JP2010505386A - Ｃｄｋｉ経路阻害剤の同定 - Google Patents
Ｃｄｋｉ経路阻害剤の同定 Download PDFInfo
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- JP2010505386A JP2010505386A JP2009511025A JP2009511025A JP2010505386A JP 2010505386 A JP2010505386 A JP 2010505386A JP 2009511025 A JP2009511025 A JP 2009511025A JP 2009511025 A JP2009511025 A JP 2009511025A JP 2010505386 A JP2010505386 A JP 2010505386A
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Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2015506376A (ja) * | 2012-02-02 | 2015-03-02 | セネックス バイオテクノロジー インク．Ｓｅｎｅｘ Ｂｉｏｔｅｃｈｎｏｌｏｇｙ Ｉｎｃ． | Ｃｄｋ８／ｃｄｋ１９選択的阻害剤、ならびに癌のための抗転移および化学防御の方法におけるそれらの使用 |
| JP2019206549A (ja) * | 2014-12-15 | 2019-12-05 | ザ リージェンツ オブ ザ ユニバーシティ オブ ミシガン | Ｅｇｆｒ及びｐｉ３ｋの小分子阻害剤 |
| JP2022544700A (ja) * | 2019-08-22 | 2022-10-20 | バイオヘイブン・セラピューティクス・リミテッド | 筋萎縮性側索硬化症および関連障害の治療のためにｔｄｐ－４３に結合する分子 |
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| US20050171172A1 (en) | 2003-11-13 | 2005-08-04 | Ambit Biosciences Corporation | Amide derivatives as PDGFR modulators |
| US7829574B2 (en) * | 2008-05-09 | 2010-11-09 | Hutchison Medipharma Enterprises Limited | Substituted quinazoline compounds and their use in treating angiogenesis-related diseases |
| KR101696936B1 (ko) * | 2008-07-10 | 2017-01-16 | 잇반샤단호우징 화루마바레프로제쿠토 시엥기코우 | 퀴놀린카르복사미드 유도체를 유효 성분으로 하는 ｓｔａｔ３ 저해제 |
| US20100190807A1 (en) * | 2008-08-26 | 2010-07-29 | Senex Biotechnology, Inc. | CDKI Pathway inhibitors and uses thereof to regulate expression to TAU protein |
| AR079814A1 (es) | 2009-12-31 | 2012-02-22 | Otsuka Pharma Co Ltd | Compuestos heterociclicos, composiciones farmaceuticas que los contienen y sus usos |
| KR20140048216A (ko) | 2011-06-29 | 2014-04-23 | 오츠카 세이야쿠 가부시키가이샤 | 치료 화합물로서의 퀴나졸린 및 관련된 사용 방법 |
| WO2018226230A1 (en) * | 2017-06-08 | 2018-12-13 | The Children's Medical Center Corporation | Compounds and methods for treatment of diamond blackfan anemia |
| RU2763347C2 (ru) * | 2018-03-01 | 2021-12-28 | Закрытое Акционерное Общество "Биокад" | Новые ингибиторы cdk8/19 |
| WO2025024311A2 (en) * | 2023-07-21 | 2025-01-30 | Icahn School Of Medicine At Mount Sinai | G9a/glp inhibitors and methods of use |
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| US5480883A (en) * | 1991-05-10 | 1996-01-02 | Rhone-Poulenc Rorer Pharmaceuticals Inc. | Bis mono- and bicyclic aryl and heteroaryl compounds which inhibit EGF and/or PDGF receptor tyrosine kinase |
| GB9603095D0 (en) * | 1996-02-14 | 1996-04-10 | Zeneca Ltd | Quinazoline derivatives |
| GB9922173D0 (en) * | 1999-09-21 | 1999-11-17 | Zeneca Ltd | Chemical compounds |
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| WO2004065392A1 (en) * | 2003-01-24 | 2004-08-05 | Smithkline Beecham Corporation | Condensed pyridines and pyrimidines and their use as alk-5 receptor ligands |
| EP1720841B1 (en) * | 2004-02-19 | 2015-11-04 | Rexahn Pharmaceuticals, Inc. | Quinazoline derivatives and therapeutic use thereof |
| AU2005238270A1 (en) * | 2004-04-28 | 2005-11-10 | Arrow Therapeutics Limited | Morpholinylanilinoquinazo- line derivatives for use as antiviral agents |
| EP1838879A4 (en) * | 2005-01-13 | 2009-09-23 | Senex Biotechnology Inc | HIGH-QUALITY SCREENING FOR CLEANING AGAINST CANCER AND AGED DISEASES |
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- 2007-05-15 WO PCT/US2007/011623 patent/WO2007133773A2/en not_active Ceased
- 2007-05-15 AU AU2007249762A patent/AU2007249762A1/en not_active Abandoned
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2015506376A (ja) * | 2012-02-02 | 2015-03-02 | セネックス バイオテクノロジー インク．Ｓｅｎｅｘ Ｂｉｏｔｅｃｈｎｏｌｏｇｙ Ｉｎｃ． | Ｃｄｋ８／ｃｄｋ１９選択的阻害剤、ならびに癌のための抗転移および化学防御の方法におけるそれらの使用 |
| JP2019206549A (ja) * | 2014-12-15 | 2019-12-05 | ザ リージェンツ オブ ザ ユニバーシティ オブ ミシガン | Ｅｇｆｒ及びｐｉ３ｋの小分子阻害剤 |
| JP2022544700A (ja) * | 2019-08-22 | 2022-10-20 | バイオヘイブン・セラピューティクス・リミテッド | 筋萎縮性側索硬化症および関連障害の治療のためにｔｄｐ－４３に結合する分子 |
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| CA2652341A1 (en) | 2007-11-22 |
| EP2021019A2 (en) | 2009-02-11 |
| US20080033000A1 (en) | 2008-02-07 |
| EP2021019A4 (en) | 2009-12-09 |
| WO2007133773A3 (en) | 2009-01-22 |
| WO2007133773A2 (en) | 2007-11-22 |
| AU2007249762A1 (en) | 2007-11-22 |
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