3- (U-3b) -4-OMe cPr 2-F-3,4-di-CF_Three
U-4a 3- (U-3b) -4-OCF_Three     cPr 2-F-3-CF_Three-4-OMe
U-4a 3-CF₂H-4-F cPr 2,4-di-F-3-OMe
U-4a 3-CF₂H-4-Cl cPr 2-F-3-OMe-4-Cl
U-4a 3-CF₂H-4-Br cPr 2-F-3-OMe-4-Br
U-4a 3-CF₂H-4-Me cPr 2-F-3-OMe-4-Me
U-4a 3-CF₂H-4-CF_Three        cPr 2-F-3-OMe-4-CF_Three
U-4a 3-CF₂H-4-OMe cPr 2-F-3,4-di-OMe
U-4a 3-CF₂H-4-OCF_Three       cPr 2,3,5-tri-F
U-4a 3-CN-4-F cPr 2,3-di-F-5-Cl
U-4a 3-CN-4-Cl cPr 2,3-di-F-5-Br
U-4a 3-CN-4-Br cPr 2,3-di-F-5-Me
U-4a 3-CN-4-Me cPr 2,3-di-F-5-CF_Three
U-4a 3-CN-4-CF_Three          cPr 2,3-di-F-5-OMe
U-4a 3-CN-4-OMe cPr 2,5-di-F-3-Cl
U-4a 3-CN-4-OCF_Three         cPr 2-F-3,5-di-Cl
U-4a 3-Et-4-F cPr 2-F-3-Cl-5-Br
U-4a 3-Et-4-Cl cPr 2-F-3-Cl-5-Me
U-4a 3-Et-4-Br cPr 2-F-3-Cl-5-CF_Three
U-4a 3-Et-4-Me cPr 2-F-3-Cl-5-OMe
U-4a 3-Et-4-CF_Three          cPr 2,5-di-F-3-Br
U-4a 3-Et-4-OMe cPr 2-F-3-Br-5-Cl
U-4a 3-Et-4-OCF_Three         cPr 2-F-3,5-di-Br
U-4a 3-OCF₂H-4-F cPr 2-F-3-Br-5-Me
U-4a 3-OCF₂H-4-Cl cPr 2-F-3-Br-5-CF_Three
U-4a 3-OCF₂H-4-Br cPr 2-F-3-Br-5-OMe
U-4a 3-OCF₂H-4-Me cPr 2,5-di-F-3-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
U-4a 3-OCF₂H-4-CF_Three       cPr 2-F-3-Me-5-Cl
U-4a 3-OCF₂H-4-OMe cPr 2-F-3-Me-5-Br
U-4a 3-OCF₂H-4-OCF_Three      cPr 2-F-3,5-di-Me
U-4a 3-OEt-4-F cPr 2-F-3-Me-5-CF_Three
U-4a 3-OEt-4-Cl cPr 2-F-3-Me-5-OMe
U-4a 3-OEt-4-Br cPr 2,5-di-F-3-CF_Three
U-4a 3-OEt-4-Me cPr 2-F-3-CF_Three-5-Cl
U-4a 3-OEt-4-CF_Three         cPr 2-F-3-CF_Three-5-Br
U-4a 3-OEt-4-OMe cPr 2-F-3-CF_Three-5-Me
U-4a 3-OEt-4-OCF_Three        cPr 2-F-3,5-di-CF_Three
U-4a 3-C (O) CF_Three-4-F cPr 2-F-3-CF_Three-5-OMe
U-4a 3-C (O) CF_Three-4-Cl cPr 2,5-di-F-3-OMe
U-4a 3-C (O) CF_Three-4-Br cPr 2-F-3-OMe-5-Cl
U-4a 3-C (O) CF_Three-4-Me cPr 2-F-3-OMe-5-Br
U-4a 3-C (O) CF_Three-4-CF_Three     cPr 2-F-3-OMe-5-Me
U-4a 3-C (O) CF_Three-4-OMe cPr 2-F-3-OMe-5-CF_Three
U-4a 3-C (O) CF_Three-4-OCF_Three    cPr 2-F-3,5-di-OMe
U-4a 3-Ac-5-F cPr 2,4,5-tri-F
U-4a 3-Ac-5-Cl cPr 2,4-di-F-5-Cl
U-4a 3-Ac-5-Br cPr 2,4-di-F-5-Br
U-4a 3-Ac-5-Me cPr 2,4-di-F-5-Me
U-4a 3-Ac-5-CF_Three          cPr 2,4-di-F-5-CF_Three
U-4a 3-Ac-5-OMe cPr 2,4-di-F-5-OMe
U-4a 3-Ac-5-OCF_Three         cPr 2,5-di-F-4-Cl
U-4a 3- (U-3b) -5-F cPr 2-F-4,5-di-Cl
U-4a 3- (U-3b) -5-Cl cPr 2-F-4-Cl-5-Br
U-4a 3- (U-3b) -5-Br cPr 2-F-4-Cl-5-Me
U-4a 3- (U-3b) -5-Me cPr 2-F-4-Cl-5-CF_Three
U-4a 3- (U-3b) -5-CF_Three      cPr 2-F-4-Cl-5-OMe
U-4a 3- (U-3b) -5-OMe cPr 2,5-di-F-4-Br
U-4a 3- (U-3b) -5-OCF_Three     cPr 2-F-4-Br-5-Cl
U-4a 3-CF₂H-5-F cPr 2-F-4,5-di-Br
U-4a 3-CF₂H-5-Cl cPr 2-F-4-Br-5-Me
U-4a 3-CF₂H-5-Br cPr 2-F-4-Br-5-CF_Three
U-4a 3-CF₂H-5-Me cPr 2-F-4-Br-5-OMe
U-4a 3-CF₂H-5-CF_Three        cPr 2,5-di-F-4-Me
U-4a 3-CF₂H-5-OMe cPr 2-F-4-Me-5-Cl
U-4a 3-CF₂H-5-OCF_Three       cPr 2-F-4-Me-5-Br
U-4a 3-CN-5-F cPr 2-F-4,5-di-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
U-4a 3-CN-5-Cl cPr 2-F-4-Me-5-CF_Three
U-4a 3-CN-5-Br cPr 2-F-4-Me-5-OMe
U-4a 3-CN-5-Me cPr 2,5-di-F-4-CF_Three
U-4a 3-CN-5-CF_Three          cPr 2-F-4-CF_Three-5-Cl
U-4a 3-CN-5-OMe cPr 2-F-4-CF_Three-5-Br
U-4a 3-CN-5-OCF_Three         cPr 2-F-4-CF_Three-5-Me
U-4a 3-Et-5-F cPr 2-F-4,5-di-CF_Three
U-4a 3-Et-5-Cl cPr 2-F-4-CF_Three-5-OMe
U-4a 3-Et-5-Br cPr 2,5-di-F-4-OMe
U-4a 3-Et-5-Me cPr 2-F-4-OMe-5-Cl
U-4a 3-Et-5-CF_Three          cPr 2-F-4-OMe-5-Br
U-4a 3-Et-5-OMe cPr 2-F-4-OMe-5-Me
U-4a 3-Et-5-OCF_Three         cPr 2-F-4-OMe-5-CF_Three
U-4a 3-OCF₂H-5-F cPr 2-F-4,5-di-OMe
U-4a 3-OCF₂H-5-Cl cPr 3,4,5-tri-F
U-4a 3-OCF₂H-5-Br cPr 3,4-di-F-5-Cl
U-4a 3-OCF₂H-5-Me cPr 3,4-di-F-5-Br
U-4a 3-OCF₂H-5-CF_Three       cPr 3,4-di-F-5-Me
U-4a 3-OCF₂H-5-OMe cPr 3,4-di-F-5-CF_Three
U-4a 3-OCF₂H-5-OCF_Three      cPr 3,4-di-F-5-OMe
U-4a 3-OEt-5-F cPr 3,5-di-F-4-Cl
U-4a 3-OEt-5-Cl cPr 3-F-4,5-di-Cl
U-4a 3-OEt-5-Br cPr 3-F-4-Cl-5-Br
U-4a 3-OEt-5-Me cPr 3-F-4-Cl-5-Me
U-4a 3-OEt-5-CF_Three         cPr 3-F-4-Cl-5-CF_Three
U-4a 3-OEt-5-OMe cPr 3-F-4-Cl-5-OMe
U-4a 3-OEt-5-OCF_Three        cPr 3,5-di-F-4-Br
U-4a 3-C (O) CF_Three-5-F cPr 3-F-4-Br-5-Cl
U-4a 3-C (O) CF_Three-5-Cl cPr 3-F-4,5-di-Br
U-4a 3-C (O) CF_Three-5-Br cPr 3-F-4-Br-5-Me
U-4a 3-C (O) CF_Three-5-Me cPr 3-F-4-Br-5-CF_Three
U-4a 3-C (O) CF_Three-5-CF_Three     cPr 3-F-4-Br-5-OMe
U-4a 3-C (O) CF_Three-5-OMe cPr 3,5-di-F-4-Me
U-4a 3-C (O) CF_Three-5-OCF_Three    cPr 3-F-4-Me-5-Cl
CF_Three   2-F-3-Ac cPr 3-F-4-Me-5-Br
CF_Three   2-F-3- (U-3b) cPr 3-F-4,5-di-Me
CF_Three   2-F-3-CF₂H cPr 3-F-4-Me-5-CF_Three
CF_Three   2-F-3-CN cPr 3-F-4-Me-5-OMe
CF_Three   2-F-3-Et cPr 3,5-di-F-4-CF_Three
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
CF_Three   2-F-3-OCF₂H cPr 3-F-4-CF_Three-5-Cl
CF_Three   2-F-3-OEt cPr 3-F-4-CF_Three-5-Br
CF_Three   2-F-3-C (O) CF_Three       cPr 3-F-4-CF_Three-5-Me
CF_Three   2-Cl-3-Ac cPr 3-F-4,5-di-CF_Three
CF_Three   2-Cl-3- (U-3b) cPr 3-F-4-CF_Three-5-OMe
CF_Three   2-Cl-3-CF₂H cPr 3,5-di-F-4-OMe
CF_Three   2-Cl-3-CN cPr 3-F-4-OMe-5-Cl
CF_Three   2-Cl-3-Et cPr 3-F-4-OMe-5-Br
CF_Three   2-Cl-3-OCF₂H cPr 3-F-4-OMe-5-Me
CF_Three   2-Cl-3-OEt cPr 3-F-4-OMe-5-CF_Three
CF_Three   2-Cl-3-C (O) CF_Three      cPr 3-F-4,5-di-OMe
CF_Three   2-Br-3-Ac cPr 2-Cl-3,4-di-F
CF_Three   2-Br-3- (U-3b) cPr 2,4-di-Cl-3-F
CF_Three   2-Br-3-CF₂H cPr 2-Cl-3-F-4-Br
CF_Three   2-Br-3-CN cPr 2-Cl-3-F-4-Me
CF_Three   2-Br-3-Et cPr 2-Cl-3-F-4-CF_Three
CF_Three   2-Br-3-OCF₂H cPr 2-Cl-3-F-4-OMe
CF_Three   2-Br-3-OEt cPr 2,3-di-Cl-4-F
CF_Three   2-Br-3-C (O) CF_Three      cPr 2,3,4-tri-Cl
CF_Three   2-Me-3-Ac cPr 2,3-di-Cl-4-Br
CF_Three   2-Me-3- (U-3b) cPr 2,3-di-Cl-4-Me
CF_Three   2-Me-3-CF₂H cPr 2,3-di-Cl-4-CF_Three
CF_Three   2-Me-3-CN cPr 2,3-di-Cl-4-OMe
CF_Three   2-Me-3-Et cPr 2-Cl-3-Br-4-F
CF_Three   2-Me-3-OCF₂H cPr 2,4-di-Cl-3-Br
CF_Three   2-Me-3-OEt cPr 2-Cl-3,4-di-Br
CF_Three   2-Me-3-C (O) CF_Three      cPr 2-Cl-3-Br-4-Me
CF_Three   2-CF_Three-3-Ac cPr 2-Cl-3-Br-4-CF_Three
CF_Three   2-CF_Three-3- (U-3b) cPr 2-Cl-3-Br-4-OMe
CF_Three   2-CF_Three-3-CF₂H cPr 2-Cl-3-Me-4-F
CF_Three   2-CF_Three-3-CN cPr 2,4-di-Cl-3-Me
CF_Three   2-CF_Three-3-Et cPr 2-Cl-3-Me-4-Br
CF_Three   2-CF_Three-3-OCF₂H cPr 2-Cl-3,4-di-Me
CF_Three   2-CF_Three-3-OEt cPr 2-Cl-3-Me-4-CF_Three
CF_Three   2-CF_Three-3-C (O) CF_Three     cPr 2-Cl-3-Me-4-OMe
CF_Three   2-OMe-3-Ac cPr 2-Cl-3-CF_Three-4-F
CF_Three   2-OMe-3- (U-3b) cPr 2,4-di-Cl-3-CF_Three
CF_Three   2-OMe-3-CF₂H cPr 2-Cl-3-CF_Three-4-Br
CF_Three   2-OMe-3-CN cPr 2-Cl-3-CF_Three-4-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
CF_Three   2-OMe-3-Et cPr 2-Cl-3,4-di-CF_Three
CF_Three   2-OMe-3-OCF₂H cPr 2-Cl-3-CF_Three-4-OMe
CF_Three   2-OMe-3-OEt cPr 2-Cl-3-OMe-4-F
CF_Three   2-OMe-3-C (O) CF_Three     cPr 2,4-di-Cl-3-OMe
CF_Three   2-OCF_Three-3-Ac cPr 2-Cl-3-OMe-4-Br
CF_Three   2-OCF_Three-3- (U-3b) cPr 2-Cl-3-OMe-4-Me
CF_Three   2-OCF_Three-3-CF₂H cPr 2-Cl-3-OMe-4-CF_Three
CF_Three   2-OCF_Three-3-CN cPr 2-Cl-3,4-di-OMe
CF_Three   2-OCF_Three-3-Et cPr 2-Cl-3,5-di-F
CF_Three   2-OCF_Three-3-OCF₂H cPr 2,5-di-Cl-3-F
CF_Three   2-OCF_Three-3-OEt cPr 2-Cl-3-F-5-Br
CF_Three   2-OCF_Three-3-C (O) CF_Three    cPr 2-Cl-3-F-5-Me
CF_Three   2-F-4-Ac cPr 2-Cl-3-F-5-CF_Three
CF_Three   2-F-4- (U-3b) cPr 2-Cl-3-F-5-OMe
CF_Three   2-F-4-CF₂H cPr 2,3-di-Cl-5-F
CF_Three   2-F-4-CN cPr 2,3,5-tri-Cl
CF_Three   2-F-4-Et cPr 2,3-di-Cl-5-Br
CF_Three   2-F-4-OCF₂H cPr 2,3-di-Cl-5-Me
CF_Three   2-F-4-OEt cPr 2,3-di-Cl-5-CF_Three
CF_Three   2-F-4-C (O) CF_Three       cPr 2,3-di-Cl-5-OMe
CF_Three   2-Cl-4-Ac cPr 2-Cl-3-Br-5-F
CF_Three   2-Cl-4- (U-3b) cPr 2,5-di-Cl-3-Br
CF_Three   2-Cl-4-CF₂H cPr 2-Cl-3,5-di-Br
CF_Three   2-Cl-4-CN cPr 2-Cl-3-Br-5-Me
CF_Three   2-Cl-4-Et cPr 2-Cl-3-Br-5-CF_Three
CF_Three   2-Cl-4-OCF₂H cPr 2-Cl-3-Br-5-OMe
CF_Three   2-Cl-4-OEt cPr 2-Cl-3-Me-5-F
CF_Three   2-Cl-4-C (O) CF_Three      cPr 2,5-di-Cl-3-Me
CF_Three   2-Br-4-Ac cPr 2-Cl-3-Me-5-Br
CF_Three   2-Br-4- (U-3b) cPr 2-Cl-3,5-di-Me
CF_Three   2-Br-4-CF₂H cPr 2-Cl-3-Me-5-CF_Three
CF_Three   2-Br-4-CN cPr 2-Cl-3-Me-5-OMe
CF_Three   2-Br-4-Et cPr 2-Cl-3-CF_Three-5-F
CF_Three   2-Br-4-OCF₂H cPr 2,5-di-Cl-3-CF_Three
CF_Three   2-Br-4-OEt cPr 2-Cl-3-CF_Three-5-Br
CF_Three   2-Br-4-C (O) CF_Three      cPr 2-Cl-3-CF_Three-5-Me
CF_Three   2-Me-4-Ac cPr 2-Cl-3,5-di-CF_Three
CF_Three   2-Me-4- (U-3b) cPr 2-Cl-3-CF_Three-5-OMe
CF_Three   2-Me-4-CF₂H cPr 2-Cl-3-OMe-5-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
CF_Three   2-Me-4-CN cPr 2,5-di-Cl-3-OMe
CF_Three   2-Me-4-Et cPr 2-Cl-3-OMe-5-Br
CF_Three   2-Me-4-OCF₂H cPr 2-Cl-3-OMe-5-Me
CF_Three   2-Me-4-OEt cPr 2-Cl-3-OMe-5-CF_Three
CF_Three   2-Me-4-C (O) CF_Three      cPr 2-Cl-3,5-di-OMe
CF_Three   2-CF_Three-4-Ac cPr 2-Cl-4,5-di-F
CF_Three   2-CF_Three-4- (U-3b) cPr 2,5-di-Cl-4-F
CF_Three   2-CF_Three-4-CF₂H cPr 2-Cl-4-F-5-Br
CF_Three   2-CF_Three-4-CN cPr 2-Cl-4-F-5-Me
CF_Three   2-CF_Three-4-Et cPr 2-Cl-4-F-5-CF_Three
CF_Three   2-CF_Three-4-OCF₂H cPr 2-Cl-4-F-5-OMe
CF_Three   2-CF_Three-4-OEt cPr 2,4-di-Cl-5-F
CF_Three   2-CF_Three-4-C (O) CF_Three     cPr 2,4,5-tri-Cl
CF_Three   2-OMe-4-Ac cPr 2,4-di-Cl-5-Br
CF_Three   2-OMe-4- (U-3b) cPr 2,4-di-Cl-5-Me
CF_Three   2-OMe-4-CF₂H cPr 2,4-di-Cl-5-CF_Three
CF_Three   2-OMe-4-CN cPr 2,4-di-Cl-5-OMe
CF_Three   2-OMe-4-Et cPr 2-Cl-4-Br-5-F
CF_Three   2-OMe-4-OCF₂H cPr 2,5-di-Cl-4-Br
CF_Three   2-OMe-4-OEt cPr 2-Cl-4,5-di-Br
CF_Three   2-OMe-4-C (O) CF_Three     cPr 2-Cl-4-Br-5-Me
CF_Three   2-OCF_Three-4-Ac cPr 2-Cl-4-Br-5-CF_Three
CF_Three   2-OCF_Three-4- (U-3b) cPr 2-Cl-4-Br-5-OMe
CF_Three   2-OCF_Three-4-CF₂H cPr 2-Cl-4-Me-5-F
CF_Three   2-OCF_Three-4-CN cPr 2,5-di-Cl-4-Me
CF_Three   2-OCF_Three-4-Et cPr 2-Cl-4-Me-5-Br
CF_Three   2-OCF_Three-4-OCF₂H cPr 2-Cl-4,5-di-Me
CF_Three   2-OCF_Three-4-OEt cPr 2-Cl-4-Me-5-CF_Three
CF_Three   2-OCF_Three-4-C (O) CF_Three    cPr 2-Cl-4-Me-5-OMe
CF_Three   2-F-5-Ac cPr 2-Cl-4-CF_Three-5-F
CF_Three   2-F-5- (U-3b) cPr 2,5-di-Cl-4-CF_Three
CF_Three   2-F-5-CF₂H cPr 2-Cl-4-CF_Three-5-Br
CF_Three   2-F-5-CN cPr 2-Cl-4-CF_Three-5-Me
CF_Three   2-F-5-Et cPr 2-Cl-4,5-di-CF_Three
CF_Three   2-F-5-OCF₂H cPr 2-Cl-4-CF_Three-5-OMe
CF_Three   2-F-5-OEt cPr 2-Cl-4-OMe-5-F
CF_Three   2-F-5-C (O) CF_Three       cPr 2,5-di-Cl-4-OMe
CF_Three   2-Cl-5-Ac cPr 2-Cl-4-OMe-5-Br
CF_Three   2-Cl-5- (U-3b) cPr 2-Cl-4-OMe-5-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
CF_Three   2-Cl-5-CF₂H cPr 2-Cl-4-OMe-5-CF_Three
CF_Three   2-Cl-5-CN cPr 2-Cl-4,5-di-OMe
CF_Three   2-Cl-5-Et cPr 3-Cl-4,5-di-F
CF_Three   2-Cl-5-OCF₂H cPr 3,5-di-Cl-4-F
CF_Three   2-Cl-5-OEt cPr 3-Cl-4-F-5-Br
CF_Three   2-Cl-5-C (O) CF_Three      cPr 3-Cl-4-F-5-Me
CF_Three   2-Br-5-Ac cPr 3-Cl-4-F-5-CF_Three
CF_Three   2-Br-5- (U-3b) cPr 3-Cl-4-F-5-OMe
CF_Three   2-Br-5-CF₂H cPr 3,4-di-Cl-5-F
CF_Three   2-Br-5-CN cPr 3,4,5-tri-Cl
CF_Three   2-Br-5-Et cPr 3,4-di-Cl-5-Br
CF_Three   2-Br-5-OCF₂H cPr 3,4-di-Cl-5-Me
CF_Three   2-Br-5-OEt cPr 3,4-di-Cl-5-CF_Three
CF_Three   2-Br-5-C (O) CF_Three      cPr 3,4-di-Cl-5-OMe
CF_Three   2-Me-5-Ac cPr 3-Cl-4-Br-5-F
CF_Three   2-Me-5- (U-3b) cPr 3,5-di-Cl-4-Br
CF_Three   2-Me-5-CF₂H cPr 3-Cl-4,5-di-Br
CF_Three   2-Me-5-CN cPr 3-Cl-4-Br-5-Me
CF_Three   2-Me-5-Et cPr 3-Cl-4-Br-5-CF_Three
CF_Three   2-Me-5-OCF₂H cPr 3-Cl-4-Br-5-OMe
CF_Three   2-Me-5-OEt cPr 3-Cl-4-Me-5-F
CF_Three   2-Me-5-C (O) CF_Three      cPr 3,5-di-Cl-4-Me
CF_Three   2-CF_Three-5-Ac cPr 3-Cl-4-Me-5-Br
CF_Three   2-CF_Three-5- (U-3b) cPr 3-Cl-4,5-di-Me
CF_Three   2-CF_Three-5-CF₂H cPr 3-Cl-4-Me-5-CF_Three
CF_Three   2-CF_Three-5-CN cPr 3-Cl-4-Me-5-OMe
CF_Three   2-CF_Three-5-Et cPr 3-Cl-4-CF_Three-5-F
CF_Three   2-CF_Three-5-OCF₂H cPr 3,5-di-Cl-4-CF_Three
CF_Three   2-CF_Three-5-OEt cPr 3-Cl-4-CF_Three-5-Br
CF_Three   2-CF_Three-5-C (O) CF_Three     cPr 3-Cl-4-CF_Three-5-Me
CF_Three   2-OMe-5-Ac cPr 3-Cl-4,5-di-CF_Three
CF_Three   2-OMe-5- (U-3b) cPr 3-Cl-4-CF_Three-5-OMe
CF_Three   2-OMe-5-CF₂H cPr 3-Cl-4-OMe-5-F
CF_Three   2-OMe-5-CN cPr 3,5-di-Cl-4-OMe
CF_Three   2-OMe-5-Et cPr 3-Cl-4-OMe-5-Br
CF_Three   2-OMe-5-OCF₂H cPr 3-Cl-4-OMe-5-Me
CF_Three   2-OMe-5-OEt cPr 3-Cl-4-OMe-5-CF_Three
CF_Three   2-OMe-5-C (O) CF_Three     cPr 3-Cl-4,5-di-OMe
CF_Three   2-OCF_Three-5-Ac cPr 2-Br-3,4-di-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
CF_Three   2-OCF_Three-5- (U-3b) cPr 2-Br-3-F-4-Cl
CF_Three   2-OCF_Three-5-CF₂H cPr 2,4-di-Br-3-F
CF_Three   2-OCF_Three-5-CN cPr 2-Br-3-F-4-Me
CF_Three   2-OCF_Three-5-Et cPr 2-Br-3-F-4-CF_Three
CF_Three   2-OCF_Three-5-OCF₂H cPr 2-Br-3-F-4-OMe
CF_Three   2-OCF_Three-5-OEt cPr 2-Br-3-Cl-4-F
CF_Three   2-OCF_Three-5-C (O) CF_Three    cPr 2-Br-3,4-di-Cl
CF_Three   3-F-4-Ac cPr 2,4-di-Br-3-Cl
CF_Three   3-F-4- (U-3b) cPr 2-Br-3-Cl-4-Me
CF_Three   3-F-4-CF₂H cPr 2-Br-3-Cl-4-CF_Three
CF_Three   3-F-4-CN cPr 2-Br-3-Cl-4-OMe
CF_Three   3-F-4-Et cPr 2,3-di-Br-4-F
CF_Three   3-F-4-OCF₂H cPr 2,3-di-Br-4-Cl
CF_Three   3-F-4-OEt cPr 2,3,4-tri-Br
CF_Three   3-F-4-C (O) CF_Three       cPr 2,3-di-Br-4-Me
CF_Three   3-Cl-4-Ac cPr 2,3-di-Br-4-CF_Three
CF_Three   3-Cl-4- (U-3b) cPr 2,3-di-Br-4-OMe
CF_Three   3-Cl-4-CF₂H cPr 2-Br-3-Me-4-F
CF_Three   3-Cl-4-CN cPr 2-Br-3-Me-4-Cl
CF_Three   3-Cl-4-Et cPr 2,4-di-Br-3-Me
CF_Three   3-Cl-4-OCF₂H cPr 2-Br-3,4-di-Me
CF_Three   3-Cl-4-OEt cPr 2-Br-3-Me-4-CF_Three
CF_Three   3-Cl-4-C (O) CF_Three      cPr 2-Br-3-Me-4-OMe
CF_Three   3-Br-4-Ac cPr 2-Br-3-CF_Three-4-F
CF_Three   3-Br-4- (U-3b) cPr 2-Br-3-CF_Three-4-Cl
CF_Three   3-Br-4-CF₂H cPr 2,4-di-Br-3-CF_Three
CF_Three   3-Br-4-CN cPr 2-Br-3-CF_Three-4-Me
CF_Three   3-Br-4-Et cPr 2-Br-3,4-di-CF_Three
CF_Three   3-Br-4-OCF₂H cPr 2-Br-3-CF_Three-4-OMe
CF_Three   3-Br-4-OEt cPr 2-Br-3-OMe-4-F
CF_Three   3-Br-4-C (O) CF_Three      cPr 2-Br-3-OMe-4-Cl
CF_Three   3-Me-4-Ac cPr 2,4-di-Br-3-OMe
CF_Three   3-Me-4- (U-3b) cPr 2-Br-3-OMe-4-Me
CF_Three   3-Me-4-CF₂H cPr 2-Br-3-OMe-4-CF_Three
CF_Three   3-Me-4-CN cPr 2-Br-3,4-di-OMe
CF_Three   3-Me-4-Et cPr 2-Br-3,5-di-F
CF_Three   3-Me-4-OCF₂H cPr 2-Br-3-F-5-Cl
CF_Three   3-Me-4-OEt cPr 2,5-di-Br-3-F
CF_Three   3-Me-4-C (O) CF_Three      cPr 2-Br-3-F-5-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
CF_Three   3-CF_Three-4-Ac cPr 2-Br-3-F-5-CF_Three
CF_Three   3-CF_Three-4- (U-3b) cPr 2-Br-3-F-5-OMe
CF_Three   3-CF_Three-4-CF₂H cPr 2-Br-3-Cl-5-F
CF_Three   3-CF_Three-4-CN cPr 2-Br-3,5-di-Cl
CF_Three   3-CF_Three-4-Et cPr 2,5-di-Br-3-Cl
CF_Three   3-CF_Three-4-OCF₂H cPr 2-Br-3-Cl-5-Me
CF_Three   3-CF_Three-4-OEt cPr 2-Br-3-Cl-5-CF_Three
CF_Three   3-CF_Three-4-C (O) CF_Three     cPr 2-Br-3-Cl-5-OMe
CF_Three   3-OMe-4-Ac cPr 2,3-di-Br-5-F
CF_Three   3-OMe-4- (U-3b) cPr 2,3-di-Br-5-Cl
CF_Three   3-OMe-4-CF₂H cPr 2,3,5-tri-Br
CF_Three   3-OMe-4-CN cPr 2,3-di-Br-5-Me
CF_Three   3-OMe-4-Et cPr 2,3-di-Br-5-CF_Three
CF_Three   3-OMe-4-OCF₂H cPr 2,3-di-Br-5-OMe
CF_Three   3-OMe-4-OEt cPr 2-Br-3-Me-5-F
CF_Three   3-OMe-4-C (O) CF_Three     cPr 2-Br-3-Me-5-Cl
CF_Three   3-OCF_Three-4-Ac cPr 2,5-di-Br-3-Me
CF_Three   3-OCF_Three-4- (U-3b) cPr 2-Br-3,5-di-Me
CF_Three   3-OCF_Three-4-CF₂H cPr 2-Br-3-Me-5-CF_Three
CF_Three   3-OCF_Three-4-CN cPr 2-Br-3-Me-5-OMe
CF_Three   3-OCF_Three-4-Et cPr 2-Br-3-CF_Three-5-F
CF_Three   3-OCF_Three-4-OCF₂H cPr 2-Br-3-CF_Three-5-Cl
CF_Three   3-OCF_Three-4-OEt cPr 2,5-di-Br-3-CF_Three
CF_Three   3-OCF_Three-4-C (O) CF_Three    cPr 2-Br-3-CF_Three-5-Me
CF_Three   3-F-5-Ac cPr 2-Br-3,5-di-CF_Three
CF_Three   3-F-5- (U-3b) cPr 2-Br-3-CF_Three-5-OMe
CF_Three   3-F-5-CF₂H cPr 2-Br-3-OMe-5-F
CF_Three   3-F-5-CN cPr 2-Br-3-OMe-5-Cl
CF_Three   3-F-5-Et cPr 2,5-di-Br-3-OMe
CF_Three   3-F-5-OCF₂H cPr 2-Br-3-OMe-5-Me
CF_Three   3-F-5-OEt cPr 2-Br-3-OMe-5-CF_Three
CF_Three   3-F-5-C (O) CF_Three       cPr 2-Br-3,5-di-OMe
CF_Three   3-Cl-5-Ac cPr 2-Br-4,5-di-F
CF_Three   3-Cl-5- (U-3b) cPr 2-Br-4-F-5-Cl
CF_Three   3-Cl-5-CF₂H cPr 2,5-di-Br-4-F
CF_Three   3-Cl-5-CN cPr 2-Br-4-F-5-Me
CF_Three   3-Cl-5-Et cPr 2-Br-4-F-5-CF_Three
CF_Three   3-Cl-5-OCF₂H cPr 2-Br-4-F-5-OMe
CF_Three   3-Cl-5-OEt cPr 2-Br-4-Cl-5-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
CF_Three   3-Cl-5-C (O) CF_Three      cPr 2-Br-4,5-di-Cl
CF_Three   3-Br-5-Ac cPr 2,5-di-Br-4-Cl
CF_Three   3-Br-5- (U-3b) cPr 2-Br-4-Cl-5-Me
CF_Three   3-Br-5-CF₂H cPr 2-Br-4-Cl-5-CF_Three
CF_Three   3-Br-5-CN cPr 2-Br-4-Cl-5-OMe
CF_Three   3-Br-5-Et cPr 2,4-di-Br-5-F
CF_Three   3-Br-5-OCF₂H cPr 2,4-di-Br-5-Cl
CF_Three   3-Br-5-OEt cPr 2,4,5-tri-Br
CF_Three   3-Br-5-C (O) CF_Three      cPr 2,4-di-Br-5-Me
CF_Three   3-Me-5-Ac cPr 2,4-di-Br-5-CF_Three
CF_Three   3-Me-5- (U-3b) cPr 2,4-di-Br-5-OMe
CF_Three   3-Me-5-CF₂H cPr 2-Br-4-Me-5-F
CF_Three   3-Me-5-CN cPr 2-Br-4-Me-5-Cl
CF_Three   3-Me-5-Et cPr 2,5-di-Br-4-Me
CF_Three   3-Me-5-OCF₂H cPr 2-Br-4,5-di-Me
CF_Three   3-Me-5-OEt cPr 2-Br-4-Me-5-CF_Three
CF_Three   3-Me-5-C (O) CF_Three      cPr 2-Br-4-Me-5-OMe
CF_Three   3-CF_Three-5-Ac cPr 2-Br-4-CF_Three-5-F
CF_Three   3-CF_Three-5- (U-3b) cPr 2-Br-4-CF_Three-5-Cl
CF_Three   3-CF_Three-5-CF₂H cPr 2,5-di-Br-4-CF_Three
CF_Three   3-CF_Three-5-CN cPr 2-Br-4-CF_Three-5-Me
CF_Three   3-CF_Three-5-Et cPr 2-Br-4,5-di-CF_Three
CF_Three   3-CF_Three-5-OCF₂H cPr 2-Br-4-CF_Three-5-OMe
CF_Three   3-CF_Three-5-OEt cPr 2-Br-4-OMe-5-F
CF_Three   3-CF_Three-5-C (O) CF_Three     cPr 2-Br-4-OMe-5-Cl
CF_Three   3-OMe-5-Ac cPr 2,5-di-Br-4-OMe
CF_Three   3-OMe-5- (U-3b) cPr 2-Br-4-OMe-5-Me
CF_Three   3-OMe-5-CF₂H cPr 2-Br-4-OMe-5-CF_Three
CF_Three   3-OMe-5-CN cPr 2-Br-4,5-di-OMe
CF_Three   3-OMe-5-Et cPr 3-Br-4,5-di-F
CF_Three   3-OMe-5-OCF₂H cPr 3-Br-4-F-5-Cl
CF_Three   3-OMe-5-OEt cPr 3,5-di-Br-4-F
CF_Three   3-OMe-5-C (O) CF_Three     cPr 3-Br-4-F-5-Me
CF_Three   3-OCF_Three-5-Ac cPr 3-Br-4-F-5-CF_Three
CF_Three   3-OCF_Three-5- (U-3b) cPr 3-Br-4-F-5-OMe
CF_Three   3-OCF_Three-5-CF₂H cPr 3-Br-4-Cl-5-F
CF_Three   3-OCF_Three-5-CN cPr 3-Br-4,5-di-Cl
CF_Three   3-OCF_Three-5-Et cPr 3,5-di-Br-4-Cl
CF_Three   3-OCF_Three-5-OCF₂H cPr 3-Br-4-Cl-5-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
CF_Three   3-OCF_Three-5-OEt cPr 3-Br-4-Cl-5-CF_Three
CF_Three   3-OCF_Three-5-C (O) CF_Three    cPr 3-Br-4-Cl-5-OMe
CF_Three   2-Ac-3-F cPr 3,4-di-Br-5-F
CF_Three   2-Ac-3-Cl cPr 3,4-di-Br-5-Cl
CF_Three   2-Ac-3-Br cPr 3,4,5-tri-Br
CF_Three   2-Ac-3-Me cPr 3,4-di-Br-5-Me
CF_Three   2-Ac-3-CF_Three          cPr 3,4-di-Br-5-CF_Three
CF_Three   2-Ac-3-OMe cPr 3,4-di-Br-5-OMe
CF_Three   2-Ac-3-OCF_Three         cPr 3-Br-4-Me-5-F
CF_Three   2- (U-3b) -3-F cPr 3-Br-4-Me-5-Cl
CF_Three   2- (U-3b) -3-Cl cPr 3,5-di-Br-4-Me
CF_Three   2- (U-3b) -3-Br cPr 3-Br-4,5-di-Me
CF_Three   2- (U-3b) -3-Me cPr 3-Br-4-Me-5-CF_Three
CF_Three   2- (U-3b) -3-CF_Three      cPr 3-Br-4-Me-5-OMe
CF_Three   2- (U-3b) -3-OMe cPr 3-Br-4-CF_Three-5-F
CF_Three   2- (U-3b) -3-OCF_Three     cPr 3-Br-4-CF_Three-5-Cl
CF_Three   2-CF₂H-3-F cPr 3,5-di-Br-4-CF_Three
CF_Three   2-CF₂H-3-Cl cPr 3-Br-4-CF_Three-5-Me
CF_Three   2-CF₂H-3-Br cPr 3-Br-4,5-di-CF_Three
CF_Three   2-CF₂H-3-Me cPr 3-Br-4-CF_Three-5-OMe
CF_Three   2-CF₂H-3-CF_Three        cPr 3-Br-4-OMe-5-F
CF_Three   2-CF₂H-3-OMe cPr 3-Br-4-OMe-5-Cl
CF_Three   2-CF₂H-3-OCF_Three       cPr 3,5-di-Br-4-OMe
CF_Three   2-CN-3-F cPr 3-Br-4-OMe-5-Me
CF_Three   2-CN-3-Cl cPr 3-Br-4-OMe-5-CF_Three
CF_Three   2-CN-3-Br cPr 3-Br-4,5-di-OMe
CF_Three   2-CN-3-Me cPr 2-Me-3,4-di-F
CF_Three   2-CN-3-CF_Three          cPr 2-Me-3-F-4-Cl
CF_Three   2-CN-3-OMe cPr 2-Me-3-F-4-Br
CF_Three   2-CN-3-OCF_Three         cPr 2,4-di-Me-3-F
CF_Three   2-Et-3-F cPr 2-Me-3-F-4-CF_Three
CF_Three   2-Et-3-Cl cPr 2-Me-3-F-4-OMe
CF_Three   2-Et-3-Br cPr 2-Me-3-Cl-4-F
CF_Three   2-Et-3-Me cPr 2-Me-3,4-di-Cl
CF_Three   2-Et-3-CF_Three          cPr 2-Me-3-Cl-4-Br
CF_Three   2-Et-3-OMe cPr 2,4-di-Me-3-Cl
CF_Three   2-Et-3-OCF_Three         cPr 2-Me-3-Cl-4-CF_Three
CF_Three   2-OCF₂H-3-F cPr 2-Me-3-Cl-4-OMe
CF_Three   2-OCF₂H-3-Cl cPr 2-Me-3-Br-4-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
CF_Three   2-OCF₂H-3-Br cPr 2-Me-3-Br-4-Cl
CF_Three   2-OCF₂H-3-Me cPr 2-Me-3,4-di-Br
CF_Three   2-OCF₂H-3-CF_Three       cPr 2,4-di-Me-3-Br
CF_Three   2-OCF₂H-3-OMe cPr 2-Me-3-Br-4-CF_Three
CF_Three   2-OCF₂H-3-OCF_Three      cPr 2-Me-3-Br-4-OMe
CF_Three   2-OEt-3-F cPr 2,3-di-Me-4-F
CF_Three   2-OEt-3-Cl cPr 2,3-di-Me-4-Cl
CF_Three   2-OEt-3-Br cPr 2,3-di-Me-4-Br
CF_Three   2-OEt-3-Me cPr 2,3,4-tri-Me
CF_Three   2-OEt-3-CF_Three         cPr 2,3-di-Me-4-CF_Three
CF_Three   2-OEt-3-OMe cPr 2,3-di-Me-4-OMe
CF_Three   2-OEt-3-OCF_Three        cPr 2-Me-3-CF_Three-4-F
CF_Three   2-C (O) CF_Three-3-F cPr 2-Me-3-CF_Three-4-Cl
CF_Three   2-C (O) CF_Three-3-Cl cPr 2-Me-3-CF_Three-4-Br
CF_Three   2-C (O) CF_Three-3-Br cPr 2,4-di-Me-3-CF_Three
CF_Three   2-C (O) CF_Three-3-Me cPr 2-Me-3,4-di-CF_Three
CF_Three   2-C (O) CF_Three-3-CF_Three     cPr 2-Me-3-CF_Three-4-OMe
CF_Three   2-C (O) CF_Three-3-OMe cPr 2-Me-3-OMe-4-F
CF_Three   2-C (O) CF_Three-3-OCF_Three    cPr 2-Me-3-OMe-4-Cl
CF_Three   2-Ac-4-F cPr 2-Me-3-OMe-4-Br
CF_Three   2-Ac-4-Cl cPr 2,4-di-Me-3-OMe
CF_Three   2-Ac-4-Br cPr 2-Me-3-OMe-4-CF_Three
CF_Three   2-Ac-4-Me cPr 2-Me-3,4-di-OMe
CF_Three   2-Ac-4-CF_Three          cPr 2-Me-3,5-di-F
CF_Three   2-Ac-4-OMe cPr 2-Me-3-F-5-Cl
CF_Three   2-Ac-4-OCF_Three         cPr 2-Me-3-F-5-Br
CF_Three   2- (U-3b) -4-F cPr 2,5-di-Me-3-F
CF_Three   2- (U-3b) -4-Cl cPr 2-Me-3-F-5-CF_Three
CF_Three   2- (U-3b) -4-Br cPr 2-Me-3-F-5-OMe
CF_Three   2- (U-3b) -4-Me cPr 2-Me-3-Cl-5-F
CF_Three   2- (U-3b) -4-CF_Three      cPr 2-Me-3,5-di-Cl
CF_Three   2- (U-3b) -4-OMe cPr 2-Me-3-Cl-5-Br
CF_Three   2- (U-3b) -4-OCF_Three     cPr 2,5-di-Me-3-Cl
CF_Three   2-CF₂H-4-F cPr 2-Me-3-Cl-5-CF_Three
CF_Three   2-CF₂H-4-Cl cPr 2-Me-3-Cl-5-OMe
CF_Three   2-CF₂H-4-Br cPr 2-Me-3-Br-5-F
CF_Three   2-CF₂H-4-Me cPr 2-Me-3-Br-5-Cl
CF_Three   2-CF₂H-4-CF_Three        cPr 2-Me-3,5-di-Br
CF_Three   2-CF₂H-4-OMe cPr 2,5-di-Me-3-Br
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
CF_Three   2-CF₂H-4-OCF_Three       cPr 2-Me-3-Br-5-CF_Three
CF_Three   2-CN-4-F cPr 2-Me-3-Br-5-OMe
CF_Three   2-CN-4-Cl cPr 2,3-di-Me-5-F
CF_Three   2-CN-4-Br cPr 2,3-di-Me-5-Cl
CF_Three   2-CN-4-Me cPr 2,3-di-Me-5-Br
CF_Three   2-CN-4-CF_Three          cPr 2,3,5-tri-Me
CF_Three   2-CN-4-OMe cPr 2,3-di-Me-5-CF_Three
CF_Three   2-CN-4-OCF_Three         cPr 2,3-di-Me-5-OMe
CF_Three   2-Et-4-F cPr 2-Me-3-CF_Three-5-F
CF_Three   2-Et-4-Cl cPr 2-Me-3-CF_Three-5-Cl
CF_Three   2-Et-4-Br cPr 2-Me-3-CF_Three-5-Br
CF_Three   2-Et-4-Me cPr 2,5-di-Me-3-CF_Three
CF_Three   2-Et-4-CF_Three          cPr 2-Me-3,5-di-CF_Three
CF_Three   2-Et-4-OMe cPr 2-Me-3-CF_Three-5-OMe
CF_Three   2-Et-4-OCF_Three         cPr 2-Me-3-OMe-5-F
CF_Three   2-OCF₂H-4-F cPr 2-Me-3-OMe-5-Cl
CF_Three   2-OCF₂H-4-Cl cPr 2-Me-3-OMe-5-Br
CF_Three   2-OCF₂H-4-Br cPr 2,5-di-Me-3-OMe
CF_Three   2-OCF₂H-4-Me cPr 2-Me-3-OMe-5-CF_Three
CF_Three   2-OCF₂H-4-CF_Three       cPr 2-Me-3,5-di-OMe
CF_Three   2-OCF₂H-4-OMe cPr 2-Me-4,5-di-F
CF_Three   2-OCF₂H-4-OCF_Three      cPr 2-Me-4-F-5-Cl
CF_Three   2-OEt-4-F cPr 2-Me-4-F-5-Br
CF_Three   2-OEt-4-Cl cPr 2,5-di-Me-4-F
CF_Three   2-OEt-4-Br cPr 2-Me-4-F-5-CF_Three
CF_Three   2-OEt-4-Me cPr 2-Me-4-F-5-OMe
CF_Three   2-OEt-4-CF_Three         cPr 2-Me-4-Cl-5-F
CF_Three   2-OEt-4-OMe cPr 2-Me-4,5-di-Cl
CF_Three   2-OEt-4-OCF_Three        cPr 2-Me-4-Cl-5-Br
CF_Three   2-C (O) CF_Three-4-F cPr 2,5-di-Me-4-Cl
CF_Three   2-C (O) CF_Three-4-Cl cPr 2-Me-4-Cl-5-CF_Three
CF_Three   2-C (O) CF_Three-4-Br cPr 2-Me-4-Cl-5-OMe
CF_Three   2-C (O) CF_Three-4-Me cPr 2-Me-4-Br-5-F
CF_Three   2-C (O) CF_Three-4-CF_Three     cPr 2-Me-4-Br-5-Cl
CF_Three   2-C (O) CF_Three-4-OMe cPr 2-Me-4,5-di-Br
CF_Three   2-C (O) CF_Three-4-OCF_Three    cPr 2,5-di-Me-4-Br
CF_Three   2-Ac-5-F cPr 2-Me-4-Br-5-CF_Three
CF_Three   2-Ac-5-Cl cPr 2-Me-4-Br-5-OMe
CF_Three   2-Ac-5-Br cPr 2,4-di-Me-5-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
CF_Three   2-Ac-5-Me cPr 2,4-di-Me-5-Cl
CF_Three   2-Ac-5-CF_Three          cPr 2,4-di-Me-5-Br
CF_Three   2-Ac-5-OMe cPr 2,4,5-tri-Me
CF_Three   2-Ac-5-OCF_Three         cPr 2,4-di-Me-5-CF_Three
CF_Three   2- (U-3b) -5-F cPr 2,4-di-Me-5-OMe
CF_Three   2- (U-3b) -5-Cl cPr 2-Me-4-CF_Three-5-F
CF_Three   2- (U-3b) -5-Br cPr 2-Me-4-CF_Three-5-Cl
CF_Three   2- (U-3b) -5-Me cPr 2-Me-4-CF_Three-5-Br
CF_Three   2- (U-3b) -5-CF_Three      cPr 2,5-di-Me-4-CF_Three
CF_Three   2- (U-3b) -5-OMe cPr 2-Me-4,5-di-CF_Three
CF_Three   2- (U-3b) -5-OCF_Three     cPr 2-Me-4-CF_Three-5-OMe
CF_Three   2-CF₂H-5-F cPr 2-Me-4-OMe-5-F
CF_Three   2-CF₂H-5-Cl cPr 2-Me-4-OMe-5-Cl
CF_Three   2-CF₂H-5-Br cPr 2-Me-4-OMe-5-Br
CF_Three   2-CF₂H-5-Me cPr 2,5-di-Me-4-OMe
CF_Three   2-CF₂H-5-CF_Three        cPr 2-Me-4-OMe-5-CF_Three
CF_Three   2-CF₂H-5-OMe cPr 2-Me-4,5-di-OMe
CF_Three   2-CF₂H-5-OCF_Three       cPr 3-Me-4,5-di-F
CF_Three   2-CN-5-F cPr 3-Me-4-F-5-Cl
CF_Three   2-CN-5-Cl cPr 3-Me-4-F-5-Br
CF_Three   2-CN-5-Br cPr 3,5-di-Me-4-F
CF_Three   2-CN-5-Me cPr 3-Me-4-F-5-CF_Three
CF_Three   2-CN-5-CF_Three          cPr 3-Me-4-F-5-OMe
CF_Three   2-CN-5-OMe cPr 3-Me-4-Cl-5-F
CF_Three   2-CN-5-OCF_Three         cPr 3-Me-4,5-di-Cl
CF_Three   2-Et-5-F cPr 3-Me-4-Cl-5-Br
CF_Three   2-Et-5-Cl cPr 3,5-di-Me-4-Cl
CF_Three   2-Et-5-Br cPr 3-Me-4-Cl-5-CF_Three
CF_Three   2-Et-5-Me cPr 3-Me-4-Cl-5-OMe
CF_Three   2-Et-5-CF_Three          cPr 3-Me-4-Br-5-F
CF_Three   2-Et-5-OMe cPr 3-Me-4-Br-5-Cl
CF_Three   2-Et-5-OCF_Three         cPr 3-Me-4,5-di-Br
CF_Three   2-OCF₂H-5-F cPr 3,5-di-Me-4-Br
CF_Three   2-OCF₂H-5-Cl cPr 3-Me-4-Br-5-CF_Three
CF_Three   2-OCF₂H-5-Br cPr 3-Me-4-Br-5-OMe
CF_Three   2-OCF₂H-5-Me cPr 3,4-di-Me-5-F
CF_Three   2-OCF₂H-5-CF_Three       cPr 3,4-di-Me-5-Cl
CF_Three   2-OCF₂H-5-OMe cPr 3,4-di-Me-5-Br
CF_Three   2-OCF₂H-5-OCF_Three      cPr 3,4,5-tri-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
CF_Three   2-OEt-5-F cPr 3,4-di-Me-5-CF_Three
CF_Three   2-OEt-5-Cl cPr 3,4-di-Me-5-OMe
CF_Three   2-OEt-5-Br cPr 3-Me-4-CF_Three-5-F
CF_Three   2-OEt-5-Me cPr 3-Me-4-CF_Three-5-Cl
CF_Three   2-OEt-5-CF_Three         cPr 3-Me-4-CF_Three-5-Br
CF_Three   2-OEt-5-OMe cPr 3,5-di-Me-4-CF_Three
CF_Three   2-OEt-5-OCF_Three        cPr 3-Me-4,5-di-CF_Three
CF_Three   2-C (O) CF_Three-5-F cPr 3-Me-4-CF_Three-5-OMe
CF_Three   2-C (O) CF_Three-5-Cl cPr 3-Me-4-OMe-5-F
CF_Three   2-C (O) CF_Three-5-Br cPr 3-Me-4-OMe-5-Cl
CF_Three   2-C (O) CF_Three-5-Me cPr 3-Me-4-OMe-5-Br
CF_Three   2-C (O) CF_Three-5-CF_Three     cPr 3,5-di-Me-4-OMe
CF_Three   2-C (O) CF_Three-5-OMe cPr 3-Me-4-OMe-5-CF_Three
CF_Three   2-C (O) CF_Three-5-OCF_Three    cPr 3-Me-4,5-di-OMe
CF_Three   3-Ac-4-F cPr 2-CF_Three-3,4-di-F
CF_Three   3-Ac-4-Cl cPr 2-CF_Three-3-F-4-Cl
CF_Three   3-Ac-4-Br cPr 2-CF_Three-3-F-4-Br
CF_Three   3-Ac-4-Me cPr 2-CF_Three-3-F-4-Me
CF_Three   3-Ac-4-CF_Three          cPr 2,4-di-CF_Three-3-F
CF_Three   3-Ac-4-OMe cPr 2-CF_Three-3-F-4-OMe
CF_Three   3-Ac-4-OCF_Three         cPr 2-CF_Three-3-Cl-4-F
CF_Three   3- (U-3b) -4-F cPr 2-CF_Three-3,4-di-Cl
CF_Three   3- (U-3b) -4-Cl cPr 2-CF_Three-3-Cl-4-Br
CF_Three   3- (U-3b) -4-Br cPr 2-CF_Three-3-Cl-4-Me
CF_Three   3- (U-3b) -4-Me cPr 2,4-di-CF_Three-3-Cl
CF_Three   3- (U-3b) -4-CF_Three      cPr 2-CF_Three-3-Cl-4-OMe
CF_Three   3- (U-3b) -4-OMe cPr 2-CF_Three-3-Br-4-F
CF_Three   3- (U-3b) -4-OCF_Three     cPr 2-CF_Three-3-Br-4-Cl
CF_Three   3-CF₂H-4-F cPr 2-CF_Three-3,4-di-Br
CF_Three   3-CF₂H-4-Cl cPr 2-CF_Three-3-Br-4-Me
CF_Three   3-CF₂H-4-Br cPr 2,4-di-CF_Three-3-Br
CF_Three   3-CF₂H-4-Me cPr 2-CF_Three-3-Br-4-OMe
CF_Three   3-CF₂H-4-CF_Three        cPr 2-CF_Three-3-Me-4-F
CF_Three   3-CF₂H-4-OMe cPr 2-CF_Three-3-Me-4-Cl
CF_Three   3-CF₂H-4-OCF_Three       cPr 2-CF_Three-3-Me-4-Br
CF_Three   3-CN-4-F cPr 2-CF_Three-3,4-di-Me
CF_Three   3-CN-4-Cl cPr 2,4-di-CF_Three-3-Me
CF_Three   3-CN-4-Br cPr 2-CF_Three-3-Me-4-OMe
CF_Three   3-CN-4-Me cPr 2,3-di-CF_Three-4-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
CF_Three   3-CN-4-CF_Three          cPr 2,3-di-CF_Three-4-Cl
CF_Three   3-CN-4-OMe cPr 2,3-di-CF_Three-4-Br
CF_Three   3-CN-4-OCF_Three         cPr 2,3-di-CF_Three-4-Me
CF_Three   3-Et-4-F cPr 2,3,4-tri-CF_Three
CF_Three   3-Et-4-Cl cPr 2,3-di-CF_Three-4-OMe
CF_Three   3-Et-4-Br cPr 2-CF_Three-3-OMe-4-F
CF_Three   3-Et-4-Me cPr 2-CF_Three-3-OMe-4-Cl
CF_Three   3-Et-4-CF_Three          cPr 2-CF_Three-3-OMe-4-Br
CF_Three   3-Et-4-OMe cPr 2-CF_Three-3-OMe-4-Me
CF_Three   3-Et-4-OCF_Three         cPr 2,4-di-CF_Three-3-OMe
CF_Three   3-OCF₂H-4-F cPr 2-CF_Three-3,4-di-OMe
CF_Three   3-OCF₂H-4-Cl cPr 2-CF_Three-3,5-di-F
CF_Three   3-OCF₂H-4-Br cPr 2-CF_Three-3-F-5-Cl
CF_Three   3-OCF₂H-4-Me cPr 2-CF_Three-3-F-5-Br
CF_Three   3-OCF₂H-4-CF_Three       cPr 2-CF_Three-3-F-5-Me
CF_Three   3-OCF₂H-4-OMe cPr 2,5-di-CF_Three-3-F
CF_Three   3-OCF₂H-4-OCF_Three      cPr 2-CF_Three-3-F-5-OMe
CF_Three   3-OEt-4-F cPr 2-CF_Three-3-Cl-5-F
CF_Three   3-OEt-4-Cl cPr 2-CF_Three-3,5-di-Cl
CF_Three   3-OEt-4-Br cPr 2-CF_Three-3-Cl-5-Br
CF_Three   3-OEt-4-Me cPr 2-CF_Three-3-Cl-5-Me
CF_Three   3-OEt-4-CF_Three         cPr 2,5-di-CF_Three-3-Cl
CF_Three   3-OEt-4-OMe cPr 2-CF_Three-3-Cl-5-OMe
CF_Three   3-OEt-4-OCF_Three        cPr 2-CF_Three-3-Br-5-F
CF_Three   3-C (O) CF_Three-4-F cPr 2-CF_Three-3-Br-5-Cl
CF_Three   3-C (O) CF_Three-4-Cl cPr 2-CF_Three-3,5-di-Br
CF_Three   3-C (O) CF_Three-4-Br cPr 2-CF_Three-3-Br-5-Me
CF_Three   3-C (O) CF_Three-4-Me cPr 2,5-di-CF_Three-3-Br
CF_Three   3-C (O) CF_Three-4-CF_Three     cPr 2-CF_Three-3-Br-5-OMe
CF_Three   3-C (O) CF_Three-4-OMe cPr 2-CF_Three-3-Me-5-F
CF_Three   3-C (O) CF_Three-4-OCF_Three    cPr 2-CF_Three-3-Me-5-Cl
CF_Three   3-Ac-5-F cPr 2-CF_Three-3-Me-5-Br
CF_Three   3-Ac-5-Cl cPr 2-CF_Three-3,5-di-Me
CF_Three   3-Ac-5-Br cPr 2,5-di-CF_Three-3-Me
CF_Three   3-Ac-5-Me cPr 2-CF_Three-3-Me-5-OMe
CF_Three   3-Ac-5-CF_Three          cPr 2,3-di-CF_Three-5-F
CF_Three   3-Ac-5-OMe cPr 2,3-di-CF_Three-5-Cl
CF_Three   3-Ac-5-OCF_Three         cPr 2,3-di-CF_Three-5-Br
CF_Three   3- (U-3b) -5-F cPr 2,3-di-CF_Three-5-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
CF_Three   3- (U-3b) -5-Cl cPr 2,3,5-tri-CF_Three
CF_Three   3- (U-3b) -5-Br cPr 2,3-di-CF_Three-5-OMe
CF_Three   3- (U-3b) -5-Me cPr 2-CF_Three-3-OMe-5-F
CF_Three   3- (U-3b) -5-CF_Three      cPr 2-CF_Three-3-OMe-5-Cl
CF_Three   3- (U-3b) -5-OMe cPr 2-CF_Three-3-OMe-5-Br
CF_Three   3- (U-3b) -5-OCF_Three     cPr 2-CF_Three-3-OMe-5-Me
CF_Three   3-CF₂H-5-F cPr 2,5-di-CF_Three-3-OMe
CF_Three   3-CF₂H-5-Cl cPr 2-CF_Three-3,5-di-OMe
CF_Three   3-CF₂H-5-Br cPr 2-CF_Three-4,5-di-F
CF_Three   3-CF₂H-5-Me cPr 2-CF_Three-4-F-5-Cl
CF_Three   3-CF₂H-5-CF_Three        cPr 2-CF_Three-4-F-5-Br
CF_Three   3-CF₂H-5-OMe cPr 2-CF_Three-4-F-5-Me
CF_Three   3-CF₂H-5-OCF_Three       cPr 2,5-di-CF_Three-4-F
CF_Three   3-CN-5-F cPr 2-CF_Three-4-F-5-OMe
CF_Three   3-CN-5-Cl cPr 2-CF_Three-4-Cl-5-F
CF_Three   3-CN-5-Br cPr 2-CF_Three-4,5-di-Cl
CF_Three   3-CN-5-Me cPr 2-CF_Three-4-Cl-5-Br
CF_Three   3-CN-5-CF_Three          cPr 2-CF_Three-4-Cl-5-Me
CF_Three   3-CN-5-OMe cPr 2,5-di-CF_Three-4-Cl
CF_Three   3-CN-5-OCF_Three         cPr 2-CF_Three-4-Cl-5-OMe
CF_Three   3-Et-5-F cPr 2-CF_Three-4-Br-5-F
CF_Three   3-Et-5-Cl cPr 2-CF_Three-4-Br-5-Cl
CF_Three  3-Et-5-Br cPr 2-CF_Three-4,5-di-Br
CF_Three   3-Et-5-Me cPr 2-CF_Three-4-Br-5-Me
CF_Three   3-Et-5-CF_Three          cPr 2,5-di-CF_Three-4-Br
CF_Three   3-Et-5-OMe cPr 2-CF_Three-4-Br-5-OMe
CF_Three   3-Et-5-OCF_Three         cPr 2-CF_Three-4-Me-5-F
CF_Three   3-OCF₂H-5-F cPr 2-CF_Three-4-Me-5-Cl
CF_Three   3-OCF₂H-5-Cl cPr 2-CF_Three-4-Me-5-Br
CF_Three   3-OCF₂H-5-Br cPr 2-CF_Three-4,5-di-Me
CF_Three   3-OCF₂H-5-Me cPr 2,5-di-CF_Three-4-Me
CF_Three   3-OCF₂H-5-CF_Three       cPr 2-CF_Three-4-Me-5-OMe
CF_Three   3-OCF₂H-5-OMe cPr 2,4-di-CF_Three-5-F
CF_Three   3-OCF₂H-5-OCF_Three      cPr 2,4-di-CF_Three-5-Cl
CF_Three   3-OEt-5-F cPr 2,4-di-CF_Three-5-Br
CF_Three   3-OEt-5-Cl cPr 2,4-di-CF_Three-5-Me
CF_Three   3-OEt-5-Br cPr 2,4,5-tri-CF_Three
CF_Three   3-OEt-5-Me cPr 2,4-di-CF_Three-5-OMe
CF_Three   3-OEt-5-CF_Three         cPr 2-CF_Three-4-OMe-5-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
CF_Three   3-OEt-5-OMe cPr 2-CF_Three-4-OMe-5-Cl
CF_Three   3-OEt-5-OCF_Three        cPr 2-CF_Three-4-OMe-5-Br
CF_Three   3-C (O) CF_Three-5-F cPr 2-CF_Three-4-OMe-5-Me
CF_Three   3-C (O) CF_Three-5-Cl cPr 2,5-di-CF_Three-4-OMe
CF_Three   3-C (O) CF_Three-5-Br cPr 2-CF_Three-4,5-di-OMe
CF_Three   3-C (O) CF_Three-5-Me cPr 3-CF_Three-4,5-di-F
CF_Three   3-C (O) CF_Three-5-CF_Three     cPr 3-CF_Three-4-F-5-Cl
CF_Three   3-C (O) CF_Three-5-OMe cPr 3-CF_Three-4-F-5-Br
CF_Three   3-C (O) CF_Three-5-OCF_Three    cPr 3-CF_Three-4-F-5-Me
cPr 2-F-3-Ac cPr 3,5-di-CF_Three-4-F
cPr 2-F-3- (U-3b) cPr 3-CF_Three-4-F-5-OMe
cPr 2-F-3-CF₂H cPr 3-CF_Three-4-Cl-5-F
cPr 2-F-3-CN cPr 3-CF_Three-4,5-di-Cl
cPr 2-F-3-Et cPr 3-CF_Three-4-Cl-5-Br
cPr 2-F-3-OCF₂H cPr 3-CF_Three-4-Cl-5-Me
cPr 2-F-3-OEt cPr 3,5-di-CF_Three-4-Cl
cPr 2-F-3-C (O) CF_Three       cPr 3-CF_Three-4-Cl-5-OMe
cPr 2-Cl-3-Ac cPr 3-CF_Three-4-Br-5-F
cPr 2-Cl-3- (U-3b) cPr 3-CF_Three-4-Br-5-Cl
cPr 2-Cl-3-CF₂H cPr 3-CF_Three-4,5-di-Br
cPr 2-Cl-3-CN cPr 3-CF_Three-4-Br-5-Me
cPr 2-Cl-3-Et cPr 3,5-di-CF_Three-4-Br
cPr 2-Cl-3-OCF₂H cPr 3-CF_Three-4-Br-5-OMe
cPr 2-Cl-3-OEt cPr 3-CF_Three-4-Me-5-F
cPr 2-Cl-3-C (O) CF_Three      cPr 3-CF_Three-4-Me-5-Cl
cPr 2-Br-3-Ac cPr 3-CF_Three-4-Me-5-Br
cPr 2-Br-3- (U-3b) cPr 3-CF_Three-4,5-di-Me
cPr 2-Br-3-CF₂H cPr 3,5-di-CF_Three-4-Me
cPr 2-Br-3-CN cPr 3-CF_Three-4-Me-5-OMe
cPr 2-Br-3-Et cPr 3,4-di-CF_Three-5-F
cPr 2-Br-3-OCF₂H cPr 3,4-di-CF_Three-5-Cl
cPr 2-Br-3-OEt cPr 3,4-di-CF_Three-5-Br
cPr 2-Br-3-C (O) CF_Three      cPr 3,4-di-CF_Three-5-Me
cPr 2-Me-3-Ac cPr 3,4,5-tri-CF_Three
cPr 2-Me-3- (U-3b) cPr 3,4-di-CF_Three-5-OMe
cPr 2-Me-3-CF₂H cPr 3-CF_Three-4-OMe-5-F
cPr 2-Me-3-CN cPr 3-CF_Three-4-OMe-5-Cl
cPr 2-Me-3-Et cPr 3-CF_Three-4-OMe-5-Br
cPr 2-Me-3-OCF₂H cPr 3-CF_Three-4-OMe-5-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
cPr 2-Me-3-OEt cPr 3,5-di-CF_Three-4-OMe
cPr 2-Me-3-C (O) CF_Three      cPr 3-CF_Three-4,5-di-OMe
cPr 2-CF_Three-3-Ac cPr 2-OMe-3,4-di-F
cPr 2-CF_Three-3- (U-3b) cPr 2-OMe-3-F-4-Cl
cPr 2-CF_Three-3-CF₂H cPr 2-OMe-3-F-4-Br
cPr 2-CF_Three-3-CN cPr 2-OMe-3-F-4-Me
cPr 2-CF_Three-3-Et cPr 2-OMe-3-F-4-CF_Three
cPr 2-CF_Three-3-OCF₂H cPr 2,4-di-OMe-3-F
cPr 2-CF_Three-3-OEt cPr 2-OMe-3-Cl-4-F
cPr 2-CF_Three-3-C (O) CF_Three     cPr 2-OMe-3,4-di-Cl
cPr 2-OMe-3-Ac cPr 2-OMe-3-Cl-4-Br
cPr 2-OMe-3- (U-3b) cPr 2-OMe-3-Cl-4-Me
cPr 2-OMe-3-CF₂H cPr 2-OMe-3-Cl-4-CF_Three
cPr 2-OMe-3-CN cPr 2,4-di-OMe-3-Cl
cPr 2-OMe-3-Et cPr 2-OMe-3-Br-4-F
cPr 2-OMe-3-OCF₂H cPr 2-OMe-3-Br-4-Cl
cPr 2-OMe-3-OEt cPr 2-OMe-3,4-di-Br
cPr 2-OMe-3-C (O) CF_Three     cPr 2-OMe-3-Br-4-Me
cPr 2-OCF_Three-3-Ac cPr 2-OMe-3-Br-4-CF_Three
cPr 2-OCF_Three-3- (U-3b) cPr 2,4-di-OMe-3-Br
cPr 2-OCF_Three-3-CF₂H cPr 2-OMe-3-Me-4-F
cPr 2-OCF_Three-3-CN cPr 2-OMe-3-Me-4-Cl
cPr 2-OCF_Three-3-Et cPr 2-OMe-3-Me-4-Br
cPr 2-OCF_Three-3-OCF₂H cPr 2-OMe-3,4-di-Me
cPr 2-OCF_Three-3-OEt cPr 2-OMe-3-Me-4-CF_Three
cPr 2-OCF_Three-3-C (O) CF_Three    cPr 2,4-di-OMe-3-Me
cPr 2-F-4-Ac cPr 2-OMe-3-CF_Three-4-F
cPr 2-F-4- (U-3b) cPr 2-OMe-3-CF_Three-4-Cl
cPr 2-F-4-CF₂H cPr 2-OMe-3-CF_Three-4-Br
cPr 2-F-4-CN cPr 2-OMe-3-CF_Three-4-Me
cPr 2-F-4-Et cPr 2-OMe-3,4-di-CF_Three
cPr 2-F-4-OCF₂H cPr 2,4-di-OMe-3-CF_Three
cPr 2-F-4-OEt cPr 2,3-di-OMe-4-F
cPr 2-F-4-C (O) CF_Three       cPr 2,3-di-OMe-4-Cl
cPr 2-Cl-4-Ac cPr 2,3-di-OMe-4-Br
cPr 2-Cl-4- (U-3b) cPr 2,3-di-OMe-4-Me
cPr 2-Cl-4-CF₂H cPr 2,3-di-OMe-4-CF_Three
cPr 2-Cl-4-CN cPr 2,3,4-tri-OMe
cPr 2-Cl-4-Et cPr 2-OMe-3,5-di-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
cPr 2-Cl-4-OCF₂H cPr 2-OMe-3-F-5-Cl
cPr 2-Cl-4-OEt cPr 2-OMe-3-F-5-Br
cPr 2-Cl-4-C (O) CF_Three      cPr 2-OMe-3-F-5-Me
cPr 2-Br-4-Ac cPr 2-OMe-3-F-5-CF_Three
cPr 2-Br-4- (U-3b) cPr 2,5-di-OMe-3-F
cPr 2-Br-4-CF₂H cPr 2-OMe-3-Cl-5-F
cPr 2-Br-4-CN cPr 2-OMe-3,5-di-Cl
cPr 2-Br-4-Et cPr 2-OMe-3-Cl-5-Br
cPr 2-Br-4-OCF₂H cPr 2-OMe-3-Cl-5-Me
cPr 2-Br-4-OEt cPr 2-OMe-3-Cl-5-CF_Three
cPr 2-Br-4-C (O) CF_Three      cPr 2,5-di-OMe-3-Cl
cPr 2-Me-4-Ac cPr 2-OMe-3-Br-5-F
cPr 2-Me-4- (U-3b) cPr 2-OMe-3-Br-5-Cl
cPr 2-Me-4-CF₂H cPr 2-OMe-3,5-di-Br
cPr 2-Me-4-CN cPr 2-OMe-3-Br-5-Me
cPr 2-Me-4-Et cPr 2-OMe-3-Br-5-CF_Three
cPr 2-Me-4-OCF₂H cPr 2,5-di-OMe-3-Br
cPr 2-Me-4-OEt cPr 2-OMe-3-Me-5-F
cPr 2-Me-4-C (O) CF_Three      cPr 2-OMe-3-Me-5-Cl
cPr 2-CF_Three-4-Ac cPr 2-OMe-3-Me-5-Br
cPr 2-CF_Three-4- (U-3b) cPr 2-OMe-3,5-di-Me
cPr 2-CF_Three-4-CF₂H cPr 2-OMe-3-Me-5-CF_Three
cPr 2-CF_Three-4-CN cPr 2,5-di-OMe-3-Me
cPr 2-CF_Three-4-Et cPr 2-OMe-3-CF_Three-5-F
cPr 2-CF_Three-4-OCF₂H cPr 2-OMe-3-CF_Three-5-Cl
cPr 2-CF_Three-4-OEt cPr 2-OMe-3-CF_Three-5-Br
cPr 2-CF_Three-4-C (O) CF_Three     cPr 2-OMe-3-CF_Three-5-Me
cPr 2-OMe-4-Ac cPr 2-OMe-3,5-di-CF_Three
cPr 2-OMe-4- (U-3b) cPr 2,5-di-OMe-3-CF_Three
cPr 2-OMe-4-CF₂H cPr 2,3-di-OMe-5-F
cPr 2-OMe-4-CN cPr 2,3-di-OMe-5-Cl
cPr 2-OMe-4-Et cPr 2,3-di-OMe-5-Br
cPr 2-OMe-4-OCF₂H cPr 2,3-di-OMe-5-Me
cPr 2-OMe-4-OEt cPr 2,3-di-OMe-5-CF_Three
cPr 2-OMe-4-C (O) CF_Three     cPr 2,3,5-tri-OMe
cPr 2-OCF_Three-4-Ac cPr 2-OMe-4,5-di-F
cPr 2-OCF_Three-4- (U-3b) cPr 2-OMe-4-F-5-Cl
cPr 2-OCF_Three-4-CF₂H cPr 2-OMe-4-F-5-Br
cPr 2-OCF_Three-4-CN cPr 2-OMe-4-F-5-Me
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
cPr 2-OCF_Three-4-Et cPr 2-OMe-4-F-5-CF_Three
cPr 2-OCF_Three-4-OCF₂H cPr 2,5-di-OMe-4-F
cPr 2-OCF_Three-4-OEt cPr 2-OMe-4-Cl-5-F
cPr 2-OCF_Three-4-C (O) CF_Three    cPr 2-OMe-4,5-di-Cl
cPr 2-F-5-Ac cPr 2-OMe-4-Cl-5-Br
cPr 2-F-5- (U-3b) cPr 2-OMe-4-Cl-5-Me
cPr 2-F-5-CF₂H cPr 2-OMe-4-Cl-5-CF_Three
cPr 2-F-5-CN cPr 2,5-di-OMe-4-Cl
cPr 2-F-5-Et cPr 2-OMe-4-Br-5-F
cPr 2-F-5-OCF₂H cPr 2-OMe-4-Br-5-Cl
cPr 2-F-5-OEt cPr 2-OMe-4,5-di-Br
cPr 2-F-5-C (O) CF_Three       cPr 2-OMe-4-Br-5-Me
cPr 2-Cl-5-Ac cPr 2-OMe-4-Br-5-CF_Three
cPr 2-Cl-5- (U-3b) cPr 2,5-di-OMe-4-Br
cPr 2-Cl-5-CF₂H cPr 2-OMe-4-Me-5-F
cPr 2-Cl-5-CN cPr 2-OMe-4-Me-5-Cl
cPr 2-Cl-5-Et cPr 2-OMe-4-Me-5-Br
cPr 2-Cl-5-OCF₂H cPr 2-OMe-4,5-di-Me
cPr 2-Cl-5-OEt cPr 2-OMe-4-Me-5-CF_Three
cPr 2-Cl-5-C (O) CF_Three      cPr 2,5-di-OMe-4-Me
cPr 2-Br-5-Ac cPr 2-OMe-4-CF_Three-5-F
cPr 2-Br-5- (U-3b) cPr 2-OMe-4-CF_Three-5-Cl
cPr 2-Br-5-CF₂H cPr 2-OMe-4-CF_Three-5-Br
cPr 2-Br-5-CN cPr 2-OMe-4-CF_Three-5-Me
cPr 2-Br-5-Et cPr 2-OMe-4,5-di-CF_Three
cPr 2-Br-5-OCF₂H cPr 2,5-di-OMe-4-CF_Three
cPr 2-Br-5-OEt cPr 2,4-di-OMe-5-F
cPr 2-Br-5-C (O) CF_Three      cPr 2,4-di-OMe-5-Cl
cPr 2-Me-5-Ac cPr 2,4-di-OMe-5-Br
cPr 2-Me-5- (U-3b) cPr 2,4-di-OMe-5-Me
cPr 2-Me-5-CF₂H cPr 2,4-di-OMe-5-CF_Three
cPr 2-Me-5-CN cPr 2,4,5-tri-OMe
cPr 2-Me-5-Et cPr 3-OMe-4,5-di-F
cPr 2-Me-5-OCF₂H cPr 3-OMe-4-F-5-Cl
cPr 2-Me-5-OEt cPr 3-OMe-4-F-5-Br
cPr 2-Me-5-C (O) CF_Three      cPr 3-OMe-4-F-5-Me
cPr 2-CF_Three-5-Ac cPr 3-OMe-4-F-5-CF_Three
cPr 2-CF_Three-5- (U-3b) cPr 3,5-di-OMe-4-F
cPr 2-CF_Three-5-CF₂H cPr 3-OMe-4-Cl-5-F
----------- -------------
[Table 1] (continued) [Table 1] (continued)
----------- -------------
R^Three     Z R^Three    Z
----------- -------------
cPr 2-CF_Three-5-CN cPr 3-OMe-4,5-di-Cl
cPr 2-CF_Three-5-Et cPr 3-OMe-4-Cl-5-Br
cPr 2-CF_Three-5-OCF₂H cPr 3-OMe-4-Cl-5-Me
cPr 2-CF_Three-5-OEt cPr 3-OMe-4-Cl-5-CF_Three
cPr 2-CF_Three-5-C (O) CF_Three     cPr 3,5-di-OMe-4-Cl
cPr 2-OMe-5-Ac cPr 3-OMe-4-Br-5-F
cPr 2-OMe-5- (U-3b) cPr 3-OMe-4-Br-5-Cl
cPr 2-OMe-5-CF₂H cPr 3-OMe-4,5-di-Br
cPr 2-OMe-5-CN cPr 3-OMe-4-Br-5-Me
cPr 2-OMe-5-Et cPr 3-OMe-4-Br-5-CF_Three
cPr 2-OMe-5-OCF₂H cPr 3,5-di-OMe-4-Br
cPr 2-OMe-5-OEt cPr 3-OMe-4-Me-5-F
cPr 2-OMe-5-C (O) CF_Three     cPr 3-OMe-4-Me-5-Cl
cPr 2-OCF_Three-5-Ac cPr 3-OMe-4-Me-5-Br
cPr 2-OCF_Three-5- (U-3b) cPr 3-OMe-4,5-di-Me
cPr 2-OCF_Three-5-CF₂H cPr 3-OMe-4-Me-5-CF_Three
cPr 2-OCF_Three-5-CN cPr 3,5-di-OMe-4-Me
cPr 2-OCF_Three-5-Et cPr 3-OMe-4-CF_Three-5-F
cPr 2-OCF_Three-5-OCF₂H cPr 3-OMe-4-CF_Three-5-Cl
cPr 2-OCF_Three-5-OEt cPr 3-OMe-4-CF_Three-5-Br
cPr 2-OCF_Three-5-C (O) CF_Three    cPr 3-OMe-4-CF_Three-5-Me
cPr 3-F-4-Ac cPr 3-OMe-4,5-di-CF_Three
cPr 3-F-4- (U-3b) cPr 3,5-di-OMe-4-CF_Three
cPr 3-F-4-CF₂H cPr 3,4-di-OMe-5-F
cPr 3-F-4-CN cPr 3,4-di-OMe-5-Cl
cPr 3-F-4-Et cPr 3,4-di-OMe-5-Br
cPr 3-F-4-OCF₂H cPr 3,4-di-OMe-5-Me
cPr 3-F-4-OEt cPr 3,4-di-OMe-5-CF_Three
cPr 3-F-4-C (O) CF_Three       cPr 3,4,5-tri-OMe
----------- -------------
[Table 2]

［第２表］［第２表］（続き）［第２表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
Me 2-F Et 2-F-3-OCF₃ U-4e 2-F-3-Me
Me 2-Cl Et 2-Cl-3-F U-4e 2-F-3-CF₃
Me 2-Br Et 2,3-di-Cl U-4e 2-F-3-OMe
Me 2-Me Et 2-Cl-3-Br U-4e 2-F-3-OCF₃
Me 2-CF₃ Et 2-Cl-3-Me U-4e 2-Cl-3-F
Me 2-OMe Et 2-Cl-3-CF₃ U-4e 2,3-di-Cl
Me 2-OCF₃ Et 2-Cl-3-OMe U-4e 2-Cl-3-Br
Me 3-F Et 2-Cl-3-OCF₃ U-4e 2-Cl-3-Me
Me 3-Cl Et 2-Br-3-F U-4e 2-Cl-3-CF₃
Me 3-Br Et 2-Br-3-Cl U-4e 2-Cl-3-OMe
Me 3-Me Et 2,3-di-Br U-4e 2-Cl-3-OCF₃
Me 3-CF₃ Et 2-Br-3-Me U-4e 2-Br-3-F
Me 3-OMe Et 2-Br-3-CF₃ U-4e 2-Br-3-Cl
Me 3-OCF₃ Et 2-Br-3-OMe U-4e 2,3-di-Br
Et 2-F Et 2-Br-3-OCF₃ U-4e 2-Br-3-Me
Et 2-Cl Et 2-Me-3-F U-4e 2-Br-3-CF₃
Et 2-Br Et 2-Me-3-Cl U-4e 2-Br-3-OMe
Et 2-Me Et 2-Me-3-Br U-4e 2-Br-3-OCF₃
Et 2-CF₃ Et 2,3-di-Me U-4e 2-Me-3-F
Et 2-OMe Et 2-Me-3-CF₃ U-4e 2-Me-3-Cl
Et 2-OCF₃ Et 2-Me-3-OMe U-4e 2-Me-3-Br
Et 3-F Et 2-Me-3-OCF₃ U-4e 2,3-di-Me
Et 3-Cl Et 2-CF₃-3-F U-4e 2-Me-3-CF₃
Et 3-Br Et 2-CF₃-3-Cl U-4e 2-Me-3-OMe
Et 3-Me Et 2-CF₃-3-Br U-4e 2-Me-3-OCF₃
Et 3-CF₃ Et 2-CF₃-3-Me U-4e 2-CF₃-3-F
Et 3-OMe Et 2,3-di-CF₃ U-4e 2-CF₃-3-Cl
Et 3-OCF₃ Et 2-CF₃-3-OMe U-4e 2-CF₃-3-Br
iPr 2-F Et 2-CF₃-3-OCF₃ U-4e 2-CF₃-3-Me
iPr 2-Cl Et 2-OMe-3-F U-4e 2,3-di-CF₃
iPr 2-Br Et 2-OMe-3-Cl U-4e 2-CF₃-3-OMe
iPr 2-Me Et 2-OMe-3-Br U-4e 2-CF₃-3-OCF₃
iPr 2-CF₃ Et 2-OMe-3-Me U-4e 2-OMe-3-F
iPr 2-OMe Et 2-OMe-3-CF₃ U-4e 2-OMe-3-Cl
iPr 2-OCF₃ Et 2,3-di-OMe U-4e 2-OMe-3-Br
iPr 3-F Et 2-OMe-3-OCF₃ U-4e 2-OMe-3-Me
iPr 3-Cl Et 2-OCF₃-3-F U-4e 2-OMe-3-CF₃
iPr 3-Br Et 2-OCF₃-3-Cl U-4e 2,3-di-OMe
iPr 3-Me Et 2-OCF₃-3-Br U-4e 2-OMe-3-OCF₃
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第２表］（続き）［第２表］（続き）［第２表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
iPr 3-CF₃ Et 2-OCF₃-3-Me U-4e 2-OCF₃-3-F
iPr 3-OMe Et 2-OCF₃-3-CF₃ U-4e 2-OCF₃-3-Cl
iPr 3-OCF₃ Et 2-OCF₃-3-OMe U-4e 2-OCF₃-3-Br
U-4a 2-F Et 2,3-di-OCF₃ U-4e 2-OCF₃-3-Me
U-4a 2-Cl iPr 2,3-di-F U-4e 2-OCF₃-3-CF₃
U-4a 2-Br iPr 2-F-3-Cl U-4e 2-OCF₃-3-OMe
U-4a 2-Me iPr 2-F-3-Br U-4e 2,3-di-OCF₃
U-4a 2-CF₃ iPr 2-F-3-Me U-4f 2,3-di-F
U-4a 2-OMe iPr 2-F-3-CF₃ U-4f 2-F-3-Cl
U-4a 2-OCF₃ iPr 2-F-3-OMe U-4f 2-F-3-Br
U-4a 3-F iPr 2-F-3-OCF₃ U-4f 2-F-3-Me
U-4a 3-Cl iPr 2-Cl-3-F U-4f 2-F-3-CF₃
U-4a 3-Br iPr 2,3-di-Cl U-4f 2-F-3-OMe
U-4a 3-Me iPr 2-Cl-3-Br U-4f 2-F-3-OCF₃
U-4a 3-CF₃ iPr 2-Cl-3-Me U-4f 2-Cl-3-F
U-4a 3-OMe iPr 2-Cl-3-CF₃ U-4f 2,3-di-Cl
U-4a 3-OCF₃ iPr 2-Cl-3-OMe U-4f 2-Cl-3-Br
CF₃ 2-F iPr 2-Cl-3-OCF₃ U-4f 2-Cl-3-Me
CF₃ 2-Cl iPr 2-Br-3-F U-4f 2-Cl-3-CF₃
CF₃ 2-Br iPr 2-Br-3-Cl U-4f 2-Cl-3-OMe
CF₃ 2-Me iPr 2,3-di-Br U-4f 2-Cl-3-OCF₃
CF₃ 2-CF₃ iPr 2-Br-3-Me U-4f 2-Br-3-F
CF₃ 2-OMe iPr 2-Br-3-CF₃ U-4f 2-Br-3-Cl
CF₃ 2-OCF₃ iPr 2-Br-3-OMe U-4f 2,3-di-Br
CF₃ 3-F iPr 2-Br-3-OCF₃ U-4f 2-Br-3-Me
CF₃ 3-Cl iPr 2-Me-3-F U-4f 2-Br-3-CF₃
CF₃ 3-Br iPr 2-Me-3-Cl U-4f 2-Br-3-OMe
CF₃ 3-Me iPr 2-Me-3-Br U-4f 2-Br-3-OCF₃
CF₃ 3-CF₃ iPr 2,3-di-Me U-4f 2-Me-3-F
CF₃ 3-OMe iPr 2-Me-3-CF₃ U-4f 2-Me-3-Cl
CF₃ 3-OCF₃ iPr 2-Me-3-OMe U-4f 2-Me-3-Br
cPr 2-F iPr 2-Me-3-OCF₃ U-4f 2,3-di-Me
cPr 2-Cl iPr 2-CF₃-3-F U-4f 2-Me-3-CF₃
cPr 2-Br iPr 2-CF₃-3-Cl U-4f 2-Me-3-OMe
cPr 2-Me iPr 2-CF₃-3-Br U-4f 2-Me-3-OCF₃
cPr 2-CF₃ iPr 2-CF₃-3-Me U-4f 2-CF₃-3-F
cPr 2-OMe iPr 2,3-di-CF₃ U-4f 2-CF₃-3-Cl
cPr 2-OCF₃ iPr 2-CF₃-3-OMe U-4f 2-CF₃-3-Br
cPr 3-F iPr 2-CF₃-3-OCF₃ U-4f 2-CF₃-3-Me
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第２表］（続き）［第２表］（続き）［第２表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
cPr 3-Cl iPr 2-OMe-3-F U-4f 2,3-di-CF₃
cPr 3-Br iPr 2-OMe-3-Cl U-4f 2-CF₃-3-OMe
cPr 3-Me iPr 2-OMe-3-Br U-4f 2-CF₃-3-OCF₃
cPr 3-CF₃ iPr 2-OMe-3-Me U-4f 2-OMe-3-F
cPr 3-OMe iPr 2-OMe-3-CF₃ U-4f 2-OMe-3-Cl
cPr 3-OCF₃ iPr 2,3-di-OMe U-4f 2-OMe-3-Br
U-4b 2-F iPr 2-OMe-3-OCF₃ U-4f 2-OMe-3-Me
U-4b 2-Cl iPr 2-OCF₃-3-F U-4f 2-OMe-3-CF₃
U-4b 2-Br iPr 2-OCF₃-3-Cl U-4f 2,3-di-OMe
U-4b 2-Me iPr 2-OCF₃-3-Br U-4f 2-OMe-3-OCF₃
U-4b 2-CF₃ iPr 2-OCF₃-3-Me U-4f 2-OCF₃-3-F
U-4b 2-OMe iPr 2-OCF₃-3-CF₃ U-4f 2-OCF₃-3-Cl
U-4b 2-OCF₃ iPr 2-OCF₃-3-OMe U-4f 2-OCF₃-3-Br
U-4b 3-F iPr 2,3-di-OCF₃ U-4f 2-OCF₃-3-Me
U-4b 3-Cl U-4a 2,3-di-F U-4f 2-OCF₃-3-CF₃
U-4b 3-Br U-4a 2-F-3-Cl U-4f 2-OCF₃-3-OMe
U-4b 3-Me U-4a 2-F-3-Br U-4f 2,3-di-OCF₃
U-4b 3-CF₃ U-4a 2-F-3-Me U-4g 2,3-di-F
U-4b 3-OMe U-4a 2-F-3-CF₃ U-4g 2-F-3-Cl
U-4b 3-OCF₃ U-4a 2-F-3-OMe U-4g 2-F-3-Br
U-4c 2-F U-4a 2-F-3-OCF₃ U-4g 2-F-3-Me
U-4c 2-Cl U-4a 2-Cl-3-F U-4g 2-F-3-CF₃
U-4c 2-Br U-4a 2,3-di-Cl U-4g 2-F-3-OMe
U-4c 2-Me U-4a 2-Cl-3-Br U-4g 2-F-3-OCF₃
U-4c 2-CF₃ U-4a 2-Cl-3-Me U-4g 2-Cl-3-F
U-4c 2-OMe U-4a 2-Cl-3-CF₃ U-4g 2,3-di-Cl
U-4c 2-OCF₃ U-4a 2-Cl-3-OMe U-4g 2-Cl-3-Br
U-4c 3-F U-4a 2-Cl-3-OCF₃ U-4g 2-Cl-3-Me
U-4c 3-Cl U-4a 2-Br-3-F U-4g 2-Cl-3-CF₃
U-4c 3-Br U-4a 2-Br-3-Cl U-4g 2-Cl-3-OMe
U-4c 3-Me U-4a 2,3-di-Br U-4g 2-Cl-3-OCF₃
U-4c 3-CF₃ U-4a 2-Br-3-Me U-4g 2-Br-3-F
U-4c 3-OMe U-4a 2-Br-3-CF₃ U-4g 2-Br-3-Cl
U-4c 3-OCF₃ U-4a 2-Br-3-OMe U-4g 2,3-di-Br
U-4d 2-F U-4a 2-Br-3-OCF₃ U-4g 2-Br-3-Me
U-4d 2-Cl U-4a 2-Me-3-F U-4g 2-Br-3-CF₃
U-4d 2-Br U-4a 2-Me-3-Cl U-4g 2-Br-3-OMe
U-4d 2-Me U-4a 2-Me-3-Br U-4g 2-Br-3-OCF₃
U-4d 2-CF₃ U-4a 2,3-di-Me U-4g 2-Me-3-F
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第２表］（続き）［第２表］（続き）［第２表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
U-4d 2-OMe U-4a 2-Me-3-CF₃ U-4g 2-Me-3-Cl
U-4d 2-OCF₃ U-4a 2-Me-3-OMe U-4g 2-Me-3-Br
U-4d 3-F U-4a 2-Me-3-OCF₃ U-4g 2,3-di-Me
U-4d 3-Cl U-4a 2-CF₃-3-F U-4g 2-Me-3-CF₃
U-4d 3-Br U-4a 2-CF₃-3-Cl U-4g 2-Me-3-OMe
U-4d 3-Me U-4a 2-CF₃-3-Br U-4g 2-Me-3-OCF₃
U-4d 3-CF₃ U-4a 2-CF₃-3-Me U-4g 2-CF₃-3-F
U-4d 3-OMe U-4a 2,3-di-CF₃ U-4g 2-CF₃-3-Cl
U-4d 3-OCF₃ U-4a 2-CF₃-3-OMe U-4g 2-CF₃-3-Br
U-4e 2-F U-4a 2-CF₃-3-OCF₃ U-4g 2-CF₃-3-Me
U-4e 2-Cl U-4a 2-OMe-3-F U-4g 2,3-di-CF₃
U-4e 2-Br U-4a 2-OMe-3-Cl U-4g 2-CF₃-3-OMe
U-4e 2-Me U-4a 2-OMe-3-Br U-4g 2-CF₃-3-OCF₃
U-4e 2-CF₃ U-4a 2-OMe-3-Me U-4g 2-OMe-3-F
U-4e 2-OMe U-4a 2-OMe-3-CF₃ U-4g 2-OMe-3-Cl
U-4e 2-OCF₃ U-4a 2,3-di-OMe U-4g 2-OMe-3-Br
U-4e 3-F U-4a 2-OMe-3-OCF₃ U-4g 2-OMe-3-Me
U-4e 3-Cl U-4a 2-OCF₃-3-F U-4g 2-OMe-3-CF₃
U-4e 3-Br U-4a 2-OCF₃-3-Cl U-4g 2,3-di-OMe
U-4e 3-Me U-4a 2-OCF₃-3-Br U-4g 2-OMe-3-OCF₃
U-4e 3-CF₃ U-4a 2-OCF₃-3-Me U-4g 2-OCF₃-3-F
U-4e 3-OMe U-4a 2-OCF₃-3-CF₃ U-4g 2-OCF₃-3-Cl
U-4e 3-OCF₃ U-4a 2-OCF₃-3-OMe U-4g 2-OCF₃-3-Br
U-4f 2-F U-4a 2,3-di-OCF₃ U-4g 2-OCF₃-3-Me
U-4f 2-Cl CF₃ 2,3-di-F U-4g 2-OCF₃-3-CF₃
U-4f 2-Br CF₃ 2-F-3-Cl U-4g 2-OCF₃-3-OMe
U-4f 2-Me CF₃ 2-F-3-Br U-4g 2,3-di-OCF₃
U-4f 2-CF₃ CF₃ 2-F-3-Me OMe 2,3-di-F
U-4f 2-OMe CF₃ 2-F-3-CF₃ OMe 2-F-3-Cl
U-4f 2-OCF₃ CF₃ 2-F-3-OMe OMe 2-F-3-Br
U-4f 3-F CF₃ 2-F-3-OCF₃ OMe 2-F-3-Me
U-4f 3-Cl CF₃ 2-Cl-3-F OMe 2-F-3-CF₃
U-4f 3-Br CF₃ 2,3-di-Cl OMe 2-F-3-OMe
U-4f 3-Me CF₃ 2-Cl-3-Br OMe 2-F-3-OCF₃
U-4f 3-CF₃ CF₃ 2-Cl-3-Me OMe 2-Cl-3-F
U-4f 3-OMe CF₃ 2-Cl-3-CF₃ OMe 2,3-di-Cl
U-4f 3-OCF₃ CF₃ 2-Cl-3-OMe OMe 2-Cl-3-Br
U-4g 2-F CF₃ 2-Cl-3-OCF₃ OMe 2-Cl-3-Me
U-4g 2-Cl CF₃ 2-Br-3-F OMe 2-Cl-3-CF₃
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第２表］（続き）［第２表］（続き）［第２表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
U-4g 2-Br CF₃ 2-Br-3-Cl OMe 2-Cl-3-OMe
U-4g 2-Me CF₃ 2,3-di-Br OMe 2-Cl-3-OCF₃
U-4g 2-CF₃ CF₃ 2-Br-3-Me OMe 2-Br-3-F
U-4g 2-OMe CF₃ 2-Br-3-CF₃ OMe 2-Br-3-Cl
U-4g 2-OCF₃ CF₃ 2-Br-3-OMe OMe 2,3-di-Br
U-4g 3-F CF₃ 2-Br-3-OCF₃ OMe 2-Br-3-Me
U-4g 3-Cl CF₃ 2-Me-3-F OMe 2-Br-3-CF₃
U-4g 3-Br CF₃ 2-Me-3-Cl OMe 2-Br-3-OMe
U-4g 3-Me CF₃ 2-Me-3-Br OMe 2-Br-3-OCF₃
U-4g 3-CF₃ CF₃ 2,3-di-Me OMe 2-Me-3-F
U-4g 3-OMe CF₃ 2-Me-3-CF₃ OMe 2-Me-3-Cl
U-4g 3-OCF₃ CF₃ 2-Me-3-OMe OMe 2-Me-3-Br
OMe 2-F CF₃ 2-Me-3-OCF₃ OMe 2,3-di-Me
OMe 2-Cl CF₃ 2-CF₃-3-F OMe 2-Me-3-CF₃
OMe 2-Br CF₃ 2-CF₃-3-Cl OMe 2-Me-3-OMe
OMe 2-Me CF₃ 2-CF₃-3-Br OMe 2-Me-3-OCF₃
OMe 2-CF₃ CF₃ 2-CF₃-3-Me OMe 2-CF₃-3-F
OMe 2-OMe CF₃ 2,3-di-CF₃ OMe 2-CF₃-3-Cl
OMe 2-OCF₃ CF₃ 2-CF₃-3-OMe OMe 2-CF₃-3-Br
OMe 3-F CF₃ 2-CF₃-3-OCF₃ OMe 2-CF₃-3-Me
OMe 3-Cl CF₃ 2-OMe-3-F OMe 2,3-di-CF₃
OMe 3-Br CF₃ 2-OMe-3-Cl OMe 2-CF₃-3-OMe
OMe 3-Me CF₃ 2-OMe-3-Br OMe 2-CF₃-3-OCF₃
OMe 3-CF₃ CF₃ 2-OMe-3-Me OMe 2-OMe-3-F
OMe 3-OMe CF₃ 2-OMe-3-CF₃ OMe 2-OMe-3-Cl
OMe 3-OCF₃ CF₃ 2,3-di-OMe OMe 2-OMe-3-Br
SMe 2-F CF₃ 2-OMe-3-OCF₃ OMe 2-OMe-3-Me
SMe 2-Cl CF₃ 2-OCF₃-3-F OMe 2-OMe-3-CF₃
SMe 2-Br CF₃ 2-OCF₃-3-Cl OMe 2,3-di-OMe
SMe 2-Me CF₃ 2-OCF₃-3-Br OMe 2-OMe-3-OCF₃
SMe 2-CF₃ CF₃ 2-OCF₃-3-Me OMe 2-OCF₃-3-F
SMe 2-OMe CF₃ 2-OCF₃-3-CF₃ OMe 2-OCF₃-3-Cl
SMe 2-OCF₃ CF₃ 2-OCF₃-3-OMe OMe 2-OCF₃-3-Br
SMe 3-F CF₃ 2,3-di-OCF₃ OMe 2-OCF₃-3-Me
SMe 3-Cl cPr 2,3-di-F OMe 2-OCF₃-3-CF₃
SMe 3-Br cPr 2-F-3-Cl OMe 2-OCF₃-3-OMe
SMe 3-Me cPr 2-F-3-Br OMe 2,3-di-OCF₃
SMe 3-CF₃ cPr 2-F-3-Me SMe 2,3-di-F
SMe 3-OMe cPr 2-F-3-CF₃ SMe 2-F-3-Cl
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第２表］（続き）［第２表］（続き）［第２表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
SMe 3-OCF₃ cPr 2-F-3-OMe SMe 2-F-3-Br
Ac 2-F cPr 2-F-3-OCF₃ SMe 2-F-3-Me
Ac 2-Cl cPr 2-Cl-3-F SMe 2-F-3-CF₃
Ac 2-Br cPr 2,3-di-Cl SMe 2-F-3-OMe
Ac 2-Me cPr 2-Cl-3-Br SMe 2-F-3-OCF₃
Ac 2-CF₃ cPr 2-Cl-3-Me SMe 2-Cl-3-F
Ac 2-OMe cPr 2-Cl-3-CF₃ SMe 2,3-di-Cl
Ac 2-OCF₃ cPr 2-Cl-3-OMe SMe 2-Cl-3-Br
Ac 3-F cPr 2-Cl-3-OCF₃ SMe 2-Cl-3-Me
Ac 3-Cl cPr 2-Br-3-F SMe 2-Cl-3-CF₃
Ac 3-Br cPr 2-Br-3-Cl SMe 2-Cl-3-OMe
Ac 3-Me cPr 2,3-di-Br SMe 2-Cl-3-OCF₃
Ac 3-CF₃ cPr 2-Br-3-Me SMe 2-Br-3-F
Ac 3-OMe cPr 2-Br-3-CF₃ SMe 2-Br-3-Cl
Ac 3-OCF₃ cPr 2-Br-3-OMe SMe 2,3-di-Br
cPen 2-F cPr 2-Br-3-OCF₃ SMe 2-Br-3-Me
cPen 2-Cl cPr 2-Me-3-F SMe 2-Br-3-CF₃
cPen 2-Br cPr 2-Me-3-Cl SMe 2-Br-3-OMe
cPen 2-Me cPr 2-Me-3-Br SMe 2-Br-3-OCF₃
cPen 2-CF₃ cPr 2,3-di-Me SMe 2-Me-3-F
cPen 2-OMe cPr 2-Me-3-CF₃ SMe 2-Me-3-Cl
cPen 2-OCF₃ cPr 2-Me-3-OMe SMe 2-Me-3-Br
cPen 3-F cPr 2-Me-3-OCF₃ SMe 2,3-di-Me
cPen 3-Cl cPr 2-CF₃-3-F SMe 2-Me-3-CF₃
cPen 3-Br cPr 2-CF₃-3-Cl SMe 2-Me-3-OMe
cPen 3-Me cPr 2-CF₃-3-Br SMe 2-Me-3-OCF₃
cPen 3-CF₃ cPr 2-CF₃-3-Me SMe 2-CF₃-3-F
cPen 3-OMe cPr 2,3-di-CF₃ SMe 2-CF₃-3-Cl
cPen 3-OCF₃ cPr 2-CF₃-3-OMe SMe 2-CF₃-3-Br
U-1e 2-F cPr 2-CF₃-3-OCF₃ SMe 2-CF₃-3-Me
U-1e 2-Cl cPr 2-OMe-3-F SMe 2,3-di-CF₃
U-1e 2-Br cPr 2-OMe-3-Cl SMe 2-CF₃-3-OMe
U-1e 2-Me cPr 2-OMe-3-Br SMe 2-CF₃-3-OCF₃
U-1e 2-CF₃ cPr 2-OMe-3-Me SMe 2-OMe-3-F
U-1e 2-OMe cPr 2-OMe-3-CF₃ SMe 2-OMe-3-Cl
U-1e 2-OCF₃ cPr 2,3-di-OMe SMe 2-OMe-3-Br
U-1e 3-F cPr 2-OMe-3-OCF₃ SMe 2-OMe-3-Me
U-1e 3-Cl cPr 2-OCF₃-3-F SMe 2-OMe-3-CF₃
U-1e 3-Br cPr 2-OCF₃-3-Cl SMe 2,3-di-OMe
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第２表］（続き）［第２表］（続き）［第２表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
U-1e 3-Me cPr 2-OCF₃-3-Br SMe 2-OMe-3-OCF₃
U-1e 3-CF₃ cPr 2-OCF₃-3-Me SMe 2-OCF₃-3-F
U-1e 3-OMe cPr 2-OCF₃-3-CF₃ SMe 2-OCF₃-3-Cl
U-1e 3-OCF₃ cPr 2-OCF₃-3-OMe SMe 2-OCF₃-3-Br
Me 2-Ac cPr 2,3-di-OCF₃ SMe 2-OCF₃-3-Me
Me 2-(U-3b) U-4b 2,3-di-F SMe 2-OCF₃-3-CF₃
Me 2-CF₂H U-4b 2-F-3-Cl SMe 2-OCF₃-3-OMe
Me 2-CN U-4b 2-F-3-Br SMe 2,3-di-OCF₃
Me 2-Et U-4b 2-F-3-Me Ac 2,3-di-F
Me 2-OCF₂H U-4b 2-F-3-CF₃ Ac 2-F-3-Cl
Me 2-OEt U-4b 2-F-3-OMe Ac 2-F-3-Br
Me 2-C(O)CF₃ U-4b 2-F-3-OCF₃ Ac 2-F-3-Me
Me 3-Ac U-4b 2-Cl-3-F Ac 2-F-3-CF₃
Me 3-(U-3b) U-4b 2,3-di-Cl Ac 2-F-3-OMe
Me 3-CF₂H U-4b 2-Cl-3-Br Ac 2-F-3-OCF₃
Me 3-CN U-4b 2-Cl-3-Me Ac 2-Cl-3-F
Me 3-Et U-4b 2-Cl-3-CF₃ Ac 2,3-di-Cl
Me 3-OCF₂H U-4b 2-Cl-3-OMe Ac 2-Cl-3-Br
Me 3-OEt U-4b 2-Cl-3-OCF₃ Ac 2-Cl-3-Me
Me 3-C(O)CF₃ U-4b 2-Br-3-F Ac 2-Cl-3-CF₃
Et 2-Ac U-4b 2-Br-3-Cl Ac 2-Cl-3-OMe
Et 2-(U-3b) U-4b 2,3-di-Br Ac 2-Cl-3-OCF₃
Et 2-CF₂H U-4b 2-Br-3-Me Ac 2-Br-3-F
Et 2-CN U-4b 2-Br-3-CF₃ Ac 2-Br-3-Cl
Et 2-Et U-4b 2-Br-3-OMe Ac 2,3-di-Br
Et 2-OCF₂H U-4b 2-Br-3-OCF₃ Ac 2-Br-3-Me
Et 2-OEt U-4b 2-Me-3-F Ac 2-Br-3-CF₃
Et 2-C(O)CF₃ U-4b 2-Me-3-Cl Ac 2-Br-3-OMe
Et 3-Ac U-4b 2-Me-3-Br Ac 2-Br-3-OCF₃
Et 3-(U-3b) U-4b 2,3-di-Me Ac 2-Me-3-F
Et 3-CF₂H U-4b 2-Me-3-CF₃ Ac 2-Me-3-Cl
Et 3-CN U-4b 2-Me-3-OMe Ac 2-Me-3-Br
Et 3-Et U-4b 2-Me-3-OCF₃ Ac 2,3-di-Me
Et 3-OCF₂H U-4b 2-CF₃-3-F Ac 2-Me-3-CF₃
Et 3-OEt U-4b 2-CF₃-3-Cl Ac 2-Me-3-OMe
Et 3-C(O)CF₃ U-4b 2-CF₃-3-Br Ac 2-Me-3-OCF₃
iPr 2-Ac U-4b 2-CF₃-3-Me Ac 2-CF₃-3-F
iPr 2-(U-3b) U-4b 2,3-di-CF₃ Ac 2-CF₃-3-Cl
iPr 2-CF₂H U-4b 2-CF₃-3-OMe Ac 2-CF₃-3-Br
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第２表］（続き）［第２表］（続き）［第２表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
iPr 2-CN U-4b 2-CF₃-3-OCF₃ Ac 2-CF₃-3-Me
iPr 2-Et U-4b 2-OMe-3-F Ac 2,3-di-CF₃
iPr 2-OCF₂H U-4b 2-OMe-3-Cl Ac 2-CF₃-3-OMe
iPr 2-OEt U-4b 2-OMe-3-Br Ac 2-CF₃-3-OCF₃
iPr 2-C(O)CF₃ U-4b 2-OMe-3-Me Ac 2-OMe-3-F
iPr 3-Ac U-4b 2-OMe-3-CF₃ Ac 2-OMe-3-Cl
iPr 3-(U-3b) U-4b 2,3-di-OMe Ac 2-OMe-3-Br
iPr 3-CF₂H U-4b 2-OMe-3-OCF₃ Ac 2-OMe-3-Me
iPr 3-CN U-4b 2-OCF₃-3-F Ac 2-OMe-3-CF₃
iPr 3-Et U-4b 2-OCF₃-3-Cl Ac 2,3-di-OMe
iPr 3-OCF₂H U-4b 2-OCF₃-3-Br Ac 2-OMe-3-OCF₃
iPr 3-OEt U-4b 2-OCF₃-3-Me Ac 2-OCF₃-3-F
iPr 3-C(O)CF₃ U-4b 2-OCF₃-3-CF₃ Ac 2-OCF₃-3-Cl
U-4a 2-Ac U-4b 2-OCF₃-3-OMe Ac 2-OCF₃-3-Br
U-4a 2-(U-3b) U-4b 2,3-di-OCF₃ Ac 2-OCF₃-3-Me
U-4a 2-CF₂H U-4c 2,3-di-F Ac 2-OCF₃-3-CF₃
U-4a 2-CN U-4c 2-F-3-Cl Ac 2-OCF₃-3-OMe
U-4a 2-Et U-4c 2-F-3-Br Ac 2,3-di-OCF₃
U-4a 2-OCF₂H U-4c 2-F-3-Me cPen 2,3-di-F
U-4a 2-OEt U-4c 2-F-3-CF₃ cPen 2-F-3-Cl
U-4a 2-C(O)CF₃ U-4c 2-F-3-OMe cPen 2-F-3-Br
U-4a 3-Ac U-4c 2-F-3-OCF₃ cPen 2-F-3-Me
U-4a 3-(U-3b) U-4c 2-Cl-3-F cPen 2-F-3-CF₃
U-4a 3-CF₂H U-4c 2,3-di-Cl cPen 2-F-3-OMe
U-4a 3-CN U-4c 2-Cl-3-Br cPen 2-F-3-OCF₃
U-4a 3-Et U-4c 2-Cl-3-Me cPen 2-Cl-3-F
U-4a 3-OCF₂H U-4c 2-Cl-3-CF₃ cPen 2,3-di-Cl
U-4a 3-OEt U-4c 2-Cl-3-OMe cPen 2-Cl-3-Br
U-4a 3-C(O)CF₃ U-4c 2-Cl-3-OCF₃ cPen 2-Cl-3-Me
CF₃ 2-Ac U-4c 2-Br-3-F cPen 2-Cl-3-CF₃
CF₃ 2-(U-3b) U-4c 2-Br-3-Cl cPen 2-Cl-3-OMe
CF₃ 2-CF₂H U-4c 2,3-di-Br cPen 2-Cl-3-OCF₃
CF₃ 2-CN U-4c 2-Br-3-Me cPen 2-Br-3-F
CF₃ 2-Et U-4c 2-Br-3-CF₃ cPen 2-Br-3-Cl
CF₃ 2-OCF₂H U-4c 2-Br-3-OMe cPen 2,3-di-Br
CF₃ 2-OEt U-4c 2-Br-3-OCF₃ cPen 2-Br-3-Me
CF₃ 2-C(O)CF₃ U-4c 2-Me-3-F cPen 2-Br-3-CF₃
CF₃ 3-Ac U-4c 2-Me-3-Cl cPen 2-Br-3-OMe
CF₃ 3-(U-3b) U-4c 2-Me-3-Br cPen 2-Br-3-OCF₃
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第２表］（続き）［第２表］（続き）［第２表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
CF₃ 3-CF₂H U-4c 2,3-di-Me cPen 2-Me-3-F
CF₃ 3-CN U-4c 2-Me-3-CF₃ cPen 2-Me-3-Cl
CF₃ 3-Et U-4c 2-Me-3-OMe cPen 2-Me-3-Br
CF₃ 3-OCF₂H U-4c 2-Me-3-OCF₃ cPen 2,3-di-Me
CF₃ 3-OEt U-4c 2-CF₃-3-F cPen 2-Me-3-CF₃
CF₃ 3-C(O)CF₃ U-4c 2-CF₃-3-Cl cPen 2-Me-3-OMe
cPr 2-Ac U-4c 2-CF₃-3-Br cPen 2-Me-3-OCF₃
cPr 2-(U-3b) U-4c 2-CF₃-3-Me cPen 2-CF₃-3-F
cPr 2-CF₂H U-4c 2,3-di-CF₃ cPen 2-CF₃-3-Cl
cPr 2-CN U-4c 2-CF₃-3-OMe cPen 2-CF₃-3-Br
cPr 2-Et U-4c 2-CF₃-3-OCF₃ cPen 2-CF₃-3-Me
cPr 2-OCF₂H U-4c 2-OMe-3-F cPen 2,3-di-CF₃
cPr 2-OEt U-4c 2-OMe-3-Cl cPen 2-CF₃-3-OMe
cPr 2-C(O)CF₃ U-4c 2-OMe-3-Br cPen 2-CF₃-3-OCF₃
cPr 3-Ac U-4c 2-OMe-3-Me cPen 2-OMe-3-F
cPr 3-(U-3b) U-4c 2-OMe-3-CF₃ cPen 2-OMe-3-Cl
cPr 3-CF₂H U-4c 2,3-di-OMe cPen 2-OMe-3-Br
cPr 3-CN U-4c 2-OMe-3-OCF₃ cPen 2-OMe-3-Me
cPr 3-Et U-4c 2-OCF₃-3-F cPen 2-OMe-3-CF₃
cPr 3-OCF₂H U-4c 2-OCF₃-3-Cl cPen 2,3-di-OMe
cPr 3-OEt U-4c 2-OCF₃-3-Br cPen 2-OMe-3-OCF₃
cPr 3-C(O)CF₃ U-4c 2-OCF₃-3-Me cPen 2-OCF₃-3-F
Me 2,3-di-F U-4c 2-OCF₃-3-CF₃ cPen 2-OCF₃-3-Cl
Me 2-F-3-Cl U-4c 2-OCF₃-3-OMe cPen 2-OCF₃-3-Br
Me 2-F-3-Br U-4c 2,3-di-OCF₃ cPen 2-OCF₃-3-Me
Me 2-F-3-Me U-4d 2,3-di-F cPen 2-OCF₃-3-CF₃
Me 2-F-3-CF₃ U-4d 2-F-3-Cl cPen 2-OCF₃-3-OMe
Me 2-F-3-OMe U-4d 2-F-3-Br cPen 2,3-di-OCF₃
Me 2-F-3-OCF₃ U-4d 2-F-3-Me U-1e 2,3-di-F
Me 2-Cl-3-F U-4d 2-F-3-CF₃ U-1e 2-F-3-Cl
Me 2,3-di-Cl U-4d 2-F-3-OMe U-1e 2-F-3-Br
Me 2-Cl-3-Br U-4d 2-F-3-OCF₃ U-1e 2-F-3-Me
Me 2-Cl-3-Me U-4d 2-Cl-3-F U-1e 2-F-3-CF₃
Me 2-Cl-3-CF₃ U-4d 2,3-di-Cl U-1e 2-F-3-OMe
Me 2-Cl-3-OMe U-4d 2-Cl-3-Br U-1e 2-F-3-OCF₃
Me 2-Cl-3-OCF₃ U-4d 2-Cl-3-Me U-1e 2-Cl-3-F
Me 2-Br-3-F U-4d 2-Cl-3-CF₃ U-1e 2,3-di-Cl
Me 2-Br-3-Cl U-4d 2-Cl-3-OMe U-1e 2-Cl-3-Br
Me 2,3-di-Br U-4d 2-Cl-3-OCF₃ U-1e 2-Cl-3-Me
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第２表］（続き）［第２表］（続き）［第２表］（続き）
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
Me 2-Br-3-Me U-4d 2-Br-3-F U-1e 2-Cl-3-CF₃
Me 2-Br-3-CF₃ U-4d 2-Br-3-Cl U-1e 2-Cl-3-OMe
Me 2-Br-3-OMe U-4d 2,3-di-Br U-1e 2-Cl-3-OCF₃
Me 2-Br-3-OCF₃ U-4d 2-Br-3-Me U-1e 2-Br-3-F
Me 2-Me-3-F U-4d 2-Br-3-CF₃ U-1e 2-Br-3-Cl
Me 2-Me-3-Cl U-4d 2-Br-3-OMe U-1e 2,3-di-Br
Me 2-Me-3-Br U-4d 2-Br-3-OCF₃ U-1e 2-Br-3-Me
Me 2,3-di-Me U-4d 2-Me-3-F U-1e 2-Br-3-CF₃
Me 2-Me-3-CF₃ U-4d 2-Me-3-Cl U-1e 2-Br-3-OMe
Me 2-Me-3-OMe U-4d 2-Me-3-Br U-1e 2-Br-3-OCF₃
Me 2-Me-3-OCF₃ U-4d 2,3-di-Me U-1e 2-Me-3-F
Me 2-CF₃-3-F U-4d 2-Me-3-CF₃ U-1e 2-Me-3-Cl
Me 2-CF₃-3-Cl U-4d 2-Me-3-OMe U-1e 2-Me-3-Br
Me 2-CF₃-3-Br U-4d 2-Me-3-OCF₃ U-1e 2,3-di-Me
Me 2-CF₃-3-Me U-4d 2-CF₃-3-F U-1e 2-Me-3-CF₃
Me 2,3-di-CF₃ U-4d 2-CF₃-3-Cl U-1e 2-Me-3-OMe
Me 2-CF₃-3-OMe U-4d 2-CF₃-3-Br U-1e 2-Me-3-OCF₃
Me 2-CF₃-3-OCF₃ U-4d 2-CF₃-3-Me U-1e 2-CF₃-3-F
Me 2-OMe-3-F U-4d 2,3-di-CF₃ U-1e 2-CF₃-3-Cl
Me 2-OMe-3-Cl U-4d 2-CF₃-3-OMe U-1e 2-CF₃-3-Br
Me 2-OMe-3-Br U-4d 2-CF₃-3-OCF₃ U-1e 2-CF₃-3-Me
Me 2-OMe-3-Me U-4d 2-OMe-3-F U-1e 2,3-di-CF₃
Me 2-OMe-3-CF₃ U-4d 2-OMe-3-Cl U-1e 2-CF₃-3-OMe
Me 2,3-di-OMe U-4d 2-OMe-3-Br U-1e 2-CF₃-3-OCF₃
Me 2-OMe-3-OCF₃ U-4d 2-OMe-3-Me U-1e 2-OMe-3-F
Me 2-OCF₃-3-F U-4d 2-OMe-3-CF₃ U-1e 2-OMe-3-Cl
Me 2-OCF₃-3-Cl U-4d 2,3-di-OMe U-1e 2-OMe-3-Br
Me 2-OCF₃-3-Br U-4d 2-OMe-3-OCF₃ U-1e 2-OMe-3-Me
Me 2-OCF₃-3-Me U-4d 2-OCF₃-3-F U-1e 2-OMe-3-CF₃
Me 2-OCF₃-3-CF₃ U-4d 2-OCF₃-3-Cl U-1e 2,3-di-OMe
Me 2-OCF₃-3-OMe U-4d 2-OCF₃-3-Br U-1e 2-OMe-3-OCF₃
Me 2,3-di-OCF₃ U-4d 2-OCF₃-3-Me U-1e 2-OCF₃-3-F
Et 2,3-di-F U-4d 2-OCF₃-3-CF₃ U-1e 2-OCF₃-3-Cl
Et 2-F-3-Cl U-4d 2-OCF₃-3-OMe U-1e 2-OCF₃-3-Br
Et 2-F-3-Br U-4d 2,3-di-OCF₃ U-1e 2-OCF₃-3-Me
Et 2-F-3-Me U-4e 2,3-di-F U-1e 2-OCF₃-3-CF₃
Et 2-F-3-CF₃ U-4e 2-F-3-Cl U-1e 2-OCF₃-3-OMe
Et 2-F-3-OMe U-4e 2-F-3-Br U-1e 2,3-di-OCF₃
−−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第２表］（続き）［第２表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−−
Me 2-F-3-Ac U-4a 2-F-3-Ac
Me 2-F-3-(U-3b) U-4a 2-F-3-(U-3b)
Me 2-F-3-CF₂H U-4a 2-F-3-CF₂H
Me 2-F-3-CN U-4a 2-F-3-CN
Me 2-F-3-Et U-4a 2-F-3-Et
Me 2-F-3-OCF₂H U-4a 2-F-3-OCF₂H
Me 2-F-3-OEt U-4a 2-F-3-OEt
Me 2-F-3-C(O)CF₃ U-4a 2-F-3-C(O)CF₃
Me 2-Cl-3-Ac U-4a 2-Cl-3-Ac
Me 2-Cl-3-(U-3b) U-4a 2-Cl-3-(U-3b)
Me 2-Cl-3-CF₂H U-4a 2-Cl-3-CF₂H
Me 2-Cl-3-CN U-4a 2-Cl-3-CN
Me 2-Cl-3-Et U-4a 2-Cl-3-Et
Me 2-Cl-3-OCF₂H U-4a 2-Cl-3-OCF₂H
Me 2-Cl-3-OEt U-4a 2-Cl-3-OEt
Me 2-Cl-3-C(O)CF₃ U-4a 2-Cl-3-C(O)CF₃
Me 2-Br-3-Ac U-4a 2-Br-3-Ac
Me 2-Br-3-(U-3b) U-4a 2-Br-3-(U-3b)
Me 2-Br-3-CF₂H U-4a 2-Br-3-CF₂H
Me 2-Br-3-CN U-4a 2-Br-3-CN
Me 2-Br-3-Et U-4a 2-Br-3-Et
Me 2-Br-3-OCF₂H U-4a 2-Br-3-OCF₂H
Me 2-Br-3-OEt U-4a 2-Br-3-OEt
Me 2-Br-3-C(O)CF₃ U-4a 2-Br-3-C(O)CF₃
Me 2-Me-3-Ac U-4a 2-Me-3-Ac
Me 2-Me-3-(U-3b) U-4a 2-Me-3-(U-3b)
Me 2-Me-3-CF₂H U-4a 2-Me-3-CF₂H
Me 2-Me-3-CN U-4a 2-Me-3-CN
Me 2-Me-3-Et U-4a 2-Me-3-Et
Me 2-Me-3-OCF₂H U-4a 2-Me-3-OCF₂H
Me 2-Me-3-OEt U-4a 2-Me-3-OEt
Me 2-Me-3-C(O)CF₃ U-4a 2-Me-3-C(O)CF₃
Me 2-CF₃-3-Ac U-4a 2-CF₃-3-Ac
Me 2-CF₃-3-(U-3b) U-4a 2-CF₃-3-(U-3b)
Me 2-CF₃-3-CF₂H U-4a 2-CF₃-3-CF₂H
Me 2-CF₃-3-CN U-4a 2-CF₃-3-CN
Me 2-CF₃-3-Et U-4a 2-CF₃-3-Et
Me 2-CF₃-3-OCF₂H U-4a 2-CF₃-3-OCF₂H
Me 2-CF₃-3-OEt U-4a 2-CF₃-3-OEt
−−−−−−−−−−− −−−−−−−−−−−−−−
［第２表］（続き）［第２表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−−
Me 2-CF₃-3-C(O)CF₃ U-4a 2-CF₃-3-C(O)CF₃
Me 2-OMe-3-Ac U-4a 2-OMe-3-Ac
Me 2-OMe-3-(U-3b) U-4a 2-OMe-3-(U-3b)
Me 2-OMe-3-CF₂H U-4a 2-OMe-3-CF₂H
Me 2-OMe-3-CN U-4a 2-OMe-3-CN
Me 2-OMe-3-Et U-4a 2-OMe-3-Et
Me 2-OMe-3-OCF₂H U-4a 2-OMe-3-OCF₂H
Me 2-OMe-3-OEt U-4a 2-OMe-3-OEt
Me 2-OMe-3-C(O)CF₃ U-4a 2-OMe-3-C(O)CF₃
Me 2-OCF₃-3-Ac U-4a 2-OCF₃-3-Ac
Me 2-OCF₃-3-(U-3b) U-4a 2-OCF₃-3-(U-3b)
Me 2-OCF₃-3-CF₂H U-4a 2-OCF₃-3-CF₂H
Me 2-OCF₃-3-CN U-4a 2-OCF₃-3-CN
Me 2-OCF₃-3-Et U-4a 2-OCF₃-3-Et
Me 2-OCF₃-3-OCF₂H U-4a 2-OCF₃-3-OCF₂H
Me 2-OCF₃-3-OEt U-4a 2-OCF₃-3-OEt
Me 2-OCF₃-3-C(O)CF₃ U-4a 2-OCF₃-3-C(O)CF₃
Me 2-Ac-3-F U-4a 2-Ac-3-F
Me 2-Ac-3-Cl U-4a 2-Ac-3-Cl
Me 2-Ac-3-Br U-4a 2-Ac-3-Br
Me 2-Ac-3-Me U-4a 2-Ac-3-Me
Me 2-Ac-3-CF₃ U-4a 2-Ac-3-CF₃
Me 2-Ac-3-OMe U-4a 2-Ac-3-OMe
Me 2-Ac-3-OCF₃ U-4a 2-Ac-3-OCF₃
Me 2-(U-3b)-3-F U-4a 2-(U-3b)-3-F
Me 2-(U-3b)-3-Cl U-4a 2-(U-3b)-3-Cl
Me 2-(U-3b)-3-Br U-4a 2-(U-3b)-3-Br
Me 2-(U-3b)-3-Me U-4a 2-(U-3b)-3-Me
Me 2-(U-3b)-3-CF₃ U-4a 2-(U-3b)-3-CF₃
Me 2-(U-3b)-3-OMe U-4a 2-(U-3b)-3-OMe
Me 2-(U-3b)-3-OCF₃ U-4a 2-(U-3b)-3-OCF₃
Me 2-CF₂H-3-F U-4a 2-CF₂H-3-F
Me 2-CF₂H-3-Cl U-4a 2-CF₂H-3-Cl
Me 2-CF₂H-3-Br U-4a 2-CF₂H-3-Br
Me 2-CF₂H-3-Me U-4a 2-CF₂H-3-Me
Me 2-CF₂H-3-CF₃ U-4a 2-CF₂H-3-CF₃
Me 2-CF₂H-3-OMe U-4a 2-CF₂H-3-OMe
Me 2-CF₂H-3-OCF₃ U-4a 2-CF₂H-3-OCF₃
Me 2-CN-3-F U-4a 2-CN-3-F
−−−−−−−−−−− −−−−−−−−−−−−−−
［第２表］（続き）［第２表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−−
Me 2-CN-3-Cl U-4a 2-CN-3-Cl
Me 2-CN-3-Br U-4a 2-CN-3-Br
Me 2-CN-3-Me U-4a 2-CN-3-Me
Me 2-CN-3-CF₃ U-4a 2-CN-3-CF₃
Me 2-CN-3-OMe U-4a 2-CN-3-OMe
Me 2-CN-3-OCF₃ U-4a 2-CN-3-OCF₃
Me 2-Et-3-F U-4a 2-Et-3-F
Me 2-Et-3-Cl U-4a 2-Et-3-Cl
Me 2-Et-3-Br U-4a 2-Et-3-Br
Me 2-Et-3-Me U-4a 2-Et-3-Me
Me 2-Et-3-CF₃ U-4a 2-Et-3-CF₃
Me 2-Et-3-OMe U-4a 2-Et-3-OMe
Me 2-Et-3-OCF₃ U-4a 2-Et-3-OCF₃
Me 2-OCF₂H-3-F U-4a 2-OCF₂H-3-F
Me 2-OCF₂H-3-Cl U-4a 2-OCF₂H-3-Cl
Me 2-OCF₂H-3-Br U-4a 2-OCF₂H-3-Br
Me 2-OCF₂H-3-Me U-4a 2-OCF₂H-3-Me
Me 2-OCF₂H-3-CF₃ U-4a 2-OCF₂H-3-CF₃
Me 2-OCF₂H-3-OMe U-4a 2-OCF₂H-3-OMe
Me 2-OCF₂H-3-OCF₃ U-4a 2-OCF₂H-3-OCF₃
Me 2-OEt-3-F U-4a 2-OEt-3-F
Me 2-OEt-3-Cl U-4a 2-OEt-3-Cl
Me 2-OEt-3-Br U-4a 2-OEt-3-Br
Me 2-OEt-3-Me U-4a 2-OEt-3-Me
Me 2-OEt-3-CF₃ U-4a 2-OEt-3-CF₃
Me 2-OEt-3-OMe U-4a 2-OEt-3-OMe
Me 2-OEt-3-OCF₃ U-4a 2-OEt-3-OCF₃
Me 2-C(O)CF₃-3-F U-4a 2-C(O)CF₃-3-F
Me 2-C(O)CF₃-3-Cl U-4a 2-C(O)CF₃-3-Cl
Me 2-C(O)CF₃-3-Br U-4a 2-C(O)CF₃-3-Br
Me 2-C(O)CF₃-3-Me U-4a 2-C(O)CF₃-3-Me
Me 2-C(O)CF₃-3-CF₃ U-4a 2-C(O)CF₃-3-CF₃
Me 2-C(O)CF₃-3-OMe U-4a 2-C(O)CF₃-3-OMe
Me 2-C(O)CF₃-3-OCF₃ U-4a 2-C(O)CF₃-3-OCF₃
Et 2-F-3-Ac CF₃ 2-F-3-Ac
Et 2-F-3-(U-3b) CF₃ 2-F-3-(U-3b)
Et 2-F-3-CF₂H CF₃ 2-F-3-CF₂H
Et 2-F-3-CN CF₃ 2-F-3-CN
Et 2-F-3-Et CF₃ 2-F-3-Et
−−−−−−−−−−− −−−−−−−−−−−−−−
［第２表］（続き）［第２表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−−
Et 2-F-3-OCF₂H CF₃ 2-F-3-OCF₂H
Et 2-F-3-OEt CF₃ 2-F-3-OEt
Et 2-F-3-C(O)CF₃ CF₃ 2-F-3-C(O)CF₃
Et 2-Cl-3-Ac CF₃ 2-Cl-3-Ac
Et 2-Cl-3-(U-3b) CF₃ 2-Cl-3-(U-3b)
Et 2-Cl-3-CF₂H CF₃ 2-Cl-3-CF₂H
Et 2-Cl-3-CN CF₃ 2-Cl-3-CN
Et 2-Cl-3-Et CF₃ 2-Cl-3-Et
Et 2-Cl-3-OCF₂H CF₃ 2-Cl-3-OCF₂H
Et 2-Cl-3-OEt CF₃ 2-Cl-3-OEt
Et 2-Cl-3-C(O)CF₃ CF₃ 2-Cl-3-C(O)CF₃
Et 2-Br-3-Ac CF₃ 2-Br-3-Ac
Et 2-Br-3-(U-3b) CF₃ 2-Br-3-(U-3b)
Et 2-Br-3-CF₂H CF₃ 2-Br-3-CF₂H
Et 2-Br-3-CN CF₃ 2-Br-3-CN
Et 2-Br-3-Et CF₃ 2-Br-3-Et
Et 2-Br-3-OCF₂H CF₃ 2-Br-3-OCF₂H
Et 2-Br-3-OEt CF₃ 2-Br-3-OEt
Et 2-Br-3-C(O)CF₃ CF₃ 2-Br-3-C(O)CF₃
Et 2-Me-3-Ac CF₃ 2-Me-3-Ac
Et 2-Me-3-(U-3b) CF₃ 2-Me-3-(U-3b)
Et 2-Me-3-CF₂H CF₃ 2-Me-3-CF₂H
Et 2-Me-3-CN CF₃ 2-Me-3-CN
Et 2-Me-3-Et CF₃ 2-Me-3-Et
Et 2-Me-3-OCF₂H CF₃ 2-Me-3-OCF₂H
Et 2-Me-3-OEt CF₃ 2-Me-3-OEt
Et 2-Me-3-C(O)CF₃ CF₃ 2-Me-3-C(O)CF₃
Et 2-CF₃-3-Ac CF₃ 2-CF₃-3-Ac
Et 2-CF₃-3-(U-3b) CF₃ 2-CF₃-3-(U-3b)
Et 2-CF₃-3-CF₂H CF₃ 2-CF₃-3-CF₂H
Et 2-CF₃-3-CN CF₃ 2-CF₃-3-CN
Et 2-CF₃-3-Et CF₃ 2-CF₃-3-Et
Et 2-CF₃-3-OCF₂H CF₃ 2-CF₃-3-OCF₂H
Et 2-CF₃-3-OEt CF₃ 2-CF₃-3-OEt
Et 2-CF₃-3-C(O)CF₃ CF₃ 2-CF₃-3-C(O)CF₃
Et 2-OMe-3-Ac CF₃ 2-OMe-3-Ac
Et 2-OMe-3-(U-3b) CF₃ 2-OMe-3-(U-3b)
Et 2-OMe-3-CF₂H CF₃ 2-OMe-3-CF₂H
Et 2-OMe-3-CN CF₃ 2-OMe-3-CN
−−−−−−−−−−− −−−−−−−−−−−−−−
［第２表］（続き）［第２表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−−
Et 2-OMe-3-Et CF₃ 2-OMe-3-Et
Et 2-OMe-3-OCF₂H CF₃ 2-OMe-3-OCF₂H
Et 2-OMe-3-OEt CF₃ 2-OMe-3-OEt
Et 2-OMe-3-C(O)CF₃ CF₃ 2-OMe-3-C(O)CF₃
Et 2-OCF₃-3-Ac CF₃ 2-OCF₃-3-Ac
Et 2-OCF₃-3-(U-3b) CF₃ 2-OCF₃-3-(U-3b)
Et 2-OCF₃-3-CF₂H CF₃ 2-OCF₃-3-CF₂H
Et 2-OCF₃-3-CN CF₃ 2-OCF₃-3-CN
Et 2-OCF₃-3-Et CF₃ 2-OCF₃-3-Et
Et 2-OCF₃-3-OCF₂H CF₃ 2-OCF₃-3-OCF₂H
Et 2-OCF₃-3-OEt CF₃ 2-OCF₃-3-OEt
Et 2-OCF₃-3-C(O)CF₃ CF₃ 2-OCF₃-3-C(O)CF₃
Et 2-Ac-3-F CF₃ 2-Ac-3-F
Et 2-Ac-3-Cl CF₃ 2-Ac-3-Cl
Et 2-Ac-3-Br CF₃ 2-Ac-3-Br
Et 2-Ac-3-Me CF₃ 2-Ac-3-Me
Et 2-Ac-3-CF₃ CF₃ 2-Ac-3-CF₃
Et 2-Ac-3-OMe CF₃ 2-Ac-3-OMe
Et 2-Ac-3-OCF₃ CF₃ 2-Ac-3-OCF₃
Et 2-(U-3b)-3-F CF₃ 2-(U-3b)-3-F
Et 2-(U-3b)-3-Cl CF₃ 2-(U-3b)-3-Cl
Et 2-(U-3b)-3-Br CF₃ 2-(U-3b)-3-Br
Et 2-(U-3b)-3-Me CF₃ 2-(U-3b)-3-Me
Et 2-(U-3b)-3-CF₃ CF₃ 2-(U-3b)-3-CF₃
Et 2-(U-3b)-3-OMe CF₃ 2-(U-3b)-3-OMe
Et 2-(U-3b)-3-OCF₃ CF₃ 2-(U-3b)-3-OCF₃
Et 2-CF₂H-3-F CF₃ 2-CF₂H-3-F
Et 2-CF₂H-3-Cl CF₃ 2-CF₂H-3-Cl
Et 2-CF₂H-3-Br CF₃ 2-CF₂H-3-Br
Et 2-CF₂H-3-Me CF₃ 2-CF₂H-3-Me
Et 2-CF₂H-3-CF₃ CF₃ 2-CF₂H-3-CF₃
Et 2-CF₂H-3-OMe CF₃ 2-CF₂H-3-OMe
Et 2-CF₂H-3-OCF₃ CF₃ 2-CF₂H-3-OCF₃
Et 2-CN-3-F CF₃ 2-CN-3-F
Et 2-CN-3-Cl CF₃ 2-CN-3-Cl
Et 2-CN-3-Br CF₃ 2-CN-3-Br
Et 2-CN-3-Me CF₃ 2-CN-3-Me
Et 2-CN-3-CF₃ CF₃ 2-CN-3-CF₃
Et 2-CN-3-OMe CF₃ 2-CN-3-OMe
−−−−−−−−−−− −−−−−−−−−−−−−−
［第２表］（続き）［第２表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−−
Et 2-CN-3-OCF₃ CF₃ 2-CN-3-OCF₃
Et 2-Et-3-F CF₃ 2-Et-3-F
Et 2-Et-3-Cl CF₃ 2-Et-3-Cl
Et 2-Et-3-Br CF₃ 2-Et-3-Br
Et 2-Et-3-Me CF₃ 2-Et-3-Me
Et 2-Et-3-CF₃ CF₃ 2-Et-3-CF₃
Et 2-Et-3-OMe CF₃ 2-Et-3-OMe
Et 2-Et-3-OCF₃ CF₃ 2-Et-3-OCF₃
Et 2-OCF₂H-3-F CF₃ 2-OCF₂H-3-F
Et 2-OCF₂H-3-Cl CF₃ 2-OCF₂H-3-Cl
Et 2-OCF₂H-3-Br CF₃ 2-OCF₂H-3-Br
Et 2-OCF₂H-3-Me CF₃ 2-OCF₂H-3-Me
Et 2-OCF₂H-3-CF₃ CF₃ 2-OCF₂H-3-CF₃
Et 2-OCF₂H-3-OMe CF₃ 2-OCF₂H-3-OMe
Et 2-OCF₂H-3-OCF₃ CF₃ 2-OCF₂H-3-OCF₃
Et 2-OEt-3-F CF₃ 2-OEt-3-F
Et 2-OEt-3-Cl CF₃ 2-OEt-3-Cl
Et 2-OEt-3-Br CF₃ 2-OEt-3-Br
Et 2-OEt-3-Me CF₃ 2-OEt-3-Me
Et 2-OEt-3-CF₃ CF₃ 2-OEt-3-CF₃
Et 2-OEt-3-OMe CF₃ 2-OEt-3-OMe
Et 2-OEt-3-OCF₃ CF₃ 2-OEt-3-OCF₃
Et 2-C(O)CF₃-3-F CF₃ 2-C(O)CF₃-3-F
Et 2-C(O)CF₃-3-Cl CF₃ 2-C(O)CF₃-3-Cl
Et 2-C(O)CF₃-3-Br CF₃ 2-C(O)CF₃-3-Br
Et 2-C(O)CF₃-3-Me CF₃ 2-C(O)CF₃-3-Me
Et 2-C(O)CF₃-3-CF₃ CF₃ 2-C(O)CF₃-3-CF₃
Et 2-C(O)CF₃-3-OMe CF₃ 2-C(O)CF₃-3-OMe
Et 2-C(O)CF₃-3-OCF₃ CF₃ 2-C(O)CF₃-3-OCF₃
iPr 2-F-3-Ac cPr 2-F-3-Ac
iPr 2-F-3-(U-3b) cPr 2-F-3-(U-3b)
iPr 2-F-3-CF₂H cPr 2-F-3-CF₂H
iPr 2-F-3-CN cPr 2-F-3-CN
iPr 2-F-3-Et cPr 2-F-3-Et
iPr 2-F-3-OCF₂H cPr 2-F-3-OCF₂H
iPr 2-F-3-OEt cPr 2-F-3-OEt
iPr 2-F-3-C(O)CF₃ cPr 2-F-3-C(O)CF₃
iPr 2-Cl-3-Ac cPr 2-Cl-3-Ac
iPr 2-Cl-3-(U-3b) cPr 2-Cl-3-(U-3b)
−−−−−−−−−−− −−−−−−−−−−−−−−
［第２表］（続き）［第２表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−−
iPr 2-Cl-3-CF₂H cPr 2-Cl-3-CF₂H
iPr 2-Cl-3-CN cPr 2-Cl-3-CN
iPr 2-Cl-3-Et cPr 2-Cl-3-Et
iPr 2-Cl-3-OCF₂H cPr 2-Cl-3-OCF₂H
iPr 2-Cl-3-OEt cPr 2-Cl-3-OEt
iPr 2-Cl-3-C(O)CF₃ cPr 2-Cl-3-C(O)CF₃
iPr 2-Br-3-Ac cPr 2-Br-3-Ac
iPr 2-Br-3-(U-3b) cPr 2-Br-3-(U-3b)
iPr 2-Br-3-CF₂H cPr 2-Br-3-CF₂H
iPr 2-Br-3-CN cPr 2-Br-3-CN
iPr 2-Br-3-Et cPr 2-Br-3-Et
iPr 2-Br-3-OCF₂H cPr 2-Br-3-OCF₂H
iPr 2-Br-3-OEt cPr 2-Br-3-OEt
iPr 2-Br-3-C(O)CF₃ cPr 2-Br-3-C(O)CF₃
iPr 2-Me-3-Ac cPr 2-Me-3-Ac
iPr 2-Me-3-(U-3b) cPr 2-Me-3-(U-3b)
iPr 2-Me-3-CF₂H cPr 2-Me-3-CF₂H
iPr 2-Me-3-CN cPr 2-Me-3-CN
iPr 2-Me-3-Et cPr 2-Me-3-Et
iPr 2-Me-3-OCF₂H cPr 2-Me-3-OCF₂H
iPr 2-Me-3-OEt cPr 2-Me-3-OEt
iPr 2-Me-3-C(O)CF₃ cPr 2-Me-3-C(O)CF₃
iPr 2-CF₃-3-Ac cPr 2-CF₃-3-Ac
iPr 2-CF₃-3-(U-3b) cPr 2-CF₃-3-(U-3b)
iPr 2-CF₃-3-CF₂H cPr 2-CF₃-3-CF₂H
iPr 2-CF₃-3-CN cPr 2-CF₃-3-CN
iPr 2-CF₃-3-Et cPr 2-CF₃-3-Et
iPr 2-CF₃-3-OCF₂H cPr 2-CF₃-3-OCF₂H
iPr 2-CF₃-3-OEt cPr 2-CF₃-3-OEt
iPr 2-CF₃-3-C(O)CF₃ cPr 2-CF₃-3-C(O)CF₃
iPr 2-OMe-3-Ac cPr 2-OMe-3-Ac
iPr 2-OMe-3-(U-3b) cPr 2-OMe-3-(U-3b)
iPr 2-OMe-3-CF₂H cPr 2-OMe-3-CF₂H
iPr 2-OMe-3-CN cPr 2-OMe-3-CN
iPr 2-OMe-3-Et cPr 2-OMe-3-Et
iPr 2-OMe-3-OCF₂H cPr 2-OMe-3-OCF₂H
iPr 2-OMe-3-OEt cPr 2-OMe-3-OEt
iPr 2-OMe-3-C(O)CF₃ cPr 2-OMe-3-C(O)CF₃
iPr 2-OCF₃-3-Ac cPr 2-OCF₃-3-Ac
−−−−−−−−−−− −−−−−−−−−−−−−−
［第２表］（続き）［第２表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−−
iPr 2-OCF₃-3-(U-3b) cPr 2-OCF₃-3-(U-3b)
iPr 2-OCF₃-3-CF₂H cPr 2-OCF₃-3-CF₂H
iPr 2-OCF₃-3-CN cPr 2-OCF₃-3-CN
iPr 2-OCF₃-3-Et cPr 2-OCF₃-3-Et
iPr 2-OCF₃-3-OCF₂H cPr 2-OCF₃-3-OCF₂H
iPr 2-OCF₃-3-OEt cPr 2-OCF₃-3-OEt
iPr 2-OCF₃-3-C(O)CF₃ cPr 2-OCF₃-3-C(O)CF₃
iPr 2-Ac-3-F cPr 2-Ac-3-F
iPr 2-Ac-3-Cl cPr 2-Ac-3-Cl
iPr 2-Ac-3-Br cPr 2-Ac-3-Br
iPr 2-Ac-3-Me cPr 2-Ac-3-Me
iPr 2-Ac-3-CF₃ cPr 2-Ac-3-CF₃
iPr 2-Ac-3-OMe cPr 2-Ac-3-OMe
iPr 2-Ac-3-OCF₃ cPr 2-Ac-3-OCF₃
iPr 2-(U-3b)-3-F cPr 2-(U-3b)-3-F
iPr 2-(U-3b)-3-Cl cPr 2-(U-3b)-3-Cl
iPr 2-(U-3b)-3-Br cPr 2-(U-3b)-3-Br
iPr 2-(U-3b)-3-Me cPr 2-(U-3b)-3-Me
iPr 2-(U-3b)-3-CF₃ cPr 2-(U-3b)-3-CF₃
iPr 2-(U-3b)-3-OMe cPr 2-(U-3b)-3-OMe
iPr 2-(U-3b)-3-OCF₃ cPr 2-(U-3b)-3-OCF₃
iPr 2-CF₂H-3-F cPr 2-CF₂H-3-F
iPr 2-CF₂H-3-Cl cPr 2-CF₂H-3-Cl
iPr 2-CF₂H-3-Br cPr 2-CF₂H-3-Br
iPr 2-CF₂H-3-Me cPr 2-CF₂H-3-Me
iPr 2-CF₂H-3-CF₃ cPr 2-CF₂H-3-CF₃
iPr 2-CF₂H-3-OMe cPr 2-CF₂H-3-OMe
iPr 2-CF₂H-3-OCF₃ cPr 2-CF₂H-3-OCF₃
iPr 2-CN-3-F cPr 2-CN-3-F
iPr 2-CN-3-Cl cPr 2-CN-3-Cl
iPr 2-CN-3-Br cPr 2-CN-3-Br
iPr 2-CN-3-Me cPr 2-CN-3-Me
iPr 2-CN-3-CF₃ cPr 2-CN-3-CF₃
iPr 2-CN-3-OMe cPr 2-CN-3-OMe
iPr 2-CN-3-OCF₃ cPr 2-CN-3-OCF₃
iPr 2-Et-3-F cPr 2-Et-3-F
iPr 2-Et-3-Cl cPr 2-Et-3-Cl
iPr 2-Et-3-Br cPr 2-Et-3-Br
iPr 2-Et-3-Me cPr 2-Et-3-Me
−−−−−−−−−−− −−−−−−−−−−−−−−
［第２表］（続き）［第２表］（続き）
−−−−−−−−−−− −−−−−−−−−−−−−−
R³ Z R³ Z
−−−−−−−−−−− −−−−−−−−−−−−−−
iPr 2-Et-3-CF₃ cPr 2-Et-3-CF₃
iPr 2-Et-3-OMe cPr 2-Et-3-OMe
iPr 2-Et-3-OCF₃ cPr 2-Et-3-OCF₃
iPr 2-OCF₂H-3-F cPr 2-OCF₂H-3-F
iPr 2-OCF₂H-3-Cl cPr 2-OCF₂H-3-Cl
iPr 2-OCF₂H-3-Br cPr 2-OCF₂H-3-Br
iPr 2-OCF₂H-3-Me cPr 2-OCF₂H-3-Me
iPr 2-OCF₂H-3-CF₃ cPr 2-OCF₂H-3-CF₃
iPr 2-OCF₂H-3-OMe cPr 2-OCF₂H-3-OMe
iPr 2-OCF₂H-3-OCF₃ cPr 2-OCF₂H-3-OCF₃
iPr 2-OEt-3-F cPr 2-OEt-3-F
iPr 2-OEt-3-Cl cPr 2-OEt-3-Cl
iPr 2-OEt-3-Br cPr 2-OEt-3-Br
iPr 2-OEt-3-Me cPr 2-OEt-3-Me
iPr 2-OEt-3-CF₃ cPr 2-OEt-3-CF₃
iPr 2-OEt-3-OMe cPr 2-OEt-3-OMe
iPr 2-OEt-3-OCF₃ cPr 2-OEt-3-OCF₃
iPr 2-C(O)CF₃-3-F cPr 2-C(O)CF₃-3-F
iPr 2-C(O)CF₃-3-Cl cPr 2-C(O)CF₃-3-Cl
iPr 2-C(O)CF₃-3-Br cPr 2-C(O)CF₃-3-Br
iPr 2-C(O)CF₃-3-Me cPr 2-C(O)CF₃-3-Me
iPr 2-C(O)CF₃-3-CF₃ cPr 2-C(O)CF₃-3-CF₃
iPr 2-C(O)CF₃-3-OMe cPr 2-C(O)CF₃-3-OMe
iPr 2-C(O)CF₃-3-OCF₃ cPr 2-C(O)CF₃-3-OCF₃
−−−−−−−−−−− −−−−−−−−−−−−−−
［第３表］ [Table 2] [Table 2] (continued) [Table 2] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
Me 2-F Et 2-F-3-OCF_Three     U-4e 2-F-3-Me
Me 2-Cl Et 2-Cl-3-F U-4e 2-F-3-CF_Three
Me 2-Br Et 2,3-di-Cl U-4e 2-F-3-OMe
Me 2-Me Et 2-Cl-3-Br U-4e 2-F-3-OCF_Three
Me 2-CF_Three          Et 2-Cl-3-Me U-4e 2-Cl-3-F
Me 2-OMe Et 2-Cl-3-CF_Three     U-4e 2,3-di-Cl
Me 2-OCF_Three         Et 2-Cl-3-OMe U-4e 2-Cl-3-Br
Me 3-F Et 2-Cl-3-OCF_Three    U-4e 2-Cl-3-Me
Me 3-Cl Et 2-Br-3-F U-4e 2-Cl-3-CF_Three
Me 3-Br Et 2-Br-3-Cl U-4e 2-Cl-3-OMe
Me 3-Me Et 2,3-di-Br U-4e 2-Cl-3-OCF_Three
Me 3-CF_Three          Et 2-Br-3-Me U-4e 2-Br-3-F
Me 3-OMe Et 2-Br-3-CF_Three     U-4e 2-Br-3-Cl
Me 3-OCF_Three         Et 2-Br-3-OMe U-4e 2,3-di-Br
Et 2-F Et 2-Br-3-OCF_Three    U-4e 2-Br-3-Me
Et 2-Cl Et 2-Me-3-F U-4e 2-Br-3-CF_Three
Et 2-Br Et 2-Me-3-Cl U-4e 2-Br-3-OMe
Et 2-Me Et 2-Me-3-Br U-4e 2-Br-3-OCF_Three
Et 2-CF_Three          Et 2,3-di-Me U-4e 2-Me-3-F
Et 2-OMe Et 2-Me-3-CF_Three     U-4e 2-Me-3-Cl
Et 2-OCF_Three         Et 2-Me-3-OMe U-4e 2-Me-3-Br
Et 3-F Et 2-Me-3-OCF_Three    U-4e 2,3-di-Me
Et 3-Cl Et 2-CF_Three-3-F U-4e 2-Me-3-CF_Three
Et 3-Br Et 2-CF_Three-3-Cl U-4e 2-Me-3-OMe
Et 3-Me Et 2-CF_Three-3-Br U-4e 2-Me-3-OCF_Three
Et 3-CF_Three          Et 2-CF_Three-3-Me U-4e 2-CF_Three-3-F
Et 3-OMe Et 2,3-di-CF_Three     U-4e 2-CF_Three-3-Cl
Et 3-OCF_Three         Et 2-CF_Three-3-OMe U-4e 2-CF_Three-3-Br
iPr 2-F Et 2-CF_Three-3-OCF_Three   U-4e 2-CF_Three-3-Me
iPr 2-Cl Et 2-OMe-3-F U-4e 2,3-di-CF_Three
iPr 2-Br Et 2-OMe-3-Cl U-4e 2-CF_Three-3-OMe
iPr 2-Me Et 2-OMe-3-Br U-4e 2-CF_Three-3-OCF_Three
iPr 2-CF_Three          Et 2-OMe-3-Me U-4e 2-OMe-3-F
iPr 2-OMe Et 2-OMe-3-CF_Three    U-4e 2-OMe-3-Cl
iPr 2-OCF_Three         Et 2,3-di-OMe U-4e 2-OMe-3-Br
iPr 3-F Et 2-OMe-3-OCF_Three   U-4e 2-OMe-3-Me
iPr 3-Cl Et 2-OCF_Three-3-F U-4e 2-OMe-3-CF_Three
iPr 3-Br Et 2-OCF_Three-3-Cl U-4e 2,3-di-OMe
iPr 3-Me Et 2-OCF_Three-3-Br U-4e 2-OMe-3-OCF_Three
--------- --------- ------------
[Table 2] (continued) [Table 2] (continued) [Table 2] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
iPr 3-CF_Three          Et 2-OCF_Three-3-Me U-4e 2-OCF_Three-3-F
iPr 3-OMe Et 2-OCF_Three-3-CF_Three   U-4e 2-OCF_Three-3-Cl
iPr 3-OCF_Three         Et 2-OCF_Three-3-OMe U-4e 2-OCF_Three-3-Br
U-4a 2-F Et 2,3-di-OCF_Three    U-4e 2-OCF_Three-3-Me
U-4a 2-Cl iPr 2,3-di-F U-4e 2-OCF_Three-3-CF_Three
U-4a 2-Br iPr 2-F-3-Cl U-4e 2-OCF_Three-3-OMe
U-4a 2-Me iPr 2-F-3-Br U-4e 2,3-di-OCF_Three
U-4a 2-CF_Three          iPr 2-F-3-Me U-4f 2,3-di-F
U-4a 2-OMe iPr 2-F-3-CF_Three      U-4f 2-F-3-Cl
U-4a 2-OCF_Three         iPr 2-F-3-OMe U-4f 2-F-3-Br
U-4a 3-F iPr 2-F-3-OCF_Three     U-4f 2-F-3-Me
U-4a 3-Cl iPr 2-Cl-3-F U-4f 2-F-3-CF_Three
U-4a 3-Br iPr 2,3-di-Cl U-4f 2-F-3-OMe
U-4a 3-Me iPr 2-Cl-3-Br U-4f 2-F-3-OCF_Three
U-4a 3-CF_Three          iPr 2-Cl-3-Me U-4f 2-Cl-3-F
U-4a 3-OMe iPr 2-Cl-3-CF_Three     U-4f 2,3-di-Cl
U-4a 3-OCF_Three         iPr 2-Cl-3-OMe U-4f 2-Cl-3-Br
CF_Three   2-F iPr 2-Cl-3-OCF_Three    U-4f 2-Cl-3-Me
CF_Three   2-Cl iPr 2-Br-3-F U-4f 2-Cl-3-CF_Three
CF_Three   2-Br iPr 2-Br-3-Cl U-4f 2-Cl-3-OMe
CF_Three   2-Me iPr 2,3-di-Br U-4f 2-Cl-3-OCF_Three
CF_Three   2-CF_Three          iPr 2-Br-3-Me U-4f 2-Br-3-F
CF_Three   2-OMe iPr 2-Br-3-CF_Three     U-4f 2-Br-3-Cl
CF_Three   2-OCF_Three         iPr 2-Br-3-OMe U-4f 2,3-di-Br
CF_Three   3-F iPr 2-Br-3-OCF_Three    U-4f 2-Br-3-Me
CF_Three   3-Cl iPr 2-Me-3-F U-4f 2-Br-3-CF_Three
CF_Three   3-Br iPr 2-Me-3-Cl U-4f 2-Br-3-OMe
CF_Three   3-Me iPr 2-Me-3-Br U-4f 2-Br-3-OCF_Three
CF_Three   3-CF_Three          iPr 2,3-di-Me U-4f 2-Me-3-F
CF_Three   3-OMe iPr 2-Me-3-CF_Three     U-4f 2-Me-3-Cl
CF_Three   3-OCF_Three         iPr 2-Me-3-OMe U-4f 2-Me-3-Br
cPr 2-F iPr 2-Me-3-OCF_Three    U-4f 2,3-di-Me
cPr 2-Cl iPr 2-CF_Three-3-F U-4f 2-Me-3-CF_Three
cPr 2-Br iPr 2-CF_Three-3-Cl U-4f 2-Me-3-OMe
cPr 2-Me iPr 2-CF_Three-3-Br U-4f 2-Me-3-OCF_Three
cPr 2-CF_Three          iPr 2-CF_Three-3-Me U-4f 2-CF_Three-3-F
cPr 2-OMe iPr 2,3-di-CF_Three     U-4f 2-CF_Three-3-Cl
cPr 2-OCF_Three         iPr 2-CF_Three-3-OMe U-4f 2-CF_Three-3-Br
cPr 3-F iPr 2-CF_Three-3-OCF_Three   U-4f 2-CF_Three-3-Me
--------- --------- ------------
[Table 2] (continued) [Table 2] (continued) [Table 2] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
cPr 3-Cl iPr 2-OMe-3-F U-4f 2,3-di-CF_Three
cPr 3-Br iPr 2-OMe-3-Cl U-4f 2-CF_Three-3-OMe
cPr 3-Me iPr 2-OMe-3-Br U-4f 2-CF_Three-3-OCF_Three
cPr 3-CF_Three          iPr 2-OMe-3-Me U-4f 2-OMe-3-F
cPr 3-OMe iPr 2-OMe-3-CF_Three    U-4f 2-OMe-3-Cl
cPr 3-OCF_Three         iPr 2,3-di-OMe U-4f 2-OMe-3-Br
U-4b 2-F iPr 2-OMe-3-OCF_Three   U-4f 2-OMe-3-Me
U-4b 2-Cl iPr 2-OCF_Three-3-F U-4f 2-OMe-3-CF_Three
U-4b 2-Br iPr 2-OCF_Three-3-Cl U-4f 2,3-di-OMe
U-4b 2-Me iPr 2-OCF_Three-3-Br U-4f 2-OMe-3-OCF_Three
U-4b 2-CF_Three          iPr 2-OCF_Three-3-Me U-4f 2-OCF_Three-3-F
U-4b 2-OMe iPr 2-OCF_Three-3-CF_Three   U-4f 2-OCF_Three-3-Cl
U-4b 2-OCF_Three         iPr 2-OCF_Three-3-OMe U-4f 2-OCF_Three-3-Br
U-4b 3-F iPr 2,3-di-OCF_Three    U-4f 2-OCF_Three-3-Me
U-4b 3-Cl U-4a 2,3-di-F U-4f 2-OCF_Three-3-CF_Three
U-4b 3-Br U-4a 2-F-3-Cl U-4f 2-OCF_Three-3-OMe
U-4b 3-Me U-4a 2-F-3-Br U-4f 2,3-di-OCF_Three
U-4b 3-CF_Three          U-4a 2-F-3-Me U-4g 2,3-di-F
U-4b 3-OMe U-4a 2-F-3-CF_Three      U-4g 2-F-3-Cl
U-4b 3-OCF_Three         U-4a 2-F-3-OMe U-4g 2-F-3-Br
U-4c 2-F U-4a 2-F-3-OCF_Three     U-4g 2-F-3-Me
U-4c 2-Cl U-4a 2-Cl-3-F U-4g 2-F-3-CF_Three
U-4c 2-Br U-4a 2,3-di-Cl U-4g 2-F-3-OMe
U-4c 2-Me U-4a 2-Cl-3-Br U-4g 2-F-3-OCF_Three
U-4c 2-CF_Three          U-4a 2-Cl-3-Me U-4g 2-Cl-3-F
U-4c 2-OMe U-4a 2-Cl-3-CF_Three     U-4g 2,3-di-Cl
U-4c 2-OCF_Three         U-4a 2-Cl-3-OMe U-4g 2-Cl-3-Br
U-4c 3-F U-4a 2-Cl-3-OCF_Three    U-4g 2-Cl-3-Me
U-4c 3-Cl U-4a 2-Br-3-F U-4g 2-Cl-3-CF_Three
U-4c 3-Br U-4a 2-Br-3-Cl U-4g 2-Cl-3-OMe
U-4c 3-Me U-4a 2,3-di-Br U-4g 2-Cl-3-OCF_Three
U-4c 3-CF_Three          U-4a 2-Br-3-Me U-4g 2-Br-3-F
U-4c 3-OMe U-4a 2-Br-3-CF_Three     U-4g 2-Br-3-Cl
U-4c 3-OCF_Three         U-4a 2-Br-3-OMe U-4g 2,3-di-Br
U-4d 2-F U-4a 2-Br-3-OCF_Three    U-4g 2-Br-3-Me
U-4d 2-Cl U-4a 2-Me-3-F U-4g 2-Br-3-CF_Three
U-4d 2-Br U-4a 2-Me-3-Cl U-4g 2-Br-3-OMe
U-4d 2-Me U-4a 2-Me-3-Br U-4g 2-Br-3-OCF_Three
U-4d 2-CF_Three          U-4a 2,3-di-Me U-4g 2-Me-3-F
--------- --------- ------------
[Table 2] (continued) [Table 2] (continued) [Table 2] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
U-4d 2-OMe U-4a 2-Me-3-CF_Three     U-4g 2-Me-3-Cl
U-4d 2-OCF_Three         U-4a 2-Me-3-OMe U-4g 2-Me-3-Br
U-4d 3-F U-4a 2-Me-3-OCF_Three    U-4g 2,3-di-Me
U-4d 3-Cl U-4a 2-CF_Three-3-F U-4g 2-Me-3-CF_Three
U-4d 3-Br U-4a 2-CF_Three-3-Cl U-4g 2-Me-3-OMe
U-4d 3-Me U-4a 2-CF_Three-3-Br U-4g 2-Me-3-OCF_Three
U-4d 3-CF_Three          U-4a 2-CF_Three-3-Me U-4g 2-CF_Three-3-F
U-4d 3-OMe U-4a 2,3-di-CF_Three     U-4g 2-CF_Three-3-Cl
U-4d 3-OCF_Three         U-4a 2-CF_Three-3-OMe U-4g 2-CF_Three-3-Br
U-4e 2-F U-4a 2-CF_Three-3-OCF_Three   U-4g 2-CF_Three-3-Me
U-4e 2-Cl U-4a 2-OMe-3-F U-4g 2,3-di-CF_Three
U-4e 2-Br U-4a 2-OMe-3-Cl U-4g 2-CF_Three-3-OMe
U-4e 2-Me U-4a 2-OMe-3-Br U-4g 2-CF_Three-3-OCF_Three
U-4e 2-CF_Three          U-4a 2-OMe-3-Me U-4g 2-OMe-3-F
U-4e 2-OMe U-4a 2-OMe-3-CF_Three    U-4g 2-OMe-3-Cl
U-4e 2-OCF_Three         U-4a 2,3-di-OMe U-4g 2-OMe-3-Br
U-4e 3-F U-4a 2-OMe-3-OCF_Three   U-4g 2-OMe-3-Me
U-4e 3-Cl U-4a 2-OCF_Three-3-F U-4g 2-OMe-3-CF_Three
U-4e 3-Br U-4a 2-OCF_Three-3-Cl U-4g 2,3-di-OMe
U-4e 3-Me U-4a 2-OCF_Three-3-Br U-4g 2-OMe-3-OCF_Three
U-4e 3-CF_Three          U-4a 2-OCF_Three-3-Me U-4g 2-OCF_Three-3-F
U-4e 3-OMe U-4a 2-OCF_Three-3-CF_Three   U-4g 2-OCF_Three-3-Cl
U-4e 3-OCF_Three         U-4a 2-OCF_Three-3-OMe U-4g 2-OCF_Three-3-Br
U-4f 2-F U-4a 2,3-di-OCF_Three    U-4g 2-OCF_Three-3-Me
U-4f 2-Cl CF_Three   2,3-di-F U-4g 2-OCF_Three-3-CF_Three
U-4f 2-Br CF_Three   2-F-3-Cl U-4g 2-OCF_Three-3-OMe
U-4f 2-Me CF_Three   2-F-3-Br U-4g 2,3-di-OCF_Three
U-4f 2-CF_Three          CF_Three   2-F-3-Me OMe 2,3-di-F
U-4f 2-OMe CF_Three   2-F-3-CF_Three      OMe 2-F-3-Cl
U-4f 2-OCF_Three         CF_Three   2-F-3-OMe OMe 2-F-3-Br
U-4f 3-F CF_Three   2-F-3-OCF_Three     OMe 2-F-3-Me
U-4f 3-Cl CF_Three   2-Cl-3-F OMe 2-F-3-CF_Three
U-4f 3-Br CF_Three   2,3-di-Cl OMe 2-F-3-OMe
U-4f 3-Me CF_Three   2-Cl-3-Br OMe 2-F-3-OCF_Three
U-4f 3-CF_Three          CF_Three   2-Cl-3-Me OMe 2-Cl-3-F
U-4f 3-OMe CF_Three   2-Cl-3-CF_Three     OMe 2,3-di-Cl
U-4f 3-OCF_Three         CF_Three   2-Cl-3-OMe OMe 2-Cl-3-Br
U-4g 2-F CF_Three   2-Cl-3-OCF_Three    OMe 2-Cl-3-Me
U-4g 2-Cl CF_Three   2-Br-3-F OMe 2-Cl-3-CF_Three
--------- --------- ------------
[Table 2] (continued) [Table 2] (continued) [Table 2] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
U-4g 2-Br CF_Three   2-Br-3-Cl OMe 2-Cl-3-OMe
U-4g 2-Me CF_Three   2,3-di-Br OMe 2-Cl-3-OCF_Three
U-4g 2-CF_Three          CF_Three   2-Br-3-Me OMe 2-Br-3-F
U-4g 2-OMe CF_Three   2-Br-3-CF_Three     OMe 2-Br-3-Cl
U-4g 2-OCF_Three         CF_Three   2-Br-3-OMe OMe 2,3-di-Br
U-4g 3-F CF_Three   2-Br-3-OCF_Three    OMe 2-Br-3-Me
U-4g 3-Cl CF_Three   2-Me-3-F OMe 2-Br-3-CF_Three
U-4g 3-Br CF_Three   2-Me-3-Cl OMe 2-Br-3-OMe
U-4g 3-Me CF_Three   2-Me-3-Br OMe 2-Br-3-OCF_Three
U-4g 3-CF_Three          CF_Three   2,3-di-Me OMe 2-Me-3-F
U-4g 3-OMe CF_Three   2-Me-3-CF_Three     OMe 2-Me-3-Cl
U-4g 3-OCF_Three         CF_Three   2-Me-3-OMe OMe 2-Me-3-Br
OMe 2-F CF_Three   2-Me-3-OCF_Three    OMe 2,3-di-Me
OMe 2-Cl CF_Three   2-CF_Three-3-F OMe 2-Me-3-CF_Three
OMe 2-Br CF_Three   2-CF_Three-3-Cl OMe 2-Me-3-OMe
OMe 2-Me CF_Three   2-CF_Three-3-Br OMe 2-Me-3-OCF_Three
OMe 2-CF_Three          CF_Three   2-CF_Three-3-Me OMe 2-CF_Three-3-F
OMe 2-OMe CF_Three   2,3-di-CF_Three     OMe 2-CF_Three-3-Cl
OMe 2-OCF_Three         CF_Three   2-CF_Three-3-OMe OMe 2-CF_Three-3-Br
OMe 3-F CF_Three   2-CF_Three-3-OCF_Three   OMe 2-CF_Three-3-Me
OMe 3-Cl CF_Three   2-OMe-3-F OMe 2,3-di-CF_Three
OMe 3-Br CF_Three   2-OMe-3-Cl OMe 2-CF_Three-3-OMe
OMe 3-Me CF_Three   2-OMe-3-Br OMe 2-CF_Three-3-OCF_Three
OMe 3-CF_Three          CF_Three   2-OMe-3-Me OMe 2-OMe-3-F
OMe 3-OMe CF_Three   2-OMe-3-CF_Three    OMe 2-OMe-3-Cl
OMe 3-OCF_Three         CF_Three   2,3-di-OMe OMe 2-OMe-3-Br
SMe 2-F CF_Three   2-OMe-3-OCF_Three   OMe 2-OMe-3-Me
SMe 2-Cl CF_Three   2-OCF_Three-3-F OMe 2-OMe-3-CF_Three
SMe 2-Br CF_Three   2-OCF_Three-3-Cl OMe 2,3-di-OMe
SMe 2-Me CF_Three   2-OCF_Three-3-Br OMe 2-OMe-3-OCF_Three
SMe 2-CF_Three          CF_Three   2-OCF_Three-3-Me OMe 2-OCF_Three-3-F
SMe 2-OMe CF_Three   2-OCF_Three-3-CF_Three   OMe 2-OCF_Three-3-Cl
SMe 2-OCF_Three         CF_Three   2-OCF_Three-3-OMe OMe 2-OCF_Three-3-Br
SMe 3-F CF_Three   2,3-di-OCF_Three    OMe 2-OCF_Three-3-Me
SMe 3-Cl cPr 2,3-di-F OMe 2-OCF_Three-3-CF_Three
SMe 3-Br cPr 2-F-3-Cl OMe 2-OCF_Three-3-OMe
SMe 3-Me cPr 2-F-3-Br OMe 2,3-di-OCF_Three
SMe 3-CF_Three          cPr 2-F-3-Me SMe 2,3-di-F
SMe 3-OMe cPr 2-F-3-CF_Three      SMe 2-F-3-Cl
--------- --------- ------------
[Table 2] (continued) [Table 2] (continued) [Table 2] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
SMe 3-OCF_Three         cPr 2-F-3-OMe SMe 2-F-3-Br
Ac 2-F cPr 2-F-3-OCF_Three     SMe 2-F-3-Me
Ac 2-Cl cPr 2-Cl-3-F SMe 2-F-3-CF_Three
Ac 2-Br cPr 2,3-di-Cl SMe 2-F-3-OMe
Ac 2-Me cPr 2-Cl-3-Br SMe 2-F-3-OCF_Three
Ac 2-CF_Three          cPr 2-Cl-3-Me SMe 2-Cl-3-F
Ac 2-OMe cPr 2-Cl-3-CF_Three     SMe 2,3-di-Cl
Ac 2-OCF_Three         cPr 2-Cl-3-OMe SMe 2-Cl-3-Br
Ac 3-F cPr 2-Cl-3-OCF_Three    SMe 2-Cl-3-Me
Ac 3-Cl cPr 2-Br-3-F SMe 2-Cl-3-CF_Three
Ac 3-Br cPr 2-Br-3-Cl SMe 2-Cl-3-OMe
Ac 3-Me cPr 2,3-di-Br SMe 2-Cl-3-OCF_Three
Ac 3-CF_Three          cPr 2-Br-3-Me SMe 2-Br-3-F
Ac 3-OMe cPr 2-Br-3-CF_Three     SMe 2-Br-3-Cl
Ac 3-OCF_Three         cPr 2-Br-3-OMe SMe 2,3-di-Br
cPen 2-F cPr 2-Br-3-OCF_Three    SMe 2-Br-3-Me
cPen 2-Cl cPr 2-Me-3-F SMe 2-Br-3-CF_Three
cPen 2-Br cPr 2-Me-3-Cl SMe 2-Br-3-OMe
cPen 2-Me cPr 2-Me-3-Br SMe 2-Br-3-OCF_Three
cPen 2-CF_Three          cPr 2,3-di-Me SMe 2-Me-3-F
cPen 2-OMe cPr 2-Me-3-CF_Three     SMe 2-Me-3-Cl
cPen 2-OCF_Three         cPr 2-Me-3-OMe SMe 2-Me-3-Br
cPen 3-F cPr 2-Me-3-OCF_Three    SMe 2,3-di-Me
cPen 3-Cl cPr 2-CF_Three-3-F SMe 2-Me-3-CF_Three
cPen 3-Br cPr 2-CF_Three-3-Cl SMe 2-Me-3-OMe
cPen 3-Me cPr 2-CF_Three-3-Br SMe 2-Me-3-OCF_Three
cPen 3-CF_Three          cPr 2-CF_Three-3-Me SMe 2-CF_Three-3-F
cPen 3-OMe cPr 2,3-di-CF_Three     SMe 2-CF_Three-3-Cl
cPen 3-OCF_Three         cPr 2-CF_Three-3-OMe SMe 2-CF_Three-3-Br
U-1e 2-F cPr 2-CF_Three-3-OCF_Three   SMe 2-CF_Three-3-Me
U-1e 2-Cl cPr 2-OMe-3-F SMe 2,3-di-CF_Three
U-1e 2-Br cPr 2-OMe-3-Cl SMe 2-CF_Three-3-OMe
U-1e 2-Me cPr 2-OMe-3-Br SMe 2-CF_Three-3-OCF_Three
U-1e 2-CF_Three          cPr 2-OMe-3-Me SMe 2-OMe-3-F
U-1e 2-OMe cPr 2-OMe-3-CF_Three    SMe 2-OMe-3-Cl
U-1e 2-OCF_Three         cPr 2,3-di-OMe SMe 2-OMe-3-Br
U-1e 3-F cPr 2-OMe-3-OCF_Three   SMe 2-OMe-3-Me
U-1e 3-Cl cPr 2-OCF_Three-3-F SMe 2-OMe-3-CF_Three
U-1e 3-Br cPr 2-OCF_Three-3-Cl SMe 2,3-di-OMe
--------- --------- ------------
[Table 2] (continued) [Table 2] (continued) [Table 2] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
U-1e 3-Me cPr 2-OCF_Three-3-Br SMe 2-OMe-3-OCF_Three
U-1e 3-CF_Three          cPr 2-OCF_Three-3-Me SMe 2-OCF_Three-3-F
U-1e 3-OMe cPr 2-OCF_Three-3-CF_Three   SMe 2-OCF_Three-3-Cl
U-1e 3-OCF_Three         cPr 2-OCF_Three-3-OMe SMe 2-OCF_Three-3-Br
Me 2-Ac cPr 2,3-di-OCF_Three    SMe 2-OCF_Three-3-Me
Me 2- (U-3b) U-4b 2,3-di-F SMe 2-OCF_Three-3-CF_Three
Me 2-CF₂H U-4b 2-F-3-Cl SMe 2-OCF_Three-3-OMe
Me 2-CN U-4b 2-F-3-Br SMe 2,3-di-OCF_Three
Me 2-Et U-4b 2-F-3-Me Ac 2,3-di-F
Me 2-OCF₂H U-4b 2-F-3-CF_Three      Ac 2-F-3-Cl
Me 2-OEt U-4b 2-F-3-OMe Ac 2-F-3-Br
Me 2-C (O) CF_Three      U-4b 2-F-3-OCF_Three     Ac 2-F-3-Me
Me 3-Ac U-4b 2-Cl-3-F Ac 2-F-3-CF_Three
Me 3- (U-3b) U-4b 2,3-di-Cl Ac 2-F-3-OMe
Me 3-CF₂H U-4b 2-Cl-3-Br Ac 2-F-3-OCF_Three
Me 3-CN U-4b 2-Cl-3-Me Ac 2-Cl-3-F
Me 3-Et U-4b 2-Cl-3-CF_Three     Ac 2,3-di-Cl
Me 3-OCF₂H U-4b 2-Cl-3-OMe Ac 2-Cl-3-Br
Me 3-OEt U-4b 2-Cl-3-OCF_Three    Ac 2-Cl-3-Me
Me 3-C (O) CF_Three      U-4b 2-Br-3-F Ac 2-Cl-3-CF_Three
Et 2-Ac U-4b 2-Br-3-Cl Ac 2-Cl-3-OMe
Et 2- (U-3b) U-4b 2,3-di-Br Ac 2-Cl-3-OCF_Three
Et 2-CF₂H U-4b 2-Br-3-Me Ac 2-Br-3-F
Et 2-CN U-4b 2-Br-3-CF_Three     Ac 2-Br-3-Cl
Et 2-Et U-4b 2-Br-3-OMe Ac 2,3-di-Br
Et 2-OCF₂H U-4b 2-Br-3-OCF_Three    Ac 2-Br-3-Me
Et 2-OEt U-4b 2-Me-3-F Ac 2-Br-3-CF_Three
Et 2-C (O) CF_Three      U-4b 2-Me-3-Cl Ac 2-Br-3-OMe
Et 3-Ac U-4b 2-Me-3-Br Ac 2-Br-3-OCF_Three
Et 3- (U-3b) U-4b 2,3-di-Me Ac 2-Me-3-F
Et 3-CF₂H U-4b 2-Me-3-CF_Three     Ac 2-Me-3-Cl
Et 3-CN U-4b 2-Me-3-OMe Ac 2-Me-3-Br
Et 3-Et U-4b 2-Me-3-OCF_Three    Ac 2,3-di-Me
Et 3-OCF₂H U-4b 2-CF_Three-3-F Ac 2-Me-3-CF_Three
Et 3-OEt U-4b 2-CF_Three-3-Cl Ac 2-Me-3-OMe
Et 3-C (O) CF_Three      U-4b 2-CF_Three-3-Br Ac 2-Me-3-OCF_Three
iPr 2-Ac U-4b 2-CF_Three-3-Me Ac 2-CF_Three-3-F
iPr 2- (U-3b) U-4b 2,3-di-CF_Three     Ac 2-CF_Three-3-Cl
iPr 2-CF₂H U-4b 2-CF_Three-3-OMe Ac 2-CF_Three-3-Br
--------- --------- ------------
[Table 2] (continued) [Table 2] (continued) [Table 2] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
iPr 2-CN U-4b 2-CF_Three-3-OCF_Three   Ac 2-CF_Three-3-Me
iPr 2-Et U-4b 2-OMe-3-F Ac 2,3-di-CF_Three
iPr 2-OCF₂H U-4b 2-OMe-3-Cl Ac 2-CF_Three-3-OMe
iPr 2-OEt U-4b 2-OMe-3-Br Ac 2-CF_Three-3-OCF_Three
iPr 2-C (O) CF_Three      U-4b 2-OMe-3-Me Ac 2-OMe-3-F
iPr 3-Ac U-4b 2-OMe-3-CF_Three    Ac 2-OMe-3-Cl
iPr 3- (U-3b) U-4b 2,3-di-OMe Ac 2-OMe-3-Br
iPr 3-CF₂H U-4b 2-OMe-3-OCF_Three   Ac 2-OMe-3-Me
iPr 3-CN U-4b 2-OCF_Three-3-F Ac 2-OMe-3-CF_Three
iPr 3-Et U-4b 2-OCF_Three-3-Cl Ac 2,3-di-OMe
iPr 3-OCF₂H U-4b 2-OCF_Three-3-Br Ac 2-OMe-3-OCF_Three
iPr 3-OEt U-4b 2-OCF_Three-3-Me Ac 2-OCF_Three-3-F
iPr 3-C (O) CF_Three      U-4b 2-OCF_Three-3-CF_Three   Ac 2-OCF_Three-3-Cl
U-4a 2-Ac U-4b 2-OCF_Three-3-OMe Ac 2-OCF_Three-3-Br
U-4a 2- (U-3b) U-4b 2,3-di-OCF_Three    Ac 2-OCF_Three-3-Me
U-4a 2-CF₂H U-4c 2,3-di-F Ac 2-OCF_Three-3-CF_Three
U-4a 2-CN U-4c 2-F-3-Cl Ac 2-OCF_Three-3-OMe
U-4a 2-Et U-4c 2-F-3-Br Ac 2,3-di-OCF_Three
U-4a 2-OCF₂H U-4c 2-F-3-Me cPen 2,3-di-F
U-4a 2-OEt U-4c 2-F-3-CF_Three      cPen 2-F-3-Cl
U-4a 2-C (O) CF_Three      U-4c 2-F-3-OMe cPen 2-F-3-Br
U-4a 3-Ac U-4c 2-F-3-OCF_Three     cPen 2-F-3-Me
U-4a 3- (U-3b) U-4c 2-Cl-3-F cPen 2-F-3-CF_Three
U-4a 3-CF₂H U-4c 2,3-di-Cl cPen 2-F-3-OMe
U-4a 3-CN U-4c 2-Cl-3-Br cPen 2-F-3-OCF_Three
U-4a 3-Et U-4c 2-Cl-3-Me cPen 2-Cl-3-F
U-4a 3-OCF₂H U-4c 2-Cl-3-CF_Three     cPen 2,3-di-Cl
U-4a 3-OEt U-4c 2-Cl-3-OMe cPen 2-Cl-3-Br
U-4a 3-C (O) CF_Three      U-4c 2-Cl-3-OCF_Three    cPen 2-Cl-3-Me
CF_Three   2-Ac U-4c 2-Br-3-F cPen 2-Cl-3-CF_Three
CF_Three   2- (U-3b) U-4c 2-Br-3-Cl cPen 2-Cl-3-OMe
CF_Three   2-CF₂H U-4c 2,3-di-Br cPen 2-Cl-3-OCF_Three
CF_Three   2-CN U-4c 2-Br-3-Me cPen 2-Br-3-F
CF_Three   2-Et U-4c 2-Br-3-CF_Three     cPen 2-Br-3-Cl
CF_Three   2-OCF₂H U-4c 2-Br-3-OMe cPen 2,3-di-Br
CF_Three   2-OEt U-4c 2-Br-3-OCF_Three    cPen 2-Br-3-Me
CF_Three   2-C (O) CF_Three      U-4c 2-Me-3-F cPen 2-Br-3-CF_Three
CF_Three   3-Ac U-4c 2-Me-3-Cl cPen 2-Br-3-OMe
CF_Three   3- (U-3b) U-4c 2-Me-3-Br cPen 2-Br-3-OCF_Three
--------- --------- ------------
[Table 2] (continued) [Table 2] (continued) [Table 2] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
CF_Three   3-CF₂H U-4c 2,3-di-Me cPen 2-Me-3-F
CF_Three   3-CN U-4c 2-Me-3-CF_Three     cPen 2-Me-3-Cl
CF_Three   3-Et U-4c 2-Me-3-OMe cPen 2-Me-3-Br
CF_Three   3-OCF₂H U-4c 2-Me-3-OCF_Three    cPen 2,3-di-Me
CF_Three   3-OEt U-4c 2-CF_Three-3-F cPen 2-Me-3-CF_Three
CF_Three   3-C (O) CF_Three      U-4c 2-CF_Three-3-Cl cPen 2-Me-3-OMe
cPr 2-Ac U-4c 2-CF_Three-3-Br cPen 2-Me-3-OCF_Three
cPr 2- (U-3b) U-4c 2-CF_Three-3-Me cPen 2-CF_Three-3-F
cPr 2-CF₂H U-4c 2,3-di-CF_Three     cPen 2-CF_Three-3-Cl
cPr 2-CN U-4c 2-CF_Three-3-OMe cPen 2-CF_Three-3-Br
cPr 2-Et U-4c 2-CF_Three-3-OCF_Three   cPen 2-CF_Three-3-Me
cPr 2-OCF₂H U-4c 2-OMe-3-F cPen 2,3-di-CF_Three
cPr 2-OEt U-4c 2-OMe-3-Cl cPen 2-CF_Three-3-OMe
cPr 2-C (O) CF_Three      U-4c 2-OMe-3-Br cPen 2-CF_Three-3-OCF_Three
cPr 3-Ac U-4c 2-OMe-3-Me cPen 2-OMe-3-F
cPr 3- (U-3b) U-4c 2-OMe-3-CF_Three    cPen 2-OMe-3-Cl
cPr 3-CF₂H U-4c 2,3-di-OMe cPen 2-OMe-3-Br
cPr 3-CN U-4c 2-OMe-3-OCF_Three   cPen 2-OMe-3-Me
cPr 3-Et U-4c 2-OCF_Three-3-F cPen 2-OMe-3-CF_Three
cPr 3-OCF₂H U-4c 2-OCF_Three-3-Cl cPen 2,3-di-OMe
cPr 3-OEt U-4c 2-OCF_Three-3-Br cPen 2-OMe-3-OCF_Three
cPr 3-C (O) CF_Three      U-4c 2-OCF_Three-3-Me cPen 2-OCF_Three-3-F
Me 2,3-di-F U-4c 2-OCF_Three-3-CF_Three   cPen 2-OCF_Three-3-Cl
Me 2-F-3-Cl U-4c 2-OCF_Three-3-OMe cPen 2-OCF_Three-3-Br
Me 2-F-3-Br U-4c 2,3-di-OCF_Three    cPen 2-OCF_Three-3-Me
Me 2-F-3-Me U-4d 2,3-di-F cPen 2-OCF_Three-3-CF_Three
Me 2-F-3-CF_Three      U-4d 2-F-3-Cl cPen 2-OCF_Three-3-OMe
Me 2-F-3-OMe U-4d 2-F-3-Br cPen 2,3-di-OCF_Three
Me 2-F-3-OCF_Three     U-4d 2-F-3-Me U-1e 2,3-di-F
Me 2-Cl-3-F U-4d 2-F-3-CF_Three      U-1e 2-F-3-Cl
Me 2,3-di-Cl U-4d 2-F-3-OMe U-1e 2-F-3-Br
Me 2-Cl-3-Br U-4d 2-F-3-OCF_Three     U-1e 2-F-3-Me
Me 2-Cl-3-Me U-4d 2-Cl-3-F U-1e 2-F-3-CF_Three
Me 2-Cl-3-CF_Three     U-4d 2,3-di-Cl U-1e 2-F-3-OMe
Me 2-Cl-3-OMe U-4d 2-Cl-3-Br U-1e 2-F-3-OCF_Three
Me 2-Cl-3-OCF_Three    U-4d 2-Cl-3-Me U-1e 2-Cl-3-F
Me 2-Br-3-F U-4d 2-Cl-3-CF_Three     U-1e 2,3-di-Cl
Me 2-Br-3-Cl U-4d 2-Cl-3-OMe U-1e 2-Cl-3-Br
Me 2,3-di-Br U-4d 2-Cl-3-OCF_Three    U-1e 2-Cl-3-Me
--------- --------- ------------
[Table 2] (continued) [Table 2] (continued) [Table 2] (continued)
--------- --------- ------------
R^Three     Z R^Three    Z R^Three    Z
--------- --------- ------------
Me 2-Br-3-Me U-4d 2-Br-3-F U-1e 2-Cl-3-CF_Three
Me 2-Br-3-CF_Three     U-4d 2-Br-3-Cl U-1e 2-Cl-3-OMe
Me 2-Br-3-OMe U-4d 2,3-di-Br U-1e 2-Cl-3-OCF_Three
Me 2-Br-3-OCF_Three    U-4d 2-Br-3-Me U-1e 2-Br-3-F
Me 2-Me-3-F U-4d 2-Br-3-CF_Three     U-1e 2-Br-3-Cl
Me 2-Me-3-Cl U-4d 2-Br-3-OMe U-1e 2,3-di-Br
Me 2-Me-3-Br U-4d 2-Br-3-OCF_Three    U-1e 2-Br-3-Me
Me 2,3-di-Me U-4d 2-Me-3-F U-1e 2-Br-3-CF_Three
Me 2-Me-3-CF_Three     U-4d 2-Me-3-Cl U-1e 2-Br-3-OMe
Me 2-Me-3-OMe U-4d 2-Me-3-Br U-1e 2-Br-3-OCF_Three
Me 2-Me-3-OCF_Three    U-4d 2,3-di-Me U-1e 2-Me-3-F
Me 2-CF_Three-3-F U-4d 2-Me-3-CF_Three     U-1e 2-Me-3-Cl
Me 2-CF_Three-3-Cl U-4d 2-Me-3-OMe U-1e 2-Me-3-Br
Me 2-CF_Three-3-Br U-4d 2-Me-3-OCF_Three    U-1e 2,3-di-Me
Me 2-CF_Three-3-Me U-4d 2-CF_Three-3-F U-1e 2-Me-3-CF_Three
Me 2,3-di-CF_Three     U-4d 2-CF_Three-3-Cl U-1e 2-Me-3-OMe
Me 2-CF_Three-3-OMe U-4d 2-CF_Three-3-Br U-1e 2-Me-3-OCF_Three
Me 2-CF_Three-3-OCF_Three   U-4d 2-CF_Three-3-Me U-1e 2-CF_Three-3-F
Me 2-OMe-3-F U-4d 2,3-di-CF_Three     U-1e 2-CF_Three-3-Cl
Me 2-OMe-3-Cl U-4d 2-CF_Three-3-OMe U-1e 2-CF_Three-3-Br
Me 2-OMe-3-Br U-4d 2-CF_Three-3-OCF_Three   U-1e 2-CF_Three-3-Me
Me 2-OMe-3-Me U-4d 2-OMe-3-F U-1e 2,3-di-CF_Three
Me 2-OMe-3-CF_Three    U-4d 2-OMe-3-Cl U-1e 2-CF_Three-3-OMe
Me 2,3-di-OMe U-4d 2-OMe-3-Br U-1e 2-CF_Three-3-OCF_Three
Me 2-OMe-3-OCF_Three   U-4d 2-OMe-3-Me U-1e 2-OMe-3-F
Me 2-OCF_Three-3-F U-4d 2-OMe-3-CF_Three    U-1e 2-OMe-3-Cl
Me 2-OCF_Three-3-Cl U-4d 2,3-di-OMe U-1e 2-OMe-3-Br
Me 2-OCF_Three-3-Br U-4d 2-OMe-3-OCF_Three   U-1e 2-OMe-3-Me
Me 2-OCF_Three-3-Me U-4d 2-OCF_Three-3-F U-1e 2-OMe-3-CF_Three
Me 2-OCF_Three-3-CF_Three   U-4d 2-OCF_Three-3-Cl U-1e 2,3-di-OMe
Me 2-OCF_Three-3-OMe U-4d 2-OCF_Three-3-Br U-1e 2-OMe-3-OCF_Three
Me 2,3-di-OCF_Three    U-4d 2-OCF_Three-3-Me U-1e 2-OCF_Three-3-F
Et 2,3-di-F U-4d 2-OCF_Three-3-CF_Three   U-1e 2-OCF_Three-3-Cl
Et 2-F-3-Cl U-4d 2-OCF_Three-3-OMe U-1e 2-OCF_Three-3-Br
Et 2-F-3-Br U-4d 2,3-di-OCF_Three    U-1e 2-OCF_Three-3-Me
Et 2-F-3-Me U-4e 2,3-di-F U-1e 2-OCF_Three-3-CF_Three
Et 2-F-3-CF_Three      U-4e 2-F-3-Cl U-1e 2-OCF_Three-3-OMe
Et 2-F-3-OMe U-4e 2-F-3-Br U-1e 2,3-di-OCF_Three
--------- --------- ------------
[Table 2] (continued) [Table 2] (continued)
----------- --------------
R^Three     Z R^Three      Z
----------- --------------
Me 2-F-3-Ac U-4a 2-F-3-Ac
Me 2-F-3- (U-3b) U-4a 2-F-3- (U-3b)
Me 2-F-3-CF₂H U-4a 2-F-3-CF₂H
Me 2-F-3-CN U-4a 2-F-3-CN
Me 2-F-3-Et U-4a 2-F-3-Et
Me 2-F-3-OCF₂H U-4a 2-F-3-OCF₂H
Me 2-F-3-OEt U-4a 2-F-3-OEt
Me 2-F-3-C (O) CF_Three       U-4a 2-F-3-C (O) CF_Three
Me 2-Cl-3-Ac U-4a 2-Cl-3-Ac
Me 2-Cl-3- (U-3b) U-4a 2-Cl-3- (U-3b)
Me 2-Cl-3-CF₂H U-4a 2-Cl-3-CF₂H
Me 2-Cl-3-CN U-4a 2-Cl-3-CN
Me 2-Cl-3-Et U-4a 2-Cl-3-Et
Me 2-Cl-3-OCF₂H U-4a 2-Cl-3-OCF₂H
Me 2-Cl-3-OEt U-4a 2-Cl-3-OEt
Me 2-Cl-3-C (O) CF_Three      U-4a 2-Cl-3-C (O) CF_Three
Me 2-Br-3-Ac U-4a 2-Br-3-Ac
Me 2-Br-3- (U-3b) U-4a 2-Br-3- (U-3b)
Me 2-Br-3-CF₂H U-4a 2-Br-3-CF₂H
Me 2-Br-3-CN U-4a 2-Br-3-CN
Me 2-Br-3-Et U-4a 2-Br-3-Et
Me 2-Br-3-OCF₂H U-4a 2-Br-3-OCF₂H
Me 2-Br-3-OEt U-4a 2-Br-3-OEt
Me 2-Br-3-C (O) CF_Three      U-4a 2-Br-3-C (O) CF_Three
Me 2-Me-3-Ac U-4a 2-Me-3-Ac
Me 2-Me-3- (U-3b) U-4a 2-Me-3- (U-3b)
Me 2-Me-3-CF₂H U-4a 2-Me-3-CF₂H
Me 2-Me-3-CN U-4a 2-Me-3-CN
Me 2-Me-3-Et U-4a 2-Me-3-Et
Me 2-Me-3-OCF₂H U-4a 2-Me-3-OCF₂H
Me 2-Me-3-OEt U-4a 2-Me-3-OEt
Me 2-Me-3-C (O) CF_Three      U-4a 2-Me-3-C (O) CF_Three
Me 2-CF_Three-3-Ac U-4a 2-CF_Three-3-Ac
Me 2-CF_Three-3- (U-3b) U-4a 2-CF_Three-3- (U-3b)
Me 2-CF_Three-3-CF₂H U-4a 2-CF_Three-3-CF₂H
Me 2-CF_Three-3-CN U-4a 2-CF_Three-3-CN
Me 2-CF_Three-3-Et U-4a 2-CF_Three-3-Et
Me 2-CF_Three-3-OCF₂H U-4a 2-CF_Three-3-OCF₂H
Me 2-CF_Three-3-OEt U-4a 2-CF_Three-3-OEt
----------- --------------
[Table 2] (continued) [Table 2] (continued)
----------- --------------
R^Three     Z R^Three      Z
----------- --------------
Me 2-CF_Three-3-C (O) CF_Three     U-4a 2-CF_Three-3-C (O) CF_Three
Me 2-OMe-3-Ac U-4a 2-OMe-3-Ac
Me 2-OMe-3- (U-3b) U-4a 2-OMe-3- (U-3b)
Me 2-OMe-3-CF₂H U-4a 2-OMe-3-CF₂H
Me 2-OMe-3-CN U-4a 2-OMe-3-CN
Me 2-OMe-3-Et U-4a 2-OMe-3-Et
Me 2-OMe-3-OCF₂H U-4a 2-OMe-3-OCF₂H
Me 2-OMe-3-OEt U-4a 2-OMe-3-OEt
Me 2-OMe-3-C (O) CF_Three     U-4a 2-OMe-3-C (O) CF_Three
Me 2-OCF_Three-3-Ac U-4a 2-OCF_Three-3-Ac
Me 2-OCF_Three-3- (U-3b) U-4a 2-OCF_Three-3- (U-3b)
Me 2-OCF_Three-3-CF₂H U-4a 2-OCF_Three-3-CF₂H
Me 2-OCF_Three-3-CN U-4a 2-OCF_Three-3-CN
Me 2-OCF_Three-3-Et U-4a 2-OCF_Three-3-Et
Me 2-OCF_Three-3-OCF₂H U-4a 2-OCF_Three-3-OCF₂H
Me 2-OCF_Three-3-OEt U-4a 2-OCF_Three-3-OEt
Me 2-OCF_Three-3-C (O) CF_Three    U-4a 2-OCF_Three-3-C (O) CF_Three
Me 2-Ac-3-F U-4a 2-Ac-3-F
Me 2-Ac-3-Cl U-4a 2-Ac-3-Cl
Me 2-Ac-3-Br U-4a 2-Ac-3-Br
Me 2-Ac-3-Me U-4a 2-Ac-3-Me
Me 2-Ac-3-CF_Three          U-4a 2-Ac-3-CF_Three
Me 2-Ac-3-OMe U-4a 2-Ac-3-OMe
Me 2-Ac-3-OCF_Three         U-4a 2-Ac-3-OCF_Three
Me 2- (U-3b) -3-F U-4a 2- (U-3b) -3-F
Me 2- (U-3b) -3-Cl U-4a 2- (U-3b) -3-Cl
Me 2- (U-3b) -3-Br U-4a 2- (U-3b) -3-Br
Me 2- (U-3b) -3-Me U-4a 2- (U-3b) -3-Me
Me 2- (U-3b) -3-CF_Three      U-4a 2- (U-3b) -3-CF_Three
Me 2- (U-3b) -3-OMe U-4a 2- (U-3b) -3-OMe
Me 2- (U-3b) -3-OCF_Three     U-4a 2- (U-3b) -3-OCF_Three
Me 2-CF₂H-3-F U-4a 2-CF₂H-3-F
Me 2-CF₂H-3-Cl U-4a 2-CF₂H-3-Cl
Me 2-CF₂H-3-Br U-4a 2-CF₂H-3-Br
Me 2-CF₂H-3-Me U-4a 2-CF₂H-3-Me
Me 2-CF₂H-3-CF_Three        U-4a 2-CF₂H-3-CF_Three
Me 2-CF₂H-3-OMe U-4a 2-CF₂H-3-OMe
Me 2-CF₂H-3-OCF_Three       U-4a 2-CF₂H-3-OCF_Three
Me 2-CN-3-F U-4a 2-CN-3-F
----------- --------------
[Table 2] (continued) [Table 2] (continued)
----------- --------------
R^Three     Z R^Three      Z
----------- --------------
Me 2-CN-3-Cl U-4a 2-CN-3-Cl
Me 2-CN-3-Br U-4a 2-CN-3-Br
Me 2-CN-3-Me U-4a 2-CN-3-Me
Me 2-CN-3-CF_Three          U-4a 2-CN-3-CF_Three
Me 2-CN-3-OMe U-4a 2-CN-3-OMe
Me 2-CN-3-OCF_Three         U-4a 2-CN-3-OCF_Three
Me 2-Et-3-F U-4a 2-Et-3-F
Me 2-Et-3-Cl U-4a 2-Et-3-Cl
Me 2-Et-3-Br U-4a 2-Et-3-Br
Me 2-Et-3-Me U-4a 2-Et-3-Me
Me 2-Et-3-CF_Three          U-4a 2-Et-3-CF_Three
Me 2-Et-3-OMe U-4a 2-Et-3-OMe
Me 2-Et-3-OCF_Three         U-4a 2-Et-3-OCF_Three
Me 2-OCF₂H-3-F U-4a 2-OCF₂H-3-F
Me 2-OCF₂H-3-Cl U-4a 2-OCF₂H-3-Cl
Me 2-OCF₂H-3-Br U-4a 2-OCF₂H-3-Br
Me 2-OCF₂H-3-Me U-4a 2-OCF₂H-3-Me
Me 2-OCF₂H-3-CF_Three       U-4a 2-OCF₂H-3-CF_Three
Me 2-OCF₂H-3-OMe U-4a 2-OCF₂H-3-OMe
Me 2-OCF₂H-3-OCF_Three      U-4a 2-OCF₂H-3-OCF_Three
Me 2-OEt-3-F U-4a 2-OEt-3-F
Me 2-OEt-3-Cl U-4a 2-OEt-3-Cl
Me 2-OEt-3-Br U-4a 2-OEt-3-Br
Me 2-OEt-3-Me U-4a 2-OEt-3-Me
Me 2-OEt-3-CF_Three         U-4a 2-OEt-3-CF_Three
Me 2-OEt-3-OMe U-4a 2-OEt-3-OMe
Me 2-OEt-3-OCF_Three        U-4a 2-OEt-3-OCF_Three
Me 2-C (O) CF_Three-3-F U-4a 2-C (O) CF_Three-3-F
Me 2-C (O) CF_Three-3-Cl U-4a 2-C (O) CF_Three-3-Cl
Me 2-C (O) CF_Three-3-Br U-4a 2-C (O) CF_Three-3-Br
Me 2-C (O) CF_Three-3-Me U-4a 2-C (O) CF_Three-3-Me
Me 2-C (O) CF_Three-3-CF_Three     U-4a 2-C (O) CF_Three-3-CF_Three
Me 2-C (O) CF_Three-3-OMe U-4a 2-C (O) CF_Three-3-OMe
Me 2-C (O) CF_Three-3-OCF_Three    U-4a 2-C (O) CF_Three-3-OCF_Three
Et 2-F-3-Ac CF_Three    2-F-3-Ac
Et 2-F-3- (U-3b) CF_Three    2-F-3- (U-3b)
Et 2-F-3-CF₂H CF_Three    2-F-3-CF₂H
Et 2-F-3-CN CF_Three    2-F-3-CN
Et 2-F-3-Et CF_Three    2-F-3-Et
----------- --------------
[Table 2] (continued) [Table 2] (continued)
----------- --------------
R^Three     Z R^Three      Z
----------- --------------
Et 2-F-3-OCF₂H CF_Three    2-F-3-OCF₂H
Et 2-F-3-OEt CF_Three    2-F-3-OEt
Et 2-F-3-C (O) CF_Three       CF_Three    2-F-3-C (O) CF_Three
Et 2-Cl-3-Ac CF_Three    2-Cl-3-Ac
Et 2-Cl-3- (U-3b) CF_Three    2-Cl-3- (U-3b)
Et 2-Cl-3-CF₂H CF_Three    2-Cl-3-CF₂H
Et 2-Cl-3-CN CF_Three    2-Cl-3-CN
Et 2-Cl-3-Et CF_Three    2-Cl-3-Et
Et 2-Cl-3-OCF₂H CF_Three    2-Cl-3-OCF₂H
Et 2-Cl-3-OEt CF_Three    2-Cl-3-OEt
Et 2-Cl-3-C (O) CF_Three      CF_Three    2-Cl-3-C (O) CF_Three
Et 2-Br-3-Ac CF_Three    2-Br-3-Ac
Et 2-Br-3- (U-3b) CF_Three    2-Br-3- (U-3b)
Et 2-Br-3-CF₂H CF_Three    2-Br-3-CF₂H
Et 2-Br-3-CN CF_Three    2-Br-3-CN
Et 2-Br-3-Et CF_Three    2-Br-3-Et
Et 2-Br-3-OCF₂H CF_Three    2-Br-3-OCF₂H
Et 2-Br-3-OEt CF_Three    2-Br-3-OEt
Et 2-Br-3-C (O) CF_Three      CF_Three    2-Br-3-C (O) CF_Three
Et 2-Me-3-Ac CF_Three    2-Me-3-Ac
Et 2-Me-3- (U-3b) CF_Three    2-Me-3- (U-3b)
Et 2-Me-3-CF₂H CF_Three    2-Me-3-CF₂H
Et 2-Me-3-CN CF_Three    2-Me-3-CN
Et 2-Me-3-Et CF_Three    2-Me-3-Et
Et 2-Me-3-OCF₂H CF_Three    2-Me-3-OCF₂H
Et 2-Me-3-OEt CF_Three    2-Me-3-OEt
Et 2-Me-3-C (O) CF_Three      CF_Three    2-Me-3-C (O) CF_Three
Et 2-CF_Three-3-Ac CF_Three    2-CF_Three-3-Ac
Et 2-CF_Three-3- (U-3b) CF_Three    2-CF_Three-3- (U-3b)
Et 2-CF_Three-3-CF₂H CF_Three    2-CF_Three-3-CF₂H
Et 2-CF_Three-3-CN CF_Three    2-CF_Three-3-CN
Et 2-CF_Three-3-Et CF_Three    2-CF_Three-3-Et
Et 2-CF_Three-3-OCF₂H CF_Three    2-CF_Three-3-OCF₂H
Et 2-CF_Three-3-OEt CF_Three    2-CF_Three-3-OEt
Et 2-CF_Three-3-C (O) CF_Three     CF_Three    2-CF_Three-3-C (O) CF_Three
Et 2-OMe-3-Ac CF_Three    2-OMe-3-Ac
Et 2-OMe-3- (U-3b) CF_Three    2-OMe-3- (U-3b)
Et 2-OMe-3-CF₂H CF_Three    2-OMe-3-CF₂H
Et 2-OMe-3-CN CF_Three    2-OMe-3-CN
----------- --------------
[Table 2] (continued) [Table 2] (continued)
----------- --------------
R^Three     Z R^Three      Z
----------- --------------
Et 2-OMe-3-Et CF_Three    2-OMe-3-Et
Et 2-OMe-3-OCF₂H CF_Three    2-OMe-3-OCF₂H
Et 2-OMe-3-OEt CF_Three    2-OMe-3-OEt
Et 2-OMe-3-C (O) CF_Three     CF_Three    2-OMe-3-C (O) CF_Three
Et 2-OCF_Three-3-Ac CF_Three    2-OCF_Three-3-Ac
Et 2-OCF_Three-3- (U-3b) CF_Three    2-OCF_Three-3- (U-3b)
Et 2-OCF_Three-3-CF₂H CF_Three    2-OCF_Three-3-CF₂H
Et 2-OCF_Three-3-CN CF_Three    2-OCF_Three-3-CN
Et 2-OCF_Three-3-Et CF_Three    2-OCF_Three-3-Et
Et 2-OCF_Three-3-OCF₂H CF_Three    2-OCF_Three-3-OCF₂H
Et 2-OCF_Three-3-OEt CF_Three    2-OCF_Three-3-OEt
Et 2-OCF_Three-3-C (O) CF_Three    CF_Three    2-OCF_Three-3-C (O) CF_Three
Et 2-Ac-3-F CF_Three    2-Ac-3-F
Et 2-Ac-3-Cl CF_Three    2-Ac-3-Cl
Et 2-Ac-3-Br CF_Three    2-Ac-3-Br
Et 2-Ac-3-Me CF_Three    2-Ac-3-Me
Et 2-Ac-3-CF_Three          CF_Three    2-Ac-3-CF_Three
Et 2-Ac-3-OMe CF_Three    2-Ac-3-OMe
Et 2-Ac-3-OCF_Three         CF_Three    2-Ac-3-OCF_Three
Et 2- (U-3b) -3-F CF_Three    2- (U-3b) -3-F
Et 2- (U-3b) -3-Cl CF_Three    2- (U-3b) -3-Cl
Et 2- (U-3b) -3-Br CF_Three    2- (U-3b) -3-Br
Et 2- (U-3b) -3-Me CF_Three    2- (U-3b) -3-Me
Et 2- (U-3b) -3-CF_Three      CF_Three    2- (U-3b) -3-CF_Three
Et 2- (U-3b) -3-OMe CF_Three    2- (U-3b) -3-OMe
Et 2- (U-3b) -3-OCF_Three     CF_Three    2- (U-3b) -3-OCF_Three
Et 2-CF₂H-3-F CF_Three    2-CF₂H-3-F
Et 2-CF₂H-3-Cl CF_Three    2-CF₂H-3-Cl
Et 2-CF₂H-3-Br CF_Three    2-CF₂H-3-Br
Et 2-CF₂H-3-Me CF_Three    2-CF₂H-3-Me
Et 2-CF₂H-3-CF_Three        CF_Three    2-CF₂H-3-CF_Three
Et 2-CF₂H-3-OMe CF_Three    2-CF₂H-3-OMe
Et 2-CF₂H-3-OCF_Three       CF_Three    2-CF₂H-3-OCF_Three
Et 2-CN-3-F CF_Three    2-CN-3-F
Et 2-CN-3-Cl CF_Three    2-CN-3-Cl
Et 2-CN-3-Br CF_Three    2-CN-3-Br
Et 2-CN-3-Me CF_Three    2-CN-3-Me
Et 2-CN-3-CF_Three          CF_Three    2-CN-3-CF_Three
Et 2-CN-3-OMe CF_Three    2-CN-3-OMe
----------- --------------
[Table 2] (continued) [Table 2] (continued)
----------- --------------
R^Three     Z R^Three      Z
----------- --------------
Et 2-CN-3-OCF_Three         CF_Three    2-CN-3-OCF_Three
Et 2-Et-3-F CF_Three    2-Et-3-F
Et 2-Et-3-Cl CF_Three    2-Et-3-Cl
Et 2-Et-3-Br CF_Three    2-Et-3-Br
Et 2-Et-3-Me CF_Three    2-Et-3-Me
Et 2-Et-3-CF_Three          CF_Three    2-Et-3-CF_Three
Et 2-Et-3-OMe CF_Three    2-Et-3-OMe
Et 2-Et-3-OCF_Three         CF_Three    2-Et-3-OCF_Three
Et 2-OCF₂H-3-F CF_Three    2-OCF₂H-3-F
Et 2-OCF₂H-3-Cl CF_Three    2-OCF₂H-3-Cl
Et 2-OCF₂H-3-Br CF_Three    2-OCF₂H-3-Br
Et 2-OCF₂H-3-Me CF_Three    2-OCF₂H-3-Me
Et 2-OCF₂H-3-CF_Three       CF_Three    2-OCF₂H-3-CF_Three
Et 2-OCF₂H-3-OMe CF_Three    2-OCF₂H-3-OMe
Et 2-OCF₂H-3-OCF_Three      CF_Three    2-OCF₂H-3-OCF_Three
Et 2-OEt-3-F CF_Three    2-OEt-3-F
Et 2-OEt-3-Cl CF_Three    2-OEt-3-Cl
Et 2-OEt-3-Br CF_Three    2-OEt-3-Br
Et 2-OEt-3-Me CF_Three    2-OEt-3-Me
Et 2-OEt-3-CF_Three         CF_Three    2-OEt-3-CF_Three
Et 2-OEt-3-OMe CF_Three    2-OEt-3-OMe
Et 2-OEt-3-OCF_Three        CF_Three    2-OEt-3-OCF_Three
Et 2-C (O) CF_Three-3-F CF_Three    2-C (O) CF_Three-3-F
Et 2-C (O) CF_Three-3-Cl CF_Three    2-C (O) CF_Three-3-Cl
Et 2-C (O) CF_Three-3-Br CF_Three    2-C (O) CF_Three-3-Br
Et 2-C (O) CF_Three-3-Me CF_Three    2-C (O) CF_Three-3-Me
Et 2-C (O) CF_Three-3-CF_Three     CF_Three    2-C (O) CF_Three-3-CF_Three
Et 2-C (O) CF_Three-3-OMe CF_Three    2-C (O) CF_Three-3-OMe
Et 2-C (O) CF_Three-3-OCF_Three    CF_Three    2-C (O) CF_Three-3-OCF_Three
iPr 2-F-3-Ac cPr 2-F-3-Ac
iPr 2-F-3- (U-3b) cPr 2-F-3- (U-3b)
iPr 2-F-3-CF₂H cPr 2-F-3-CF₂H
iPr 2-F-3-CN cPr 2-F-3-CN
iPr 2-F-3-Et cPr 2-F-3-Et
iPr 2-F-3-OCF₂H cPr 2-F-3-OCF₂H
iPr 2-F-3-OEt cPr 2-F-3-OEt
iPr 2-F-3-C (O) CF_Three       cPr 2-F-3-C (O) CF_Three
iPr 2-Cl-3-Ac cPr 2-Cl-3-Ac
iPr 2-Cl-3- (U-3b) cPr 2-Cl-3- (U-3b)
----------- --------------
[Table 2] (continued) [Table 2] (continued)
----------- --------------
R^Three     Z R^Three      Z
----------- --------------
iPr 2-Cl-3-CF₂H cPr 2-Cl-3-CF₂H
iPr 2-Cl-3-CN cPr 2-Cl-3-CN
iPr 2-Cl-3-Et cPr 2-Cl-3-Et
iPr 2-Cl-3-OCF₂H cPr 2-Cl-3-OCF₂H
iPr 2-Cl-3-OEt cPr 2-Cl-3-OEt
iPr 2-Cl-3-C (O) CF_Three      cPr 2-Cl-3-C (O) CF_Three
iPr 2-Br-3-Ac cPr 2-Br-3-Ac
iPr 2-Br-3- (U-3b) cPr 2-Br-3- (U-3b)
iPr 2-Br-3-CF₂H cPr 2-Br-3-CF₂H
iPr 2-Br-3-CN cPr 2-Br-3-CN
iPr 2-Br-3-Et cPr 2-Br-3-Et
iPr 2-Br-3-OCF₂H cPr 2-Br-3-OCF₂H
iPr 2-Br-3-OEt cPr 2-Br-3-OEt
iPr 2-Br-3-C (O) CF_Three      cPr 2-Br-3-C (O) CF_Three
iPr 2-Me-3-Ac cPr 2-Me-3-Ac
iPr 2-Me-3- (U-3b) cPr 2-Me-3- (U-3b)
iPr 2-Me-3-CF₂H cPr 2-Me-3-CF₂H
iPr 2-Me-3-CN cPr 2-Me-3-CN
iPr 2-Me-3-Et cPr 2-Me-3-Et
iPr 2-Me-3-OCF₂H cPr 2-Me-3-OCF₂H
iPr 2-Me-3-OEt cPr 2-Me-3-OEt
iPr 2-Me-3-C (O) CF_Three      cPr 2-Me-3-C (O) CF_Three
iPr 2-CF_Three-3-Ac cPr 2-CF_Three-3-Ac
iPr 2-CF_Three-3- (U-3b) cPr 2-CF_Three-3- (U-3b)
iPr 2-CF_Three-3-CF₂H cPr 2-CF_Three-3-CF₂H
iPr 2-CF_Three-3-CN cPr 2-CF_Three-3-CN
iPr 2-CF_Three-3-Et cPr 2-CF_Three-3-Et
iPr 2-CF_Three-3-OCF₂H cPr 2-CF_Three-3-OCF₂H
iPr 2-CF_Three-3-OEt cPr 2-CF_Three-3-OEt
iPr 2-CF_Three-3-C (O) CF_Three     cPr 2-CF_Three-3-C (O) CF_Three
iPr 2-OMe-3-Ac cPr 2-OMe-3-Ac
iPr 2-OMe-3- (U-3b) cPr 2-OMe-3- (U-3b)
iPr 2-OMe-3-CF₂H cPr 2-OMe-3-CF₂H
iPr 2-OMe-3-CN cPr 2-OMe-3-CN
iPr 2-OMe-3-Et cPr 2-OMe-3-Et
iPr 2-OMe-3-OCF₂H cPr 2-OMe-3-OCF₂H
iPr 2-OMe-3-OEt cPr 2-OMe-3-OEt
iPr 2-OMe-3-C (O) CF_Three     cPr 2-OMe-3-C (O) CF_Three
iPr 2-OCF_Three-3-Ac cPr 2-OCF_Three-3-Ac
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[Table 2] (continued) [Table 2] (continued)
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R^Three     Z R^Three      Z
----------- --------------
iPr 2-OCF_Three-3- (U-3b) cPr 2-OCF_Three-3- (U-3b)
iPr 2-OCF_Three-3-CF₂H cPr 2-OCF_Three-3-CF₂H
iPr 2-OCF_Three-3-CN cPr 2-OCF_Three-3-CN
iPr 2-OCF_Three-3-Et cPr 2-OCF_Three-3-Et
iPr 2-OCF_Three-3-OCF₂H cPr 2-OCF_Three-3-OCF₂H
iPr 2-OCF_Three-3-OEt cPr 2-OCF_Three-3-OEt
iPr 2-OCF_Three-3-C (O) CF_Three    cPr 2-OCF_Three-3-C (O) CF_Three
iPr 2-Ac-3-F cPr 2-Ac-3-F
iPr 2-Ac-3-Cl cPr 2-Ac-3-Cl
iPr 2-Ac-3-Br cPr 2-Ac-3-Br
iPr 2-Ac-3-Me cPr 2-Ac-3-Me
iPr 2-Ac-3-CF_Three          cPr 2-Ac-3-CF_Three
iPr 2-Ac-3-OMe cPr 2-Ac-3-OMe
iPr 2-Ac-3-OCF_Three         cPr 2-Ac-3-OCF_Three
iPr 2- (U-3b) -3-F cPr 2- (U-3b) -3-F
iPr 2- (U-3b) -3-Cl cPr 2- (U-3b) -3-Cl
iPr 2- (U-3b) -3-Br cPr 2- (U-3b) -3-Br
iPr 2- (U-3b) -3-Me cPr 2- (U-3b) -3-Me
iPr 2- (U-3b) -3-CF_Three      cPr 2- (U-3b) -3-CF_Three
iPr 2- (U-3b) -3-OMe cPr 2- (U-3b) -3-OMe
iPr 2- (U-3b) -3-OCF_Three     cPr 2- (U-3b) -3-OCF_Three
iPr 2-CF₂H-3-F cPr 2-CF₂H-3-F
iPr 2-CF₂H-3-Cl cPr 2-CF₂H-3-Cl
iPr 2-CF₂H-3-Br cPr 2-CF₂H-3-Br
iPr 2-CF₂H-3-Me cPr 2-CF₂H-3-Me
iPr 2-CF₂H-3-CF_Three        cPr 2-CF₂H-3-CF_Three
iPr 2-CF₂H-3-OMe cPr 2-CF₂H-3-OMe
iPr 2-CF₂H-3-OCF_Three       cPr 2-CF₂H-3-OCF_Three
iPr 2-CN-3-F cPr 2-CN-3-F
iPr 2-CN-3-Cl cPr 2-CN-3-Cl
iPr 2-CN-3-Br cPr 2-CN-3-Br
iPr 2-CN-3-Me cPr 2-CN-3-Me
iPr 2-CN-3-CF_Three          cPr 2-CN-3-CF_Three
iPr 2-CN-3-OMe cPr 2-CN-3-OMe
iPr 2-CN-3-OCF_Three         cPr 2-CN-3-OCF_Three
iPr 2-Et-3-F cPr 2-Et-3-F
iPr 2-Et-3-Cl cPr 2-Et-3-Cl
iPr 2-Et-3-Br cPr 2-Et-3-Br
iPr 2-Et-3-Me cPr 2-Et-3-Me
----------- --------------
[Table 2] (continued) [Table 2] (continued)
----------- --------------
R^Three     Z R^Three      Z
----------- --------------
iPr 2-Et-3-CF_Three          cPr 2-Et-3-CF_Three
iPr 2-Et-3-OMe cPr 2-Et-3-OMe
iPr 2-Et-3-OCF_Three         cPr 2-Et-3-OCF_Three
iPr 2-OCF₂H-3-F cPr 2-OCF₂H-3-F
iPr 2-OCF₂H-3-Cl cPr 2-OCF₂H-3-Cl
iPr 2-OCF₂H-3-Br cPr 2-OCF₂H-3-Br
iPr 2-OCF₂H-3-Me cPr 2-OCF₂H-3-Me
iPr 2-OCF₂H-3-CF_Three       cPr 2-OCF₂H-3-CF_Three
iPr 2-OCF₂H-3-OMe cPr 2-OCF₂H-3-OMe
iPr 2-OCF₂H-3-OCF_Three      cPr 2-OCF₂H-3-OCF_Three
iPr 2-OEt-3-F cPr 2-OEt-3-F
iPr 2-OEt-3-Cl cPr 2-OEt-3-Cl
iPr 2-OEt-3-Br cPr 2-OEt-3-Br
iPr 2-OEt-3-Me cPr 2-OEt-3-Me
iPr 2-OEt-3-CF_Three         cPr 2-OEt-3-CF_Three
iPr 2-OEt-3-OMe cPr 2-OEt-3-OMe
iPr 2-OEt-3-OCF_Three        cPr 2-OEt-3-OCF_Three
iPr 2-C (O) CF_Three-3-F cPr 2-C (O) CF_Three-3-F
iPr 2-C (O) CF_Three-3-Cl cPr 2-C (O) CF_Three-3-Cl
iPr 2-C (O) CF_Three-3-Br cPr 2-C (O) CF_Three-3-Br
iPr 2-C (O) CF_Three-3-Me cPr 2-C (O) CF_Three-3-Me
iPr 2-C (O) CF_Three-3-CF_Three     cPr 2-C (O) CF_Three-3-CF_Three
iPr 2-C (O) CF_Three-3-OMe cPr 2-C (O) CF_Three-3-OMe
iPr 2-C (O) CF_Three-3-OCF_Three    cPr 2-C (O) CF_Three-3-OCF_Three
----------- --------------
[Table 3]

［第３表］ −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
Me 2-F Et 2-Br-4-F Me 2-Cl Et 2-Br-4-Cl Me 2-Br Et 2,4-di-Br Me 2-Me Et 2-Br-4-Me Me 2-CF₃ Me 2-OMe Et 2-Br-4-OMe Me 2-OCF₃ Me 3-F Et 2-Me-4-F Me 3-Cl Et 2-Me-4-Cl Me 3-Br Et 2-Me-4-Br Me 3-Me Et 2,4-di-Me Me 3-CF₃ Me 3-OMe Et 2-Me-4-OMe Me 3-OCF₃ Me 4-F Et Me 4-Cl Et Me 4-Br Et Me 4-Me Et Me 4-CF₃ Me 4-OMe Et Me 4-OCF₃ Et 2-F Et 2-OMe-4-F Et 2-Cl Et 2-OMe-4-Cl Et 2-Br Et 2-OMe-4-Br Et 2-Me Et 2-OMe-4-Me Et 2-CF₃ Et 2-OMe Et 2,4-di-OMe Et 2-OCF₃ Et 3-F Et Et 3-Cl Et Et 3-Br Et Et 3-Me Et Et 3-CF₃ Et 3-OMe Et Et 3-OCF₃ Et 4-F Et 3,4-di-F Et 4-Cl Et 3-F-4-Cl Et 4-Br Et 3-F-4-Br Et 4-Me Et 3-F-4-Me −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第３表］（続き） −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
Et 4-CF₃ Et 4-OMe Et 3-F-4-OMe Et 4-OCF₃ iPr 2-F Et 3-Cl-4-F iPr 2-Cl Et 3,4-di-Cl iPr 2-Br Et 3-Cl-4-Br iPr 2-Me Et 3-Cl-4-Me iPr 2-CF₃ iPr 2-OMe Et 3-Cl-4-OMe iPr 2-OCF₃ iPr 3-F Et 3-Br-4-F iPr 3-Cl Et 3-Br-4-Cl iPr 3-Br Et 3,4-di-Br iPr 3-Me Et 3-Br-4-Me iPr 3-CF₃ iPr 3-OMe Et 3-Br-4-OMe iPr 3-OCF₃ iPr 4-F Et 3-Me-4-F iPr 4-Cl Et 3-Me-4-Cl iPr 4-Br Et 3-Me-4-Br iPr 4-Me Et 3,4-di-Me iPr 4-CF₃ iPr 4-OMe Et 3-Me-4-OMe iPr 4-OCF₃ U-4a 2-F Et U-4a 2-Cl Et U-4a 2-Br Et U-4a 2-Me Et U-4a 2-CF₃ U-4a 2-OMe Et U-4a 2-OCF₃ U-4a 3-F Et 3-OMe-4-F U-4a 3-Cl Et 3-OMe-4-Cl U-4a 3-Br Et 3-OMe-4-Br U-4a 3-Me Et 3-OMe-4-Me U-4a 3-CF₃ U-4a 3-OMe Et 3,4-di-OMe U-4a 3-OCF₃ U-4a 4-F Et −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第３表］（続き） −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
U-4a 4-Cl Et U-4a 4-Br Et U-4a 4-Me Et U-4a 4-CF₃ U-4a 4-OMe Et U-4a 4-OCF₃ CF₃ 2-F CF₃ 2-Cl CF₃ 2-Br CF₃ 2-Me CF₃ 2-CF₃ CF₃ 2-OMe CF₃ 2-OCF₃ CF₃ 3-F CF₃ 3-Cl CF₃ 3-Br CF₃ 3-Me CF₃ 3-CF₃ CF₃ 3-OMe CF₃ 3-OCF₃ CF₃ 4-F CF₃ 4-Cl CF₃ 4-Br CF₃ 4-Me CF₃ 4-CF₃ CF₃ 4-OMe CF₃ 4-OCF₃ cPr 2-F iPr 2-Me-3-F cPr 2-Cl iPr 2-Me-3-Cl cPr 2-Br iPr 2-Me-3-Br cPr 2-Me iPr 2,3-di-Me cPr 2-CF₃ cPr 2-OMe iPr 2-Me-3-OMe cPr 2-OCF₃ cPr 3-F cPr 3-Cl cPr 3-Br cPr 3-Me cPr 3-CF₃ −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第３表］（続き） −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
cPr 3-OMe cPr 3-OCF₃ cPr 4-F iPr 2-OMe-3-F cPr 4-Cl iPr 2-OMe-3-Cl cPr 4-Br iPr 2-OMe-3-Br cPr 4-Me iPr 2-OMe-3-Me cPr 4-CF₃ cPr 4-OMe iPr 2,3-di-OMe cPr 4-OCF₃ Me 2,3-di-F Me 2-F-3-Cl Me 2-F-3-Br Me 2-F-3-Me Me 2-F-3-CF₃ Me 2-F-3-OMe Me 2-F-3-OCF₃ Me 2-Cl-3-F iPr 2,4-di-F Me 2,3-di-Cl iPr 2-F-4-Cl Me 2-Cl-3-Br iPr 2-F-4-Br Me 2-Cl-3-Me iPr 2-F-4-Me Me 2-Cl-3-CF₃ Me 2-Cl-3-OMe iPr 2-F-4-OMe Me 2-Cl-3-OCF₃ Me 2-Br-3-F iPr 2-Cl-4-F Me 2-Br-3-Cl iPr 2,4-di-Cl Me 2,3-di-Br iPr 2-Cl-4-Br Me 2-Br-3-Me iPr 2-Cl-4-Me Me 2-Br-3-CF₃ Me 2-Br-3-OMe iPr 2-Cl-4-OMe Me 2-Br-3-OCF₃ Me 2-Me-3-F iPr 2-Br-4-F Me 2-Me-3-Cl iPr 2-Br-4-Cl Me 2-Me-3-Br iPr 2,4-di-Br Me 2,3-di-Me iPr 2-Br-4-Me Me 2-Me-3-CF₃ Me 2-Me-3-OMe iPr 2-Br-4-OMe Me 2-Me-3-OCF₃ Me 2-CF₃-3-F Me 2-CF₃-3-Cl −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第３表］（続き） −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
Me 2-CF₃-3-Br Me 2-CF₃-3-Me Me 2,3-di-CF₃ Me 2-CF₃-3-OMe Me 2-CF₃-3-OCF₃ Me 2-OMe-3-F Me 2-OMe-3-Cl Me 2-OMe-3-Br Me 2-OMe-3-Me Me 2-OMe-3-CF₃ Me 2,3-di-OMe Me 2-OMe-3-OCF₃ Me 2-OCF₃-3-F Me 2-OCF₃-3-Cl Me 2-OCF₃-3-Br Me 2-OCF₃-3-Me Me 2-OCF₃-3-CF₃ Me 2-OCF₃-3-OMe Me 2,3-di-OCF₃ Me 2,4-di-F Me 2-F-4-Cl Me 2-F-4-Br Me 2-F-4-Me Me 2-F-4-CF₃ Me 2-F-4-OMe Me 2-F-4-OCF₃ Me 2-Cl-4-F iPr 3,4-di-F Me 2,4-di-Cl iPr 3-F-4-Cl Me 2-Cl-4-Br iPr 3-F-4-Br Me 2-Cl-4-Me iPr 3-F-4-Me Me 2-Cl-4-CF₃ Me 2-Cl-4-OMe iPr 3-F-4-OMe Me 2-Cl-4-OCF₃ Me 2-Br-4-F iPr 3-Cl-4-F Me 2-Br-4-Cl iPr 3,4-di-Cl Me 2,4-di-Br iPr 3-Cl-4-Br Me 2-Br-4-Me iPr 3-Cl-4-Me Me 2-Br-4-CF₃ Me 2-Br-4-OMe iPr 3-Cl-4-OMe −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第３表］（続き） −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
Me 2-Br-4-OCF₃ Me 2-Me-4-F iPr 3-Br-4-F Me 2-Me-4-Cl iPr 3-Br-4-Cl Me 2-Me-4-Br iPr 3,4-di-Br Me 2,4-di-Me iPr 3-Br-4-Me Me 2-Me-4-CF₃ Me 2-Me-4-OMe iPr 3-Br-4-OMe Me 2-Me-4-OCF₃ Me 2-CF₃-4-F Me 2-CF₃-4-Cl Me 2-CF₃-4-Br Me 2-CF₃-4-Me Me 2,4-di-CF₃ Me 2-CF₃-4-OMe Me 2-CF₃-4-OCF₃ Me 2-OMe-4-F Me 2-OMe-4-Cl Me 2-OMe-4-Br Me 2-OMe-4-Me Me 2-OMe-4-CF₃ Me 2,4-di-OMe Me 2-OMe-4-OCF₃ Me 2-OCF₃-4-F Me 2-OCF₃-4-Cl Me 2-OCF₃-4-Br Me 2-OCF₃-4-Me Me 2-OCF₃-4-CF₃ Me 2-OCF₃-4-OMe Me 2,4-di-OCF₃ Me 3,4-di-F Me 3-F-4-Cl Me 3-F-4-Br Me 3-F-4-Me Me 3-F-4-CF₃ Me 3-F-4-OMe Me 3-F-4-OCF₃ Me 3-Cl-4-F U-4a 2,3-di-F Me 3,4-di-Cl U-4a 2-F-3-Cl Me 3-Cl-4-Br U-4a 2-F-3-Br −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第３表］（続き） −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
Me 3-Cl-4-Me U-4a 2-F-3-Me Me 3-Cl-4-CF₃ Me 3-Cl-4-OMe U-4a 2-F-3-OMe Me 3-Cl-4-OCF₃ Me 3-Br-4-F U-4a 2-Cl-3-F Me 3-Br-4-Cl U-4a 2,3-di-Cl Me 3,4-di-Br U-4a 2-Cl-3-Br Me 3-Br-4-Me U-4a 2-Cl-3-Me Me 3-Br-4-CF₃ Me 3-Br-4-OMe U-4a 2-Cl-3-OMe Me 3-Br-4-OCF₃ Me 3-Me-4-F U-4a 2-Br-3-F Me 3-Me-4-Cl U-4a 2-Br-3-Cl Me 3-Me-4-Br U-4a 2,3-di-Br Me 3,4-di-Me U-4a 2-Br-3-Me Me 3-Me-4-CF₃ Me 3-Me-4-OMe U-4a 2-Br-3-OMe Me 3-Me-4-OCF₃ Me 3-CF₃-4-F Me 3-CF₃-4-Cl Me 3-CF₃-4-Br Me 3-CF₃-4-Me Me 3,4-di-CF₃ Me 3-CF₃-4-OMe Me 3-CF₃-4-OCF₃ Me 3-OMe-4-F Me 3-OMe-4-Cl Me 3-OMe-4-Br Me 3-OMe-4-Me Me 3-OMe-4-CF₃ Me 3,4-di-OMe Me 3-OMe-4-OCF₃ Me 3-OCF₃-4-F Me 3-OCF₃-4-Cl Me 3-OCF₃-4-Br Me 3-OCF₃-4-Me Me 3-OCF₃-4-CF₃ Me 3-OCF₃-4-OMe Me 3,4-di-OCF₃ −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第３表］（続き） −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
Et 2,3-di-F Et 2-F-3-Cl Et 2-F-3-Br Et 2-F-3-Me Et 2-F-3-CF₃ Et 2-F-3-OMe Et 2-F-3-OCF₃ Et 2-Cl-3-F U-4a 2,4-di-F Et 2,3-di-Cl U-4a 2-F-4-Cl Et 2-Cl-3-Br U-4a 2-F-4-Br Et 2-Cl-3-Me U-4a 2-F-4-Me Et 2-Cl-3-CF₃ Et 2-Cl-3-OMe U-4a 2-F-4-OMe Et 2-Cl-3-OCF₃ Et 2-Br-3-F U-4a 2-Cl-4-F Et 2-Br-3-Cl U-4a 2,4-di-Cl Et 2,3-di-Br U-4a 2-Cl-4-Br Et 2-Br-3-Me U-4a 2-Cl-4-Me Et 2-Br-3-CF₃ Et 2-Br-3-OMe U-4a 2-Cl-4-OMe Et 2-Br-3-OCF₃ Et 2-Me-3-F U-4a 2-Br-4-F Et 2-Me-3-Cl U-4a 2-Br-4-Cl Et 2-Me-3-Br U-4a 2,4-di-Br Et 2,3-di-Me U-4a 2-Br-4-Me Et 2-Me-3-CF₃ Et 2-Me-3-OMe U-4a 2-Br-4-OMe Et 2-Me-3-OCF₃ Et 2-CF₃-3-F Et 2-CF₃-3-Cl Et 2-CF₃-3-Br Et 2-CF₃-3-Me Et 2,3-di-CF₃ Et 2-CF₃-3-OMe Et 2-CF₃-3-OCF₃ Et 2-OMe-3-F Et 2-OMe-3-Cl Et 2-OMe-3-Br Et 2-OMe-3-Me −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第３表］（続き） −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
Et 2-OMe-3-CF₃ Et 2,3-di-OMe Et 2-OMe-3-OCF₃ Et 2-OCF₃-3-F Et 2-OCF₃-3-Cl Et 2-OCF₃-3-Br Et 2-OCF₃-3-Me Et 2-OCF₃-3-CF₃ Et 2-OCF₃-3-OMe Et 2,3-di-OCF₃ Et 2,4-di-F Et 2-F-4-Cl Et 2-F-4-Br Et 2-F-4-Me Et 2-F-4-CF₃ Et 2-F-4-OMe Et 2-F-4-OCF₃ Et 2-Cl-4-F U-4a 3,4-di-F Et 2,4-di-Cl U-4a 3-F-4-Cl Et 2-Cl-4-Br U-4a 3-F-4-Br Et 2-Cl-4-Me U-4a 3-F-4-Me Et 2-Cl-4-CF₃ Et 2-Cl-4-OMe U-4a 3-F-4-OMe Et 2-Cl-4-OCF₃ −−−−−−−−− −−−−−−−−− −−−−−−−−−−−
［第４表］ [Table 3] [Table ［第３表］（続き）［第３表］（続き）
R³ Z R³ Z
U-4a 3-Cl-4-F
U-4a 3,4-di-Cl
U-4a 3-Cl-4-Br
U-4a 3-Cl-4-Me
Et 2-Br-4-CF₃ U-4a 3-Cl-4-CF₃
U-4a 3-Cl-4-OMe
Et 2-Br-4-OCF₃ U-4a 3-Cl-4-OCF₃
U-4a 3-Br-4-F
U-4a 3-Br-4-Cl
U-4a 3,4-di-Br
U-4a 3-Br-4-Me
Et 2-Me-4-CF₃ U-4a 3-Br-4-CF₃
U-4a 3-Br-4-OMe
Et 2-Me-4-OCF₃ U-4a 3-Br-4-OCF₃
2-CF₃-4-F U-4a 3-Me-4-F
2-CF₃-4-Cl U-4a 3-Me-4-Cl
2-CF₃-4-Br U-4a 3-Me-4-Br
2-CF₃-4-Me U-4a 3,4-di-Me
Et 2,4-di-CF₃ U-4a 3-Me-4-CF₃
2-CF₃-4-OMe U-4a 3-Me-4-OMe
Et 2-CF₃-4-OCF₃ U-4a 3-Me-4-OCF₃
U-4a 3-CF₃-4-F
U-4a 3-CF₃-4-Cl
U-4a 3-CF₃-4-Br
U-4a 3-CF₃-4-Me
Et 2-OMe-4-CF₃ U-4a 3,4-di-CF₃
U-4a 3-CF₃-4-OMe
Et 2-OMe-4-OCF₃ U-4a 3-CF₃-4-OCF₃
2-OCF₃-4-F U-4a 3-OMe-4-F
2-OCF₃-4-Cl U-4a 3-OMe-4-Cl
2-OCF₃-4-Br U-4a 3-OMe-4-Br
2-OCF₃-4-Me U-4a 3-OMe-4-Me
Et 2-OCF₃-4-CF₃ U-4a 3-OMe-4-CF₃
2-OCF₃-4-OMe U-4a 3,4-di-OMe
Et 2,4-di-OCF₃ U-4a 3-OMe-4-OCF₃
U-4a 3-OCF₃-4-F
U-4a 3-OCF₃-4-Cl
U-4a 3-OCF₃-4-Br
U-4a 3-OCF₃-4-Me
［第３表］（続き）［第３表］（続き）
R³ Z R³ Z
Et 3-F-4-CF₃ U-4a 3-OCF₃-4-CF₃
U-4a 3-OCF₃-4-OMe
Et 3-F-4-OCF₃ U-4a 3,4-di-OCF₃
CF₃ 2,3-di-F
CF₃ 2-F-3-Cl
CF₃ 2-F-3-Br
CF₃ 2-F-3-Me
Et 3-Cl-4-CF₃ CF₃ 2-F-3-CF₃
CF₃ 2-F-3-OMe
Et 3-Cl-4-OCF₃ CF₃ 2-F-3-OCF₃
CF₃ 2-Cl-3-F
CF₃ 2,3-di-Cl
CF₃ 2-Cl-3-Br
CF₃ 2-Cl-3-Me
Et 3-Br-4-CF₃ CF₃ 2-Cl-3-CF₃
CF₃ 2-Cl-3-OMe
Et 3-Br-4-OCF₃ CF₃ 2-Cl-3-OCF₃
CF₃ 2-Br-3-F
CF₃ 2-Br-3-Cl
CF₃ 2,3-di-Br
CF₃ 2-Br-3-Me
Et 3-Me-4-CF₃ CF₃ 2-Br-3-CF₃
CF₃ 2-Br-3-OMe
Et 3-Me-4-OCF₃ CF₃ 2-Br-3-OCF₃
3-CF₃-4-F CF₃ 2-Me-3-F
3-CF₃-4-Cl CF₃ 2-Me-3-Cl
3-CF₃-4-Br CF₃ 2-Me-3-Br
3-CF₃-4-Me CF₃ 2,3-di-Me
Et 3,4-di-CF₃ CF₃ 2-Me-3-CF₃
3-CF₃-4-OMe CF₃ 2-Me-3-OMe
Et 3-CF₃-4-OCF₃ CF₃ 2-Me-3-OCF₃
CF₃ 2-CF₃-3-F
CF₃ 2-CF₃-3-Cl
CF₃ 2-CF₃-3-Br
CF₃ 2-CF₃-3-Me
Et 3-OMe-4-CF₃ CF₃ 2,3-di-CF₃
CF₃ 2-CF₃-3-OMe
Et 3-OMe-4-OCF₃ CF₃ 2-CF₃-3-OCF₃
3-OCF₃-4-F CF₃ 2-OMe-3-F
［第３表］（続き）［第３表］（続き）
R³ Z R³ Z
3-OCF₃-4-Cl CF₃ 2-OMe-3-Cl
3-OCF₃-4-Br CF₃ 2-OMe-3-Br
3-OCF₃-4-Me CF₃ 2-OMe-3-Me
Et 3-OCF₃-4-CF₃ CF₃ 2-OMe-3-CF₃
3-OCF₃-4-OMe CF₃ 2,3-di-OMe
Et 3,4-di-OCF₃ CF₃ 2-OMe-3-OCF₃
iPr 2,3-di-F CF₃ 2-OCF₃-3-F
iPr 2-F-3-Cl CF₃ 2-OCF₃-3-Cl
iPr 2-F-3-Br CF₃ 2-OCF₃-3-Br
iPr 2-F-3-Me CF₃ 2-OCF₃-3-Me
iPr 2-F-3-CF₃ CF₃ 2-OCF₃-3-CF₃
iPr 2-F-3-OMe CF₃ 2-OCF₃-3-OMe
iPr 2-F-3-OCF₃ CF₃ 2,3-di-OCF₃
iPr 2-Cl-3-F CF₃ 2,4-di-F
iPr 2,3-di-Cl CF₃ 2-F-4-Cl
iPr 2-Cl-3-Br CF₃ 2-F-4-Br
iPr 2-Cl-3-Me CF₃ 2-F-4-Me
iPr 2-Cl-3-CF₃ CF₃ 2-F-4-CF₃
iPr 2-Cl-3-OMe CF₃ 2-F-4-OMe
iPr 2-Cl-3-OCF₃ CF₃ 2-F-4-OCF₃
iPr 2-Br-3-F CF₃ 2-Cl-4-F
iPr 2-Br-3-Cl CF₃ 2,4-di-Cl
iPr 2,3-di-Br CF₃ 2-Cl-4-Br
iPr 2-Br-3-Me CF₃ 2-Cl-4-Me
iPr 2-Br-3-CF₃ CF₃ 2-Cl-4-CF₃
iPr 2-Br-3-OMe CF₃ 2-Cl-4-OMe
iPr 2-Br-3-OCF₃ CF₃ 2-Cl-4-OCF₃
CF₃ 2-Br-4-F
CF₃ 2-Br-4-Cl
CF₃ 2,4-di-Br
CF₃ 2-Br-4-Me
iPr 2-Me-3-CF₃ CF₃ 2-Br-4-CF₃
CF₃ 2-Br-4-OMe
iPr 2-Me-3-OCF₃ CF₃ 2-Br-4-OCF₃
iPr 2-CF₃-3-F CF₃ 2-Me-4-F
iPr 2-CF₃-3-Cl CF₃ 2-Me-4-Cl
iPr 2-CF₃-3-Br CF₃ 2-Me-4-Br
iPr 2-CF₃-3-Me CF₃ 2,4-di-Me
iPr 2,3-di-CF₃ CF₃ 2-Me-4-CF₃
［第３表］（続き）［第３表］（続き）
R³ Z R³ Z
iPr 2-CF₃-3-OMe CF₃ 2-Me-4-OMe
iPr 2-CF₃-3-OCF₃ CF₃ 2-Me-4-OCF₃
CF₃ 2-CF₃-4-F
CF₃ 2-CF₃-4-Cl
CF₃ 2-CF₃-4-Br
CF₃ 2-CF₃-4-Me
iPr 2-OMe-3-CF₃ CF₃ 2,4-di-CF₃
CF₃ 2-CF₃-4-OMe
iPr 2-OMe-3-OCF₃ CF₃ 2-CF₃-4-OCF₃
iPr 2-OCF₃-3-F CF₃ 2-OMe-4-F
iPr 2-OCF₃-3-Cl CF₃ 2-OMe-4-Cl
iPr 2-OCF₃-3-Br CF₃ 2-OMe-4-Br
iPr 2-OCF₃-3-Me CF₃ 2-OMe-4-Me
iPr 2-OCF₃-3-CF₃ CF₃ 2-OMe-4-CF₃
iPr 2-OCF₃-3-OMe CF₃ 2,4-di-OMe
iPr 2,3-di-OCF₃ CF₃ 2-OMe-4-OCF₃
CF₃ 2-OCF₃-4-F
CF₃ 2-OCF₃-4-Cl
CF₃ 2-OCF₃-4-Br
CF₃ 2-OCF₃-4-Me
iPr 2-F-4-CF₃ CF₃ 2-OCF₃-4-CF₃
CF₃ 2-OCF₃-4-OMe
iPr 2-F-4-OCF₃ CF₃ 2,4-di-OCF₃
CF₃ 3,4-di-F
CF₃ 3-F-4-Cl
CF₃ 3-F-4-Br
CF₃ 3-F-4-Me
iPr 2-Cl-4-CF₃ CF₃ 3-F-4-CF₃
CF₃ 3-F-4-OMe
iPr 2-Cl-4-OCF₃ CF₃ 3-F-4-OCF₃
CF₃ 3-Cl-4-F
CF₃ 3,4-di-Cl
CF₃ 3-Cl-4-Br
CF₃ 3-Cl-4-Me
iPr 2-Br-4-CF₃ CF₃ 3-Cl-4-CF₃
CF₃ 3-Cl-4-OMe
iPr 2-Br-4-OCF₃ CF₃ 3-Cl-4-OCF₃
iPr 2-Me-4-F CF₃ 3-Br-4-F
iPr 2-Me-4-Cl CF₃ 3-Br-4-Cl
［第３表］（続き）［第３表］（続き）
R³ Z R³ Z
iPr 2-Me-4-Br CF₃ 3,4-di-Br
iPr 2,4-di-Me CF₃ 3-Br-4-Me
iPr 2-Me-4-CF₃ CF₃ 3-Br-4-CF₃
iPr 2-Me-4-OMe CF₃ 3-Br-4-OMe
iPr 2-Me-4-OCF₃ CF₃ 3-Br-4-OCF₃
iPr 2-CF₃-4-F CF₃ 3-Me-4-F
iPr 2-CF₃-4-Cl CF₃ 3-Me-4-Cl
iPr 2-CF₃-4-Br CF₃ 3-Me-4-Br
iPr 2-CF₃-4-Me CF₃ 3,4-di-Me
iPr 2,4-di-CF₃ CF₃ 3-Me-4-CF₃
iPr 2-CF₃-4-OMe CF₃ 3-Me-4-OMe
iPr 2-CF₃-4-OCF₃ CF₃ 3-Me-4-OCF₃
iPr 2-OMe-4-F CF₃ 3-CF₃-4-F
iPr 2-OMe-4-Cl CF₃ 3-CF₃-4-Cl
iPr 2-OMe-4-Br CF₃ 3-CF₃-4-Br
iPr 2-OMe-4-Me CF₃ 3-CF₃-4-Me
iPr 2-OMe-4-CF₃ CF₃ 3,4-di-CF₃
iPr 2,4-di-OMe CF₃ 3-CF₃-4-OMe
iPr 2-OMe-4-OCF₃ CF₃ 3-CF₃-4-OCF₃
iPr 2-OCF₃-4-F CF₃ 3-OMe-4-F
iPr 2-OCF₃-4-Cl CF₃ 3-OMe-4-Cl
iPr 2-OCF₃-4-Br CF₃ 3-OMe-4-Br
iPr 2-OCF₃-4-Me CF₃ 3-OMe-4-Me
iPr 2-OCF₃-4-CF₃ CF₃ 3-OMe-4-CF₃
iPr 2-OCF₃-4-OMe CF₃ 3,4-di-OMe
iPr 2,4-di-OCF₃ CF₃ 3-OMe-4-OCF₃
CF₃ 3-OCF₃-4-F
CF₃ 3-OCF₃-4-Cl
CF₃ 3-OCF₃-4-Br
CF₃ 3-OCF₃-4-Me
iPr 3-F-4-CF₃ CF₃ 3-OCF₃-4-CF₃
CF₃ 3-OCF₃-4-OMe
iPr 3-F-4-OCF₃ CF₃ 3,4-di-OCF₃
cPr 2,3-di-F
cPr 2-F-3-Cl
cPr 2-F-3-Br
cPr 2-F-3-Me
iPr 3-Cl-4-CF₃ cPr 2-F-3-CF₃
cPr 2-F-3-OMe
［第３表］（続き）［第３表］（続き）
R³ Z R³ Z
iPr 3-Cl-4-OCF₃ cPr 2-F-3-OCF₃
cPr 2-Cl-3-F
cPr 2,3-di-Cl
cPr 2-Cl-3-Br
cPr 2-Cl-3-Me
iPr 3-Br-4-CF₃ cPr 2-Cl-3-CF₃
cPr 2-Cl-3-OMe
iPr 3-Br-4-OCF₃ cPr 2-Cl-3-OCF₃
iPr 3-Me-4-F cPr 2-Br-3-F
iPr 3-Me-4-Cl cPr 2-Br-3-Cl
iPr 3-Me-4-Br cPr 2,3-di-Br
iPr 3,4-di-Me cPr 2-Br-3-Me
iPr 3-Me-4-CF₃ cPr 2-Br-3-CF₃
iPr 3-Me-4-OMe cPr 2-Br-3-OMe
iPr 3-Me-4-OCF₃ cPr 2-Br-3-OCF₃
iPr 3-CF₃-4-F cPr 2-Me-3-F
iPr 3-CF₃-4-Cl cPr 2-Me-3-Cl
iPr 3-CF₃-4-Br cPr 2-Me-3-Br
iPr 3-CF₃-4-Me cPr 2,3-di-Me
iPr 3,4-di-CF₃ cPr 2-Me-3-CF₃
iPr 3-CF₃-4-OMe cPr 2-Me-3-OMe
iPr 3-CF₃-4-OCF₃ cPr 2-Me-3-OCF₃
iPr 3-OMe-4-F cPr 2-CF₃-3-F
iPr 3-OMe-4-Cl cPr 2-CF₃-3-Cl
iPr 3-OMe-4-Br cPr 2-CF₃-3-Br
iPr 3-OMe-4-Me cPr 2-CF₃-3-Me
iPr 3-OMe-4-CF₃ cPr 2,3-di-CF₃
iPr 3,4-di-OMe cPr 2-CF₃-3-OMe
iPr 3-OMe-4-OCF₃ cPr 2-CF₃-3-OCF₃
iPr 3-OCF₃-4-F cPr 2-OMe-3-F
iPr 3-OCF₃-4-Cl cPr 2-OMe-3-Cl
iPr 3-OCF₃-4-Br cPr 2-OMe-3-Br
iPr 3-OCF₃-4-Me cPr 2-OMe-3-Me
iPr 3-OCF₃-4-CF₃ cPr 2-OMe-3-CF₃
iPr 3-OCF₃-4-OMe cPr 2,3-di-OMe
iPr 3,4-di-OCF₃ cPr 2-OMe-3-OCF₃
cPr 2-OCF₃-3-F
cPr 2-OCF₃-3-Cl
cPr 2-OCF₃-3-Br
［第３表］（続き）［第３表］（続き）
R³ Z R³ Z
cPr 2-OCF₃-3-Me
U-4a 2-F-3-CF₃ cPr 2-OCF₃-3-CF₃
cPr 2-OCF₃-3-OMe
U-4a 2-F-3-OCF₃ cPr 2,3-di-OCF₃
cPr 2,4-di-F
cPr 2-F-4-Cl
cPr 2-F-4-Br
cPr 2-F-4-Me
U-4a 2-Cl-3-CF₃ cPr 2-F-4-CF₃
cPr 2-F-4-OMe
U-4a 2-Cl-3-OCF₃ cPr 2-F-4-OCF₃
cPr 2-Cl-4-F
cPr 2,4-di-Cl
cPr 2-Cl-4-Br
cPr 2-Cl-4-Me
U-4a 2-Br-3-CF₃ cPr 2-Cl-4-CF₃
cPr 2-Cl-4-OMe
U-4a 2-Br-3-OCF₃ cPr 2-Cl-4-OCF₃
U-4a 2-Me-3-F cPr 2-Br-4-F
U-4a 2-Me-3-Cl cPr 2-Br-4-Cl
U-4a 2-Me-3-Br cPr 2,4-di-Br
U-4a 2,3-di-Me cPr 2-Br-4-Me
U-4a 2-Me-3-CF₃ cPr 2-Br-4-CF₃
U-4a 2-Me-3-OMe cPr 2-Br-4-OMe
U-4a 2-Me-3-OCF₃ cPr 2-Br-4-OCF₃
U-4a 2-CF₃-3-F cPr 2-Me-4-F
U-4a 2-CF₃-3-Cl cPr 2-Me-4-Cl
U-4a 2-CF₃-3-Br cPr 2-Me-4-Br
U-4a 2-CF₃-3-Me cPr 2,4-di-Me
U-4a 2,3-di-CF₃ cPr 2-Me-4-CF₃
U-4a 2-CF₃-3-OMe cPr 2-Me-4-OMe
U-4a 2-CF₃-3-OCF₃ cPr 2-Me-4-OCF₃
U-4a 2-OMe-3-F cPr 2-CF₃-4-F
U-4a 2-OMe-3-Cl cPr 2-CF₃-4-Cl
U-4a 2-OMe-3-Br cPr 2-CF₃-4-Br
U-4a 2-OMe-3-Me cPr 2-CF₃-4-Me
U-4a 2-OMe-3-CF₃ cPr 2,4-di-CF₃
U-4a 2,3-di-OMe cPr 2-CF₃-4-OMe
U-4a 2-OMe-3-OCF₃ cPr 2-CF₃-4-OCF₃
［第３表］（続き）［第３表］（続き）
R³ Z R³ Z
U-4a 2-OCF₃-3-F cPr 2-OMe-4-F
U-4a 2-OCF₃-3-Cl cPr 2-OMe-4-Cl
U-4a 2-OCF₃-3-Br cPr 2-OMe-4-Br
U-4a 2-OCF₃-3-Me cPr 2-OMe-4-Me
U-4a 2-OCF₃-3-CF₃ cPr 2-OMe-4-CF₃
U-4a 2-OCF₃-3-OMe cPr 2,4-di-OMe
U-4a 2,3-di-OCF₃ cPr 2-OMe-4-OCF₃
cPr 2-OCF₃-4-F
cPr 2-OCF₃-4-Cl
cPr 2-OCF₃-4-Br
cPr 2-OCF₃-4-Me
U-4a 2-F-4-CF₃ cPr 2-OCF₃-4-CF₃
cPr 2-OCF₃-4-OMe
U-4a 2-F-4-OCF₃ cPr 2,4-di-OCF₃
cPr 3,4-di-F
cPr 3-F-4-Cl
cPr 3-F-4-Br
cPr 3-F-4-Me
U-4a 2-Cl-4-CF₃ cPr 3-F-4-CF₃
cPr 3-F-4-OMe
U-4a 2-Cl-4-OCF₃ cPr 3-F-4-OCF₃
cPr 3-Cl-4-F
cPr 3,4-di-Cl
cPr 3-Cl-4-Br
cPr 3-Cl-4-Me
U-4a 2-Br-4-CF₃ cPr 3-Cl-4-CF₃
cPr 3-Cl-4-OMe
U-4a 2-Br-4-OCF₃ cPr 3-Cl-4-OCF₃
U-4a 2-Me-4-F cPr 3-Br-4-F
U-4a 2-Me-4-Cl cPr 3-Br-4-Cl
U-4a 2-Me-4-Br cPr 3,4-di-Br
U-4a 2,4-di-Me cPr 3-Br-4-Me
U-4a 2-Me-4-CF₃ cPr 3-Br-4-CF₃
U-4a 2-Me-4-OMe cPr 3-Br-4-OMe
U-4a 2-Me-4-OCF₃ cPr 3-Br-4-OCF₃
U-4a 2-CF₃-4-F cPr 3-Me-4-F
U-4a 2-CF₃-4-Cl cPr 3-Me-4-Cl
U-4a 2-CF₃-4-Br cPr 3-Me-4-Br
U-4a 2-CF₃-4-Me cPr 3,4-di-Me
［第３表］（続き）［第３表］（続き）
R³ Z R³ Z
U-4a 2,4-di-CF₃ cPr 3-Me-4-CF₃
U-4a 2-CF₃-4-OMe cPr 3-Me-4-OMe
U-4a 2-CF₃-4-OCF₃ cPr 3-Me-4-OCF₃
U-4a 2-OMe-4-F cPr 3-CF₃-4-F
U-4a 2-OMe-4-Cl cPr 3-CF₃-4-Cl
U-4a 2-OMe-4-Br cPr 3-CF₃-4-Br
U-4a 2-OMe-4-Me cPr 3-CF₃-4-Me
U-4a 2-OMe-4-CF₃ cPr 3,4-di-CF₃
U-4a 2,4-di-OMe cPr 3-CF₃-4-OMe
U-4a 2-OMe-4-OCF₃ cPr 3-CF₃-4-OCF₃
U-4a 2-OCF₃-4-F cPr 3-OMe-4-F
U-4a 2-OCF₃-4-Cl cPr 3-OMe-4-Cl
U-4a 2-OCF₃-4-Br cPr 3-OMe-4-Br
U-4a 2-OCF₃-4-Me cPr 3-OMe-4-Me
U-4a 2-OCF₃-4-CF₃ cPr 3-OMe-4-CF₃
U-4a 2-OCF₃-4-OMe cPr 3,4-di-OMe
U-4a 2,4-di-OCF₃ cPr 3-OMe-4-OCF₃
cPr 3-OCF₃-4-F
cPr 3-OCF₃-4-Cl
cPr 3-OCF₃-4-Br
cPr 3-OCF₃-4-Me
U-4a 3-F-4-CF₃ cPr 3-OCF₃-4-CF₃
cPr 3-OCF₃-4-OMe
U-4a 3-F-4-OCF₃ cPr 3,4-di-OCF₃
3] (continued) [Table 3] (continued)
--------- --------- --------
R ³ ZR ³ ZR ³ Z
--------- --------- --------
Me 2-F Et 2-Br-4-F U-4a 3-Cl-4-F
Me 2-Cl Et 2-Br-4-Cl U-4a 3,4-di-Cl
Me 2-Br Et 2,4-di-Br U-4a 3-Cl-4-Br
Me 2-Me Et 2-Br-4-Me U-4a 3-Cl-4-Me
Me 2-CF ₃ Et 2-Br-4-CF ₃ U-4a 3-Cl-4-CF ₃
Me 2-OMe Et 2-Br-4-OMe U-4a 3-Cl-4-OMe
Me 2-OCF ₃ Et 2-Br-4-OCF ₃ U-4a 3-Cl-4-OCF ₃
Me 3-F Et 2-Me-4-F U-4a 3-Br-4-F
Me 3-Cl Et 2-Me-4-Cl U-4a 3-Br-4-Cl
Me 3-Br Et 2-Me-4-Br U-4a 3,4-di-Br
Me 3-Me Et 2,4-di-Me U-4a 3-Br-4-Me
Me 3-CF ₃ Et 2-Me-4-CF ₃ U-4a 3-Br-4-CF ₃
Me 3-OMe Et 2-Me-4-OMe U-4a 3-Br-4-OMe
Me 3-OCF ₃ Et 2-Me-4-OCF ₃ U-4a 3-Br-4-OCF ₃
Me 4-F Et 2-CF ₃ -4-F U-4a 3-Me-4-F
Me 4-Cl Et 2-CF ₃ -4-Cl U-4a 3-Me-4-Cl
Me 4-Br Et 2-CF ₃ -4-Br U-4a 3-Me-4-Br
Me 4-Me Et 2-CF ₃ -4-Me U-4a 3,4-di-Me
Me 4-CF ₃ Et 2,4-di-CF ₃ U-4a 3-Me-4-CF ₃
Me 4-OMe Et 2-CF ₃ -4-OMe U-4a 3-Me-4-OMe
Me 4-OCF ₃ Et 2-CF ₃ -4-OCF ₃ U-4a 3-Me-4-OCF ₃
Et 2-F Et 2-OMe-4-F U-4a 3-CF ₃ -4-F
Et 2-Cl Et 2-OMe-4-Cl U-4a 3-CF ₃ -4-Cl
Et 2-Br Et 2-OMe-4-Br U-4a 3-CF ₃ -4-Br
Et 2-Me Et 2-OMe-4-Me U-4a 3-CF ₃ -4-Me
Et 2-CF ₃ Et 2-OMe-4-CF ₃ U-4a 3,4-di-CF ₃
Et 2-OMe Et 2,4-di-OMe U-4a 3-CF ₃ -4-OMe
Et 2-OCF ₃ Et 2-OMe-4-OCF ₃ U-4a 3-CF ₃ -4-OCF ₃
Et 3-F Et 2-OCF ₃ -4-F U-4a 3-OMe-4-F
Et 3-Cl Et 2-OCF ₃ -4-Cl U-4a 3-OMe-4-Cl
Et 3-Br Et 2-OCF ₃ -4-Br U-4a 3-OMe-4-Br
Et 3-Me Et 2-OCF ₃ -4-Me U-4a 3-OMe-4-Me
Et 3-CF ₃ Et 2-OCF ₃ -4-CF ₃ U-4a 3-OMe-4-CF ₃
Et 3-OMe Et 2-OCF ₃ -4-OMe U-4a 3,4-di-OMe
Et 3-OCF ₃ Et 2,4-di-OCF ₃ U-4a 3-OMe-4-OCF ₃
Et 4-F Et 3,4-di-F U-4a 3-OCF ₃ -4-F
Et 4-Cl Et 3-F-4-Cl U-4a 3-OCF ₃ -4-Cl
Et 4-Br Et 3-F-4-Br U-4a 3-OCF ₃ -4-Br
Et 4-Me Et 3-F-4-Me U-4a 3-OCF ₃ -4-Me
--------- --------- --------
[Table 3] (continued) [Table 3] (continued) [Table 3] (continued)
--------- --------- --------
R ³ ZR ³ ZR ³ Z
--------- --------- --------
Et 4-CF ₃ Et 3-F-4-CF ₃ U-4a 3-OCF ₃ -4-CF ₃
Et 4-OMe Et 3-F-4-OMe U-4a 3-OCF ₃ -4-OMe
Et 4-OCF ₃ Et 3-F-4-OCF ₃ U-4a 3,4-di-OCF ₃
iPr 2-F Et 3-Cl-4-F CF ₃ 2,3-di-F
iPr 2-Cl Et 3,4-di-Cl CF ₃ 2-F-3-Cl
iPr 2-Br Et 3-Cl-4-Br CF ₃ 2-F-3-Br
iPr 2-Me Et 3-Cl-4-Me CF ₃ 2-F-3-Me
iPr 2-CF ₃ Et 3-Cl-4-CF ₃ CF ₃ 2-F-3-CF ₃
iPr 2-OMe Et 3-Cl-4-OMe CF ₃ 2-F-3-OMe
iPr 2-OCF ₃ Et 3-Cl-4-OCF ₃ CF ₃ 2-F-3-OCF ₃
iPr 3-F Et 3-Br-4-F CF ₃ 2-Cl-3-F
iPr 3-Cl Et 3-Br-4-Cl CF ₃ 2,3-di-Cl
iPr 3-Br Et 3,4-di-Br CF ₃ 2-Cl-3-Br
iPr 3-Me Et 3-Br-4-Me CF ₃ 2-Cl-3-Me
iPr 3-CF ₃ Et 3-Br-4-CF ₃ CF ₃ 2-Cl-3-CF ₃
iPr 3-OMe Et 3-Br-4-OMe CF ₃ 2-Cl-3-OMe
iPr 3-OCF ₃ Et 3-Br-4-OCF ₃ CF ₃ 2-Cl-3-OCF ₃
iPr 4-F Et 3-Me-4-F CF ₃ 2-Br-3-F
iPr 4-Cl Et 3-Me-4-Cl CF ₃ 2-Br-3-Cl
iPr 4-Br Et 3-Me-4-Br CF ₃ 2,3-di-Br
iPr 4-Me Et 3,4-di-Me CF ₃ 2-Br-3-Me
iPr 4-CF ₃ Et 3-Me-4-CF ₃ CF ₃ 2-Br-3-CF ₃
iPr 4-OMe Et 3-Me-4-OMe CF ₃ 2-Br-3-OMe
iPr 4-OCF ₃ Et 3-Me-4-OCF ₃ CF ₃ 2-Br-3-OCF ₃
U-4a 2-F Et 3-CF ₃ -4-F CF ₃ 2-Me-3-F
U-4a 2-Cl Et 3-CF ₃ -4-Cl CF ₃ 2-Me-3-Cl
U-4a 2-Br Et 3-CF ₃ -4-Br CF ₃ 2-Me-3-Br
U-4a 2-Me Et 3-CF ₃ -4-Me CF ₃ 2,3-di-Me
U-4a 2-CF ₃ Et 3,4-di-CF ₃ CF ₃ 2-Me-3-CF ₃
U-4a 2-OMe Et 3-CF ₃ -4-OMe CF ₃ 2-Me-3-OMe
U-4a 2-OCF ₃ Et 3-CF ₃ -4-OCF ₃ CF ₃ 2-Me-3-OCF ₃
U-4a 3-F Et 3-OMe-4-F CF ₃ 2-CF ₃ -3-F
U-4a 3-Cl Et 3-OMe-4-Cl CF ₃ 2-CF ₃ -3-Cl
U-4a 3-Br Et 3-OMe-4-Br CF ₃ 2-CF ₃ -3-Br
U-4a 3-Me Et 3-OMe-4-Me CF ₃ 2-CF ₃ -3-Me
U-4a 3-CF ₃ Et 3-OMe-4-CF ₃ CF ₃ 2,3-di-CF ₃
U-4a 3-OMe Et 3,4-di-OMe CF ₃ 2-CF ₃ -3-OMe
U-4a 3-OCF ₃ Et 3-OMe-4-OCF ₃ CF ₃ 2-CF ₃ -3-OCF ₃
U-4a 4-F Et 3-OCF ₃ -4-F CF ₃ 2-OMe-3-F
--------- --------- --------
[Table 3] (continued) [Table 3] (continued) [Table 3] (continued)
--------- --------- --------
R ³ ZR ³ ZR ³ Z
--------- --------- --------
U-4a 4-Cl Et 3-OCF ₃ -4-Cl CF ₃ 2-OMe-3-Cl
U-4a 4-Br Et 3-OCF ₃ -4-Br CF ₃ 2-OMe-3-Br
U-4a 4-Me Et 3-OCF ₃ -4-Me CF ₃ 2-OMe-3-Me
U-4a 4-CF ₃ Et 3-OCF ₃ -4-CF ₃ CF ₃ 2-OMe-3-CF ₃
U-4a 4-OMe Et 3-OCF ₃ -4-OMe CF ₃ 2,3-di-OMe
U-4a 4-OCF ₃ Et 3,4-di-OCF ₃ CF ₃ 2-OMe-3-OCF ₃
CF ₃ 2-F iPr 2,3-di-F CF ₃ 2-OCF ₃ -3-F
CF ₃ 2-Cl iPr 2-F-3-Cl CF ₃ 2-OCF ₃ -3-Cl
CF ₃ 2-Br iPr 2-F-3-Br CF ₃ 2-OCF ₃ -3-Br
CF ₃ 2-Me iPr 2-F-3-Me CF ₃ 2-OCF ₃ -3-Me
CF ₃ 2-CF ₃ iPr 2-F-3-CF ₃ CF ₃ 2-OCF ₃ -3-CF ₃
CF ₃ 2-OMe iPr 2-F-3-OMe CF ₃ 2-OCF ₃ -3-OMe
CF ₃ 2-OCF ₃ iPr 2-F-3-OCF ₃ CF ₃ 2,3-di-OCF ₃
CF ₃ 3-F iPr 2-Cl-3-F CF ₃ 2,4-di-F
CF ₃ 3-Cl iPr 2,3-di-Cl CF ₃ 2-F-4-Cl
CF ₃ 3-Br iPr 2-Cl-3-Br CF ₃ 2-F-4-Br
CF ₃ 3-Me iPr 2-Cl-3-Me CF ₃ 2-F-4-Me
CF ₃ 3-CF ₃ iPr 2-Cl-3-CF ₃ CF ₃ 2-F-4-CF ₃
CF ₃ 3-OMe iPr 2-Cl-3-OMe CF ₃ 2-F-4-OMe
CF ₃ 3-OCF ₃ iPr 2-Cl-3-OCF ₃ CF ₃ 2-F-4-OCF ₃
CF ₃ 4-F iPr 2-Br-3-F CF ₃ 2-Cl-4-F
CF ₃ 4-Cl iPr 2-Br-3-Cl CF ₃ 2,4-di-Cl
CF ₃ 4-Br iPr 2,3-di-Br CF ₃ 2-Cl-4-Br
CF ₃ 4-Me iPr 2-Br-3-Me CF ₃ 2-Cl-4-Me
CF ₃ 4-CF ₃ iPr 2-Br-3-CF ₃ CF ₃ 2-Cl-4-CF ₃
CF ₃ 4-OMe iPr 2-Br-3-OMe CF ₃ 2-Cl-4-OMe
CF ₃ 4-OCF ₃ iPr 2-Br-3-OCF ₃ CF ₃ 2-Cl-4-OCF ₃
cPr 2-F iPr 2-Me-3-F CF ₃ 2-Br-4-F
cPr 2-Cl iPr 2-Me-3-Cl CF ₃ 2-Br-4-Cl
cPr 2-Br iPr 2-Me-3-Br CF ₃ 2,4-di-Br
cPr 2-Me iPr 2,3-di-Me CF ₃ 2-Br-4-Me
cPr 2-CF ₃ iPr 2-Me-3-CF ₃ CF ₃ 2-Br-4-CF ₃
cPr 2-OMe iPr 2-Me-3-OMe CF ₃ 2-Br-4-OMe
cPr 2-OCF ₃ iPr 2-Me-3-OCF ₃ CF ₃ 2-Br-4-OCF ₃
cPr 3-F iPr 2-CF ₃ -3-F CF ₃ 2-Me-4-F
cPr 3-Cl iPr 2-CF ₃ -3-Cl CF ₃ 2-Me-4-Cl
cPr 3-Br iPr 2-CF ₃ -3-Br CF ₃ 2-Me-4-Br
cPr 3-Me iPr 2-CF ₃ -3-Me CF ₃ 2,4-di-Me
cPr 3-CF ₃ iPr 2,3-di-CF ₃ CF ₃ 2-Me-4-CF ₃
--------- --------- --------
[Table 3] (continued) [Table 3] (continued) [Table 3] (continued)
--------- --------- --------
R ³ ZR ³ ZR ³ Z
--------- --------- --------
cPr 3-OMe iPr 2-CF ₃ -3-OMe CF ₃ 2-Me-4-OMe
cPr 3-OCF ₃ iPr 2-CF ₃ -3-OCF ₃ CF ₃ 2-Me-4-OCF ₃
cPr 4-F iPr 2-OMe-3-F CF ₃ 2-CF ₃ -4-F
cPr 4-Cl iPr 2-OMe-3-Cl CF ₃ 2-CF ₃ -4-Cl
cPr 4-Br iPr 2-OMe-3-Br CF ₃ 2-CF ₃ -4-Br
cPr 4-Me iPr 2-OMe-3-Me CF ₃ 2-CF ₃ -4-Me
cPr 4-CF ₃ iPr 2-OMe-3-CF ₃ CF ₃ 2,4-di-CF ₃
cPr 4-OMe iPr 2,3-di-OMe CF ₃ 2-CF ₃ -4-OMe
cPr 4-OCF ₃ iPr 2-OMe-3-OCF ₃ CF ₃ 2-CF ₃ -4-OCF ₃
Me 2,3-di-F iPr 2-OCF ₃ -3-F CF ₃ 2-OMe-4-F
Me 2-F-3-Cl iPr 2-OCF ₃ -3-Cl CF ₃ 2-OMe-4-Cl
Me 2-F-3-Br iPr 2-OCF ₃ -3-Br CF ₃ 2-OMe-4-Br
Me 2-F-3-Me iPr 2-OCF ₃ -3-Me CF ₃ 2-OMe-4-Me
Me 2-F-3-CF ₃ iPr 2-OCF ₃ -3-CF ₃ CF ₃ 2-OMe-4-CF ₃
Me 2-F-3-OMe iPr 2-OCF ₃ -3-OMe CF ₃ 2,4-di-OMe
Me 2-F-3-OCF ₃ iPr 2,3-di-OCF ₃ CF ₃ 2-OMe-4-OCF ₃
Me 2-Cl-3-F iPr 2,4-di-F CF ₃ 2-OCF ₃ -4-F
Me 2,3-di-Cl iPr 2-F-4-Cl CF ₃ 2-OCF ₃ -4-Cl
Me 2-Cl-3-Br iPr 2-F-4-Br CF ₃ 2-OCF ₃ -4-Br
Me 2-Cl-3-Me iPr 2-F-4-Me CF ₃ 2-OCF ₃ -4-Me
Me 2-Cl-3-CF ₃ iPr 2-F-4-CF ₃ CF ₃ 2-OCF ₃ -4-CF ₃
Me 2-Cl-3-OMe iPr 2-F-4-OMe CF ₃ 2-OCF ₃ -4-OMe
Me 2-Cl-3-OCF ₃ iPr 2-F-4-OCF ₃ CF ₃ 2,4-di-OCF ₃
Me 2-Br-3-F iPr 2-Cl-4-F CF ₃ 3,4-di-F
Me 2-Br-3-Cl iPr 2,4-di-Cl CF ₃ 3-F-4-Cl
Me 2,3-di-Br iPr 2-Cl-4-Br CF ₃ 3-F-4-Br
Me 2-Br-3-Me iPr 2-Cl-4-Me CF ₃ 3-F-4-Me
Me 2-Br-3-CF ₃ iPr 2-Cl-4-CF ₃ CF ₃ 3-F-4-CF ₃
Me 2-Br-3-OMe iPr 2-Cl-4-OMe CF ₃ 3-F-4-OMe
Me 2-Br-3-OCF ₃ iPr 2-Cl-4-OCF ₃ CF ₃ 3-F-4-OCF ₃
Me 2-Me-3-F iPr 2-Br-4-F CF ₃ 3-Cl-4-F
Me 2-Me-3-Cl iPr 2-Br-4-Cl CF ₃ 3,4-di-Cl
Me 2-Me-3-Br iPr 2,4-di-Br CF ₃ 3-Cl-4-Br
Me 2,3-di-Me iPr 2-Br-4-Me CF ₃ 3-Cl-4-Me
Me 2-Me-3-CF ₃ iPr 2-Br-4-CF ₃ CF ₃ 3-Cl-4-CF ₃
Me 2-Me-3-OMe iPr 2-Br-4-OMe CF ₃ 3-Cl-4-OMe
Me 2-Me-3-OCF ₃ iPr 2-Br-4-OCF ₃ CF ₃ 3-Cl-4-OCF ₃
Me 2-CF ₃ -3-F iPr 2-Me-4-F CF ₃ 3-Br-4-F
Me 2-CF ₃ -3-Cl iPr 2-Me-4-Cl CF ₃ 3-Br-4-Cl
--------- --------- --------
[Table 3] (continued) [Table 3] (continued) [Table 3] (continued)
--------- --------- --------
R ³ ZR ³ ZR ³ Z
--------- --------- --------
Me 2-CF ₃ -3-Br iPr 2-Me-4-Br CF ₃ 3,4-di-Br
Me 2-CF ₃ -3-Me iPr 2,4-di-Me CF ₃ 3-Br-4-Me
Me 2,3-di-CF ₃ iPr 2-Me-4-CF ₃ CF ₃ 3-Br-4-CF ₃
Me 2-CF ₃ -3-OMe iPr 2-Me-4-OMe CF ₃ 3-Br-4-OMe
Me 2-CF ₃ -3-OCF ₃ iPr 2-Me-4-OCF ₃ CF ₃ 3-Br-4-OCF ₃
Me 2-OMe-3-F iPr 2-CF ₃ -4-F CF ₃ 3-Me-4-F
Me 2-OMe-3-Cl iPr 2-CF ₃ -4-Cl CF ₃ 3-Me-4-Cl
Me 2-OMe-3-Br iPr 2-CF ₃ -4-Br CF ₃ 3-Me-4-Br
Me 2-OMe-3-Me iPr 2-CF ₃ -4-Me CF ₃ 3,4-di-Me
Me 2-OMe-3-CF ₃ iPr 2,4-di-CF ₃ CF ₃ 3-Me-4-CF ₃
Me 2,3-di-OMe iPr 2-CF ₃ -4-OMe CF ₃ 3-Me-4-OMe
Me 2-OMe-3-OCF ₃ iPr 2-CF ₃ -4-OCF ₃ CF ₃ 3-Me-4-OCF ₃
Me 2-OCF ₃ -3-F iPr 2-OMe-4-F CF ₃ 3-CF ₃ -4-F
Me 2-OCF ₃ -3-Cl iPr 2-OMe-4-Cl CF ₃ 3-CF ₃ -4-Cl
Me 2-OCF ₃ -3-Br iPr 2-OMe-4-Br CF ₃ 3-CF ₃ -4-Br
Me 2-OCF ₃ -3-Me iPr 2-OMe-4-Me CF ₃ 3-CF ₃ -4-Me
Me 2-OCF ₃ -3-CF ₃ iPr 2-OMe-4-CF ₃ CF ₃ 3,4-di-CF ₃
Me 2-OCF ₃ -3-OMe iPr 2,4-di-OMe CF ₃ 3-CF ₃ -4-OMe
Me 2,3-di-OCF ₃ iPr 2-OMe-4-OCF ₃ CF ₃ 3-CF ₃ -4-OCF ₃
Me 2,4-di-F iPr 2-OCF ₃ -4-F CF ₃ 3-OMe-4-F
Me 2-F-4-Cl iPr 2-OCF ₃ -4-Cl CF ₃ 3-OMe-4-Cl
Me 2-F-4-Br iPr 2-OCF ₃ -4-Br CF ₃ 3-OMe-4-Br
Me 2-F-4-Me iPr 2-OCF ₃ -4-Me CF ₃ 3-OMe-4-Me
Me 2-F-4-CF ₃ iPr 2-OCF ₃ -4-CF ₃ CF ₃ 3-OMe-4-CF ₃
Me 2-F-4-OMe iPr 2-OCF ₃ -4-OMe CF ₃ 3,4-di-OMe
Me 2-F-4-OCF ₃ iPr 2,4-di-OCF ₃ CF ₃ 3-OMe-4-OCF ₃
Me 2-Cl-4-F iPr 3,4-di-F CF ₃ 3-OCF ₃ -4-F
Me 2,4-di-Cl iPr 3-F-4-Cl CF ₃ 3-OCF ₃ -4-Cl
Me 2-Cl-4-Br iPr 3-F-4-Br CF ₃ 3-OCF ₃ -4-Br
Me 2-Cl-4-Me iPr 3-F-4-Me CF ₃ 3-OCF ₃ -4-Me
Me 2-Cl-4-CF ₃ iPr 3-F-4-CF ₃ CF ₃ 3-OCF ₃ -4-CF ₃
Me 2-Cl-4-OMe iPr 3-F-4-OMe CF ₃ 3-OCF ₃ -4-OMe
Me 2-Cl-4-OCF ₃ iPr 3-F-4-OCF ₃ CF ₃ 3,4-di-OCF ₃
Me 2-Br-4-F iPr 3-Cl-4-F cPr 2,3-di-F
Me 2-Br-4-Cl iPr 3,4-di-Cl cPr 2-F-3-Cl
Me 2,4-di-Br iPr 3-Cl-4-Br cPr 2-F-3-Br
Me 2-Br-4-Me iPr 3-Cl-4-Me cPr 2-F-3-Me
Me 2-Br-4-CF ₃ iPr 3-Cl-4-CF ₃ cPr 2-F-3-CF ₃
Me 2-Br-4-OMe iPr 3-Cl-4-OMe cPr 2-F-3-OMe
--------- --------- --------
[Table 3] (continued) [Table 3] (continued) [Table 3] (continued)
--------- --------- --------
R ³ ZR ³ ZR ³ Z
--------- --------- --------
Me 2-Br-4-OCF ₃ iPr 3-Cl-4-OCF ₃ cPr 2-F-3-OCF ₃
Me 2-Me-4-F iPr 3-Br-4-F cPr 2-Cl-3-F
Me 2-Me-4-Cl iPr 3-Br-4-Cl cPr 2,3-di-Cl
Me 2-Me-4-Br iPr 3,4-di-Br cPr 2-Cl-3-Br
Me 2,4-di-Me iPr 3-Br-4-Me cPr 2-Cl-3-Me
Me 2-Me-4-CF ₃ iPr 3-Br-4-CF ₃ cPr 2-Cl-3-CF ₃
Me 2-Me-4-OMe iPr 3-Br-4-OMe cPr 2-Cl-3-OMe
Me 2-Me-4-OCF ₃ iPr 3-Br-4-OCF ₃ cPr 2-Cl-3-OCF ₃
Me 2-CF ₃ -4-F iPr 3-Me-4-F cPr 2-Br-3-F
Me 2-CF ₃ -4-Cl iPr 3-Me-4-Cl cPr 2-Br-3-Cl
Me 2-CF ₃ -4-Br iPr 3-Me-4-Br cPr 2,3-di-Br
Me 2-CF ₃ -4-Me iPr 3,4-di-Me cPr 2-Br-3-Me
Me 2,4-di-CF ₃ iPr 3-Me-4-CF ₃ cPr 2-Br-3-CF ₃
Me 2-CF ₃ -4-OMe iPr 3-Me-4-OMe cPr 2-Br-3-OMe
Me 2-CF ₃ -4-OCF ₃ iPr 3-Me-4-OCF ₃ cPr 2-Br-3-OCF ₃
Me 2-OMe-4-F iPr 3-CF ₃ -4-F cPr 2-Me-3-F
Me 2-OMe-4-Cl iPr 3-CF ₃ -4-Cl cPr 2-Me-3-Cl
Me 2-OMe-4-Br iPr 3-CF ₃ -4-Br cPr 2-Me-3-Br
Me 2-OMe-4-Me iPr 3-CF ₃ -4-Me cPr 2,3-di-Me
Me 2-OMe-4-CF ₃ iPr 3,4-di-CF ₃ cPr 2-Me-3-CF ₃
Me 2,4-di-OMe iPr 3-CF ₃ -4-OMe cPr 2-Me-3-OMe
Me 2-OMe-4-OCF ₃ iPr 3-CF ₃ -4-OCF ₃ cPr 2-Me-3-OCF ₃
Me 2-OCF ₃ -4-F iPr 3-OMe-4-F cPr 2-CF ₃ -3-F
Me 2-OCF ₃ -4-Cl iPr 3-OMe-4-Cl cPr 2-CF ₃ -3-Cl
Me 2-OCF ₃ -4-Br iPr 3-OMe-4-Br cPr 2-CF ₃ -3-Br
Me 2-OCF ₃ -4-Me iPr 3-OMe-4-Me cPr 2-CF ₃ -3-Me
Me 2-OCF ₃ -4-CF ₃ iPr 3-OMe-4-CF ₃ cPr 2,3-di-CF ₃
Me 2-OCF ₃ -4-OMe iPr 3,4-di-OMe cPr 2-CF ₃ -3-OMe
Me 2,4-di-OCF ₃ iPr 3-OMe-4-OCF ₃ cPr 2-CF ₃ -3-OCF ₃
Me 3,4-di-F iPr 3-OCF ₃ -4-F cPr 2-OMe-3-F
Me 3-F-4-Cl iPr 3-OCF ₃ -4-Cl cPr 2-OMe-3-Cl
Me 3-F-4-Br iPr 3-OCF ₃ -4-Br cPr 2-OMe-3-Br
Me 3-F-4-Me iPr 3-OCF ₃ -4-Me cPr 2-OMe-3-Me
Me 3-F-4-CF ₃ iPr 3-OCF ₃ -4-CF ₃ cPr 2-OMe-3-CF ₃
Me 3-F-4-OMe iPr 3-OCF ₃ -4-OMe cPr 2,3-di-OMe
Me 3-F-4-OCF ₃ iPr 3,4-di-OCF ₃ cPr 2-OMe-3-OCF ₃
Me 3-Cl-4-F U-4a 2,3-di-F cPr 2-OCF ₃ -3-F
Me 3,4-di-Cl U-4a 2-F-3-Cl cPr 2-OCF ₃ -3-Cl
Me 3-Cl-4-Br U-4a 2-F-3-Br cPr 2-OCF ₃ -3-Br
--------- --------- --------
[Table 3] (continued) [Table 3] (continued) [Table 3] (continued)
--------- --------- --------
R ³ ZR ³ ZR ³ Z
--------- --------- --------
Me 3-Cl-4-Me U-4a 2-F-3-Me cPr 2-OCF ₃ -3-Me
Me 3-Cl-4-CF ₃ U-4a 2-F-3-CF ₃ cPr 2-OCF ₃ -3-CF ₃
Me 3-Cl-4-OMe U-4a 2-F-3-OMe cPr 2-OCF ₃ -3-OMe
Me 3-Cl-4-OCF ₃ U-4a 2-F-3-OCF ₃ cPr 2,3-di-OCF ₃
Me 3-Br-4-F U-4a 2-Cl-3-F cPr 2,4-di-F
Me 3-Br-4-Cl U-4a 2,3-di-Cl cPr 2-F-4-Cl
Me 3,4-di-Br U-4a 2-Cl-3-Br cPr 2-F-4-Br
Me 3-Br-4-Me U-4a 2-Cl-3-Me cPr 2-F-4-Me
Me 3-Br-4-CF ₃ U-4a 2-Cl-3-CF ₃ cPr 2-F-4-CF ₃
Me 3-Br-4-OMe U-4a 2-Cl-3-OMe cPr 2-F-4-OMe
Me 3-Br-4-OCF ₃ U-4a 2-Cl-3-OCF ₃ cPr 2-F-4-OCF ₃
Me 3-Me-4-F U-4a 2-Br-3-F cPr 2-Cl-4-F
Me 3-Me-4-Cl U-4a 2-Br-3-Cl cPr 2,4-di-Cl
Me 3-Me-4-Br U-4a 2,3-di-Br cPr 2-Cl-4-Br
Me 3,4-di-Me U-4a 2-Br-3-Me cPr 2-Cl-4-Me
Me 3-Me-4-CF ₃ U-4a 2-Br-3-CF ₃ cPr 2-Cl-4-CF ₃
Me 3-Me-4-OMe U-4a 2-Br-3-OMe cPr 2-Cl-4-OMe
Me 3-Me-4-OCF ₃ U-4a 2-Br-3-OCF ₃ cPr 2-Cl-4-OCF ₃
Me 3-CF ₃ -4-F U-4a 2-Me-3-F cPr 2-Br-4-F
Me 3-CF ₃ -4-Cl U-4a 2-Me-3-Cl cPr 2-Br-4-Cl
Me 3-CF ₃ -4-Br U-4a 2-Me-3-Br cPr 2,4-di-Br
Me 3-CF ₃ -4-Me U-4a 2,3-di-Me cPr 2-Br-4-Me
Me 3,4-di-CF ₃ U-4a 2-Me-3-CF ₃ cPr 2-Br-4-CF ₃
Me 3-CF ₃ -4-OMe U-4a 2-Me-3-OMe cPr 2-Br-4-OMe
Me 3-CF ₃ -4-OCF ₃ U-4a 2-Me-3-OCF ₃ cPr 2-Br-4-OCF ₃
Me 3-OMe-4-F U-4a 2-CF ₃ -3-F cPr 2-Me-4-F
Me 3-OMe-4-Cl U-4a 2-CF ₃ -3-Cl cPr 2-Me-4-Cl
Me 3-OMe-4-Br U-4a 2-CF ₃ -3-Br cPr 2-Me-4-Br
Me 3-OMe-4-Me U-4a 2-CF ₃ -3-Me cPr 2,4-di-Me
Me 3-OMe-4-CF ₃ U-4a 2,3-di-CF ₃ cPr 2-Me-4-CF ₃
Me 3,4-di-OMe U-4a 2-CF ₃ -3-OMe cPr 2-Me-4-OMe
Me 3-OMe-4-OCF ₃ U-4a 2-CF ₃ -3-OCF ₃ cPr 2-Me-4-OCF ₃
Me 3-OCF ₃ -4-F U-4a 2-OMe-3-F cPr 2-CF ₃ -4-F
Me 3-OCF ₃ -4-Cl U-4a 2-OMe-3-Cl cPr 2-CF ₃ -4-Cl
Me 3-OCF ₃ -4-Br U-4a 2-OMe-3-Br cPr 2-CF ₃ -4-Br
Me 3-OCF ₃ -4-Me U-4a 2-OMe-3-Me cPr 2-CF ₃ -4-Me
Me 3-OCF ₃ -4-CF ₃ U-4a 2-OMe-3-CF ₃ cPr 2,4-di-CF ₃
Me 3-OCF ₃ -4-OMe U-4a 2,3-di-OMe cPr 2-CF ₃ -4-OMe
Me 3,4-di-OCF ₃ U-4a 2-OMe-3-OCF ₃ cPr 2-CF ₃ -4-OCF ₃
--------- --------- --------
[Table 3] (continued) [Table 3] (continued) [Table 3] (continued)
--------- --------- --------
R ³ ZR ³ ZR ³ Z
--------- --------- --------
Et 2,3-di-F U-4a 2-OCF ₃ -3-F cPr 2-OMe-4-F
Et 2-F-3-Cl U-4a 2-OCF ₃ -3-Cl cPr 2-OMe-4-Cl
Et 2-F-3-Br U-4a 2-OCF ₃ -3-Br cPr 2-OMe-4-Br
Et 2-F-3-Me U-4a 2-OCF ₃ -3-Me cPr 2-OMe-4-Me
Et 2-F-3-CF ₃ U-4a 2-OCF ₃ -3-CF ₃ cPr 2-OMe-4-CF ₃
Et 2-F-3-OMe U-4a 2-OCF ₃ -3-OMe cPr 2,4-di-OMe
Et 2-F-3-OCF ₃ U-4a 2,3-di-OCF ₃ cPr 2-OMe-4-OCF ₃
Et 2-Cl-3-F U-4a 2,4-di-F cPr 2-OCF ₃ -4-F
Et 2,3-di-Cl U-4a 2-F-4-Cl cPr 2-OCF ₃ -4-Cl
Et 2-Cl-3-Br U-4a 2-F-4-Br cPr 2-OCF ₃ -4-Br
Et 2-Cl-3-Me U-4a 2-F-4-Me cPr 2-OCF ₃ -4-Me
Et 2-Cl-3-CF ₃ U-4a 2-F-4-CF ₃ cPr 2-OCF ₃ -4-CF ₃
Et 2-Cl-3-OMe U-4a 2-F-4-OMe cPr 2-OCF ₃ -4-OMe
Et 2-Cl-3-OCF ₃ U-4a 2-F-4-OCF ₃ cPr 2,4-di-OCF ₃
Et 2-Br-3-F U-4a 2-Cl-4-F cPr 3,4-di-F
Et 2-Br-3-Cl U-4a 2,4-di-Cl cPr 3-F-4-Cl
Et 2,3-di-Br U-4a 2-Cl-4-Br cPr 3-F-4-Br
Et 2-Br-3-Me U-4a 2-Cl-4-Me cPr 3-F-4-Me
Et 2-Br-3-CF ₃ U-4a 2-Cl-4-CF ₃ cPr 3-F-4-CF ₃
Et 2-Br-3-OMe U-4a 2-Cl-4-OMe cPr 3-F-4-OMe
Et 2-Br-3-OCF ₃ U-4a 2-Cl-4-OCF ₃ cPr 3-F-4-OCF ₃
Et 2-Me-3-F U-4a 2-Br-4-F cPr 3-Cl-4-F
Et 2-Me-3-Cl U-4a 2-Br-4-Cl cPr 3,4-di-Cl
Et 2-Me-3-Br U-4a 2,4-di-Br cPr 3-Cl-4-Br
Et 2,3-di-Me U-4a 2-Br-4-Me cPr 3-Cl-4-Me
Et 2-Me-3-CF ₃ U-4a 2-Br-4-CF ₃ cPr 3-Cl-4-CF ₃
Et 2-Me-3-OMe U-4a 2-Br-4-OMe cPr 3-Cl-4-OMe
Et 2-Me-3-OCF ₃ U-4a 2-Br-4-OCF ₃ cPr 3-Cl-4-OCF ₃
Et 2-CF ₃ -3-F U-4a 2-Me-4-F cPr 3-Br-4-F
Et 2-CF ₃ -3-Cl U-4a 2-Me-4-Cl cPr 3-Br-4-Cl
Et 2-CF ₃ -3-Br U-4a 2-Me-4-Br cPr 3,4-di-Br
Et 2-CF ₃ -3-Me U-4a 2,4-di-Me cPr 3-Br-4-Me
Et 2,3-di-CF ₃ U-4a 2-Me-4-CF ₃ cPr 3-Br-4-CF ₃
Et 2-CF ₃ -3-OMe U-4a 2-Me-4-OMe cPr 3-Br-4-OMe
Et 2-CF ₃ -3-OCF ₃ U-4a 2-Me-4-OCF ₃ cPr 3-Br-4-OCF ₃
Et 2-OMe-3-F U-4a 2-CF ₃ -4-F cPr 3-Me-4-F
Et 2-OMe-3-Cl U-4a 2-CF ₃ -4-Cl cPr 3-Me-4-Cl
Et 2-OMe-3-Br U-4a 2-CF ₃ -4-Br cPr 3-Me-4-Br
Et 2-OMe-3-Me U-4a 2-CF ₃ -4-Me cPr 3,4-di-Me
--------- --------- --------
[Table 3] (continued) [Table 3] (continued) [Table 3] (continued)
--------- --------- --------
R ³ ZR ³ ZR ³ Z
--------- --------- --------
Et 2-OMe-3-CF ₃ U-4a 2,4-di-CF ₃ cPr 3-Me-4-CF ₃
Et 2,3-di-OMe U-4a 2-CF ₃ -4-OMe cPr 3-Me-4-OMe
Et 2-OMe-3-OCF ₃ U-4a 2-CF ₃ -4-OCF ₃ cPr 3-Me-4-OCF ₃
Et 2-OCF ₃ -3-F U-4a 2-OMe-4-F cPr 3-CF ₃ -4-F
Et 2-OCF ₃ -3-Cl U-4a 2-OMe-4-Cl cPr 3-CF ₃ -4-Cl
Et 2-OCF ₃ -3-Br U-4a 2-OMe-4-Br cPr 3-CF ₃ -4-Br
Et 2-OCF ₃ -3-Me U-4a 2-OMe-4-Me cPr 3-CF ₃ -4-Me
Et 2-OCF ₃ -3-CF ₃ U-4a 2-OMe-4-CF ₃ cPr 3,4-di-CF ₃
Et 2-OCF ₃ -3-OMe U-4a 2,4-di-OMe cPr 3-CF ₃ -4-OMe
Et 2,3-di-OCF ₃ U-4a 2-OMe-4-OCF ₃ cPr 3-CF ₃ -4-OCF ₃
Et 2,4-di-F U-4a 2-OCF ₃ -4-F cPr 3-OMe-4-F
Et 2-F-4-Cl U-4a 2-OCF ₃ -4-Cl cPr 3-OMe-4-Cl
Et 2-F-4-Br U-4a 2-OCF ₃ -4-Br cPr 3-OMe-4-Br
Et 2-F-4-Me U-4a 2-OCF ₃ -4-Me cPr 3-OMe-4-Me
Et 2-F-4-CF ₃ U-4a 2-OCF ₃ -4-CF ₃ cPr 3-OMe-4-CF ₃
Et 2-F-4-OMe U-4a 2-OCF ₃ -4-OMe cPr 3,4-di-OMe
Et 2-F-4-OCF ₃ U-4a 2,4-di-OCF ₃ cPr 3-OMe-4-OCF ₃
Et 2-Cl-4-F U-4a 3,4-di-F cPr 3-OCF ₃ -4-F
Et 2,4-di-Cl U-4a 3-F-4-Cl cPr 3-OCF ₃ -4-Cl
Et 2-Cl-4-Br U-4a 3-F-4-Br cPr 3-OCF ₃ -4-Br
Et 2-Cl-4-Me U-4a 3-F-4-Me cPr 3-OCF ₃ -4-Me
Et 2-Cl-4-CF ₃ U-4a 3-F-4-CF ₃ cPr 3-OCF ₃ -4-CF ₃
Et 2-Cl-4-OMe U-4a 3-F-4-OMe cPr 3-OCF ₃ -4-OMe
Et 2-Cl-4-OCF ₃ U-4a 3-F-4-OCF ₃ cPr 3,4-di-OCF ₃
--------- --------- --------
[Table 4]

［第４表］［第４表］（続き）［第４表］（続き）
−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−− −−−−−−−−− −−−−−−−−−−−
Me Me cPen CF₃ CF(CF₃)₂ nPr
Me Et cPen cPr CF(CF₃)₂ CH₂OMe
Me iPr cHex Me CF(CF₃)₂ CF₃
Me nPr cHex Et CF(CF₃)₂ cPr
Me CH₂OMe cHex iPr CH=CH₂ Me
Me CF₃ cHex nPr CH=CH₂ Et
Me cPr cHex CH₂OMe CH=CH₂ iPr
Et Me cHex CF₃ CH=CH₂ nPr
Et Et cHex cPr CH=CH₂ CH₂OMe
Et iPr CF₃ Me CH=CH₂ CF₃
Et nPr CF₃ Et CH=CH₂ cPr
Et CH₂OMe CF₃ iPr CH₂CH=CH₂ Me
Et CF₃ CF₃ nPr CH₂CH=CH₂ Et
Et cPr CF₃ CH₂OMe CH₂CH=CH₂ iPr
nPr Me CF₃ CF₃ CH₂CH=CH₂ nPr
nPr Et CF₃ cPr CH₂CH=CH₂ CH₂OMe
nPr iPr CF₂H Me CH₂CH=CH₂ CF₃
nPr nPr CF₂H Et CH₂CH=CH₂ cPr
nPr CH₂OMe CF₂H iPr C(Me)=CH₂ Me
nPr CF₃ CF₂H nPr C(Me)=CH₂ Et
nPr cPr CF₂H CH₂OMe C(Me)=CH₂ iPr
iPr Me CF₂H CF₃ C(Me)=CH₂ nPr
iPr Et CF₂H cPr C(Me)=CH₂ CH₂OMe
iPr iPr CCl₃ Me C(Me)=CH₂ CF₃
iPr nPr CCl₃ Et C(Me)=CH₂ cPr
iPr CH₂OMe CCl₃ iPr C(Me)CH=CH₂ Me
iPr CF₃ CCl₃ nPr C(Me)CH=CH₂ Et
iPr cPr CCl₃ CH₂OMe C(Me)CH=CH₂ iPr
nBu Me CCl₃ CF₃ C(Me)CH=CH₂ nPr
nBu Et CCl₃ cPr C(Me)CH=CH₂ CH₂OMe
nBu iPr CCl₂H Me C(Me)CH=CH₂ CF₃
nBu nPr CCl₂H Et C(Me)CH=CH₂ cPr
nBu CH₂OMe CCl₂H iPr OMe Me
nBu CF₃ CCl₂H nPr OMe Et
nBu cPr CCl₂H CH₂OMe OMe iPr
cPr Me CCl₂H CF₃ OMe nPr
cPr Et CCl₂H cPr OMe CH₂OMe
cPr iPr CClH₂ Me OMe CF₃
cPr nPr CClH₂ Et OMe cPr
−−−−−−− −−−−−−−−−− −−−−−−−−−−−
［第４表］（続き）［第４表］（続き）［第４表］（続き）
−−−−−−− −−−−−−−−− −−−−−−−−−−−
R³ Z R³ Z R³ Z
−−−−−−− −−−−−−−−− −−−−−−−−−−−
cPr CH₂OMe CClH₂ iPr OEt Me
cPr CF₃ CClH₂ nPr OEt Et
cPr cPr CClH₂ CH₂OMe OEt iPr
U-1a Me CClH₂ CF₃ OEt nPr
U-1a Et CClH₂ cPr OEt CH₂OMe
U-1a iPr CH₂CF₃ Me OEt CF₃
U-1a nPr CH₂CF₃ Et OEt cPr
U-1a CH₂OMe CH₂CF₃ iPr OnPr Me
U-1a CF₃ CH₂CF₃ nPr OnPr Et
U-1a cPr CH₂CF₃ CH₂OMe OnPr iPr
U-1b Me CH₂CF₃ CF₃ OnPr nPr
U-1b Et CH₂CF₃ cPr OnPr CH₂OMe
U-1b iPr CH₂CCl₃ Me OnPr CF₃
U-1b nPr CH₂CCl₃ Et OnPr cPr
U-1b CH₂OMe CH₂CCl₃ iPr OiPr Me
U-1b CF₃ CH₂CCl₃ nPr OiPr Et
U-1b cPr CH₂CCl₃ CH₂OMe OiPr iPr
cBu Me CH₂CCl₃ CF₃ OiPr nPr
cBu Et CH₂CCl₃ cPr OiPr CH₂OMe
cBu iPr CF₂CF₃ Me OiPr CF₃
cBu nPr CF₂CF₃ Et OiPr cPr
cBu CH₂OMe CF₂CF₃ iPr Ph Me
cBu CF₃ CF₂CF₃ nPr Ph Et
cBu cPr CF₂CF₃ CH₂OMe Ph iPr
cPen Me CF₂CF₃ CF₃ Ph nPr
cPen Et CF₂CF₃ cPr Ph CH₂OMe
cPen iPr CF(CF₃)₂ Me Ph CF₃
cPen nPr CF(CF₃)₂ Et Ph cPr
cPen CH₂OMe CF(CF₃)₂ iPr −−−−−−−−−−−
−−−−−−− −−−−−−−−−
本発明化合物を植物病害及び植物害虫防除剤として施用するにあたっては、通常適当な固体担体又は液体担体と混合し、更に所望により界面活性剤、浸透剤、展着剤、増粘剤、凍結防止剤、結合剤、固結防止剤、崩壊剤及び分解防止剤等を添加して、液剤（ｓｏｌｕｂｌｅｃｏｎｃｅｎｔｒａｔｅ）、乳剤（ｅｍｕｌｓｉｆｉａｂｌｅｃｏｎｃｅｎｔｒａｔｅ）、水和剤（ｗｅｔｔａｂｌｅｐｏｗｄｅｒ）、水溶剤（ｗａｔｅｒｓｏｌｕｂｌｅｐｏｗｄｅｒ）、顆粒水和剤（ｗａｔｅｒｄｉｓｐｅｒｓｉｂｌｅｇｒａｎｕｌｅ）、顆粒水溶剤（ｗａｔｅｒｓｏｌｕｂｌｅｇｒａｎｕｌｅ）、懸濁剤（ｓｕｓｐｅｎｓｉｏｎｃｏｎｃｅｎｔｒａｔｅ）、乳濁剤（ｃｏｎｃｅｎｔｒａｔｅｄｅｍｕｌｓｉｏｎ）、サスポエマルジョン（ｓｕｓｐｏｅｍｕｌｓｉｏｎ）、マイクロエマルジョン（ｍｉｃｒｏｅｍｕｌｓｉｏｎ）、粉剤（ｄｕｓｔａｂｌｅｐｏｗｄｅｒ）、粒剤（ｇｒａｎｕｌｅ）及びゲル剤（ｇｅｌ）等任意の剤型の製剤にて実用に供することができる。また、省力化及び安全性向上の観点から、上記任意の剤型の製剤を水溶性包装体に封入して供することもできる。 [Table 4] [Table 4] (continued) [Table 4] (continued)
------- --------- ------------
R ³ ZR ³ ZR ³ Z
------- --------- ------------
Me Me cPen CF ₃ CF (CF ₃ ) ₂ nPr
Me Et cPen cPr CF (CF ₃ ) ₂ CH ₂ OMe
Me iPr cHex Me CF (CF ₃ ) ₂ CF ₃
Me nPr cHex Et CF (CF ₃ ) ₂ cPr
Me CH ₂ OMe cHex iPr CH = CH ₂ Me
Me CF ₃ cHex nPr CH = CH ₂ Et
Me cPr cHex CH ₂ OMe CH = CH ₂ iPr
Et Me cHex CF ₃ CH = CH ₂ nPr
Et Et cHex cPr CH = CH ₂ CH ₂ OMe
Et iPr CF ₃ Me CH = CH ₂ CF ₃
Et nPr CF ₃ Et CH = CH ₂ cPr
Et CH ₂ OMe CF ₃ iPr CH ₂ CH = CH ₂ Me
Et CF ₃ CF ₃ nPr CH ₂ CH = CH ₂ Et
Et cPr CF ₃ CH ₂ OMe CH ₂ CH = CH ₂ iPr
nPr Me CF ₃ CF ₃ CH ₂ CH = CH ₂ nPr
nPr Et CF ₃ cPr CH ₂ CH = CH ₂ CH ₂ OMe
nPr iPr CF ₂ H Me CH ₂ CH = CH ₂ CF ₃
nPr nPr CF ₂ H Et CH ₂ CH = CH ₂ cPr
nPr CH ₂ OMe CF ₂ H iPr C (Me) = CH ₂ Me
nPr CF ₃ CF ₂ H nPr C (Me) = CH ₂ Et
nPr cPr CF ₂ H CH ₂ OMe C (Me) = CH ₂ iPr
iPr Me CF ₂ H CF ₃ C (Me) = CH ₂ nPr
iPr Et CF ₂ H cPr C (Me) = CH ₂ CH ₂ OMe
iPr iPr CCl ₃ Me C (Me) = CH ₂ CF ₃
iPr nPr CCl ₃ Et C (Me) = CH ₂ cPr
iPr CH ₂ OMe CCl ₃ iPr C (Me) CH = CH ₂ Me
iPr CF ₃ CCl ₃ nPr C (Me) CH = CH ₂ Et
iPr cPr CCl ₃ CH ₂ OMe C (Me) CH = CH ₂ iPr
nBu Me CCl ₃ CF ₃ C (Me) CH = CH ₂ nPr
nBu Et CCl ₃ cPr C (Me) CH = CH ₂ CH ₂ OMe
nBu iPr CCl ₂ H Me C (Me) CH = CH ₂ CF ₃
nBu nPr CCl ₂ H Et C (Me) CH = CH ₂ cPr
nBu CH ₂ OMe CCl ₂ H iPr OMe Me
nBu CF ₃ CCl ₂ H nPr OMe Et
nBu cPr CCl ₂ H CH ₂ OMe OMe iPr
cPr Me CCl ₂ H CF ₃ OMe nPr
cPr Et CCl ₂ H cPr OMe CH ₂ OMe
cPr iPr CClH ₂ Me OMe CF ₃
cPr nPr CClH ₂ Et OMe cPr
------- ---------- ------------
[Table 4] (continued) [Table 4] (continued) [Table 4] (continued)
------- --------- ------------
R ³ ZR ³ ZR ³ Z
------- --------- ------------
cPr CH ₂ OMe CClH ₂ iPr OEt Me
cPr CF ₃ CClH ₂ nPr OEt Et
cPr cPr CClH ₂ CH ₂ OMe OEt iPr
U-1a Me CClH ₂ CF ₃ OEt nPr
U-1a Et CClH ₂ cPr OEt CH ₂ OMe
U-1a iPr CH ₂ CF ₃ Me OEt CF ₃
U-1a nPr CH ₂ CF ₃ Et OEt cPr
U-1a CH ₂ OMe CH ₂ CF ₃ iPr OnPr Me
U-1a CF ₃ CH ₂ CF ₃ nPr OnPr Et
U-1a cPr CH ₂ CF ₃ CH ₂ OMe OnPr iPr
U-1b Me CH ₂ CF ₃ CF ₃ OnPr nPr
U-1b Et CH ₂ CF ₃ cPr OnPr CH ₂ OMe
U-1b iPr CH ₂ CCl ₃ Me OnPr CF ₃
U-1b nPr CH ₂ CCl ₃ Et OnPr cPr
U-1b CH ₂ OMe CH ₂ CCl ₃ iPr OiPr Me
U-1b CF ₃ CH ₂ CCl ₃ nPr OiPr Et
U-1b cPr CH ₂ CCl ₃ CH ₂ OMe OiPr iPr
cBu Me CH ₂ CCl ₃ CF ₃ OiPr nPr
cBu Et CH ₂ CCl ₃ cPr OiPr CH ₂ OMe
cBu iPr CF ₂ CF ₃ Me OiPr CF ₃
cBu nPr CF ₂ CF ₃ Et OiPr cPr
cBu CH ₂ OMe CF ₂ CF ₃ iPr Ph Me
cBu CF ₃ CF ₂ CF ₃ nPr Ph Et
cBu cPr CF ₂ CF ₃ CH ₂ OMe Ph iPr
cPen Me CF ₂ CF ₃ CF ₃ Ph nPr
cPen Et CF ₂ CF ₃ cPr Ph CH ₂ OMe
cPen iPr CF (CF ₃ ) ₂ Me Ph CF ₃
cPen nPr CF (CF ₃ ) ₂ Et Ph cPr
cPen CH ₂ OMe CF (CF ₃ ) ₂ iPr ------------
----------------
When the compound of the present invention is applied as a plant disease or plant pest control agent, it is usually mixed with a suitable solid carrier or liquid carrier, and if desired, a surfactant, penetrant, spreading agent, thickener, antifreeze agent. , Binders, anti-caking agents, disintegrants, anti-decomposition agents, etc., to add liquid concentrates, emulsion concentrates, wettable powders, water soluble powders, granules Water dispersible granule, water soluble granule, suspension (concentrated emulsion), emulsion (suspension emulsion), suspension emulsion spoemulsion), microemulsion (microemulsion), dusts (dustable powder), can be put into practical use in granules (granule) and gels (gel) like any dosage form of the formulation. In addition, from the viewpoint of labor saving and safety improvement, the preparation of any of the above dosage forms can be enclosed in a water-soluble package.

固体担体としては、例えば石英、カオリナイト、パイロフィライト、セリサイト、タルク、ベントナイト、酸性白土、アタパルジャイト、ゼオライト及び珪藻土等の天然鉱物質類、炭酸カルシウム、硫酸アンモニウム、硫酸ナトリウム及び塩化カリウム等の無機塩類、合成珪酸ならびに合成珪酸塩が挙げられる。 Examples of solid carriers include quartz, kaolinite, pyrophyllite, sericite, talc, bentonite, acid clay, attapulgite, zeolite, and diatomaceous earth, and other minerals, calcium carbonate, ammonium sulfate, sodium sulfate, and potassium chloride. Examples include salts, synthetic silicic acid and synthetic silicates.

液体担体としては、例えばエチレングリコール、プロピレングリコール及びイソプロパノール等のアルコール類、キシレン、アルキルベンゼン及びアルキルナフタレン等の芳香族炭化水素類、ブチルセロソルブ等のエーテル類、シクロヘキサノン等のケトン類、γ−ブチロラクトン等のエステル類、Ｎ−メチルピロリドン、Ｎ−オクチルピロリドン等の酸アミド類、大豆油、ナタネ油、綿実油及びヒマシ油等の植物油ならびに水が挙げられる。 Examples of the liquid carrier include alcohols such as ethylene glycol, propylene glycol and isopropanol, aromatic hydrocarbons such as xylene, alkylbenzene and alkylnaphthalene, ethers such as butyl cellosolve, ketones such as cyclohexanone, and esters such as γ-butyrolactone. And acid amides such as N-methylpyrrolidone and N-octylpyrrolidone, vegetable oils such as soybean oil, rapeseed oil, cottonseed oil and castor oil, and water.

これら固体及び液体担体は、単独で用いても２種以上を併用してもよい。 These solid and liquid carriers may be used alone or in combination of two or more.

界面活性剤としては、例えばポリオキシエチレンアルキルエーテル、ポリオキシエチレンアルキルアリールエーテル、ポリオキシエチレンスチリルフェニルエーテル、ポリオキシエチレンポリオキシプロピレンブロックコポリマー、ポリオキシエチレン脂肪酸エステル、ソルビタン脂肪酸エステル及びポリオキシエチレンソルビタン脂肪酸エステル等のノニオン性界面活性剤、アルキル硫酸塩、アルキルベンゼンスルホン酸塩、リグニンスルホン酸塩、アルキルスルホコハク酸塩、ナフタレンスルホン酸塩、アルキルナフタレンスルホン酸塩、ナフタレンスルホン酸のホルマリン縮合物の塩、アルキルナフタレンスルホン酸のホルマリン縮合物の塩、ポリオキシエチレンアルキルアリールエーテル硫酸及び燐酸塩、ポリオキシエチレンスチリルフェニルエーテル硫酸及び燐酸塩、ポリカルボン酸塩及びポリスチレンスルホン酸塩等のアニオン性界面活性剤、アルキルアミン塩及びアルキル４級アンモニウム塩等のカチオン性界面活性剤ならびにアミノ酸型及びベタイン型等の両性界面活性剤が挙げられる。 Examples of the surfactant include polyoxyethylene alkyl ether, polyoxyethylene alkyl aryl ether, polyoxyethylene styryl phenyl ether, polyoxyethylene polyoxypropylene block copolymer, polyoxyethylene fatty acid ester, sorbitan fatty acid ester and polyoxyethylene sorbitan. Nonionic surfactant such as fatty acid ester, alkyl sulfate, alkylbenzene sulfonate, lignin sulfonate, alkyl sulfosuccinate, naphthalene sulfonate, alkyl naphthalene sulfonate, salt of formalin condensate of naphthalene sulfonate, Salt of formalin condensate of alkylnaphthalenesulfonic acid, polyoxyethylene alkylaryl ether sulfate and phosphate, polyoxyethylene polystyrene Anionic surfactants such as phenyl ether sulfate and phosphate, polycarboxylate and polystyrene sulfonate, cationic surfactants such as alkylamine salt and alkyl quaternary ammonium salt, and amphoteric interfaces such as amino acid type and betaine type An activator is mentioned.

これら界面活性剤の含有量は、特に限定されるものではないが、本発明の製剤１００重量部に対し、通常０．０５〜２０重量部の範囲が望ましい。また、これら界面活性剤は、単独で用いても２種以上を併用してもよい。 The content of these surfactants is not particularly limited, but is usually preferably in the range of 0.05 to 20 parts by weight with respect to 100 parts by weight of the preparation of the present invention. These surfactants may be used alone or in combination of two or more.

また、本発明化合物を農薬として使用する場合には必要に応じて製剤時又は散布時に他種の除草剤、各種殺虫剤、殺ダニ剤、殺線虫剤、殺菌剤、植物生長調節剤、共力剤、肥料、土壌改良剤等と混合施用してもよい。 In addition, when the compound of the present invention is used as an agrochemical, other types of herbicides, various insecticides, acaricides, nematicides, fungicides, plant growth regulators, co-agents, and the like, can be used when formulated or sprayed. You may mix and apply it with a power agent, a fertilizer, a soil conditioner, etc.

特に他の農薬或いは植物ホルモンと混合施用することにより、施用薬量の減少による低コスト化、混合薬剤の相乗作用による殺菌殺虫スペクトラムの拡大や、より高い有害生物防除効果が期待できる。この際、同時に複数の公知農薬との組み合わせも可能である。本発明化合物と混合使用する農薬の種類としては、例えば、ファーム・ケミカルズ・ハンドブック（ＦａｒｍＣｈｅｍｉｃａｌｓＨａｎｄｂｏｏｋ）１９９９年版に記載されている化合物等がある。具体的にその一般名を例示すれば次の通りであるが、必ずしもこれらのみに限定されるものではない。 In particular, by applying it in combination with other agricultural chemicals or plant hormones, it can be expected to reduce costs by reducing the amount of applied medicine, expand the bactericidal insecticidal spectrum due to the synergistic action of the mixed drugs, and higher pest control effects. At this time, a combination with a plurality of known agricultural chemicals is also possible. Examples of the type of agrochemical used in combination with the compound of the present invention include compounds described in the 1999 edition of Farm Chemicals Handbook (Farm Chemicals Handbook). Specific examples of common names are as follows, but the general names are not necessarily limited to these.

殺菌剤：アシベンゾラル−Ｓ−メチル（ａｃｉｂｅｎｚｏｌａｒ−Ｓ−ｍｅｔｈｙｌ）、アシペタックス（ａｃｙｐｅｔａｃｓ）、アルジモルフ（ａｌｄｉｍｏｒｐｈ）、アリルアルコール（ａｌｌｙｌａｌｃｏｈｏｌ）、アメトクトラジン（ａｍｅｔｏｃｔｒａｄｉｎ）、アミスルブロム（ａｍｉｓｕｌｂｒｏｍ）、アンバム（ａｍｏｂａｍ）、アムプロピルホス（ａｍｐｒｏｐｙｌｆｏｓ）、アニラジン（ａｎｉｌａｚｉｎｅ）、アザコナゾール（ａｚａｃｏｎａｚｏｌｅ）、アジチラム（ａｚｉｔｈｉｒａｍ）、アゾキシストロビン（ａｚｏｘｙｓｔｒｏｂｉｎ）、バリウムポリサルファイド（ｂａｒｉｕｍｐｏｌｙｓｕｌｆｉｄｅ）、ベナラキシル（ｂｅｎａｌａｘｙｌ）、ベナラキシル−Ｍ（ｂｅｎａｌａｘｙｌ−Ｍ）、ベノダニル（ｂｅｎｏｄａｎｉｌ）、ベノミル（ｂｅｎｏｍｙｌ）、ベンキノックス（ｂｅｎｑｕｉｎｏｘ）、ベンタルロン（ｂｅｎｔａｌｕｒｏｎ）、ベンチアバリカルブ−イソプロピル（ｂｅｎｔｈｉａｖａｌｉｃａｒｂ−ｉｓｏｐｒｏｐｙｌ）、ベンチアゾール（ｂｅｎｔｈｉａｚｏｌｅ）、ベンザマクリル（ｂｅｎｚａｍａｃｒｉｌ）、ベンザモルフ（ｂｅｎｚａｍｏｒｆ）、ベンゾビンディフルピル（ｂｅｎｚｏｖｉｎｄｉｆｌｕｐｙｒ）、ビナパクリル（ｂｉｎａｐａｃｒｙｌ）、ビフェニル（ｂｉｐｈｅｎｙｌ）、ビテルタノール（ｂｉｔｅｒｔａｎｏｌ）、ビキサフェン（ｂｉｘａｆｅｎ）、ブラストサイジン−Ｓ（ｂｌａｓｔｉｃｉｄｉｎ−Ｓ）、ボルドー液（ｂｏｒｄｅａｕｘｍｉｘｔｕｒｅ）、ボスカリド（ｂｏｓｃａｌｉｄ）、ブロムコナゾール（ｂｒｏｍｏｃｏｎａｚｏｌｅ）、ブピリメート（ｂｕｐｉｒｉｍａｔｅ）、ブチオベート（ｂｕｔｈｉｏｂａｔｅ）、ブチルアミン（ｂｕｔｙｌａｍｉｎｅ）、石灰硫黄合剤（ｃａｌｃｉｕｍｐｏｌｙｓｕｌｆｉｄｅ）、キャプタフォール（ｃａｐｔａｆｏｌ）、キャプタン（ｃａｐｔａｎ）、カルバモルフ（ｃａｒｂａｍｏｒｐｈ）、カルベンダジム（ｃａｒｂｅｎｄａｚｉｍ）、カルボキシン（ｃａｒｂｏｘｉｎ）、カルプロパミド（ｃａｒｐｒｏｐａｍｉｄ）、カルボン（ｃａｒｖｏｎｅ）、チェシュントミクスチャ（ｃｈｅｓｈｕｎｔｍｉｘｔｕｒｅ）、キノメチオネート（ｃｈｉｎｏｍｅｔｈｉｏｎａｔ）、クロベンチアゾン（ｃｈｌｏｂｅｎｔｈｉａｚｏｎｅ）、クロラニフォルメタン（ｃｈｌｏｒａｎｉｆｏｒｍｅｔｈａｎｅ）、クロラニル（ｃｈｌｏｒａｎｉｌ）、クロルフェナゾール（ｃｈｌｏｒｆｅｎａｚｏｌｅ）、クロロネブ（ｃｈｌｏｒｏｎｅｂ）、クロルピクリン（ｃｈｌｏｒｏｐｉｃｒｉｎ）、クロロタロニル（ｃｈｌｏｒｏｔｈａｌｏｎｉｌ）、クロルキノックス（ｃｈｌｏｒｑｕｉｎｏｘ）、クロゾリネート（ｃｈｌｏｚｏｌｉｎａｔｅ）、クリムバゾール（ｃｌｉｍｂａｚｏｌｅ）、カッパーアセテイト（ｃｏｐｐｅｒａｃｅｔａｔｅ）、塩基性炭酸銅（ｃｏｐｐｅｒｃａｒｂｏｎａｔｅ，ｂａｓｉｃ）、水酸化第二銅（ｃｏｐｐｅｒｈｙｄｒｏｘｉｄｅ）、カッパーナフテネート（ｃｏｐｐｅｒｎａｐｈｔｈｅｎａｔｅ）、カッパーオレエート（ｃｏｐｐｅｒｏｌｅａｔｅ）、塩基性塩化銅（ｃｏｐｐｅｒｏｘｙｃｈｌｏｒｉｄｅ）、硫酸銅（ｃｏｐｐｅｒｓｕｌｆａｔｅ）、塩基性硫酸銅（ｃｏｐｐｅｒｓｕｌｆａｔｅ，ｂａｓｉｃ）、カッパージンククロメイト（ｃｏｐｐｅｒｚｉｎｃｃｈｒｏｍａｔｅ）、クレゾール（ｃｒｅｓｏｌ）、クフラネブ（ｃｕｆｒａｎｅｂ）、クプロバム（ｃｕｐｒｏｂａｍ）、シアゾファミド（ｃｙａｚｏｆａｍｉｄ）、シクラフラミド（ｃｙｃｌａｆｕｒａｍｉｄ）、シクロヘキシミド（ｃｙｃｌｏｈｅｘｉｍｉｄｅ）、シフルフェナミド（ｃｙｆｌｕｆｅｎａｍｉｄ）、シモキサニル（ｃｙｍｏｘａｎｉｌ）、シペンダゾール（ｃｙｐｅｎｄａｚｏｌｅ）、シプロコナゾール（ｃｙｐｒｏｃｏｎａｚｏｌｅ）、シプロジニル（ｃｙｐｒｏｄｉｎｉｌ）、シプロフラム（ｃｙｐｒｏｆｕｒａｍ）、ダゾメット（ｄａｚｏｍｅｔ）、デバカルブ（ｄｅｂａｃａｒｂ）、デカフェンチン（ｄｅｃａｆｅｎｔｉｎ）、デハイドロアセテイト（ｄｅｈｙｄｒｏａｃｅｔｉｃａｃｉｄ）、ジクロフルアニド（ｄｉｃｈｌｏｆｌｕａｎｉｄ）、ジクロン（ｄｉｃｈｌｏｎｅ）、ジクロロフェン（ｄｉｃｈｌｏｒｏｐｈｅｎ）、ジクロゾリン（ｄｉｃｈｌｏｚｏｌｉｎｅ）、ジクロブトラゾール（ｄｉｃｌｏｂｕｔｒａｚｏｌ）、ジクロシメット（ｄｉｃｌｏｃｙｍｅｔ）、ジクロメジン（ｄｉｃｌｏｍｅｚｉｎｅ）、ジクロラン（ｄｉｃｌｏｒａｎ）、ジエトフェンカルブ（ｄｉｅｔｈｏｆｅｎｃａｒｂ）、ジフェノコナゾール（ｄｉｆｅｎｏｃｏｎａｚｏｌｅ）、ジフルメトリム（ｄｉｆｌｕｍｅｔｏｒｉｍ）、ジメチリモール（ｄｉｍｅｔｈｉｒｉｍｏｌ）、ジメトモルフ（ｄｉｍｅｔｈｏｍｏｒｐｈ）、ジモキシストロビン（ｄｉｍｏｘｙｓｔｒｏｂｉｎ）、ジニコナゾール（ｄｉｎｉｃｏｎａｚｏｌｅ）、ジニコナゾール−Ｍ（ｄｉｎｉｃｏｎａｚｏｌｅ−Ｍ）、ジノブトン（ｄｉｎｏｂｕｔｏｎ）、ジノカップ（ｄｉｎｏｃａｐ）、ジノカップ−４（ｄｉｎｏｃａｐ−４）、ジノカップ−６（ｄｉｎｏｃａｐ−６）、ジノクトン（ｄｉｎｏｃｔｏｎ）、ジノスルフォン（ｄｉｎｏｓｕｌｆｏｎ）、ジノテルボン（ｄｉｎｏｔｅｒｂｏｎ）、ジフェニルアミン（ｄｉｐｈｅｎｙｌａｍｉｎｅ）、ジピメチトロン（ｄｉｐｙｍｅｔｉｔｒｏｎｅ）、ジピリチオン（ｄｉｐｙｒｉｔｈｉｏｎｅ）、ジスルフィラム（ｄｉｓｕｌｆｉｒａｍ）、ジタリムホス（ｄｉｔａｌｉｍｆｏｓ）、ジチアノン（ｄｉｔｈｉａｎｏｎ）、デーエヌオーシー（ＤＮＯＣ）、ドデモルフ（ｄｏｄｅｍｏｒｐｈ）、ドジン（ｄｏｄｉｎｅ）、ドラゾキソロン（ｄｒａｚｏｘｏｌｏｎ）、エディフェンホス（ｅｄｉｆｅｎｐｈｏｓ）、エネストロビン（ｅｎｅｓｔｒｏｂｉｎ）、エポキシコナゾール（ｅｐｏｘｉｃｏｎａｚｏｌｅ）、エタボキサム（ｅｔｈａｂｏｘａｍ）、エタコナゾール（ｅｔａｃｏｎａｚｏｌｅ）、エテム（ｅｔｅｍ）、エチリモール（ｅｔｈｉｒｉｍｏｌ）、エトキシキン（ｅｔｈｏｘｙｑｕｉｎ）、エトリジアゾール（ｅｔｒｉｄｉａｚｏｌｅ）、ファモキサドン（ｆａｍｏｘａｄｏｎｅ）、フェナミドン（ｆｅｎａｍｉｄｏｎｅ）、フェナミノスルフ（ｆｅｎａｍｉｎｏｓｕｌｆ）、フェナパニル（ｆｅｎａｐａｎｉｌ）、フェナリモル（ｆｅｎａｒｉｍｏｌ）、フェンブコナゾール（ｆｅｎｂｕｃｏｎａｚｏｌｅ）、フェンフラム（ｆｅｎｆｕｒａｍ）、フェンヘキサミド（ｆｅｎｈｅｘａｍｉｄ）、フェニトロパン（ｆｅｎｉｔｒｏｐａｎ）、フェノキサニル（ｆｅｎｏｘａｎｉｌ）、フェンピクロニル（ｆｅｎｐｉｃｌｏｎｉｌ）、フェンプロピジン（ｆｅｎｐｒｏｐｉｄｉｎ）、フェンプロピモルフ（ｆｅｎｐｒｏｐｉｍｏｒｐｈ）、フェンピラザミン（ｆｅｎｐｙｒａｚａｍｉｎｅ）、フェンチン（ｆｅｎｔｉｎ）、ファーバム（ｆｅｒｂａｍ）、フェリムゾン（ｆｅｒｉｍｚｏｎｅ）、フルアジナム（ｆｌｕａｚｉｎａｍ）、フルジオキソニル（ｆｌｕｄｉｏｘｏｎｉｌ）、フルフェノキシストロビン（ｆｌｕｆｅｎｏｘｙｓｔｒｏｂｉｎ）、フルメトベル（ｆｌｕｍｅｔｏｖｅｒ）、フルモルフ（ｆｌｕｍｏｒｐｈ）、フルオピコリド（ｆｌｕｏｐｉｃｏｌｉｄｅ）、フルオピラム（ｆｌｕｏｐｙｒａｍ）、フルオルイミド（ｆｌｕｏｒｏｉｍｉｄｅ）、フルオトリマゾール（ｆｌｕｏｔｒｉｍａｚｏｌｅ）、フルオキサストロビン（ｆｌｕｏｘａｓｔｒｏｂｉｎ）、フルキンコナゾール（ｆｌｕｑｕｉｎｃｏｎａｚｏｌｅ）、フルシラゾール（ｆｌｕｓｉｌａｚｏｌｅ）、フルスルファミド（ｆｌｕｓｕｌｆａｍｉｄｅ）、
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Bactericides: acibenzolar-S-methyl, acipetacs, aldimorph, allyl alcohol, ametoctradin, amisulbrom, amisulbrom Phos (ampropropylfos), anilazine (anilazine), azaconazole, azithyram, azoxystrobin, barium polysulfide (barium polysulfide), benalaxylb Benodanil, benomyl, benquinox, bentaluron, benchavaricarb-isopropyl, benhiazole, bezmamol (ben), benzacril (ben) Vindiflupyr, binapacryl, biphenyl, bitertanol, bixafen, blasticidin-S (blasticin-S), borde liquor (x) ), Bromconazole, bupirimate, butiobate, butyramine, butyl sulfur, calc sulfur, capta b, captan b, capta c Carbendazim, carboxin, carpropamide, carvone, cheshunt mixture, chinomethionate, clobenchon, clobenchazone ifmetane), chloranil, chlorfenazol, chloroneb, chloropicrin, chlorquinolate, chlorquinolate, chlorquinolate, chlorquinolate, chlorquinolate, chlorquinolate (Copper acetate), basic copper carbonate (basic), cupric hydroxide, copper naphthenate, copper oleate, basic copper chloride (copper x) chloride, copper sulfate, copper sulfate, basic, copper zinc chromate, cresol, cufraneb, cuprobum, cuprobum , Cyclfuramid, Cyclofenamide, Cyxendroyl, Cyprodazole, Cyprodazole, Cyprodane, Cyprodane (Dazomet), debacarb, decafentin, dehydroacetic acid, dichlorfluanid, dichlone, dichlorofen, diclozoline, diclozoline Diclobutrazol, diclocymet, diclomezine, dichloran, diethofencarb, difenoconazole, diflumetrim, diflumetrim, diflumetrim , Dimethomorph, dimoxystrobin, diniconazole, diniconazole-M, dinobuton, dinocap-4, dinocap-4, dinocap-4, dinocap-4 (Dinocap-6), dinocton, dinosulfone, dinoterbon, diphenylamine, dipymetitrone, dipyrithione, dipyrithione, dipyrithione, dipyrithione, dipyrithione, dipyrithione, dipyrithione. itianon, DNOOC, dodemorph, dodine, drazoxolone, edifenphos, enestrobine, epoxiconazole epoxiconazole epoxiconazole (Etaconazole), etem, etirimol, ethoxyquin, etridiazole, famoxadone, fenamidone, fenaminul (fenaminul) Fenarimol, fenbuconazole, fenfuram, fenhexamid, fenitropan, fenoxanil, fenpiclonil, fenpropidin f (Fenpropimorph), fenpyrazamine, fentin, ferbam, ferimzone, fluazinam, fludioxonil, flufenoxystrobin (flumenoxtrobin) lumover, flumorph, fluopicolide, fluopyram, fluorimide, fluotrizole, fluoxastrobin, fluoxastrobnol, fluoxastrobnol Flulsulfamide,
Flutolanil, flutianil, flutriafol, fluxapyroxad, folpetto, fosetyl-aluminum, fotalidol, buverizole Furalaxyl, furametopyr, furcarbanil, fluconazole, furconazole-cis, furmecylur, phlophanate, phlophanate Ofluvin (griseofulvin), guazatine (halacrinete), hexachlorobenzene (hexachloroazole), hexylthiofos (hexylthiofos), oxyquinoline (hixylol) Imazalil, imibenconazole, iminoctadin-albesylate, iminoctadate-triacetate, iodocarba, iodocarb Ipconazole, iprobenfos, iprodione, iprovalicalcarb, isofetamid, isothiaisone, isoprotialine, isoprothiazole , Kresoxim-methyl, laminarin, mancopper, mancozeb, mandestrobin, mandipropamide, manneprop aneb), mebenil, mecarbinzid, mepanipyrim, mepronil, metalaxyl, metalaxyl-M (metaxyl-M), metamol (Metconazole), metasulfocarb (methasulfocarb), metfuroxam (metfuroxam), metyram (methinostrobin), metrafenone (metrafone), metsulfobene (metsulfoven) nil), microzoline, nabam, naphthifine, natamycin, nickel bis (dimethythythiocarbamate), nitrostyrene (nitro-propylene) (Nuarimol), octinoline, offase, oryastrobine, oxadixyl, oxathiapiprolin, oxyquinoline copper (oxine copperx) oconazole fumarate, oxycarboxin, pefurazoate, penconazole, pencycuron, penflurophenol, pentochlorophenol, pentachlorophenol 2-phenylphenol, phosdiphen, phthalide, picarbutrazox, picoxystrobin, piperalin, polycarbam te), polyoxins (polyoxins), polyoxin-D (polyoxorim), potassium azide (potassium hydrogen carbonate), pro salt (pro) zole (pro) azole, procazole (pro salt) propamocarb hydrochloride), propiconazole, propineb, proquinazid, prothiocarb, pyradipyramidopyrazopyromido Pyribencarb-methyl, pyrifenox, pyrimethanil, pyriminostrobin, pyroquiolon, prothiocarb, prothiofluol, prothiofol. ), Pyracarbolido, pyraclostrobin, pyridinitrile, pyriophenone, pyrisoxazole, pyroxyluroxy, piroxychlor ), Quinacetol-sulfate, quinazamid, quinconazole, quinoxyphene, quintoxene, benzazole, benzazole. silthiofam, simeconazole, sodium hydrogen carbonate, sodium hypochlorite, spiroxamine, sulfurazole, tebuna ole), tebufloquin, tefloftalam, technazene, tecolam, tetraconazole, thiabendazole, thiadifluol, thiadifluol. ), Thiochlorfenhim, thiophanate, thiophanate-methyl, thiuram, thiadinyl, thioxymid, tolcrophos-methyl s-methyl), tolprocarb, tolylfluanid, triadimethon, triadimenol, triamifos, triazil, triazylr, triazylr , Tributyltin oxide, trichlamide, tricyclazole, tridemorph, trifloxystrobin, trifluritrifoline , Triticonazole, validamycin, valifenalate, vinclozolin, zalamamide, zinc naphthenate, zinc sulphate, zinc sulphate Ziram, zoxamide, shiitake mycelium extract, shiitake fruiting body extract, MIF-1002 (test name), OAF-211 (test name), SB-4303 (test name), NF-180 ( Test name), S-2399 (test name), AKD-5195 (test name), and the like.

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Insecticides: abamectin, acephate, acetamiprid, aphidopyropen, afoxalaner, phosphine, alancarb, aldharb Ethyl (azinphos-ethyl), azinephos-methyl, bacillus thuringiensis, bendiocarb, benfluthrin, benfurcarb Sultap, bifenthrin, bioallethrin, bioresmethrin, bistrifluron, carbofurine c, buprofromine, buprofroin (bu) Carbofuran, carbosulfan, cartap, chloranthraniprole, chlorethoxyfos, chlorfenapyfen, chlorfenapyfen Chlorfenvinphos, Chlorfluazuron, Chlormefos, Chlorpyrifos, Chlorpyrifos-methyl, Chromaphenozine, Chromaphenozine Roll, cyclaniprole, cycloprothrin, cyfluthrin, beta-cyfluthrin, cyhalothrin, cyhalothrin Gamma-cyhalothrin, lambda-cyhalothrin, cypermethrin, alpha-cypermethrin, beta-cypermethrin (betamethrin) -Cypermethrin, cyphenothrin, cyromazine, deltamethrin, diafenthiuron, diazinon, dichlorvozur, dichlorvozur ethoate, dimethylvinphos, dinotefuran, diophenolan, disulfoton, emamectin-benzoate, empentinulsulfane, pententrin (empentrin) ), EPN (EPN), esfenvalerate, etiofencarb, ethiprole, etofenprox, etrimfos, fenitrothion (fen) ithrothion, fenobucarb, phenoxycarb, fenthion, fenvalerate, fipronil, flometoluin, flonicamudron , Flucycloxuron, flucytrinate, flufenerim, flufenoxuron, flufiprole, flumethrin, flupyrithuron (fl) pyradifurone, fluralaner, fluvalinate, fluxamethamide, tau-fluvalinate, fofofos, furothiofedi, halothiophene , Hexaflumuron, hydramethylnon, imidacloprid, imiprothrin, indoxacarb, indoxacarb-MP, indoxacarb-MP Rupro (isoprocarb), isoxathion (isoxathion), lepimectin (lepimectin), lufenuron (lufenuron), malathion (malathion), meperfluthrin (me) fluthine (meta), meta hydride (meta), meta hydride (meta) , Methidathion, methomyl, methoprene, methoxychlor, methoxyphenozide, methoflutrin, muscalua (mus) calure, nitenpyram, novaluron, noviflumuron, ometoate, oxydemeton-methyl, parathion-methrin, parathion-methyl, parathion-methrin , Phentoate, folate, fosalone, phosmet, phoxim, pirimicarb, pirimiphos-methyl, profenophos (profenfos) prothiofos), pymetrozine, pyraclofos, pyrethrins, pyridalyl, pyriquinquinone, pyriproline, pyriproline, Silafluofen, spinetoram, spinosad, spirotetramat, sulfotep, sulfoxaflor, tebufenozide Teflubenzuron, tefluthrin, terbufos, tetrachlorovinphos, tetramethrin, d-T-80-phthalthrin (d-tetramethrin), tetramethylfluthrin Tetraniliprole, thiacloprid, thiamethoxam, thiocyclam, thiodicarb, thiofanox, thioetonto, f pyrad), tralomethrin, transfluthrin, triazamate, trichlorfon, trichlorfon, triflumuron, ME5382 (test name), NC-515DI .

殺ダニ剤：アセキノシル（ａｃｅｑｕｉｎｏｃｙｌ）、アクリナトリン（ａｃｒｉｎａｔｈｒｉｎ）、アミドフルメット（ａｍｉｄｏｆｌｕｍｅｔ）、アミトラズ（ａｍｉｔｒａｚ）、アゾシクロチン（ａｚｏｃｙｃｌｏｔｉｎ）、ベンゾキシメート（ｂｅｎｚｏｘｉｍａｔｅ）、ビフェナゼート（ｂｉｆｅｎａｚａｔｅ）、ブロモプロピレート（ｂｒｏｍｏｐｒｏｐｙｌａｔｅ）、クロフェンテジン（ｃｌｏｆｅｎｔｅｚｉｎｅ）、シエノピラフェン（ｃｙｅｎｏｐｙｒａｆｅｎ）、シフルメトフェン（ｃｙｆｌｕｍｅｔｏｆｅｎ）、ジコホール（ｄｉｃｏｆｏｌ）、ジエノクロル（ｄｉｅｎｏｃｈｌｏｒ）、エトキサゾール（ｅｔｏｘａｚｏｌｅ）、フェナザキン（ｆｅｎａｚａｑｕｉｎ）、フェンブタチン−オキシド（ｆｅｎｂｕｔａｔｉｎｏｘｉｄｅ）、フェノチオカルブ（ｆｅｎｏｔｈｉｏｃａｒｂ）、フェンプロパトリン（ｆｅｎｐｒｏｐａｔｈｒｉｎ）、フェンピロキシメート（ｆｅｎｐｙｒｏｘｉｍａｔｅ）、フルアクリピリム（ｆｌｕａｃｒｙｐｙｒｉｍ）、ホルメタネート（ｆｏｒｍｅｔａｎａｔｅ）、ハルフェンプロックス（ｈａｌｆｅｎｐｒｏｘ）、ヘキシチアゾクス（ｈｅｘｙｔｈｉａｚｏｘ）、ミルベメクチン（ｍｉｌｂｅｍｅｃｔｉｎ）、プロパルギット（ｐｒｏｐａｒｇｉｔｅ）、ピフルブミド（ｐｙｆｌｕｂｕｍｉｄｅ）、ピリダベン（ｐｙｒｉｄａｂｅｎ）、ピリミジフェン（ｐｙｒｉｍｉｄｉｆｅｎ）、スピロジクロフェン（ｓｐｉｒｏｄｉｃｌｏｆｅｎ）、スピロメシフェン（ｓｐｉｒｏｍｅｓｉｆｅｎ）、テブフェンピラド（ｔｅｂｕｆｅｎｐｙｒａｄ）及びＮＡ−８９（試験名）など。 Acaricides: acequinocyl, acrinathrin, amidoflumet, amitraz, azocyclotin, benzoximate, benzopromate Phentezine, cyenopyrafen, cyflumethofen, dicophor, dienochlor, etoxazole, fenazafen in oxide, phenothiocarb, fenpropathrin, fenpyroximate, fluripyrim, flumethyx, fenfroximate propargite, pyruvumide, pyridaben, pyrimidifene, spirodiclofen, spiromesifen, tebufenpyrad (tebufenpyrad) fenpyrad) and NA-89 (test name).

殺線虫剤：カズサホス（ｃａｄｕｓａｆｏｓ）、ジクロフェンチオン（ｄｉｃｈｌｏｆｅｎｔｈｉｏｎ）、エトプロホス（ｅｔｈｏｐｒｏｐｈｏｓ）、フェナミホス（ｆｅｎａｍｉｐｈｏｓ）、フルエンスルフォン（ｆｌｕｅｎｓｕｌｆｏｎｅ）、ホスチアゼート（ｆｏｓｔｈｉａｚａｔｅ）、フォスチエタン（ｆｏｓｔｈｉｅｔａｎ）、イミシアホス（ｉｍｉｃｙａｆｏｓ）、イサミドホス（ｉｓａｍｉｄｏｆｏｓ）、イサゾホス（ｉｓａｚｏｆｏｓ）、臭化メチル（ｍｅｔｈｙｌｂｒｏｍｉｄｅ）、メチルイソチオシアネート（ｍｅｔｈｙｌｉｓｏｔｈｉｏｃｙａｎａｔｅ）、オキサミル（ｏｘａｍｙｌ）、アジ化ナトリウム（ｓｏｄｉｕｍａｚｉｄｅ）、ＢＹＩ−１９２１（試験名）及びＭＡＩ−０８０１５（試験名）など。 Nematicides: kazusafos, diclofenthion, ethoprofos, fenamifos, fluensulfos, fluthiafos, fosthiat, fosthiasto , Isazofos, methyl bromide, methyl isothiocyanate, oxamyl, sodium azide, BYI-1921 (test name) and MAI-08015 Such.

駆虫剤：アクリフラビン（ａｃｒｉｆｌａｖｉｎｅ）、アルベンダゾール（ａｌｂｅｎｄａｚｏｌｅ）、アトバコン（ａｔｏｖａｇｕｏｎｅ）、アジスロマイシン（ａｚｉｔｈｒｏｍｙｃｉｎ）、ビチオノール（ｂｉｔｈｉｏｎｏｌ）、ブロムフェノホス（ｂｒｏｍｏｆｅｎｏｆｏｓ）、カンベンダゾール（ｃａｍｂｅｎｄａｚｏｌｅ）、カルニダゾール（ｃａｒｎｉｄａｚｏｌｅ）、クロロキン（ｃｈｌｏｒｏｑｕｉｎｅ）、クラズリル（ｃｌａｚｕｒｉｌ）、クリンダマイシン（ｃｌｉｎｄａｍｙｃｉｎｈｙｄｒｏｃｈｌｏｒｉｄｅ）、クロルスロン（ｃｌｏｒｓｕｌｏｎ）、クロサンテル（ｃｌｏｓａｎｔｅｌ）、クマホス（ｃｏｕｍａｐｈｏｓ）、シミアゾル（ｃｙｍｉａｚｏｌ）、ジクロロフェン（ｄｉｃｈｌｏｒｏｐｈｅｎ）、ジエチルカルバマジン（ｄｉｅｔｈｙｌｃａｒｂａｍａｚｉｎｅ）、ジミナゼン（ｄｉｍｉｎａｚｅｎｅ）、ジソフェノール（ｄｉｓｏｐｈｅｎｏｌ）、ヨウ化ジチアザニン（ｄｉｔｈｉａｚａｎｉｎｅｉｏｄｉｄｅ）、ドキシサイクリン（ｄｏｘｙｃｙｃｌｉｎｅｈｙｄｒｏｃｈｌｏｒｉｄｅ）、ドラメクチン（ｄｏｒａｍｅｃｔｉｎ）、エモデプシド（ｅｍｏｄｅｐｓｉｄｅ）、エプリノメクチン（ｅｐｒｉｎｏｍｅｃｔｉｎ）、フェバンテル（ｆｅｂａｎｔｅｌ）、フェンベンダゾール（ｆｅｎｂｅｎｄａｚｏｌｅ）、フルベンダゾール（ｆｌｕｂｅｎｄａｚｏｌｅ）、フラゾリドン（ｆｕｒａｚｏｌｉｄｏｎｅ）、グリカルピラミド（ｇｌｙｃａｌｐｙｒａｍｉｄｅ）、イミドカルブ（ｉｍｉｄｏｃａｒｂ）、イベルメクチン（ｉｖｅｒｍｅｃｔｉｎ）、レバミゾール（ｌｅｖａｍｉｓｏｌｅ）、メベンダゾール（ｍｅｂｅｎｄａｚｏｌｅ）、メフロキン（ｍｅｆｌｏｑｕｉｎｅ）、メラルソミン二塩酸塩（ｍｅｌａｒｓａｍｉｎｅｈｙｄｒｏｃｈｌｏｒｉｄｅ）、メトロニダゾール（ｍｅｔｒｏｎｉｄａｚｏｌｅ）、メチリジン（ｍｅｔｙｒｉｄｉｎｅ）、ミルベマイシンオキシム（ｍｉｌｂｅｍｙｃｉｎｏｘｉｍｅ）、モネパンテル（ｍｏｎｅｐａｎｔｅｌ）、酒石酸モランテル（ｍｏｒａｎｔｅｌｔａｒｔｒａｔｅ）、モキシデクチン（ｍｏｘｉｄｅｃｔｉｎ）、ナイカルバジン（ｎｉｃａｒｂａｚｉｎ）、ニクロサミド（ｎｉｃｌｏｓａｍｉｄｅ）、ニトロスカネート（ｎｉｔｒｏｓｃａｎａｔｅ）、ニトロキシニル（ｎｉｔｒｏｘｙｎｉｌ）、オムファロチン（ｏｍｐｈａｌｏｔｉｎ）、パモ酸オキサンテル（ｏｘａｎｔｅｌｐａｍｏａｔｅ）、酒石酸オキサンテル（ｏｘａｎｔｅｌｔａｒｔｒａｔｅ）、オクスフェンダゾール（ｏｘｆｅｎｄａｚｏｌｅｅ）、オキシベンダゾール（ｏｘｉｂｅｎｄａｚｏｌｅ）、オキシクロザニド（ｏｘｙｃｌｏｚａｎｉｄｅ）、パマキン（ｐａｍａｑｕｉｎｅ）、フェノチアジン（ｐｈｅｎｏｔｈｉａｚｉｎｅ）、アジピン酸ピペラジン（ｐｉｐｅｒａｚｉｎｅａｄｉｐａｔｅ）、クエン酸ピペラジン（ｐｉｐｅｒａｚｉｎｅｃｉｔｒａｔｅ）、リン酸ピペラジン（ｐｉｐｅｒａｚｉｎｅｐｈｏｓｐｈａｔｅ）、ＰＮＵ−９７３３３（ｐａｒａｈｅｒｑｕａｍｉｄｅＡ）、ＰＮＵ−１４１９６２（２−ｄｅｏｘｙｐａｒａｈｅｒｑｕａｍｉｄｅ）、プラジクアンテル（ｐｒａｚｉｑｕａｎｔｅｌ）、プリマキン（ｐｒｉｍａｑｕｉｎｅ）、プロペタムホス（ｐｒｏｐｅｔａｍｐｈｏｓ）、プロポクスル（ｐｒｏｐｏｘｕｒ）、パモ酸ピランテル（ｐｙｒａｎｔｅｌｐａｍｏａｔｅ）、ピリメタミン（ｐｙｒｉｍｅｔｈａｍｉｎｅ）、サントニン（ｓａｎｔｏｎｉｎ）、セラメクチン（ｓｅｌａｍｅｃｔｉｎ）、スルファジメトキシン（ｓｕｌｆａｄｉｍｅｔｈｏｘｉｎｅ）、スルファドキシン（ｓｕｌｆａｄｏｘｉｎｅ）、スルファメラジン（ｓｕｌｆａｍｅｒａｚｉｎｅ）、スルファモノメトキシン（ｓｕｌｆａｍｏｎｏｍｅｔｈｏｘｉｎｅ）、スルファモイルダプソン（ｓｕｌｆａｍｏｉｌｄａｐｓｏｎｅ）、チアベンダゾール（ｔｈｉａｂｅｎｄａｚｏｌｅ）、チニダゾール（ｔｉｎｉｄａｚｏｌｅ）、トルトラズリル（ｔｏｌｔｒａｚｕｒｉｌ）、トリブロムサラン（ｔｒｉｂｒｏｍｓａｌａｎ）及びトリクラベンダゾール（ｔｒｉｃｌａｂｅｎｄａｚｏｌｅ）など。 Anthelmintic: acriflavine, albendazole, atovagone, azithromycin, bisionol, bromfenodac, bromofenfos chloroquine, clazuril, clindamycin, chlorsulon, closantel, coumafos, chlorofendi, dichlorophenol Diethylcarbamazine, diminazene, disophenol, dithizanine iodide, ect, decine, decide, decide, decide ), Fenbendazole, flubendazole, furazolidone, glycalpyramide, imidocarb, ivermectin ( vermectin, levamisole, mebendazole, mefloquine, melarsamine hydrochloride, methiridine, methiridine, metridine Morantel (morantel), moxidectin, nicarbazin, niclosamide, nitroskanate, nitroxynil, omphalo Oxphaltine, oxantellate, oxendazole, oxclodide, oxclodide Piperazine acid, piperazine citrate, piperazine phosphate, PNU-97333 (paraherquamide A), PNU-141962 (2-dexapuy, 2-dex) Radiquaantel, primaquine, propetamphos, dipoxur, sulphine, sulphine, selenium, selenium Sulfadoxine, sulfamerazine, sulfamonomethoxine, sulfamoyldapson, thiabendazole, tinidazole (ti) such as nidazole, toltrazuril, tribromsalan, and triclabendazole.

抗真菌剤：ケトコナゾール（ｋｅｔｏｃｏｎａｚｏｌｅ）及びミコナゾール硝酸塩（ｍｉｃｏｎａｚｏｌｅｎｉｔｒａｔｅ）など。 Antifungal agents: ketoconazole and miconazole nitrate.

抗菌剤：アモキシシリン（ａｍｏｘｉｃｉｌｌｉｎ）、アンピシリン（ａｍｐｉｃｉｌｌｉｎ）、ベトキサジン（ｂｅｔｈｏｘａｚｉｎ）、ビチオノール（ｂｉｔｈｉｏｎｏｌ）、ブロノポール（ｂｒｏｎｏｐｏｌ）、セファピリン（ｃｅｆａｐｉｒｉｎ）、セファゾリン（ｃｅｆａｚｏｌｉｎ）、セフキノム（ｃｅｆｑｕｉｎｏｍｅ）、セフチオフル（ｃｅｆｔｉｏｆｕｒ）、クロルテトラサイクリン（ｃｈｌｏｒｔｅｔｒａｃｙｃｌｉｎｅ）、クラブラン酸（ｃｌａｖｕｌａｎｉｃａｃｉｄ）、ダノフロキサシン（ｄａｎｏｆｌｏｘａｃｉｎ）、ジフロキサシン（ｄｉｆｌｏｘａｃｉｎ）、ジニトルミド（ｄｉｎｉｔｏｌｍｉｄｅ）、エンロフロキサシン（ｅｎｒｏｆｌｏｘａｃｉｎ）、フロルフェニコール（ｆｌｏｒｆｅｎｉｃｏｌ）、リンコマイシン（ｌｉｎｃｏｍｙｃｉｎ）、ロメフロキサシン（ｌｏｍｅｆｌｏｘａｃｉｎ）、マルボフロキサシン（ｍａｒｂｏｆｌｏｘａｃｉｎ）、ミロキサシン（ｍｉｌｏｘａｃｉｎ）、ミロサマイシン（ｍｉｒｏｓａｍｙｃｉｎ）、ニトラピリン（ｎｉｔｒａｐｙｒｉｎ）、ノルフロキサシン（ｎｏｒｆｌｏｘａｃｉｎ）、オクチリノン（ｏｃｔｈｉｌｉｎｏｎｅ）、オフロキサシン（ｏｆｌｏｘａｃｉｎ）、オルビフロキサシン（ｏｒｂｉｆｌｏｘａｃｉｎ）、オキソリニック酸（ｏｘｏｌｉｎｉｃａｃｉｄ）、オキシテトラサイクリン（ｏｘｙｔｅｔｒａｃｙｃｌｉｎｅ）、ペニシリン（ｐｅｎｉｃｉｌｌｉｎ）、ストレプトマイシン（ｓｔｒｅｐｔｏｍｙｃｉｎ）、チアンフェニコール（ｔｈｉａｍｐｈｅｎｉｃｏｌ）、フマル酸チアムリン（ｔｉａｍｕｌｉｎｆｕｍａｒａｔｅ）、リン酸チルミコシン（ｔｉｌｍｉｃｏｓｉｎｐｈｏｓｐｈａｔｅ）、酢酸イソ吉草酸タイロシン（ａｃｅｔｙｌｉｓｏｖａｌｅｒｙｌｔｙｌｏｓｉｎ）、リン酸タイロシン（ｔｙｌｏｓｉｎｐｈｏｓｐｈａｔｅ）、ツラスロマイシン（ｔｕｌａｔｈｒｏｍｙｃｉｎ）、バルネムリン（ｖａｌｎｅｍｕｌｉｎ）、貝殻焼成カルシウム（酸化カルシウム）、タラロマイセス属菌、トリコデルマ属菌及びユニオチリウム属菌など。 Antibacterial agents: amoxicillin, ampicillin, betoxazine, bitionol, bronopol, cefapirin, cefazolin, cefazolin, cefazolin, cefazolin, cefazolin, cefazolin (Chlortetracycline), clavulanic acid, danofloxacin, difloxacin, dinitroxine, enrofloxacin, florfenicol (florenicol) , Lincomycin, lomefloxacin, marbofloxacin, miloxacin, milosamycin, nitrapirin, inloxin, norfloxacin (nor) Orbifloxacin, oxolinic acid, oxytetracycline, penicillin, streptomycin, thiamphenicol, thiamphenicol Tiamulin fumarate, tilmicosin phosphate, tylosin isovaleric acid, tyrosin phosphate, turathrneuminum shell Calcium), Talalomyces spp., Trichoderma spp. And Unioniolium spp.

本発明化合物の施用薬量は適用場面、施用時期、施用方法、栽培作物等により差異はあるが一般には有効成分量としてヘクタール（ｈａ）当たり０．００５〜５０ｋｇ程度が適当である。 The application amount of the compound of the present invention varies depending on the application scene, the application time, the application method, the cultivated crops, etc., but generally the amount of the active ingredient is suitably about 0.005 to 50 kg per hectare (ha).

次に本発明化合物を用いる場合の製剤の配合例を示す。但し本発明の配合例は、これらのみに限定されるものではない。なお、以下の配合例において「部」は重量部を意味する。
〔水和剤〕
本発明化合物０．１〜８０部
固体担体５〜９８．９部
界面活性剤１〜１０部
その他０〜５部
その他として、例えば固結防止剤、分解防止剤等が挙げられる。
〔乳剤〕
本発明化合物０．１〜３０部
液体担体４５〜９５部
界面活性剤４．９〜１５部
その他０〜１０部
その他として、例えば展着剤、分解防止剤等が挙げられる。
〔懸濁剤〕
本発明化合物０．１〜７０部
液体担体１５〜９８．８９部
界面活性剤１〜１２部
その他０．０１〜３０部
その他として、例えば凍結防止剤、増粘剤等が挙げられる。
〔顆粒水和剤〕
本発明化合物０．１〜９０部
固体担体０〜９８．９部
界面活性剤１〜２０部
その他０〜１０部
その他として、例えば結合剤、分解防止剤等が挙げられる。
〔液剤〕
本発明化合物０．０１〜７０部
液体担体２０〜９９．９９部
その他０〜１０部
その他として、例えば凍結防止剤、展着剤等が挙げられる。
〔粒剤〕
本発明化合物０．０１〜８０部
固体担体１０〜９９．９９部
その他０〜１０部
その他として、例えば結合剤、分解防止剤等が挙げられる。
〔粉剤〕
本発明化合物０．０１〜３０部
固体担体６５〜９９．９９部
その他０〜５部
その他として、例えばドリフト防止剤、分解防止剤等が挙げられる。 Next, formulation examples of the preparation when the compound of the present invention is used are shown. However, the formulation examples of the present invention are not limited to these. In the following formulation examples, “parts” means parts by weight.
[Wettable powder]
Compound of the present invention 0.1 to 80 parts Solid carrier 5 to 98.9 parts Surfactant 1 to 10 parts Others 0 to 5 parts Others include, for example, anti-caking agents and decomposition inhibitors.
〔emulsion〕
Compound of the present invention 0.1-30 parts Liquid carrier 45-95 parts Surfactant 4.9-15 parts Others 0-10 parts Others include, for example, spreading agents, decomposition inhibitors and the like.
[Suspension]
Compounds of the present invention 0.1 to 70 parts Liquid carrier 15 to 98.89 parts Surfactant 1 to 12 parts Others 0.01 to 30 parts Others include, for example, antifreezing agents and thickeners.
(Granule wettable powder)
Compound of the present invention 0.1 to 90 parts Solid carrier 0 to 98.9 parts Surfactant 1 to 20 parts Others 0 to 10 parts Others include, for example, binders and decomposition inhibitors.
[Liquid]
Compound of the present invention 0.01 to 70 parts Liquid carrier 20 to 99.99 parts Others 0 to 10 parts Other examples include antifreezing agents and spreading agents.
[Granule]
Compound of the present invention 0.01 to 80 parts Solid carrier 10 to 99.99 parts Others 0 to 10 parts Others include, for example, binders, decomposition inhibitors and the like.
[Dust]
Compound of the present invention 0.01 to 30 parts Solid support 65 to 99.99 parts Others 0 to 5 parts Other examples include a drift inhibitor and a decomposition inhibitor.

使用に際しては上記製剤を水で１〜１００００倍に希釈して又は希釈せずに散布する。 In use, the preparation is sprayed diluted with water 1 to 10,000 times or without dilution.

次に、本発明化合物を有効成分とする農園芸用殺菌剤の製剤例を具体的に示すが、これらのみに限定されるものではない。なお、以下の製剤例において「部」は重量部を意味する。
〔製剤例１〕乳剤
本発明化合物Ｎｏ．Ａ−１２０部
メチルナフタレン５５部
シクロヘキサノン２０部
ソルポール２６８０５部
（非イオン性界面活性剤とアニオン性界面活性剤との混合物：東邦化学工業（株）商品名）
以下を均一に混合して乳剤とする。使用に際しては上記乳剤を５０〜２００００倍に希釈して有効成分量がヘクタール当たり０．００５〜５０ｋｇになるように散布する。
〔製剤例２〕水和剤
本発明化合物Ｎｏ．Ａ−１２５部
パイロフィライト６６部
ソルポール５０３９４部
（アニオン性界面活性剤：東邦化学工業（株）商品名）
カープレックス＃８０Ｄ３部
（ホワイトカーボン：塩野義製薬（株）商品名）
リグニンスルホン酸カルシウム２部
以上を均一に混合粉砕して水和剤とする。 Next, although the formulation example of the agricultural and horticultural fungicide which uses this invention compound as an active ingredient is shown concretely, it is not limited only to these. In the following formulation examples, “parts” means parts by weight.
[Formulation Example 1] Emulsion This invention Compound No. A-1 20 parts Methylnaphthalene 55 parts Cyclohexanone 20 parts Solpol 2680 5 parts (Mixture of nonionic surfactant and anionic surfactant: Toho Chemical Industries, Ltd. trade name)
The following are uniformly mixed to obtain an emulsion. In use, the emulsion is diluted 50 to 20000 times and sprayed so that the amount of the active ingredient is 0.005 to 50 kg per hectare.
[Formulation Example 2] Wetting agent Compound No. of the present invention. A-1 25 parts Pyrophyllite 66 parts Solpol 5039 4 parts (Anionic surfactant: Toho Chemical Industries, Ltd. trade name)
Carplex # 80D 3 parts (White Carbon: Shionogi & Co., Ltd. trade name)
2 parts or more of calcium lignin sulfonate are mixed and ground uniformly to obtain a wettable powder.

使用に際しては上記水和剤を５０〜２００００倍に希釈して有効成分量がヘクタール当たり０．００５〜５０ｋｇになるように散布する。
〔製剤例３〕粉剤
本発明化合物Ｎｏ．Ａ−１３部
カープレックス＃８０Ｄ０．５部
（ホワイトカーボン：塩野義製薬（株）商品名）
カオリナイト９５部
リン酸ジイソプロピル１．５部
以上を均一に混合粉砕して粉剤とする。使用に際して上記粉剤を有効成分量がヘクタール当たり０．００５〜５０ｋｇになるように散布する。
〔製剤例４〕粒剤
本発明化合物Ｎｏ．Ａ−１５部
ベントナイト３０部
タルク６４部
リグニンスルホン酸カルシウム１部
以上を均一に混合粉砕して少量の水を加えて撹拌混合し、押出式造粒機で造粒し、乾燥して粒剤とする。使用に際して上記粒剤を有効成分量がヘクタール当たり０．００５〜５０ｋｇになるように散布する。
〔製剤例５〕懸濁剤
本発明化合物Ｎｏ．Ａ−１２５部
ソルポール３３５３５部
（非イオン性界面活性剤：東邦化学工業（株）商品名）
ルノックス１０００Ｃ０．５部
（陰イオン界面活性剤：東邦化学工業（株）商品名）
ザンサンガム（天然高分子）０．２部
安息香酸ソーダ０．４部
プロピレングリコール１０部
水５８．９部
有効成分（本発明化合物）を除く上記の成分を均一に溶解し、ついで本発明化合物を加えよく撹拌した後、サンドミルにて湿式粉砕してフロアブル剤を得る。使用に際しては、上記フロアブル剤を５０〜２００００倍に希釈して有効成分量がヘクタール当たり０．００５〜５０ｋｇになるように散布する。
〔製剤例６〕粒状水和剤
本発明化合物Ｎｏ．Ａ−１７５部
ハイテノールＮＥ−１５５部
（アニオン性界面活性剤：第一工業製薬（株）商品名）
バニレックスＮ１０部
（アニオン性界面活性剤：日本製紙（株）商品名）
カープレックス＃８０Ｄ１０部
（ホワイトカーボン：塩野義製薬（株）商品名）
以上を均一に混合微粉砕して少量の水を加えて撹拌混合し、押出式造粒機で造粒し、乾燥してドライフロアブル剤とする。使用に際しては水で５０〜２００００倍に希釈して、有効成分が１ヘクタール当たり０．００５〜５０ｋｇになるように散布する。 In use, the wettable powder is diluted 50 to 20000 times and sprayed so that the amount of the active ingredient is 0.005 to 50 kg per hectare.
[Formulation Example 3] Powder Compound Nos. A-1 3 parts Carplex # 80D 0.5 part (White carbon: Shionogi & Co., Ltd. trade name)
Kaolinite 95 parts Diisopropyl phosphate 1.5 parts or more uniformly mixed and pulverized to form a powder. In use, the powder is sprayed so that the amount of the active ingredient is 0.005 to 50 kg per hectare.
[Formulation Example 4] Granules of the present compound No. A-1 5 parts Bentonite 30 parts Talc 64 parts Calcium lignin sulfonate 1 part The above mixture is uniformly mixed and ground, a small amount of water is added and mixed with stirring, granulated with an extrusion granulator, dried and granulated. And In use, the above granule is sprayed so that the amount of the active ingredient is 0.005 to 50 kg per hectare.
[Formulation Example 5] Suspending Agent Compound No. A-1 25 parts Solpol 3353 5 parts (Nonionic surfactant: Toho Chemical Co., Ltd. trade name)
Lnox 1000C 0.5 part (Anionic surfactant: Toho Chemical Co., Ltd. trade name)
Xanthan gum (natural polymer) 0.2 parts Sodium benzoate 0.4 parts Propylene glycol 10 parts Water 58.9 parts The above ingredients except the active ingredient (the compound of the present invention) are uniformly dissolved, and then the compound of the present invention is added. After thorough stirring, a flowable agent is obtained by wet grinding with a sand mill. In use, the flowable agent is diluted 50 to 20000 times and sprayed so that the amount of the active ingredient is 0.005 to 50 kg per hectare.
[Formulation Example 6] Granular wettable powder Compound No. A-1 75 parts Hightenol NE-15 5 parts (Anionic surfactant: trade name of Daiichi Kogyo Seiyaku Co., Ltd.)
Vanillex N 10 parts (anionic surfactant: Nippon Paper Industries Co., Ltd. trade name)
Carplex # 80D 10 parts (White Carbon: Shionogi & Co., Ltd. trade name)
The above mixture is uniformly mixed and pulverized, a small amount of water is added, mixed with stirring, granulated with an extrusion granulator, and dried to obtain a dry flowable agent. In use, it is diluted 50 to 20000 times with water and sprayed so that the active ingredient is 0.005 to 50 kg per hectare.

本発明化合物の施用方法としては、茎葉散布、土壌処理、種子消毒等が挙げられるが、通常当業者が利用する一般的な方法においても有効である。 Application methods of the compound of the present invention include foliage spraying, soil treatment, seed disinfection and the like, but they are also effective in general methods usually used by those skilled in the art.

以下に本発明化合物の合成例、試験例を実施例として具体的に述べることで、本発明をさらに詳しく説明するが、本発明はこれらによって限定されるものではない。 Hereinafter, the present invention will be described in more detail by specifically describing synthesis examples and test examples of the compounds of the present invention as examples, but the present invention is not limited thereto.

［合成例］
合成例１
（Ｅ）−Ｎ’−（１−（４−フルオロフェニル）エチリデン）−Ｎ−（２−（４−メチル−５−オキソ−４，５−ジヒドロ−１Ｈ−テトラゾール−１−イル）ベンジル）シクロプロパンカルボヒドラジドの製造（本発明化合物Ｎｏ．Ａ−５）
（Ｅ）−Ｎ’−（１−（４−フルオロフェニル）エチリデン）シクロプロパンカルボヒドラジド０．１５ｇ（０．７０ｍｍｏｌ）のＮ，Ｎ−ジメチルホルムアミド２ｍｌ溶液にカリウムｔｅｒｔ−ブトキシド０．８６ｇ（０．７７ｍｍｏｌ）を室温にて添加し、３０分間攪拌した。攪拌終了後、該反応混合物に１−（２−（ブロモメチル）フェニル）−４−メチル−１Ｈ−テトラゾール−５（４Ｈ）−オン０．１７ｇ（０．６４ｍｍｏｌ）を室温にて添加し、５時間攪拌を継続した。反応完結後、該反応混合物に水１０ｍｌを添加し、反応を停止させた後、該反応液を酢酸エチルにて抽出（１０ｍｌ×１）した。得られた有機層を水洗した後、飽和食塩水次いで無水硫酸ナトリウムにて脱水・乾燥、減圧下にて溶媒を留去した。得られた残渣をシリカゲルカラムクロマトグラフィー｛ｎ−ヘキサン：酢酸エチル＝２：１（体積比）｝にて精製し、目的物０．１４ｇを白色結晶として得た。
融点：１４７〜１４９℃
本発明化合物は、前記製造法及び実施例に準じて製造することができる。合成例１と同様に製造した本発明に包含されるアシルヒドラゾン誘導体の例を第５表乃至第１０表に示すが、本発明に包含されるアシルヒドラゾン誘導体はこれらのみに限定されるものではない。 [Synthesis example]
Synthesis example 1
(E) -N ′-(1- (4-Fluorophenyl) ethylidene) -N- (2- (4-methyl-5-oxo-4,5-dihydro-1H-tetrazol-1-yl) benzyl) cyclo Production of propanecarbohydrazide (present compound No. A-5)
(E) -N ′-(1- (4-fluorophenyl) ethylidene) cyclopropanecarbohydrazide 0.15 g (0.70 mmol) in 2 ml of N, N-dimethylformamide 0.86 g of potassium tert-butoxide (0. 77 mmol) was added at room temperature and stirred for 30 minutes. After the stirring was completed, 0.17 g (0.64 mmol) of 1- (2- (bromomethyl) phenyl) -4-methyl-1H-tetrazol-5 (4H) -one was added to the reaction mixture at room temperature for 5 hours. Stirring was continued. After completion of the reaction, 10 ml of water was added to the reaction mixture to stop the reaction, and the reaction solution was extracted with ethyl acetate (10 ml × 1). The obtained organic layer was washed with water, dehydrated and dried over saturated brine and then anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure. The obtained residue was purified by silica gel column chromatography {n-hexane: ethyl acetate = 2: 1 (volume ratio)} to obtain 0.14 g of the desired product as white crystals.
Melting point: 147-149 ° C
This invention compound can be manufactured according to the said manufacturing method and an Example. Examples of acyl hydrazone derivatives included in the present invention produced in the same manner as in Synthesis Example 1 are shown in Tables 5 to 10, but the acyl hydrazone derivatives included in the present invention are not limited to these. .

尚、表中、Ｍｅはメチル基を、Ｅｔはエチル基を、ｉＰｒはｉ−プロピル基を、ｃＰｒはシクロプロピル基を、ｔＢｕはｔｅｒｔ−ブチル基を、ｃＢｕはシクロブチル基を、Ｐｈはフェニル基を、Ｂｎはベンジル基を、Ａｃはアセチル基を、＝は２重結合をそれぞれ表す。 In the table, Me represents a methyl group, Et represents an ethyl group, iPr represents an i-propyl group, cPr represents a cyclopropyl group, tBu represents a tert-butyl group, cBu represents a cyclobutyl group, and Ph represents a phenyl group. , Bn represents a benzyl group, Ac represents an acetyl group, and = represents a double bond.

また、「＊１」は化合物の性状が油状又は樹脂状であったことを意味する。
［第５表］ “* 1” means that the property of the compound was oily or resinous.
[Table 5]

−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−
No. (Z)_m R² R³ (Y)_n 融点(℃)
−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−
A-1 4-F Me Me 3-Cl 148-150
A-2 4-F Me Me 3-Me 129-134
A-3 3-F Me Me 3-Me 131-133
A-4 4-F Me OMe 3-Me 153-158
A-5 4-F Me cPr - 147-149
A-6 4-F Me H 3-Me 104-108
A-7 4-F Me iPr - *1
A-8 - Me Et 3-Me 107-113
A-9 4-F Me cPr 3-Me 171-174
A-10 4-F Me CH₂OMe 3-Me 125-127
A-11 4-F Me Et 3-Me 119-125
A-12 4-F Me Et - 82-86
A-13 - Me Et - 70-73
A-14 2-OMe Me Et 3-Me 149-151
A-15 4-Ph Me Me 3-Me 173-176
A-16 - Me cPr 3-Me 149-151
A-17 3-OMe Me Et 3-Me 116-118
A-18 4-OMe Me Et 3-Me 130-134
A-19 - Ph Me 3-Me 165-167
A-20 - Ph Et 3-Me 126-129
A-21 4-CO₂Me Me Et 3-Me 132-135
A-22 3-Cl-4-F Me Et 3-Me 133-135
A-23 3-Br Me Et 3-Me 126-128
A-24 3-OCF₃ Me Et 3-Me 105-107
A-25 3-CF₃ Me Et 3-Me 116-118
A-26 3-CN Me Et 3-Me 126-128
A-27 4-F Me cBu 3-Me 151-153
A-28 4-Me Me CH₂OEt 3-Me 128-130
A-29 4-F Me tBu 3-Me 107-110
A-30 4-F Me C(O)OEt 3-Me 120-124
A-31 4-C(=NOMe)Me Me Et 3-Me 103-105
A-32 4-tBu Me Et 3-Me 158-160
A-33 3,5-di-F Me Et 3-Me 105-108
A-34 4-F Me cPr 3-Me 177-179
A-35 4-F Me CH₂OAc 3-Me 122-124
A-36 3-Cl-4-F Me cPr 3-Me 155-160
A-37 4-F Me C(Me)(OMe)₂ 3-Me 128-134
A-38 4-F Me Et 3-Me 130-132
A-39 4-F Me cPr 3-Me 135-138
A-40 3-Cl Me Et 3-Me 116-119
A-41 4-F Me CH₂SMe 3-Me 138-140
A-42 3-Br Me Et 3-Me 103-105
A-43 4-Cl Me cPr 3-Me 153-155
A-44 3-Br Me cPr 3-Me 139-140
A-45 3-Br Me Me 3-Me 147-149
A-46 3-Ac Me Et 3-Me 124-130
A-47 4-F Me Et 3-Me 125-127
A-48 3-Br-4-F Me Et 3-Me 124-126
A-49 4-OCF₃ Me Et 3-Me 140-141
A-50 3-Br-4-Me Me Et 3-Me 105-106
A-51 3-I Me Et 3-Me 131-132
A-52 4-F Me CF₂H 3-Me 160-162
A-53 3-Br-4-F Me cPr 3-Me 148-150
A-54 3,5-di-Cl Me Et 3-Me 125-127
A-55 3-Br-4-Cl Me Et 3-Me 146-148
A-56 3-Br-4-Cl Me cPr 3-Me 154-155
A-57 3-Me Me Et 3-Me 118-119
A-58 4-F Me Et 3-Me 85-87
A-59 4-F Me cPr 3-Me 104-108
A-60 3-CF₂H Me Et 3-Me 140-142
A-61 3-SMe Me cPr 3-Me *1
A-62 3-OBn Me Et 3-Me 124-130
A-63 3-Br-5-Cl Me Et 3-Me 139-143
A-64 3-Cl Me cPr - 93-94
A-65 3-OMe Me cPr - *1
A-66 3-Cl Me Et - *1
A-67 3-Cl-4-F Me Et - 90-92
A-68 4-Br Me Me - 127-128
A-69 4-Br Me cPr - 127-128
A-70 3,5-di-Cl Me Et - 72-104
A-71 4-F Me Et 6-F 147-149
−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−
［第６表］ ------------------------------
No. (Z) _m R ² R ³ (Y) _n Melting point (° C)
------------------------------
A-1 4-F Me Me 3-Cl 148-150
A-2 4-F Me Me 3-Me 129-134
A-3 3-F Me Me 3-Me 131-133
A-4 4-F Me OMe 3-Me 153-158
A-5 4-F Me cPr-147-149
A-6 4-F Me H 3-Me 104-108
A-7 4-F Me iPr-* 1
A-8-Me Et 3-Me 107-113
A-9 4-F Me cPr 3-Me 171-174
A-10 4-F Me CH ₂ OMe 3-Me 125-127
A-11 4-F Me Et 3-Me 119-125
A-12 4-F Me Et-82-86
A-13-Me Et-70-73
A-14 2-OMe Me Et 3-Me 149-151
A-15 4-Ph Me Me 3-Me 173-176
A-16-Me cPr 3-Me 149-151
A-17 3-OMe Me Et 3-Me 116-118
A-18 4-OMe Me Et 3-Me 130-134
A-19-Ph Me 3-Me 165-167
A-20-Ph Et 3-Me 126-129
A-21 4-CO ₂ Me Me Et 3-Me 132-135
A-22 3-Cl-4-F Me Et 3-Me 133-135
A-23 3-Br Me Et 3-Me 126-128
A-24 3-OCF ₃ Me Et 3-Me 105-107
A-25 3-CF ₃ Me Et 3-Me 116-118
A-26 3-CN Me Et 3-Me 126-128
A-27 4-F Me cBu 3-Me 151-153
A-28 4-Me Me CH ₂ OEt 3-Me 128-130
A-29 4-F Me tBu 3-Me 107-110
A-30 4-F Me C (O) OEt 3-Me 120-124
A-31 4-C (= NOMe) Me Me Et 3-Me 103-105
A-32 4-tBu Me Et 3-Me 158-160
A-33 3,5-di-F Me Et 3-Me 105-108
A-34 4-F Me cPr 3-Me 177-179
A-35 4-F Me CH ₂ OAc 3-Me 122-124
A-36 3-Cl-4-F Me cPr 3-Me 155-160
A-37 4-F Me C (Me) (OMe) ₂ 3-Me 128-134
A-38 4-F Me Et 3-Me 130-132
A-39 4-F Me cPr 3-Me 135-138
A-40 3-Cl Me Et 3-Me 116-119
A-41 4-F Me CH ₂ SMe 3-Me 138-140
A-42 3-Br Me Et 3-Me 103-105
A-43 4-Cl Me cPr 3-Me 153-155
A-44 3-Br Me cPr 3-Me 139-140
A-45 3-Br Me Me 3-Me 147-149
A-46 3-Ac Me Et 3-Me 124-130
A-47 4-F Me Et 3-Me 125-127
A-48 3-Br-4-F Me Et 3-Me 124-126
A-49 4-OCF ₃ Me Et 3-Me 140-141
A-50 3-Br-4-Me Me Et 3-Me 105-106
A-51 3-I Me Et 3-Me 131-132
A-52 4-F Me CF ₂ H 3-Me 160-162
A-53 3-Br-4-F Me cPr 3-Me 148-150
A-54 3,5-di-Cl Me Et 3-Me 125-127
A-55 3-Br-4-Cl Me Et 3-Me 146-148
A-56 3-Br-4-Cl Me cPr 3-Me 154-155
A-57 3-Me Me Et 3-Me 118-119
A-58 4-F Me Et 3-Me 85-87
A-59 4-F Me cPr 3-Me 104-108
A-60 3-CF ₂ H Me Et 3-Me 140-142
A-61 3-SMe Me cPr 3-Me * 1
A-62 3-OBn Me Et 3-Me 124-130
A-63 3-Br-5-Cl Me Et 3-Me 139-143
A-64 3-Cl Me cPr-93-94
A-65 3-OMe Me cPr-* 1
A-66 3-Cl Me Et-* 1
A-67 3-Cl-4-F Me Et-90-92
A-68 4-Br Me Me-127-128
A-69 4-Br Me cPr-127-128
A-70 3,5-di-Cl Me Et-72-104
A-71 4-F Me Et 6-F 147-149
------------------------------
[Table 6]

−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−
No. (Z)_n R² R³ (Y)_n 融点(℃)
−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−
B-1 6-Br Me Et - *1
B-2 4,6-di-Cl Me Et 3-OMe 61-64
B-3 6-Cl Me Et 3-Me 120-123
B-4 6-Cl Me cPr 3-Me 147-150
B-5 6-OMe Me Et 3-Me 108-110
B-6 6-Br Me Et 3-Me 126-128
B-7 6-Cl Me cPr 3-F 126-128
B-8 4-Me Me Et 3-Me 149-150
B-9 5,6-di-Me Me Et 3-Me 121-124
B-10 6-Br Me cPr 3-Me 150-153
B-11 6-F Me Et 3-Me 113-116
−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−
［第７表］ ------------------------------
No. (Z) _n R ² R ³ (Y) _n Melting point (° C)
------------------------------
B-1 6-Br Me Et-* 1
B-2 4,6-di-Cl Me Et 3-OMe 61-64
B-3 6-Cl Me Et 3-Me 120-123
B-4 6-Cl Me cPr 3-Me 147-150
B-5 6-OMe Me Et 3-Me 108-110
B-6 6-Br Me Et 3-Me 126-128
B-7 6-Cl Me cPr 3-F 126-128
B-8 4-Me Me Et 3-Me 149-150
B-9 5,6-di-Me Me Et 3-Me 121-124
B-10 6-Br Me cPr 3-Me 150-153
B-11 6-F Me Et 3-Me 113-116
------------------------------
[Table 7]

−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−
No. (Z)_p R² R³ (Y)_n 融点(℃)
−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−
C-1 5-Cl Me cPr 3-Me 163-165
C-2 5-Cl Me Et 3-Me 136-138
−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−
［第８表］ ------------------------------
No. (Z) _p R ² R ³ (Y) _n Melting point (° C)
------------------------------
C-1 5-Cl Me cPr 3-Me 163-165
C-2 5-Cl Me Et 3-Me 136-138
------------------------------
[Table 8]

−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−
No. (Z)_p R² R³ (Y)_n 融点(℃)
−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−
D-1 2,5-di-Cl Me Et 3-Me 119-122
−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−
［第９表］ ------------------------------
No. (Z) _p R ² R ³ (Y) _n Melting point (° C)
------------------------------
D-1 2,5-di-Cl Me Et 3-Me 119-122
------------------------------
[Table 9]

−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−
No. (Z)_m R² R³ (Y)_n 融点(℃)
−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−
E-1 4-Cl Me Et 3-Me 162-165
−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−
［第１０表］ ------------------------------
No. (Z) _m R ² R ³ (Y) _n Melting point (° C)
------------------------------
E-1 4-Cl Me Et 3-Me 162-165
------------------------------
[Table 10]

−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−
No. R¹ R² R³ (Y)_n 融点(℃)
−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−
F-1 Me Me Et 3-Me 67-71
−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−
第５表〜第１０表の本発明化合物のうち、融点の記載のない化合物の^１Ｈ−ＮＭＲデータを第１１表に示す。 ------------------------------
No. R ¹ R ² R ³ (Y) _n Melting point (° C)
------------------------------
F-1 Me Me Et 3-Me 67-71
------------------------------
Among the compounds of the present invention shown in Tables 5 to 10, ¹ H-NMR data of compounds having no melting point are shown in Table 11.

表中の記号は下記の意味を表す。
ｓ：シングレット、ｄ：ダブレット、ｍ：マルチプレット。 The symbols in the table have the following meanings.
s: singlet, d: doublet, m: multiplet.

なお、プロトン核磁気共鳴ケミカルシフト値は、基準物質としてＭｅ_４Ｓｉ（テトラメチルシラン）を用い、重クロロホルム溶媒中で、３００ＭＨｚにて測定した。
［第１１表］
−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−
No. ¹H-NMR (CDCl₃, Me₄Si, 300MHz)
−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−
A-7 δ7.85-7.70 (m, 2H), 7.60-7.25 (m, 4H),
7.20-7.00 (m, 2H), 4.92 (s, 2H),
3.48 (s, 3H), 2.62-2.42 (m, 1H),
2.01 (s, 3H), 1.01 (d, 6H, J=6.9Hz)。
A-61 δ7.75-7.65 (m, 1H), 7.55-7.10 (m, 6H),
5.08 (s, 2H), 3.61 (s, 3H),
2.51 (s, 3H), 2.43 (s, 3H),
1.89 (s, 3H), 1.50-1.20 (m, 1H),
1.00-0.82 (m, 2H), 0.72-0.56 (m, 2H)。
A-65 δ7.65-7.15 (m, 7H), 7.10-6.95 (m, 1H),
5.00 (s, 2H), 3.86 (s, 3H),
3.50 (s, 3H), 2.00 (s, 3H),
1.60-1.40 (m, 1H), 1.05-0.90 (m, 2H),
0.75-0.60 (m, 2H)。
A-66 δ7.80-7.70 (m, 1H), 7.70-7.25 (m, 7H),
4.94 (s, 2H), 3.53 (s, 3H),
2.25-2.00 (m, 2H), 1.97 (s, 3H),
1.15-0.95 (m, 3H)。
B-1 δ8.04-7.92 (m, 1H), 7.74-7.25 (m, 6H),
5.00 (s, 2H), 3.62 (s, 3H),
2.35-2.10 (m, 2H), 2.19 (s, 3H),
1.20-1.00 (m, 3H)。
−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−−
［試験例］
次に、本発明化合物の有害生物防除剤としての有用性について、以下の試験例において具体的に説明するが、本発明はこれらのみに限定されるものではない。 The proton nuclear magnetic resonance chemical shift value was measured at 300 MHz in deuterated chloroform solvent using Me ₄ Si (tetramethylsilane) as a reference substance.
[Table 11]
------------------------------
No. ¹ H-NMR (CDCl ₃ , Me ₄ Si, 300 MHz)
------------------------------
A-7 δ7.85-7.70 (m, 2H), 7.60-7.25 (m, 4H),
7.20-7.00 (m, 2H), 4.92 (s, 2H),
3.48 (s, 3H), 2.62-2.42 (m, 1H),
2.01 (s, 3H), 1.01 (d, 6H, J = 6.9Hz).
A-61 δ7.75-7.65 (m, 1H), 7.55-7.10 (m, 6H),
5.08 (s, 2H), 3.61 (s, 3H),
2.51 (s, 3H), 2.43 (s, 3H),
1.89 (s, 3H), 1.50-1.20 (m, 1H),
1.00-0.82 (m, 2H), 0.72-0.56 (m, 2H).
A-65 δ7.65-7.15 (m, 7H), 7.10-6.95 (m, 1H),
5.00 (s, 2H), 3.86 (s, 3H),
3.50 (s, 3H), 2.00 (s, 3H),
1.60-1.40 (m, 1H), 1.05-0.90 (m, 2H),
0.75-0.60 (m, 2H).
A-66 δ7.80-7.70 (m, 1H), 7.70-7.25 (m, 7H),
4.94 (s, 2H), 3.53 (s, 3H),
2.25-2.00 (m, 2H), 1.97 (s, 3H),
1.15-0.95 (m, 3H).
B-1 δ8.04-7.92 (m, 1H), 7.74-7.25 (m, 6H),
5.00 (s, 2H), 3.62 (s, 3H),
2.35-2.10 (m, 2H), 2.19 (s, 3H),
1.20-1.00 (m, 3H).
------------------------------
[Test example]
Next, the usefulness of the compound of the present invention as a pest control agent will be specifically described in the following test examples, but the present invention is not limited to these.

本発明化合物乳剤の調製；本発明化合物を乳化白試料（ソルポール（登録商標）３００５ＸＬ（東邦化学工業製）：Ｎ−メチルピロリドン：ソルベッソ（登録商標）２００（エクソンモービル製）＝１：５：２混合物）中に溶解し、２０％濃度の乳剤を調製した。この乳剤を以下の試験例１〜試験例２に供試した。 Preparation of the present compound emulsion; emulsified white sample of the present compound (Solpol (registered trademark) 3005XL (manufactured by Toho Chemical Industry): N-methylpyrrolidone: Solvesso (registered trademark) 200 (produced by ExxonMobil)) = 1: 5: 2 To give a 20% emulsion. This emulsion was subjected to the following Test Examples 1 and 2.

試験例１ダイズさび病防除効果試験
２葉期のダイズ（品種：エンレイ）を植えた９０ｃｍ^３のプラスチックポットに、本発明化合物乳剤を水で希釈し、５００ｐｐｍに調製した薬液を５ｍｌ散布処理した。散布１日後、ダイズさび病菌（Ｐｈａｋｏｐｓｏｒａｐａｃｈｙｒｈｉｚｉ）の胞子懸濁液をダイズに噴霧接種し、温度２３℃、湿度１００％の接種箱内に１日間入れた。その後、空調温室（２３℃）に置き、１４日間保持した。形成された病斑の接種葉に占める割合を測定し、下記の計算式に従い、防除価を算出した。 Test Example 1 Soybean Rust Disease Control Effect Test A 90 cm ³ plastic pot planted with 2-leaf soybean (variety: Enrei) was diluted with water and sprayed with 5 ml of a chemical solution prepared to 500 ppm. One day after spraying, spore suspension of soybean rust fungus (Phakopsora pachyrhizi) was spray-inoculated on soybean and placed in an inoculation box at a temperature of 23 ° C. and a humidity of 100% for one day. Thereafter, it was placed in an air-conditioned greenhouse (23 ° C.) and held for 14 days. The ratio of the formed lesions to the inoculated leaves was measured, and the control value was calculated according to the following formula.

防除価＝〔１−（処理区病斑面積率／無処理区病斑面積率）〕×１００
その結果、供試した化合物の内、以下の化合物が防除価７０％以上を示した。
本発明化合物；Ｎｏ．Ａ−１〜Ａ−１４，Ａ−１６〜１８，Ａ−２０〜２５，Ａ−２７〜２９，Ａ−３２〜３４，Ａ−３６〜４８，Ａ−５０〜５２，Ａ−５４〜６１，Ａ−６４〜６６，Ａ−６８，Ａ−６９，Ａ−７１，Ｂ−３，Ｂ−４，Ｂ−６〜８，Ｂ−１０，Ｂ−１１，Ｃ−１，Ｃ−２，Ｄ−１，Ｅ−１
試験例２キュウリ炭そ病防除効果試験
９０ｃｍ^３のプラスチックポットにキュウリ（品種：相模半白）を植え、子葉期に本発明化合物乳剤を水で希釈し、５００ｐｐｍに調製した薬液５ｍｌを散布処理した。散布１日後、キュウリ炭そ病菌（Ｃｏｌｌｅｔｏｔｒｉｃｈｕｍｌａｇｅｎａｒｉｕｍ）の分生胞子懸濁液をキュウリに噴霧接種し、温度２５℃、湿度１００％の接種箱内に２日間入れた。その後、空調温室（２３℃）に置き、７日間保持した。形成された病斑の接種葉に占める割合を測定し、試験例１と同様の計算式から防除価を算出した。 Control value = [1- (treatment area lesion area ratio / non-treatment area lesion area ratio)] × 100
As a result, among the compounds tested, the following compounds showed a control value of 70% or more.
Compound of the present invention; A-1 to A-14, A-16 to 18, A-20 to 25, A-27 to 29, A-32 to 34, A-36 to 48, A-50 to 52, A-54 to 61, A-64 to 66, A-68, A-69, A-71, B-3, B-4, B-6 to 8, B-10, B-11, C-1, C-2, D- 1, E-1
Test Example 2 Cucumber Anthracnose Control Effect Test Cucumber (variety: Sagamihanjiro) was planted in a 90 cm ³ plastic pot, and the compound emulsion of the present invention was diluted with water at the cotyledon stage and sprayed with 5 ml of a chemical solution prepared to 500 ppm. . One day after spraying, a conidial spore suspension of cucumber anthracnose fungus (Colletotrichum lagenarium) was spray-inoculated on cucumber and placed in an inoculation box at a temperature of 25 ° C. and a humidity of 100% for 2 days. Thereafter, it was placed in an air-conditioned greenhouse (23 ° C.) and held for 7 days. The ratio of the formed lesions to the inoculated leaves was measured, and the control value was calculated from the same calculation formula as in Test Example 1.

その結果、供試した化合物の内、以下の化合物が防除価７０％以上を示した。
本発明化合物；Ｎｏ．Ａ−４，Ａ−５，Ａ−７，Ａ−１０，Ａ−２６，Ｂ−２〜４，Ｃ−１
試験例３抗真菌活性測定試験
滅菌された試験管に滅菌水を１ｍｌ加え、その水の一部を、黒麹菌の培養されたシャーレに落とし、先を曲げたパスツールピペットの平らな所で上部をこすり、水と混ぜることによって、黒麹菌（Ａｓｐｅｒｇｉｌｌｕｓｎｉｇｅｒ）の胞子を採集した。黒麹菌の胞子を含む水を試験管に戻し、よく混ぜ合わせて黒麹菌胞子溶液を調製して、顕微鏡観察下で、胞子数を計測した。次いで、温めて溶かしたポテト・デキストロース寒天培地（寒天を０．２５重量％含む）を、滅菌された試験管に１４ｍｌ加え、黒麹菌胞子溶液を加えて混合した。本発明化合物をジメチルスルホキシド（ＤＭＳＯ）で溶解し、終濃度が１０μＭになるように調製した薬液を、９６ウェルプレートに１０μｌずつ加え、その上から、黒麹菌胞子を含むＰＤＡ寒天培地を３０μｌずつ加えて、２５℃で２日間培養した。黒麹菌胞子は１ウェルにつき、１０，０００個とした。同一プレート上の未処理サンプルと処理サンプルとの間で黒麹菌の生育を比較して１０段階で評価した。 As a result, among the compounds tested, the following compounds showed a control value of 70% or more.
Compound of the present invention; A-4, A-5, A-7, A-10, A-26, B-2 to 4, C-1
Test example 3 Antifungal activity measurement test Add 1 ml of sterilized water to a sterilized test tube, drop a part of the water into a petri dish where black koji molds are cultured, and place it on the flat surface of a bent Pasteur pipette. The spores of Aspergillus niger were collected by rubbing and mixing with water. Water containing spore of black koji mold was returned to the test tube, mixed well to prepare a black koji mold spore solution, and the number of spores was counted under a microscope. Next, 14 ml of potato-dextrose agar medium (containing 0.25% by weight of agar), which was warmed and dissolved, was added to a sterilized test tube, and a black koji fungus spore solution was added and mixed. A chemical solution prepared by dissolving the compound of the present invention in dimethyl sulfoxide (DMSO) to a final concentration of 10 μM is added to a 96-well plate by 10 μl, and then a PDA agar medium containing black koji fungus spores is added by 30 μl. And cultured at 25 ° C. for 2 days. The number of black bacillus spores was 10,000 per well. The growth of Aspergillus niger was compared between an untreated sample and a treated sample on the same plate and evaluated in 10 stages.

その結果、以下の化合物が１０μＭにて、５０％以上の生育阻害作用を示した。 As a result, the following compounds showed 50% or more growth inhibitory action at 10 μM.

本発明化合物；Ｎｏ．Ａ−１７，Ａ−７０
試験例４抗内部寄生虫測定試験
ショ糖密度勾配遠心法により、ヤギの糞中から捻転胃虫（Ｈａｅｍｏｎｃｈｕｓｃｏｎｔｏｒｔｕｓ）の卵を、以下の方法で、収集及び殺菌処理した。ヤギの糞１００ｇを蒸留水１００ｍｌ中で攪拌し、ガーゼにて濾過した。濾液を１５００ｇにて５分間遠心し、得られた沈殿に、５０重量％ショ糖水溶液を１００ｍｌ加え、３０分間攪拌した。その後、再び、１５００ｇにて５分間遠心した。上清を３０μｍのステンレス製網にて濾過し、集卵した。得られた卵を７重量％次亜塩素酸ナトリウム水溶液に、５分間浸漬することにより殺菌処理し、滅菌水にて洗浄することにより、捻転胃虫の消毒卵を得た。 Compound of the present invention; A-17, A-70
Test Example 4 Anti-Internal Parasite Measurement Test By a sucrose density gradient centrifugation, eggs of a haemomonchus contortus were collected and sterilized by the following method from goat feces. 100 g of goat feces was stirred in 100 ml of distilled water and filtered with gauze. The filtrate was centrifuged at 1500 g for 5 minutes, and 100 ml of a 50% by weight aqueous sucrose solution was added to the resulting precipitate, followed by stirring for 30 minutes. Thereafter, it was centrifuged again at 1500 g for 5 minutes. The supernatant was filtered through a 30 μm stainless steel net and collected. The obtained eggs were sterilized by immersing them in a 7% by weight aqueous sodium hypochlorite solution for 5 minutes, and washed with sterilized water to obtain disinfected eggs of torsion gastritis.

９６ウェルプレートに、温めて溶かしたポテト・デキストロース寒天培地（寒天を１重量％含む）を、１ウエルあたり６０μｌずつ分注した。その後、卵を含む滅菌水を、１ウエルあたり３０μｌずつ加えた。卵の数は、１ウェルあたり１００個とした。この上から、本発明化合物をジメチルスルホキシド（ＤＭＳＯ）で溶解し、終濃度が１００ｐｐｍになるように調製した薬液を、１０μｌずつ添加した。暗黒条件下２５℃にて、７日間静置した。孵化後、生きている捻転胃虫の数（孵化後生存虫数）を計測し、下記の計算式に従い、無処理区に対する不活動率を算出した。 In a 96-well plate, 60 μl of potato dextrose agar medium (containing 1 wt% agar) was dispensed per well. Thereafter, sterilized water containing eggs was added at 30 μl per well. The number of eggs was 100 per well. From this, the compound of the present invention was dissolved in dimethyl sulfoxide (DMSO), and 10 μl of a chemical solution prepared so that the final concentration was 100 ppm was added. It was allowed to stand for 7 days at 25 ° C. under dark conditions. After hatching, the number of live torsion stomach insects (the number of live insects after hatching) was counted, and the inactivity rate for the untreated area was calculated according to the following formula.

不活動率（％）＝［１−（孵化後生存虫数／無処理区の孵化後生存虫数）］×１００
その結果、以下の化合物が１００ｐｐｍ処理にて、不活動率５０％以上を示した。 Inactivity rate (%) = [1- (number of surviving insects after hatching / number of surviving insects after hatching in non-treated area)] × 100
As a result, the following compounds showed an inactivity rate of 50% or more after 100 ppm treatment.

本発明化合物；Ｎｏ．Ａ−６１，Ａ−６２ Compound of the present invention; A-61, A-62

本発明に係るアシルヒドラゾン誘導体は、優れた有害生物防除活性、特に殺菌活性を示し、且つ、ホ乳動物、魚類及び有用昆虫等の非標的生物に対してほとんど悪影響の無い、極めて有用な化合物である。 The acyl hydrazone derivative according to the present invention is an extremely useful compound that exhibits excellent pest control activity, particularly bactericidal activity, and has almost no adverse effect on non-target organisms such as mammals, fish and useful insects. is there.

Claims

Formula (I):

[Wherein W represents an oxygen atom or a sulfur atom,
A represents an oxygen atom or a sulfur atom,
R ¹ _is, C 1 -C ₆ alkyl, halo _(C 1 ~C ₆₎ ^alkyl, optionally substituted by ^{R a1} _(C 1 ~C ₆₎ _alkyl, C 3 -C ₆ _cycloalkyl, C 2 -C ₆ alkenyl, (C ₂ -C ₆ ) alkenyl optionally substituted by R ^b , C ₁ -C ₆ alkoxy, phenyl, phenyl substituted by (Z) _m , pyridin-2-yl, (Z) _n Substituted pyridin-2-yl, pyridin-3-yl, pyridin-3-yl substituted by (Z) _n , pyridin-4-yl, pyridin-4-yl substituted by (Z) _n , thiophene 2-yl, _(Z) is replaced by _p thiophene-2-yl, thiophen-3-yl, _(Z) thiophene was replaced by _p-3-yl, thiazol-2-yl, (Z replaced by _r thiazol-2-yl, thiazol-4-yl, _(Z) is replaced by _r thiazol-4-yl, thiazol-5-yl, _(Z) thiazol-5-yl which is substituted by _r , Naphthalen-1-yl, naphthalen-1-yl substituted by (Z) _q , naphthalen-2-yl or naphthalen-2-yl substituted by (Z) _q ,
R ² represents a hydrogen atom, a halogen atom, nitro, _cyano, C 1 -C ₆ alkyl, halo _(C 1 ~C ₆₎ ^alkyl, optionally substituted by ^{R b1} _(C 1 ~C ₆₎ alkyl, _{C 3} -C ₆ _cycloalkyl, C 2 -C ₆ _alkenyl, C 2 -C ₆ _alkynyl, C 1 -C ₆ _alkoxy, C 1 -C ₆ _alkylthio, C 1 -C ₆ _{alkylcarbonyl,} C 1 -C ₆ alkoxycarbonyl, Represents phenyl or phenyl substituted by (Y ¹ ) _t1 ;
when t1 represents an integer of 2, 3, 4 or 5, each Y ¹ may be the same as or different from each other;
R ³ is hydrogen atom, halogen atom, nitro, cyano, C ₁ -C ₆ alkyl, C ₃ -C ₆ cycloalkyl, halo (C ₁ -C ₆ ) alkyl, R ^a optionally substituted (C ₁ -C ₆₎ alkyl, halo _(C 3 ~C ₆₎ cycloalkyl, optionally substituted by ^{R b} _(C 3 ~C ₆₎ _cycloalkyl, C 2 -C ₆ alkenyl, halo _{_(C} 2 _~C 6) _alkenyl, C 2 -C ₆ alkynyl, halo _(C 2 ~C ₆₎ _alkynyl, C 1 -C ₆ _alkoxy, C 1 -C ₆ _alkylthio, C 1 -C ₆ _{alkylcarbonyl,} C 1 -C ₆ alkoxycarbonyl, - ^{C (= NOR c) C (} = NOR c1) R d, ^phenyl, (Y ₂₎ phenyl substituted by _t2, pyridin-2-yl, pyridin-3-yl, pyridin-4-yl Represent oxetane-2-yl or tetrahydrofuran-2-yl,
when t2 represents an integer of 2, 3, 4 or 5, each Y ² may be the same as or different from each other;
R ⁴ and R ⁵ each independently represent a hydrogen atom, a halogen atom, C ₁ -C ₆ alkyl, halo (C ₁ -C ₆ ) alkyl, C ₁ -C ₆ alkoxy or C ₁ -C ₆ alkylthio. Or R ⁴ and R ⁵ together form a C _{2 to} C ₅ alkylene chain to form a 3 to 6 membered ring with the carbon atom to which R ⁴ and R ⁵ are bonded. ,
R ⁶ , R ⁷ , R ⁸ and R ⁹ are independently of one another optionally selected from a hydrogen atom, halogen atom, nitro, cyano, C ₁ -C ₆ alkyl, halo (C ₁ -C ₆ ) alkyl, R ^b2 Substituted (C ₁ -C ₆ ) alkyl, C ₃ -C ₆ cycloalkyl, halo (C ₃ -C ₆ ) cycloalkyl, C ₂ -C ₆ alkenyl, halo (C ₂ -C ₆ ) alkenyl, C ₂ -C ₆ alkynyl, halo _(C 2 ~C ₆₎ _alkynyl, C 1 -C ₆ alkoxy, halo _(C 1 ~C ₆₎ _alkoxy, C 1 -C ₆ _alkylthio, C 1 -C ₆ alkylsulfinyl or _C 1 ~ It represents C ₆ alkylsulfonyl,
R ¹⁰ is a hydrogen atom, C ₁ -C ₆ alkyl, halo (C ₁ -C ₆ ) alkyl, (C ₁ -C ₆ ) alkyl, C ₂ -C ₆ alkenyl, or C ₂ optionally substituted with R ^b3 . ~C ₆ alkynyl,
Z is a halogen atom, nitro, cyano, formyl, hydroxy, carboxy, mercapto, _amino, C 1 -C ₆ alkyl, halo _(C 1 ~C ₆₎ ^alkyl, optionally substituted by ^{R b4} _(C 1 ~C ₆₎ _alkyl, C 3 -C ₆ cycloalkyl, halo _(C 3 -C ₆₎ _cycloalkyl, C 2 -C ₆ alkenyl, halo _(C 2 -C ₆₎ _alkenyl, C 1 -C ₆ alkoxy, halo (C ₁ -C ₆₎ ^alkoxy, optionally substituted by ^{R b4} _(C 1 ~C ₆₎ _alkoxy, C 3 -C ₆ _cycloalkoxy, C 2 -C ₆ alkenyloxy, halo _(C 2 ~C ₆₎ alkenyloxy , _C 2 -C ₆ alkynyloxy, halo _(C 2 ~C ₆₎ _alkynyloxy, C 1 -C ₆ _alkylthio, C 2 -C ₆ _{alkenylthio, C} 2 ~ ₆ alkynylthio, halo _(C 1 -C ₆₎ _alkylthio, C 1 -C ₆ _{alkylsulfinyl,} C 2 -C ₆ _{alkenylsulfinyl,} C 2 -C ₆ alkynylsulfinyl, halo _(C 1 -C ₆₎ alkylsulfinyl, C ₁ -C ₆ _{alkylsulfonyl,} C 2 -C ₆ _{alkenylsulfonyl,} C 2 -C ₆ alkynylsulfonyl, halo _(C 1 ~C ₆₎ _{alkylsulfonyl,} C 1 -C ₆ alkylamino, di _{_(C} 1 ~C 6) _alkylamino, C 1 -C ₆ alkylcarbonyl, halo _(C 1 ~C ₆₎ _{alkylcarbonyl,} C 1 -C ₆ _{alkoxycarbonyl,} C 1 -C ₆ alkylaminocarbonyl, di _(C 1 ~C ₆₎ alkylaminocarbonyl , _C 1 -C ₆ alkoxy _(C 1 ~C ₆₎ _alkyl, C 1 -C ₆ alkoxy _(C 1 ~C ₆₎ ^{^{alkoxy, -C (= NOR c) R}} d, -C≡CR e, ^phenyl, phenoxy which is substituted by the (Z ₁₎ phenyl substituted by _m1, phenoxy or ^(Z _{1) m1} Represents
m represents an integer of 2, 3, 4 or 5, n represents an integer of 2, 3 or 4, p represents an integer of 2 or 3, q is 2, 3, 4, 5, 6 Or when R represents an integer of 7, or when r represents an integer of 2, each Z may be the same as or different from each other;
when m1 represents an integer of 2, 3, 4 or 5, each Z ¹ may be the same as or different from each other;
Z ¹ , Z ² , Z ³ , Z ⁴ , Z ⁵ , Y ¹ and Y ² each independently represent a halogen atom, C ₁ -C ₆ alkyl or C ₁ -C ₆ alkoxy,
R ^a is nitro, cyano, hydroxy, C ₃ -C ₆ cycloalkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ alkylsulfonyl, C ₁ -C ₆ alkylcarbonyloxy, phenyl substituted by phenyl or _{(Z) m,}
R ^a1 represents phenyl, phenoxy which is substituted by phenyl which is substituted, phenoxy or _{(Z) m} by _{(Z) m,}
^Rb was substituted by phenyl, phenyl substituted by (Z) _m , pyridin-2-yl, pyridin-2-yl substituted by (Z) _n , pyridin-3-yl, (Z) _n Represents pyridin-4-yl substituted by pyridin-3-yl, pyridin-4-yl or (Z) _n ;
R ^b1 is hydroxy, C ₃ -C ₆ cycloalkyl, halo (C ₁ -C ₆ ) alkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ _{alkylsulfonyl,} C 1 -C ₆ alkylcarbonyloxy, phenyl substituted by phenyl or ^(Z _{2) m @ 2,}
when m2 represents an integer of 2, 3, 4 or 5, each Z ² may be the same as or different from each other;
R ^b2 is hydroxy, C ₃ -C ₆ cycloalkyl, halo (C ₁ -C ₆ ) alkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ alkylsulfonyl, C ₁ -C ₆ alkylcarbonyloxy, phenyl or phenyl substituted by (Z ³ ) _m3
when m3 represents an integer of 2, 3, 4 or 5, each Z ³ may be the same as or different from each other;
R ^b3 is hydroxy, C ₃ -C ₆ cycloalkyl, halo (C ₁ -C ₆ ) alkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ _{alkylsulfonyl,} C 1 -C ₆ alkylcarbonyloxy, phenyl substituted by phenyl or ^(Z _{4) m4,}
when m4 represents an integer of 2, 3, 4 or 5, each Z ⁴ may be the same as or different from each other;
R ^b4 is hydroxy, C ₃ -C ₆ cycloalkyl, halo (C ₁ -C ₆ ) alkyl, C ₁ -C ₆ alkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ alkylsulfonyl, C _1- C ₆ alkylcarbonyloxy, phenyl or phenyl substituted by (Z ⁵ ) _m5
when m5 represents an integer of 2, 3, 4 or 5, each Z ⁵ may be the same as or different from each other;
R ^c , R ^c1 and R ^d each independently represent a hydrogen atom or C ₁ -C ₆ alkyl;
R ^e represents a hydrogen atom, a halogen atom, C ₁ -C ₆ alkyl, C ₃ -C ₆ cycloalkyl or tri (C ₁ -C ₆ ) alkylsilyl;
p represents an integer of 1, 2 or 3,
q represents an integer of 1, 2, 3, 4, 5, 6 or 7,
r represents an integer of 1 or 2,
m, m1, m2, m3, m4, m5, t1 and t2 each independently represent an integer of 1, 2, 3, 4 or 5;
n represents an integer of 1, 2, 3 or 4. ] The acyl hydrazone derivative represented by these, its salt, or those N-oxides.

W represents an oxygen atom,
A represents an oxygen atom,
R ¹ is C ₁ -C ₆ alkyl, (C ₁ -C ₆ ) alkyl optionally substituted by R ^a1 , C ₃ -C ₆ cycloalkyl, optionally substituted by R ^b (C ₂ -C ₆ ) Alkenyl, phenyl, phenyl substituted by (Z) _m , pyridin-2-yl, pyridin-2-yl substituted by (Z) _n , pyridin-3-yl, pyridine substituted by (Z) _n -3-yl, pyridin-4-yl, (Z) _n- substituted pyridin-4-yl, thiophen-2-yl, (Z) _p- substituted thiophen-2-yl, thiophen-3-yl , _(Z) thiophene was replaced by _p-3-yl, thiazol-2-yl, _(Z) is replaced by _r thiazol-2-yl, Chiazo substituted by _{(Z) r} It represents 4-yl, thiazol-5-yl, naphthalene-1-yl or naphthalen-2-yl,
R ² is a hydrogen _atom, C 1 -C ₆ alkyl, halo _(C 1 ~C ₆₎ ^alkyl, optionally substituted by ^{R b1} _(C 1 ~C ₆₎ _alkyl, C 3 -C ₆ cycloalkyl alkyl, C ₁ -C ₆ alkoxy or phenyl,
R ³ represents a hydrogen _atom, C 1 -C ₆ _alkyl, C 3 -C ₆ cycloalkyl, halo _(C 1 ~C ₆₎ alkyl, optionally substituted by R ^a _(C 1 ~C ₆₎ alkyl, halo (C ₃ -C ₆ ) cycloalkyl, C ₂ -C ₆ alkenyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ alkoxycarbonyl, -C (= NOR ^c ) C (= NOR ^{c 1} ) R ^d , phenyl, Represents pyridin-2-yl, pyridin-3-yl or pyridin-4-yl,
R ⁴ and R ⁵ represent a hydrogen atom,
R ⁶ is a hydrogen atom, halogen atom, cyano, C ₁ -C ₆ alkyl, halo (C ₁ -C ₆ ) alkyl, C ₂ -C ₆ alkenyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ alkylthio or C ₁ -C ₆ alkyl sulfinyl,
R ¹⁰ represents C ₁ -C ₆ alkyl,
Z is a halogen atom, nitro, cyano, hydroxy, _carboxy, C 1 -C ₆ alkyl, halo _(C 1 ~C ₆₎ _alkyl, C 3 -C ₆ _cycloalkyl, C 2 -C ₆ _alkenyl, C 1 -C ₆ alkoxy, halo _(C 1 -C ₆₎ ^alkoxy, optionally substituted by ^{R b4} _(C 1 ~C ₆₎ _alkoxy, C 2 -C ₆ _alkenyloxy, C 2 -C ₆ _alkynyloxy, C 1 -C ₆ alkylthio, halo (C ₁ -C ₆ ) alkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ alkylsulfonyl, di (C ₁ -C ₆ ) alkylamino, C ₁ -C ₆ alkylcarbonyl, C ₁ -C ₆ _{alkoxycarbonyl,} C 1 -C ₆ _{alkylaminocarbonyl,} C 1 -C ₆ alkoxy _(C 1 ~C ₆₎ alkoxy, -C (= N Represents ^{^{^{OR c) R d, -C≡CR e}}} , ^phenyl, phenoxy which is substituted by the (Z ₁₎ phenyl or substituted by _{_m1} ^(Z ₁₎ _m1,
R ^a is hydroxy, C ₃ -C ₆ cycloalkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ alkylcarbonyloxy or (Z) _m Represents substituted phenyl,
R ^a1 represents phenyl or phenoxy substituted by (Z) _m ,
R ^b represents phenyl substituted by (Z) _m or pyridin-2-yl substituted by (Z) _n ;
R ^b1 represents C ₁ -C ₆ alkoxy;
R ^b4 represents phenyl,
The acyl hydrazone derivative or a salt thereof or an N-oxide thereof according to claim 1, wherein R ^c , R ^c1 and R ^d each independently represent C _{1 to} C ₆ alkyl.

R ¹ is C ₁ -C ₆ alkyl, (C ₂ -C ₆ ) alkenyl optionally substituted by R ^b , phenyl, phenyl substituted by (Z) _m , pyridine- substituted by (Z) _n 2-yl, represents a thiophene-3-yl substituted by the _(Z) thiophene was replaced by _p-2-yl or _{(Z) p,}
R ² represents C ₁ -C ₆ alkyl or phenyl,
R ³ represents a hydrogen _atom, C 1 -C ₆ _alkyl, C 3 -C ₆ cycloalkyl, halo _(C 1 ~C ₆₎ alkyl, optionally substituted by ^{R a} _(C 1 ~C ₆₎ alkyl, C Represents ₁ -C ₆ alkoxy or C ₁ -C ₆ alkoxycarbonyl,
R ⁶ represents a hydrogen atom, a halogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ alkoxy,
R ⁷ and R ⁸ represent a hydrogen atom,
R ⁹ represents a hydrogen atom or a halogen atom,
Z is optionally substituted with a halogen atom, cyano, C ₁ -C ₆ alkyl, halo (C ₁ -C ₆ ) alkyl, C ₁ -C ₆ alkoxy, halo (C ₁ -C ₆ ) alkoxy, R ^b4 _(C 1 _~C ₆₎ _-alkoxy, C 1 -C ₆ _alkylthio, C 1 -C ₆ _{alkylcarbonyl,} C 1 -C ₆ alkoxycarbonyl, -C a (= ^NOR c) ^{R d} or phenyl,
R ^b represents (Z) phenyl substituted by _m ;
The acyl hydrazone derivative or a salt thereof, or an N-oxide thereof according to claim 2, wherein R ^a represents C ₁ -C ₆ alkoxy, C ₁ -C ₆ alkylthio, or C ₁ -C ₆ alkylcarbonyloxy.

An agrochemical containing one or more selected from the acylhydrazone derivatives or salts thereof according to claims 1 to 3 or N-oxides thereof as active ingredients.

A fungicide containing, as an active ingredient, one or more selected from the acylhydrazone derivatives or salts thereof according to claims 1 to 3 or their N-oxides.

An agricultural and horticultural fungicide containing, as an active ingredient, one or more selected from the acylhydrazone derivatives or salts thereof according to claims 1 to 3 or their N-oxides.

The antifungal agent which contains as an active ingredient 1 type, or 2 or more types chosen from the acyl hydrazone derivative in any one of Claims 1-3, its salt, or those N-oxides.

An endoparasite control agent comprising, as an active ingredient, one or more selected from the acylhydrazone derivative according to any one of claims 1 to 3 or a salt thereof, or an N-oxide thereof.