JP2013530942A5 - - Google Patents

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Publication number
JP2013530942A5
JP2013530942A5 JP2013510192A JP2013510192A JP2013530942A5 JP 2013530942 A5 JP2013530942 A5 JP 2013530942A5 JP 2013510192 A JP2013510192 A JP 2013510192A JP 2013510192 A JP2013510192 A JP 2013510192A JP 2013530942 A5 JP2013530942 A5 JP 2013530942A5
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JP
Japan
Prior art keywords
formula
compound
alkyl
methyl
analog
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Pending
Application number
JP2013510192A
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English (en)
Japanese (ja)
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JP2013530942A (ja
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Priority claimed from PCT/US2011/035654 external-priority patent/WO2011140527A2/en
Publication of JP2013530942A publication Critical patent/JP2013530942A/ja
Publication of JP2013530942A5 publication Critical patent/JP2013530942A5/ja
Pending legal-status Critical Current

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JP2013510192A 2010-05-07 2011-05-06 移行型小胞体ａｔｐアーゼの阻害のための方法および組成物 Pending JP2013530942A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US33266710P 2010-05-07 2010-05-07
US61/332,667 2010-05-07
PCT/US2011/035654 WO2011140527A2 (en) 2010-05-07 2011-05-06 Methods and compositions for inhibition of the transitional endoplasmic reticulum atpase

Publications (2)

Publication Number Publication Date
JP2013530942A JP2013530942A (ja) 2013-08-01
JP2013530942A5 true JP2013530942A5 (enExample) 2014-06-26

Family

ID=44904519

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2013510192A Pending JP2013530942A (ja) 2010-05-07 2011-05-06 移行型小胞体ａｔｐアーゼの阻害のための方法および組成物

Country Status (8)

Country Link
US (1) US8865708B2 (enExample)
EP (1) EP2566480A4 (enExample)
JP (1) JP2013530942A (enExample)
KR (1) KR20130128308A (enExample)
CN (1) CN103068393A (enExample)
AU (1) AU2011249859B2 (enExample)
CA (1) CA2798698A1 (enExample)
WO (1) WO2011140527A2 (enExample)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2011140527A2 (en) 2010-05-07 2011-11-10 California Institute Of Technology And The University Of Kansas Methods and compositions for inhibition of the transitional endoplasmic reticulum atpase
US8906918B1 (en) * 2012-03-23 2014-12-09 University Of South Florida (A Florida Non-Profit Corporation) Compositions, methods of use, and methods of treatment
KR101862912B1 (ko) 2012-07-20 2018-05-30 클리브 바이오사이언스 인코포레이티드 (클리브) p97 복합체의 저해제로서의 축합된 피리미딘
EP2938610A2 (en) * 2012-12-28 2015-11-04 The U.S.A. as represented by the Secretary, Department of Health and Human Services Inhibitors of the usp1/uaf1 deubiquitinase complex and uses thereof
JP6441334B2 (ja) 2013-07-16 2018-12-19 ビーエーエスエフ ソシエタス・ヨーロピアＢａｓｆ Ｓｅ 除草性アジン
DE102013110714A1 (de) * 2013-09-27 2015-04-02 Eberhard Karls Universität Tübingen Medizinische Fakultät Prophylaxe und Behandlung einer nicht auf einer Proteinfaltungsstörung beruhenden neurodegenerativen Erkrankung
ES2739435T3 (es) 2013-10-18 2020-01-31 Univ Indiana Res & Tech Corp Efectores del ensamblaje viral de la hepatitis B
US9868722B2 (en) 2013-12-10 2018-01-16 Cleave Biosciences, Inc. Monocyclic pyrimidine/pyridine compounds as inhibitors of P97 complex
WO2015109285A1 (en) * 2014-01-20 2015-07-23 Cleave Biosciences, Inc. FUSED PYRIMIDINES AS INHIBITORS OF p97 COMPLEX
WO2015155272A1 (en) 2014-04-11 2015-10-15 Basf Se Diaminotriazine derivatives as herbicides
BR112016022782B1 (pt) 2014-04-23 2020-01-28 Basf Se composto de diaminotriazina, composição agroquímica e uso de um composto
US10029992B2 (en) 2014-04-23 2018-07-24 Basf Se Diaminotriazine compounds and their use as herbicides
CN107922377A (zh) 2015-04-17 2018-04-17 美国印第安纳大学研究和技术公司 乙肝病毒组装效应子
CN106518849B (zh) * 2016-10-27 2019-08-16 上海人类基因组研究中心 喹唑啉类化合物及其制备方法和用途
US20230096028A1 (en) * 2019-03-01 2023-03-30 Revolution Medicines, Inc. Bicyclic heterocyclyl compounds and uses thereof
EP4617262A1 (en) * 2022-11-07 2025-09-17 Kyoto University Nitrogen-containing heterocyclic compound

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1992014716A1 (en) * 1991-02-20 1992-09-03 Pfizer Inc. 2,4-diaminoquinazolines derivatives for enhancing antitumor activity
AU2002361846A1 (en) * 2001-12-21 2003-07-15 Bayer Pharmaceuticals Corporation Quinazoline and quinoline derivative compounds as inhibitors of prolylpeptidase, inducers of apoptosis and cancer treatment agents
AU2003255482A1 (en) * 2002-10-02 2004-04-23 Merck Patent Gmbh Use of 4 amino-quinazolines as anti cancer agents
US20060025406A1 (en) * 2004-07-06 2006-02-02 Angion Biomedica Corporation Modulators of hepatocyte growth factor/c- Met activity
WO2006105056A2 (en) * 2005-03-28 2006-10-05 Fmc Corporation Insecticidal 2,4-diaminoquinazolines and related derivatives
WO2007041282A2 (en) * 2005-09-29 2007-04-12 The Johns Hopkins University Methods and compositions for treatment of cystic fibrosis
WO2008157500A1 (en) * 2007-06-17 2008-12-24 Kalypsys, Inc. Aminoquinazoline cannabinoid receptor modulators for treatment of disease
US20100317607A1 (en) * 2007-06-27 2010-12-16 Infectious Disease Research Institute Use of compounds for preparing anti-tuberculosis agents
WO2009011910A2 (en) * 2007-07-18 2009-01-22 Government Of The United States Of America, As Represented By The Secretary, Department Of Health And Human Serices Imidazolidinone compounds, methods to inhibit deubiquitination and methods of treatment
US9089572B2 (en) * 2008-01-17 2015-07-28 California Institute Of Technology Inhibitors of p97
WO2010003908A1 (en) * 2008-07-08 2010-01-14 Jakobsson, Andreas Screening assay for compounds targeting the p97 aaa-atpase complex in the ubiquitin proteasome system.
WO2011140527A2 (en) 2010-05-07 2011-11-10 California Institute Of Technology And The University Of Kansas Methods and compositions for inhibition of the transitional endoplasmic reticulum atpase

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