JP2012504603A - 炎症および免疫関連の使用のための化合物 - Google Patents

炎症および免疫関連の使用のための化合物 Download PDF

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JP2012504603A
JP2012504603A JP2011530047A JP2011530047A JP2012504603A JP 2012504603 A JP2012504603 A JP 2012504603A JP 2011530047 A JP2011530047 A JP 2011530047A JP 2011530047 A JP2011530047 A JP 2011530047A JP 2012504603 A JP2012504603 A JP 2012504603A
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compound
disease
cells
immune
compounds
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JP2012504603A5 (OSRAM
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ボーナート，ゲイリー
シャー，ジージェン
チェン，ショウジュン
サン，リージュン
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シンタ ファーマシューティカルズ コーポレーション
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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965—Non-condensed pyrazines
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  • Health & Medical Sciences (AREA)
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  • Life Sciences & Earth Sciences (AREA)
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  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
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  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Engineering & Computer Science (AREA)
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  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Diabetes (AREA)
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  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Endocrinology (AREA)
  • Epidemiology (AREA)
  • Virology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Obesity (AREA)
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  • Psychology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pain & Pain Management (AREA)
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  • Molecular Biology (AREA)
JP2011530047A 2008-10-01 2009-10-01 炎症および免疫関連の使用のための化合物 Pending JP2012504603A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US19482908P 2008-10-01 2008-10-01
US61/194,829 2008-10-01
PCT/US2009/005406 WO2010039236A1 (en) 2008-10-01 2009-10-01 Compounds for inflammation and immune-related uses

Publications (2)

Publication Number Publication Date
JP2012504603A true JP2012504603A (ja) 2012-02-23
JP2012504603A5 JP2012504603A5 (OSRAM) 2012-11-15

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JP2011530047A Pending JP2012504603A (ja) 2008-10-01 2009-10-01 炎症および免疫関連の使用のための化合物

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US (3) US20110118281A9 (OSRAM)
EP (1) EP2350004A1 (OSRAM)
JP (1) JP2012504603A (OSRAM)
AU (1) AU2009300316A1 (OSRAM)
CA (1) CA2739321A1 (OSRAM)
TW (1) TW201018666A (OSRAM)
WO (1) WO2010039236A1 (OSRAM)

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Publication number Priority date Publication date Assignee Title
US8377970B2 (en) 2009-10-08 2013-02-19 Rhizen Pharmaceuticals Sa Modulators of calcium release-activated calcium channel
US8993612B2 (en) 2009-10-08 2015-03-31 Rhizen Pharmaceuticals Sa Modulators of calcium release-activated calcium channel and methods for treatment of non-small cell lung cancer
KR20120130104A (ko) * 2010-02-01 2012-11-28 닛뽕 케미파 가부시키가이샤 Ｇｐｒ119 작동약
WO2012064808A1 (en) * 2010-11-09 2012-05-18 Synta Pharmaceuticals Corp Tetrazolyl - tetrahydropyridine compounds for inflammation and immune - related uses
JP5985611B2 (ja) * 2011-05-03 2016-09-06 シンタ ファーマシューティカルズ コーポレーション 炎症および免疫関連用途のための化合物
CA2868164A1 (en) * 2012-04-13 2013-10-17 Mitsubishi Tanabe Pharma Corporation Amidopyridine derivative and use thereof
CA2940237C (en) 2014-02-21 2023-03-07 Frost Biologic, Inc. Antimitotic amides for the treatment of cancer and proliferative disorders
US20170114060A1 (en) * 2014-06-03 2017-04-27 The Trustees Of The University Of Pennsylvania Novel effective antiviral compounds and methods using same
EP3849552A1 (en) 2018-09-14 2021-07-21 Rhizen Pharmaceuticals AG Compositions comprising a crac inhibitor and a corticosteroid and methods of use thereof
MX2022008627A (es) 2020-01-13 2022-11-08 Verge Analytics Inc Pirazolo-pirimidinas sustituidas y usos de las mismas.

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2007087443A2 (en) * 2006-01-25 2007-08-02 Synta Pharmaceuticals Corp. Vinyl-phenyl derivatives for inflammation and immune-related uses
WO2008063504A2 (en) * 2006-11-13 2008-05-29 Synta Pharmaceuticals Corp. Cyclohexenyl-aryl compounds for inflammation and immune-related uses

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2008282737A1 (en) * 2007-08-01 2009-02-05 Synta Pharmaceuticals Corp. Vinyl-aryl derivatives for inflammation and immune-related uses

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2007087443A2 (en) * 2006-01-25 2007-08-02 Synta Pharmaceuticals Corp. Vinyl-phenyl derivatives for inflammation and immune-related uses
WO2008063504A2 (en) * 2006-11-13 2008-05-29 Synta Pharmaceuticals Corp. Cyclohexenyl-aryl compounds for inflammation and immune-related uses

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EP2350004A1 (en) 2011-08-03
TW201018666A (en) 2010-05-16
US20100125080A1 (en) 2010-05-20
US20130303542A1 (en) 2013-11-14
US20110118281A9 (en) 2011-05-19
AU2009300316A8 (en) 2011-06-16
AU2009300316A1 (en) 2010-04-08
US20120183579A1 (en) 2012-07-19
CA2739321A1 (en) 2010-04-08
WO2010039236A1 (en) 2010-04-08

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