JP2013505253A - 三環式化合物およびその薬学的使用 - Google Patents
三環式化合物およびその薬学的使用 Download PDFInfo
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| UA121098C2 (uk) | 2013-01-15 | 2020-04-10 | Інсайт Холдинґс Корпорейшн | Тіазолкарбоксаміди і піридинкарбоксаміди, які використовуються як інгібітори рім-кінази |
| WO2015027124A1 (en) | 2013-08-23 | 2015-02-26 | Incyte Corporation | Furo- and thieno-pyridine carboxamide compounds useful as pim kinase inhibitors |
| WO2016010897A1 (en) | 2014-07-14 | 2016-01-21 | Incyte Corporation | Bicyclic heteroaromatic carboxamide compounds useful as pim kinase inhibitors |
| US9580418B2 (en) | 2014-07-14 | 2017-02-28 | Incyte Corporation | Bicyclic aromatic carboxamide compounds useful as Pim kinase inhibitors |
| US9388181B2 (en) | 2014-10-07 | 2016-07-12 | Allergan, Inc. | Substituted 1,2,3,4-tetrahydropyrido[3,4-E] pyrrolo[1,2-A]pyrimidines as kinase |
| WO2016133860A1 (en) * | 2015-02-16 | 2016-08-25 | Board Of Regents Of The University Of Nebraska | Cancer biomarkers and methods of use thereof |
| WO2016196244A1 (en) | 2015-05-29 | 2016-12-08 | Incyte Corporation | Pyridineamine compounds useful as pim kinase inhibitors |
| TWI734699B (zh) | 2015-09-09 | 2021-08-01 | 美商英塞特公司 | Ｐｉｍ激酶抑制劑之鹽 |
| WO2017059251A1 (en) | 2015-10-02 | 2017-04-06 | Incyte Corporation | Heterocyclic compounds useful as pim kinase inhibitors |
| JP7096817B2 (ja) * | 2016-11-04 | 2022-07-06 | オークランド ユニサービシーズ リミティド | 三環式複素環式誘導体及びその使用 |
| EP3666774B1 (en) * | 2017-08-11 | 2022-05-11 | Shengke Pharmaceuticals (Jiangsu) Ltd. | 1h-pyrazolo[4,3-h]quinazoline compound serving as protein kinase inhibitor |
| AR113922A1 (es) | 2017-12-08 | 2020-07-01 | Incyte Corp | Terapia de combinación de dosis baja para el tratamiento de neoplasias mieloproliferativas |
| US11071727B2 (en) | 2018-01-26 | 2021-07-27 | Northwestern University | Therapeutic targeting of proteolytic cleavage of the mixed lineage leukemia gene product (MLL1) by taspase1 using kinase inhibitors |
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2010
- 2010-09-16 CA CA2774148A patent/CA2774148A1/en not_active Abandoned
- 2010-09-16 BR BR112012005957A patent/BR112012005957A2/pt not_active IP Right Cessation
- 2010-09-16 CN CN2010800499560A patent/CN102647906A/zh active Pending
- 2010-09-16 JP JP2012529901A patent/JP2013505253A/ja active Pending
- 2010-09-16 WO PCT/US2010/049116 patent/WO2011035022A1/en not_active Ceased
- 2010-09-16 MX MX2012003316A patent/MX2012003316A/es not_active Application Discontinuation
- 2010-09-16 US US12/883,703 patent/US20110065712A1/en not_active Abandoned
- 2010-09-16 EP EP10817825A patent/EP2477495A1/en not_active Withdrawn
- 2010-09-16 KR KR1020127009466A patent/KR20120103763A/ko not_active Withdrawn
- 2010-09-16 IN IN3213DEN2012 patent/IN2012DN03213A/en unknown
- 2010-09-16 SG SG2012018438A patent/SG179161A1/en unknown
- 2010-09-16 AU AU2010295622A patent/AU2010295622A1/en not_active Abandoned
-
2012
- 2012-03-14 IL IL218632A patent/IL218632A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2011035022A1 (en) | 2011-03-24 |
| US20110065712A1 (en) | 2011-03-17 |
| IN2012DN03213A (cg-RX-API-DMAC7.html) | 2015-10-23 |
| KR20120103763A (ko) | 2012-09-19 |
| IL218632A0 (en) | 2012-05-31 |
| MX2012003316A (es) | 2012-07-23 |
| AU2010295622A1 (en) | 2012-05-10 |
| CN102647906A (zh) | 2012-08-22 |
| BR112012005957A2 (pt) | 2019-09-24 |
| CA2774148A1 (en) | 2011-03-24 |
| SG179161A1 (en) | 2012-04-27 |
| EP2477495A1 (en) | 2012-07-25 |
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