JP2010535218A5 - - Google Patents

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Publication number
JP2010535218A5
JP2010535218A5 JP2010519949A JP2010519949A JP2010535218A5 JP 2010535218 A5 JP2010535218 A5 JP 2010535218A5 JP 2010519949 A JP2010519949 A JP 2010519949A JP 2010519949 A JP2010519949 A JP 2010519949A JP 2010535218 A5 JP2010535218 A5 JP 2010535218A5
Authority
JP
Japan
Prior art keywords
optionally substituted
compound according
compound
halo
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2010519949A
Other languages
English (en)
Japanese (ja)
Other versions
JP2010535218A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2008/009346 external-priority patent/WO2009017831A1/en
Publication of JP2010535218A publication Critical patent/JP2010535218A/ja
Publication of JP2010535218A5 publication Critical patent/JP2010535218A5/ja
Pending legal-status Critical Current

Links

JP2010519949A 2007-08-01 2008-07-31 炎症および免疫関連用途のためのビニル−アリール誘導体 Pending JP2010535218A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US96282307P 2007-08-01 2007-08-01
PCT/US2008/009346 WO2009017831A1 (en) 2007-08-01 2008-07-31 Vinyl-aryl derivatives for inflammation and immune-related uses

Publications (2)

Publication Number Publication Date
JP2010535218A JP2010535218A (ja) 2010-11-18
JP2010535218A5 true JP2010535218A5 (cg-RX-API-DMAC7.html) 2012-11-08

Family

ID=40304694

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010519949A Pending JP2010535218A (ja) 2007-08-01 2008-07-31 炎症および免疫関連用途のためのビニル−アリール誘導体

Country Status (7)

Country Link
US (2) US8349841B2 (cg-RX-API-DMAC7.html)
EP (1) EP2185514A4 (cg-RX-API-DMAC7.html)
JP (1) JP2010535218A (cg-RX-API-DMAC7.html)
AU (1) AU2008282737A1 (cg-RX-API-DMAC7.html)
CA (1) CA2695156A1 (cg-RX-API-DMAC7.html)
TW (1) TW200914440A (cg-RX-API-DMAC7.html)
WO (1) WO2009017831A1 (cg-RX-API-DMAC7.html)

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CA2595000C (en) 2005-01-25 2013-10-15 Synta Pharmaceuticals Corp. Thiophene compounds for inflammation and immune-related uses
AU2007208239B2 (en) 2006-01-25 2013-04-18 Synta Pharmaceuticals Corp. Substituted aromatic compounds for inflammation and immune-related uses
AU2007208151B2 (en) 2006-01-25 2013-04-18 Synta Pharmaceuticals Corp. Vinyl-phenyl derivatives for inflammation and immune-related uses
EP1998612A4 (en) 2006-01-25 2010-11-24 Synta Pharmaceuticals Corp SUBSTITUTED BIARYL COMPOUNDS FOR USE AGAINST INFLAMMATION AND IMMUNE DISORDERS
US8119643B2 (en) 2006-03-20 2012-02-21 Synta Pharmaceuticals Corp. Benzoimidazolyl-pyrazine compounds for inflammation and immune-related uses
US8779154B2 (en) 2006-09-26 2014-07-15 Qinglin Che Fused ring compounds for inflammation and immune-related uses
JP2010535218A (ja) * 2007-08-01 2010-11-18 シンタ ファーマシューティカルズ コーポレーション 炎症および免疫関連用途のためのビニル−アリール誘導体
JP2012504603A (ja) * 2008-10-01 2012-02-23 シンタ ファーマシューティカルズ コーポレーション 炎症および免疫関連の使用のための化合物
US8993612B2 (en) 2009-10-08 2015-03-31 Rhizen Pharmaceuticals Sa Modulators of calcium release-activated calcium channel and methods for treatment of non-small cell lung cancer
US8377970B2 (en) 2009-10-08 2013-02-19 Rhizen Pharmaceuticals Sa Modulators of calcium release-activated calcium channel
JPWO2011093501A1 (ja) * 2010-02-01 2013-06-06 日本ケミファ株式会社 Gpr119作動薬
WO2011139765A2 (en) 2010-04-27 2011-11-10 Calcimedica, Inc. Compounds that modulate intracellular calcium
WO2011139489A2 (en) 2010-04-27 2011-11-10 Calcimedica Inc. Compounds that modulate intracellular calcium
US10703722B2 (en) 2010-04-27 2020-07-07 Calcimedica, Inc. Compounds that modulate intracellular calcium
CA2809830C (en) 2010-08-27 2019-09-10 Calcimedica, Inc. Compounds comprising n-acyl-2-amino-1,3-thiazole for modulating intracellular calcium
EP2638032A1 (en) * 2010-11-09 2013-09-18 Synta Pharmaceuticals Corp. Tetrazolyl - tetrahydropyridine compounds for inflammation and immune - related uses
US20120316182A1 (en) 2011-06-10 2012-12-13 Calcimedica, Inc. Compounds that modulate intracellular calcium
US9856240B2 (en) 2011-10-19 2018-01-02 Calcimedica, Inc. Compounds that modulate intracellular calcium
US9512116B2 (en) 2012-10-12 2016-12-06 Calcimedica, Inc. Compounds that modulate intracellular calcium
TWI835179B (zh) 2015-02-27 2024-03-11 美商鈣系醫藥公司 胰腺炎治療
WO2017027400A1 (en) 2015-08-07 2017-02-16 Calcimedica, Inc. Use of crac channel inhibitors for the treatment of stroke and traumatic brain injury
EP3849552A1 (en) 2018-09-14 2021-07-21 Rhizen Pharmaceuticals AG Compositions comprising a crac inhibitor and a corticosteroid and methods of use thereof
EP4090426B1 (en) 2020-01-13 2025-12-31 Verge Analytics, Inc. Substitutes for pyrazolos and pyrimidines and their uses

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US8518950B2 (en) 2005-01-25 2013-08-27 Synta Pharmaceuticals Corp. 2-amido pyrazines for inflammation and immune related uses
AU2007208151B2 (en) * 2006-01-25 2013-04-18 Synta Pharmaceuticals Corp. Vinyl-phenyl derivatives for inflammation and immune-related uses
EP2086326B1 (en) * 2006-11-13 2014-01-08 Synta Pharmaceuticals Corp. Cyclohexenyl-aryl compounds for inflammation and immune-related uses
JO2972B1 (en) * 2007-06-08 2016-03-15 جانسين فارماسوتيكا ان. في Piperidine / piperazine derivatives
JP2010535218A (ja) * 2007-08-01 2010-11-18 シンタ ファーマシューティカルズ コーポレーション 炎症および免疫関連用途のためのビニル−アリール誘導体

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