JP2009513710A - ジアゾンアミドａ類似体 - Google Patents

ジアゾンアミドａ類似体 Download PDF

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Publication number
JP2009513710A
JP2009513710A JP2008538978A JP2008538978A JP2009513710A JP 2009513710 A JP2009513710 A JP 2009513710A JP 2008538978 A JP2008538978 A JP 2008538978A JP 2008538978 A JP2008538978 A JP 2008538978A JP 2009513710 A JP2009513710 A JP 2009513710A
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JP
Japan
Prior art keywords
compound
added
cells
paclitaxel
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2008538978A
Other languages
English (en)
Japanese (ja)
Other versions
JP2009513710A5 (https=
Inventor
ハラン、パトリック
ウィリアムズ、ノエル
バーゲット、アンソニー
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
University of Texas System
Original Assignee
University of Texas System
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US11/264,502 external-priority patent/US7517895B2/en
Application filed by University of Texas System filed Critical University of Texas System
Publication of JP2009513710A publication Critical patent/JP2009513710A/ja
Publication of JP2009513710A5 publication Critical patent/JP2009513710A5/ja
Withdrawn legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/22—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Medicinal Preparation (AREA)
JP2008538978A 2005-10-31 2006-10-31 ジアゾンアミドａ類似体 Withdrawn JP2009513710A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US11/264,502 US7517895B2 (en) 2001-08-24 2005-10-31 Synthetic diazonamides
US81465106P 2006-06-16 2006-06-16
PCT/US2006/042565 WO2007053650A2 (en) 2005-10-31 2006-10-31 Diazonamide a analog

Publications (2)

Publication Number Publication Date
JP2009513710A true JP2009513710A (ja) 2009-04-02
JP2009513710A5 JP2009513710A5 (https=) 2009-11-26

Family

ID=38006479

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2008538978A Withdrawn JP2009513710A (ja) 2005-10-31 2006-10-31 ジアゾンアミドａ類似体

Country Status (8)

Country Link
US (1) US7538129B2 (https=)
EP (1) EP1948169A4 (https=)
JP (1) JP2009513710A (https=)
AU (1) AU2006308849A1 (https=)
BR (1) BRPI0618136A2 (https=)
CR (1) CR10038A (https=)
EA (1) EA013692B1 (https=)
WO (1) WO2007053650A2 (https=)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008154441A1 (en) * 2007-06-07 2008-12-18 Joyant Pharmaceuticals, Inc. Methods for preparing diazonamides
WO2009086170A1 (en) * 2007-12-21 2009-07-09 Joyant Pharmaceuticals, Inc. Diazonamide analogs with improved solubility
AU2009243056B2 (en) * 2008-04-29 2015-05-14 Joyant Pharmaceuticals, Inc. Indoline anti-cancer agents
WO2009143485A1 (en) * 2008-05-22 2009-11-26 Joyant Pharmaceuticals, Inc. Diazonamide analogs
HRP20171930T1 (hr) 2011-04-22 2018-02-09 Joyant Pharmaceuticals, Inc. Analozi diazonamida
US10353032B2 (en) * 2015-10-27 2019-07-16 Halliburton Energy Services, Inc. Viscosity determination apparatus, systems, and methods

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7022720B2 (en) * 2001-08-24 2006-04-04 Board Of Regents, The University Of Texas System Synthetic diazonamides as novel anti-mitotic agents
US7517895B2 (en) * 2001-08-24 2009-04-14 Board Of Regents, The University Of Texas System Synthetic diazonamides

Also Published As

Publication number Publication date
EA013692B1 (ru) 2010-06-30
EA200801238A1 (ru) 2008-12-30
EP1948169A2 (en) 2008-07-30
AU2006308849A1 (en) 2007-05-10
US20070149583A1 (en) 2007-06-28
CR10038A (es) 2008-09-12
WO2007053650A2 (en) 2007-05-10
EP1948169A4 (en) 2009-11-04
US7538129B2 (en) 2009-05-26
WO2007053650A3 (en) 2007-11-22
BRPI0618136A2 (pt) 2011-08-16

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