JP2010504995A5 - - Google Patents
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- Publication number
- JP2010504995A5 JP2010504995A5 JP2009530554A JP2009530554A JP2010504995A5 JP 2010504995 A5 JP2010504995 A5 JP 2010504995A5 JP 2009530554 A JP2009530554 A JP 2009530554A JP 2009530554 A JP2009530554 A JP 2009530554A JP 2010504995 A5 JP2010504995 A5 JP 2010504995A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- effective amount
- hydrogen
- formula
- pharmaceutical composition
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
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- 0 *1C(CC2)C3C2C13 Chemical compound *1C(CC2)C3C2C13 0.000 description 3
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US84880306P | 2006-09-28 | 2006-09-28 | |
| PCT/US2007/079384 WO2008039754A1 (en) | 2006-09-28 | 2007-09-25 | 2-methylene-(20r,25s)-19,27-dinor-(22e)-vitamin d analogs |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2010504995A JP2010504995A (ja) | 2010-02-18 |
| JP2010504995A5 true JP2010504995A5 (https=) | 2010-10-21 |
Family
ID=38860081
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009530554A Pending JP2010504995A (ja) | 2006-09-28 | 2007-09-25 | ２−メチレン−（２０ｒ，２５ｓ）−１９，２７−ジノル−（２２ｅ）−ビタミンｄ類縁体 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US7741314B2 (https=) |
| EP (1) | EP2069297A1 (https=) |
| JP (1) | JP2010504995A (https=) |
| AU (1) | AU2007300214A1 (https=) |
| CA (1) | CA2662992A1 (https=) |
| MX (1) | MX2009003241A (https=) |
| NZ (1) | NZ575111A (https=) |
| WO (1) | WO2008039754A1 (https=) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8193170B2 (en) * | 2008-07-10 | 2012-06-05 | Wisconsin Alumni Research Foundation | 2-methylene-19,26-dinor-(20R,22E,25R)-vitamin D analogs |
| US8399439B2 (en) * | 2008-07-10 | 2013-03-19 | Wisconsin Alumni Research Foundation | 2-methylene-19,26-dinor-(20S,22E,25R)-vitamin D analogs |
| EP2525799B1 (en) * | 2009-10-02 | 2014-09-03 | Wisconsin Alumni Research Foundation | (20s,22e)-2-methylene-19-nor-22-ene-1alpha,25-dihydroxyvitamin d3 analogs |
| US8664206B2 (en) | 2010-03-23 | 2014-03-04 | Wisconsin Alumni Research Foundation | Diastereomers of 2-methylene-19-nor-22-methyl-1α,25-dihydroxyvitamin D3 |
| AU2011232633B2 (en) * | 2010-03-23 | 2014-05-29 | Wisconsin Alumni Research Foundation | (20S)-2-methylene-19-nor-22-dimethyl-1alpha,25- dihydroxyvitamin D3 and (20R)-2-methylene-19-nor-22- dimethyl-1alpha,25-hydroxyvitamin D3 |
| JP5931845B2 (ja) * | 2010-03-23 | 2016-06-08 | ウイスコンシン アラムニ リサーチ ファンデーション | ２−メチレン−１９−ノル−２２−メチル−１α，２５−ジヒドロキシビタミンＤ３のジアステレオマー |
| JP6035331B2 (ja) * | 2011-06-14 | 2016-11-30 | ウイスコンシン アラムニ リサーチ ファンデーション | ３−デスオキシ−２−メチレン−１９−ノル−ビタミンｄ類似体およびそれらの使用 |
| US8410080B1 (en) * | 2011-10-21 | 2013-04-02 | Wisconsin Alumni Research Foundation | 2-methylene-vitamin D analogs and their uses |
Family Cites Families (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4486333A (en) * | 1981-04-10 | 1984-12-04 | Felix Sebba | Preparation of biliquid foam compositions |
| US4666634A (en) * | 1984-12-05 | 1987-05-19 | Chugai Seiyaku Kabushiki Kaisha | vitamin D3 derivatives having a substituent at 2-position |
| US5086191A (en) * | 1991-05-28 | 1992-02-04 | Wisconsin Alumni Research Foundation | Intermediates for the synthesis of 19-nor vitamin D compounds |
| DE69400495T2 (de) * | 1993-04-05 | 1997-04-30 | Wisconsin Alumni Res Found | 19-Nor-vitamin-D3-Verbindung mit einem Substituent an die 2. Stelle |
| US5945410A (en) * | 1997-03-17 | 1999-08-31 | Wisconsin Alumni Research Foundation | 2-alkyl-19-nor-vitamin D compounds |
| US5843928A (en) * | 1997-03-17 | 1998-12-01 | Wisconsin Alumni Research Foundation | 2-alkylidene-19-nor-vitamin D compounds |
| PT3146969T (pt) * | 1999-04-23 | 2018-10-18 | Leo Pharma As | Composição farmacêutica para aplicação dérmica para uso no tratamento da psoríase compreendendo vitamina d e um corticosteroide |
| US6806262B2 (en) * | 2000-05-31 | 2004-10-19 | Wisconsin Alumni Research Foundation | 2-ethyl and 2-ethylidene-19-nor-vitamin D compounds |
| KR20020033182A (ko) | 2000-07-21 | 2002-05-04 | 요트.게.아. 롤페즈 | 이용자 프로필을 결정하는 방법 및 시스템 |
| WO2002020021A1 (en) * | 2000-09-08 | 2002-03-14 | Wisconsin Alumni Research Foundation | 1alpha-hydroxy-2-methylene-19-nor-homopregnacalciferol and its therapeutic applications |
| US6627622B2 (en) * | 2002-02-18 | 2003-09-30 | Wisconsin Alumni Research Foundation | (20S)-1α-hydroxy-2-methylene-19-nor-bishomopregnacalciferol and its uses |
| US6566352B1 (en) * | 2002-02-18 | 2003-05-20 | Wisconsin Alumni Research Foudation | 1 α-hydroxy-2-methylene-19-nor-pregnacalciferol and its uses |
| GB0305332D0 (en) | 2003-03-10 | 2003-04-09 | Leuven K U Res & Dev | Biological evaluation of novel vitamin D analogues |
| US20050009792A1 (en) | 2003-07-08 | 2005-01-13 | Deluca Hector F. | (20S)-1alpha-hydroxy-2-methylene-19-nor-vitamin D3 and its uses |
| CA2544502A1 (en) | 2003-11-25 | 2005-06-09 | Wisconsin Alumni Research Foundation | Vitamin d analogs for obesity prevention and treatment |
| JP2008520689A (ja) * | 2004-11-22 | 2008-06-19 | ウィスコンシン・アルムニ・リサーチ・ファウンデーション | １９，２６，２７−トリノル−（２０Ｓ）−１α−ヒドロキシビタミンＤ３の２α−メチルおよび２β−メチル類似体およびそれらの使用 |
| AU2006213727B2 (en) * | 2005-02-11 | 2011-08-18 | Wisconsin Alumni Research Foundation | 2-methylene-19-nor- (20S-24S) - 1alpha, 25-dihydroxyvitamin-D2 |
| US7528122B2 (en) | 2006-02-02 | 2009-05-05 | Wisconsin Alumni Research Foundation | Vitamin D analog—NEL, methods and uses thereof |
| CA2646909A1 (en) * | 2006-04-06 | 2008-03-27 | Hector F. Deluca | 2-methylene-1alpha-hydroxy-19,21-dinorvitamin d3 analogs and uses thereof |
-
2007
- 2007-09-25 MX MX2009003241A patent/MX2009003241A/es active IP Right Grant
- 2007-09-25 US US11/860,870 patent/US7741314B2/en not_active Expired - Fee Related
- 2007-09-25 EP EP07843120A patent/EP2069297A1/en not_active Withdrawn
- 2007-09-25 AU AU2007300214A patent/AU2007300214A1/en not_active Abandoned
- 2007-09-25 NZ NZ575111A patent/NZ575111A/en not_active IP Right Cessation
- 2007-09-25 CA CA002662992A patent/CA2662992A1/en not_active Abandoned
- 2007-09-25 JP JP2009530554A patent/JP2010504995A/ja active Pending
- 2007-09-25 WO PCT/US2007/079384 patent/WO2008039754A1/en not_active Ceased
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