JP2010509205A - Ｐｏｓｈ及びｐｏｓｈ−ａｐ阻害剤としてのピリミジン誘導体 - Google Patents
Ｐｏｓｈ及びｐｏｓｈ−ａｐ阻害剤としてのピリミジン誘導体 Download PDFInfo
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- JP2010509205A JP2010509205A JP2009535189A JP2009535189A JP2010509205A JP 2010509205 A JP2010509205 A JP 2010509205A JP 2009535189 A JP2009535189 A JP 2009535189A JP 2009535189 A JP2009535189 A JP 2009535189A JP 2010509205 A JP2010509205 A JP 2010509205A
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| US85737806P | 2006-11-07 | 2006-11-07 | |
| US95983107P | 2007-07-17 | 2007-07-17 | |
| PCT/IL2007/001356 WO2008056356A2 (en) | 2006-11-07 | 2007-11-07 | Pyrimidine derivatives as posh and posh-ap inhibitors |
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| JP2010509205A true JP2010509205A (ja) | 2010-03-25 |
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| EP2509601A4 (en) * | 2009-11-30 | 2013-05-29 | Proteologics Ltd | SMALL PYRIMIDINE DERIVATIVES AND METHOD OF USE THEREOF |
| WO2013088445A1 (en) * | 2011-12-13 | 2013-06-20 | Proteologics Ltd | Pyrimidine derivatives for treatment of inflammatory diseases |
| GB201415688D0 (en) * | 2014-09-04 | 2014-10-22 | Univ Edinburgh | Method and Systems |
| CN108025034B (zh) * | 2015-07-15 | 2022-09-30 | 新加坡科技研究局 | 乙型肝炎病毒复制的调控 |
| WO2018085208A1 (en) | 2016-11-02 | 2018-05-11 | The Research Foundation For The State University Of New York | Methods of inhibiting viruses using compositions targeting tsg101-ubiquitin interaction |
| AU2019297402B2 (en) * | 2018-07-05 | 2024-05-02 | Bayer Aktiengesellschaft | Substituted thiophenecarboxamides and analogues as antibacterials agents |
| KR102459858B1 (ko) * | 2019-04-02 | 2022-10-27 | 연세대학교 산학협력단 | 신규 화합물 및 이를 유효성분으로 포함하는 호흡기 질환의 예방 또는 치료용 조성물 |
| CN110760597B (zh) * | 2019-11-22 | 2022-08-23 | 西北农林科技大学 | 一种检测黄牛ncstn基因拷贝数变异的方法及其应用 |
| TW202527955A (zh) * | 2023-11-27 | 2025-07-16 | 美商尼坎醫療公司 | 用於經由泛素蛋白酶體途徑降解週期蛋白依賴性激酶２和週期蛋白依賴性激酶４的含有２，５－取代的嘧啶衍生物的雙功能化合物 |
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| WO2005013914A2 (en) * | 2003-08-08 | 2005-02-17 | Vertex Pharmaceuticals Incorporated | Heteroarylaminosulfonylphenyl derivatives for use as sodium or calcium channel blockers in the treatment of pain |
| US20060014807A1 (en) * | 2004-07-19 | 2006-01-19 | Lin Leu-Fen H | Neuroprotective small organic molecules, compositions and uses related thereto |
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| US5734081A (en) | 1994-08-05 | 1998-03-31 | Warner-Lambert Company | Arylthio compounds |
| EP1341817A2 (en) | 2000-12-08 | 2003-09-10 | Novo Nordisk A/S | Tff peptides |
| FI116940B (fi) * | 2001-07-20 | 2006-04-13 | Juvantia Pharma Ltd Oy | Alfa-2B-adrenoseptorivälitteisen sairauden hoitoon tai ehkäisyyn käyttökelpoiset yhdisteet |
| EP1422228A1 (en) * | 2001-08-08 | 2004-05-26 | Takeda Chemical Industries, Ltd. | BENZAZEPINE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE |
| FR2845382A1 (fr) * | 2002-10-02 | 2004-04-09 | Sanofi Synthelabo | Derives d'indazolecarboxamides, leur preparation et leur utilisation en therapeutique |
| US20050214751A1 (en) * | 2004-03-02 | 2005-09-29 | Proteologics, Inc. | Inhibition of viral maturation, methods and compositions related thereto |
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Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2005013914A2 (en) * | 2003-08-08 | 2005-02-17 | Vertex Pharmaceuticals Incorporated | Heteroarylaminosulfonylphenyl derivatives for use as sodium or calcium channel blockers in the treatment of pain |
| US20060014807A1 (en) * | 2004-07-19 | 2006-01-19 | Lin Leu-Fen H | Neuroprotective small organic molecules, compositions and uses related thereto |
Non-Patent Citations (4)
| Title |
|---|
| JPN6013000717; 'Ｓｙｎｔｈｅｓｉｓ ｏｆ ｓｏｍｅ ｎｅｗ ｈｅｔｅｒｏｂｉｃｙｃｌｉｃ ｃｏｍｐｏｕｎｄ ｂｅａｒｉｎｇ ｃｈｒｏｍｏｎ-３-ｙｌ ｍｏｉｅｔｙ ａｎｄ ｒｅｌａｔｅｄ ｃｏｍｐｏｕｎｄａ ａｓ ａ' Ｃｈｅｍｉｃａｌ ａｂｓｔｒａｃｔｓ Ｖｏｌ．１２７, 1997, ３４１７０ｈ，３４１７１ａ * |
| JPN6013000719; Ｒｅｇｉｓｔｒｙ Ｎｏ．３２６０２６-７５-９，Ｒｅｇｉｓｔｒｙ ［ｏｎｌｉｎｅ］； Ｒｅｔｒｉｅｖｅｄ ｆｒｏｍ ＳＴＮ , 20010307 * |
| JPN6013000721; Ｊｏｕｒｎａｌ ｏｆ Ｃｏｍｂｉｎａｔｏｒｉａｌ Ｃｈｅｍｉｓｔｒｙ Ｖｏｌ．８， Ｎｏ．３, 2006, ｐ．３２６-３３７ * |
| JPN6013000723; Ｓｕｌｆｕｒ Ｌｅｔｔｅｒｓ Ｖｏｌ．２４， Ｎｏ．４, 2001, ｐ．１５１-１７９ * |
Also Published As
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| EP2083826A2 (en) | 2009-08-05 |
| US20130131094A1 (en) | 2013-05-23 |
| AU2007318922C1 (en) | 2013-09-12 |
| WO2008056356A2 (en) | 2008-05-15 |
| WO2008056356A3 (en) | 2009-09-03 |
| EP2083826A4 (en) | 2010-09-22 |
| AU2007318922A1 (en) | 2008-05-15 |
| US20100179178A1 (en) | 2010-07-15 |
| CA2668859A1 (en) | 2008-05-15 |
| AU2007318922B2 (en) | 2013-01-10 |
| US8283355B2 (en) | 2012-10-09 |
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