JP2009539838A - マクロファージ転位阻害因子阻害剤としてのオキシム誘導体 - Google Patents

マクロファージ転位阻害因子阻害剤としてのオキシム誘導体 Download PDF

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JP2009539838A
JP2009539838A JP2009514326A JP2009514326A JP2009539838A JP 2009539838 A JP2009539838 A JP 2009539838A JP 2009514326 A JP2009514326 A JP 2009514326A JP 2009514326 A JP2009514326 A JP 2009514326A JP 2009539838 A JP2009539838 A JP 2009539838A
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compound
branched
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mammal
halogen
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JP2009539838A5 (enExample
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オール−アベド、ユウセフ
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Feinstein Institutes for Medical Research
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    • C07C291/02—Compounds containing carbon and nitrogen and having functional groups not covered by groups C07C201/00 - C07C281/00 containing nitrogen-oxide bonds
    • C07C291/04—Compounds containing carbon and nitrogen and having functional groups not covered by groups C07C201/00 - C07C281/00 containing nitrogen-oxide bonds containing amino-oxide bonds
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    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14—The ring being saturated

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Molecular Biology (AREA)
  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Cardiology (AREA)
  • Neurology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Neurosurgery (AREA)
  • Diabetes (AREA)
  • Biomedical Technology (AREA)
  • Toxicology (AREA)
  • Biotechnology (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Psychiatry (AREA)
JP2009514326A 2006-06-05 2007-06-04 マクロファージ転位阻害因子阻害剤としてのオキシム誘導体 Pending JP2009539838A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US81125806P 2006-06-05 2006-06-05
PCT/US2007/013139 WO2007145888A2 (en) 2006-06-05 2007-06-04 Oxime derivatives as inhibitors of macrophage migration inhibitory factor

Publications (2)

Publication Number Publication Date
JP2009539838A true JP2009539838A (ja) 2009-11-19
JP2009539838A5 JP2009539838A5 (enExample) 2013-04-18

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ID=38832310

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JP2009514326A Pending JP2009539838A (ja) 2006-06-05 2007-06-04 マクロファージ転位阻害因子阻害剤としてのオキシム誘導体

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Country Link
US (1) US20090318509A1 (enExample)
EP (1) EP2023732A4 (enExample)
JP (1) JP2009539838A (enExample)
AU (1) AU2007258731B2 (enExample)
CA (1) CA2653646A1 (enExample)
WO (1) WO2007145888A2 (enExample)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8362053B2 (en) * 2006-03-24 2013-01-29 The Feinstein Institute For Medical Research Modified macrophage migration inhibitory factor inhibitors
JP5186303B2 (ja) * 2008-07-31 2013-04-17 東京応化工業株式会社 レジスト組成物およびレジストパターン形成方法
US8987504B2 (en) 2010-06-18 2015-03-24 Victoria Link Limited Aminohydroxylation of alkenes
CN102190598B (zh) * 2011-03-28 2014-01-29 浙江工业大学 环丙烷肟酯衍生物及其制备方法和用途
US9567306B2 (en) 2014-06-17 2017-02-14 The Feinstein Institute For Medical Research Inhibition of macrophage migration inhibitory factor in melanoma and colon cancer
CA3196362A1 (en) * 2020-10-28 2022-05-05 University Health Network (Uhn) Methods of treating spondyloarthritis or symptoms thereof

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3918973A (en) * 1973-01-31 1975-11-11 Agfa Gevaert Process and materials for the information-wise production of amino compounds
JPS62148471A (ja) * 1985-12-23 1987-07-02 バスフ　アクチェン　ゲゼルシャフト 置換されたキノリン−８−カルボン酸のオキシムエステル、その製法及び該化合物を含有する除草剤
JPH07196629A (ja) * 1993-11-13 1995-08-01 Lucky Co Ltd ピリミジン誘導体、その製造方法及び除草剤
JPH11106371A (ja) * 1997-07-04 1999-04-20 Nisshin Flour Milling Co Ltd アシルヒドラゾン誘導体

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IT1110460B (it) * 1977-03-02 1985-12-23 Ciba Geigy Ag Prodotti che favoriscono la crescita delle piante e prodotti che proteggono le piante a base di eteri di ossime e di esteri di ossime loro preparazione e loro impiego
FR2623190B1 (fr) * 1987-11-12 1990-02-23 Rhone Poulenc Agrochimie Nicotinates d'oximes fongicides
AU1235601A (en) * 1999-10-29 2001-05-14 Cytokine Pharmasciences, Inc. Compounds having mif antagonist activity
WO2002100332A2 (en) * 2001-06-08 2002-12-19 Cytokine Pharmasciences, Inc. Isoxazoline compounds having mif antagonist activity
US7842835B2 (en) * 2003-07-07 2010-11-30 Georgetown University Histone deacetylase inhibitors and methods of use thereof
US20050222123A1 (en) * 2004-01-27 2005-10-06 North Shore-Long Island Jewish Research Institute Cholinesterase inhibitors for treating inflammation
KR100784337B1 (ko) * 2004-11-12 2007-12-13 한국생명공학연구원 신규한 ｏ-아실옥심 유도체, 그의 제조방법 및 이를유효성분으로 하는 심장순환계 질환의 예방 및 치료용약학 조성물

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3918973A (en) * 1973-01-31 1975-11-11 Agfa Gevaert Process and materials for the information-wise production of amino compounds
JPS62148471A (ja) * 1985-12-23 1987-07-02 バスフ　アクチェン　ゲゼルシャフト 置換されたキノリン−８−カルボン酸のオキシムエステル、その製法及び該化合物を含有する除草剤
JPH07196629A (ja) * 1993-11-13 1995-08-01 Lucky Co Ltd ピリミジン誘導体、その製造方法及び除草剤
JPH11106371A (ja) * 1997-07-04 1999-04-20 Nisshin Flour Milling Co Ltd アシルヒドラゾン誘導体

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AU2007258731A1 (en) 2007-12-21
WO2007145888A3 (en) 2008-07-17
AU2007258731B2 (en) 2013-01-31
EP2023732A4 (en) 2011-10-05
CA2653646A1 (en) 2007-12-21
WO2007145888A2 (en) 2007-12-21
US20090318509A1 (en) 2009-12-24
EP2023732A2 (en) 2009-02-18

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