JP2011006431A5 - - Google Patents

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Publication number
JP2011006431A5
JP2011006431A5 JP2010177518A JP2010177518A JP2011006431A5 JP 2011006431 A5 JP2011006431 A5 JP 2011006431A5 JP 2010177518 A JP2010177518 A JP 2010177518A JP 2010177518 A JP2010177518 A JP 2010177518A JP 2011006431 A5 JP2011006431 A5 JP 2011006431A5
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JP
Japan
Prior art keywords
ataxia
adenosine
medicament
prevention
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2010177518A
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English (en)
Japanese (ja)
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JP2011006431A (ja
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Publication date
Application filed filed Critical
Publication of JP2011006431A publication Critical patent/JP2011006431A/ja
Publication of JP2011006431A5 publication Critical patent/JP2011006431A5/ja
Pending legal-status Critical Current

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JP2010177518A 2002-12-19 2010-08-06 アデノシンＡ２ａレセプターアンタゴニストの使用 Pending JP2011006431A (ja)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US43532102P 2002-12-19 2002-12-19

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2005510511A Division JP2006514697A (ja) 2002-12-19 2003-12-17 アデノシンＡ２ａレセプターアンタゴニストの使用

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2013013961A Division JP2013136592A (ja) 2002-12-19 2013-01-29 アデノシンＡ２ａレセプターアンタゴニストの使用

Publications (2)

Publication Number Publication Date
JP2011006431A JP2011006431A (ja) 2011-01-13
JP2011006431A5 true JP2011006431A5 (enExample) 2011-09-15

Family

ID=34572685

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2005510511A Withdrawn JP2006514697A (ja) 2002-12-19 2003-12-17 アデノシンＡ２ａレセプターアンタゴニストの使用
JP2010177518A Pending JP2011006431A (ja) 2002-12-19 2010-08-06 アデノシンＡ２ａレセプターアンタゴニストの使用
JP2013013961A Withdrawn JP2013136592A (ja) 2002-12-19 2013-01-29 アデノシンＡ２ａレセプターアンタゴニストの使用

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2005510511A Withdrawn JP2006514697A (ja) 2002-12-19 2003-12-17 アデノシンＡ２ａレセプターアンタゴニストの使用

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2013013961A Withdrawn JP2013136592A (ja) 2002-12-19 2013-01-29 アデノシンＡ２ａレセプターアンタゴニストの使用

Country Status (15)

Country Link
US (2) US7414058B2 (enExample)
EP (3) EP1578409B1 (enExample)
JP (3) JP2006514697A (enExample)
CN (2) CN101310724A (enExample)
AT (1) ATE490775T1 (enExample)
AU (2) AU2003304527B2 (enExample)
BR (1) BR0317436A (enExample)
DE (1) DE60335294D1 (enExample)
ES (1) ES2354875T3 (enExample)
MX (1) MXPA05006790A (enExample)
NO (1) NO20053509L (enExample)
NZ (1) NZ540493A (enExample)
TW (1) TWI331036B (enExample)
WO (1) WO2005044245A1 (enExample)
ZA (1) ZA200504478B (enExample)

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DE10064453A1 (de) * 2000-12-16 2002-07-04 Schering Ag Verwendung eines dopaminergen Wirkstoffes zur Behandlung von dopaminerg behandelbaren Erkrankungen
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EP1794157B1 (en) 2004-09-22 2014-02-26 H. Lundbeck A/S 2-acylaminothiazole derivatives
US8455437B2 (en) * 2005-02-04 2013-06-04 The United States Of America, As Represented By The Secretary Of The Department Of Health And Human Services Method to predict and prevent oxygen-induced inflammatory tissue injury
US7674912B2 (en) * 2005-04-25 2010-03-09 H. Lundbeck A/S Pro-drugs of N-thiazol-2-yl-benzamide derivatives
ES2385702T3 (es) * 2005-06-07 2012-07-30 Kyowa Hakko Kirin Co., Ltd. Antagonistas de A2A para uso en el tratamiento de trastornos de la motricidad
AR057817A1 (es) 2005-09-19 2007-12-19 Schering Corp Antagonistas del receptor a2a de 2-heteroaril-pirazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pirimidin adenosina. composiciones farmaceuticas
AR056080A1 (es) 2005-09-23 2007-09-19 Schering Corp 7-[2-[4-(6-fluoro-3-metil-1,2-benciosoxazol-5-il)-1-piperazinil]etil]-2-(1-propinil)-7h-pirazol-[4,3-e]-[1,2,4]-triazol-[1,5-c] -pirimidin-5-amine
ES2273599B1 (es) 2005-10-14 2008-06-01 Universidad De Barcelona Compuestos para el tratamiento de la fibrilacion auricular.
JP2011513417A (ja) 2008-03-04 2011-04-28 シェーリング コーポレイション アデノシンＡ２ａ受容体アンタゴニストとして使用するための１，２，４−トリアゾロ［４，３−ｃ］ピリミジン−３−オンおよびピラゾロ［４，３−ｅ］−１，２，４−トリアゾロ［４，３−ｃ］ピリミジン−３−オン化合物
TWI473614B (zh) * 2008-05-29 2015-02-21 Kyowa Hakko Kirin Co Ltd Anti-analgesic inhibitors
JP5765239B2 (ja) 2009-03-13 2015-08-19 アドヴィナス・セラピューティックス・リミテッド 置換縮合ピリミジン化合物
WO2011055391A1 (en) 2009-11-09 2011-05-12 Advinus Therapeutics Private Limited Substituted fused pyrimidine compounds, its preparation and uses thereof
EP2509983B1 (en) 2009-11-16 2014-09-17 Merck Sharp & Dohme Corp. FUSED TRICYCLIC COMPOUNDS WITH ADENOSINE A2a RECEPTOR ANTAGONIST ACTIVITY
US8473582B2 (en) * 2009-12-16 2013-06-25 International Business Machines Corporation Disconnected file operations in a scalable multi-node file system cache for a remote cluster file system
WO2011101861A1 (en) 2010-01-29 2011-08-25 Msn Laboratories Limited Process for preparation of dpp-iv inhibitors
KR101838093B1 (ko) 2010-02-05 2018-03-13 헵테얼즈 테라퓨틱스 리미티드 1,2,4-트리아진-4-아민 유도체들
JP5843869B2 (ja) * 2010-09-24 2016-01-13 アドヴィナス・セラピューティックス・リミテッド アデノシン受容体拮抗薬としての縮合三環化合物
WO2012066330A1 (en) 2010-11-17 2012-05-24 Heptares Therapeutics Limited Compounds useful as a2a receptor inhibitors
WO2012135084A1 (en) * 2011-03-31 2012-10-04 Merck Sharp & Dohme Corp. METABOLITES OF 2-(FURAN-2-YL)-7-(2-(4-(4-(2-METHOXYETHOXY)PHENYL)PIPERAZIN-1-YL)ETHYL)-7H-PYRAZOLO[4,3-e][1,2,4]TRIAZOLO[1,5-c]PYRIMIDIN-5-AMINE AND THEIR UTILITY AS ADENOSINE A2a RECEPTOR ANTAGONISTS
WO2014101113A1 (en) 2012-12-28 2014-07-03 Merck Sharp & Dohme Corp. Piperazine-substituted 7-methoxy-[1,2,4]triazolo[1,5-c]quinazolin-5-amine compounds with a2a antagonist properties
CN105025899B (zh) * 2012-12-28 2017-08-18 默沙东公司 具有A2A拮抗剂性质的杂二环取代的‑[1,2,4]三唑并[1,5‑c]喹唑啉‑5‑胺化合物
WO2014101120A1 (en) 2012-12-28 2014-07-03 Merck Sharp & Dohme Corp. Heterobicyclo-substituted-7-methoxy-[1,2,4]triazolo[1,5-c]quinazolin-5-amine compounds with a2a antagonist properties
US11246871B2 (en) 2016-07-15 2022-02-15 Northwestern University Targeting adenosine A2A receptors for the treatment of levodopa-induced dyskinesias
CA3067765A1 (en) * 2017-06-30 2019-01-03 Bobowska (Nee Witkowska), Aneta Imidazo[1,2-a]pyrazine modulators of the adenosine a2a receptor
JP7391022B2 (ja) 2017-12-19 2023-12-04 インペティス・バイオサイエンシーズ・リミテッド がんの処置のための医薬組成物
ES2928238T3 (es) 2018-01-04 2022-11-16 Impetis Biosciences Ltd Compuestos tricíclicos, composiciones y aplicaciones medicinales de los mismos
DE102019116986A1 (de) 2019-06-24 2020-12-24 Helmholtz-Zentrum Dresden-Rossendorf E. V. Deuterierte 7-(3-(4-(2-([18F]Fluor)ethoxy)phenyl)propyl)-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amin-Derivate
CN114667287A (zh) * 2019-07-17 2022-06-24 泰昂治疗公司 腺苷a2a受体拮抗剂及其用途
US11806350B2 (en) * 2020-11-19 2023-11-07 Ildong Pharmaceutical Co., Ltd. Prevention and/or treatment of CNS disorders

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MXPA04002389A (es) * 2001-09-13 2004-05-31 Schering Corp Combinacion de un antagonista del receptor de adenosian a2a y un antidepresivo o ansiolitico.
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MXPA04007299A (es) * 2002-01-28 2004-10-29 Kyowa Hakko Kogyo Kk Metodos de tratamiento de pacientes que sufren de trastornos de movimiento.
WO2004019949A1 (en) * 2002-08-30 2004-03-11 Kyowa Hakko Kogyo Co. Ltd. Adenosine a2a receptor antagonists for treating restless legs syndrome or related disorders
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