EA200801238A1 - Аналог диазонамида а - Google Patents

Аналог диазонамида а

Info

Publication number
EA200801238A1
EA200801238A1 EA200801238A EA200801238A EA200801238A1 EA 200801238 A1 EA200801238 A1 EA 200801238A1 EA 200801238 A EA200801238 A EA 200801238A EA 200801238 A EA200801238 A EA 200801238A EA 200801238 A1 EA200801238 A1 EA 200801238A1
Authority
EA
Eurasian Patent Office
Prior art keywords
diazonamide
analogue
conjugates
salts
effective
Prior art date
Application number
EA200801238A
Other languages
English (en)
Other versions
EA013692B1 (ru
Inventor
Патрик Харран
Ноэлль Уилльямс
Энтони Берджетт
Original Assignee
Борд Оф Риджентс, Дзе Юниверсити Оф Техас Систем
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US11/264,502 external-priority patent/US7517895B2/en
Application filed by Борд Оф Риджентс, Дзе Юниверсити Оф Техас Систем filed Critical Борд Оф Риджентс, Дзе Юниверсити Оф Техас Систем
Publication of EA200801238A1 publication Critical patent/EA200801238A1/ru
Publication of EA013692B1 publication Critical patent/EA013692B1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/22—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Особый аналог диазонамида А и его соли и конъюгаты являются действенными в лечении пролиферативных расстройств.
EA200801238A 2005-10-31 2006-10-31 Аналог диазонамида а EA013692B1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US11/264,502 US7517895B2 (en) 2001-08-24 2005-10-31 Synthetic diazonamides
US81465106P 2006-06-16 2006-06-16
PCT/US2006/042565 WO2007053650A2 (en) 2005-10-31 2006-10-31 Diazonamide a analog

Publications (2)

Publication Number Publication Date
EA200801238A1 true EA200801238A1 (ru) 2008-12-30
EA013692B1 EA013692B1 (ru) 2010-06-30

Family

ID=38006479

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200801238A EA013692B1 (ru) 2005-10-31 2006-10-31 Аналог диазонамида а

Country Status (8)

Country Link
US (1) US7538129B2 (ru)
EP (1) EP1948169A4 (ru)
JP (1) JP2009513710A (ru)
AU (1) AU2006308849A1 (ru)
BR (1) BRPI0618136A2 (ru)
CR (1) CR10038A (ru)
EA (1) EA013692B1 (ru)
WO (1) WO2007053650A2 (ru)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7851620B2 (en) * 2007-06-07 2010-12-14 Board Of Regents, The University Of Texas System Methods for preparing diazonamides
WO2009086170A1 (en) * 2007-12-21 2009-07-09 Joyant Pharmaceuticals, Inc. Diazonamide analogs with improved solubility
CA2720516C (en) * 2008-04-29 2013-10-01 Joyant Pharmaceuticals, Inc. Indoline anti-cancer agents
US8153619B2 (en) * 2008-05-22 2012-04-10 Joyant Pharmaceuticals, Inc. Diazonamide analogs
DK2699580T3 (en) 2011-04-22 2018-01-08 Joyant Pharmaceuticals Inc DIAZONAMI DISEASES
WO2017074316A1 (en) * 2015-10-27 2017-05-04 Halliburton Energy Services, Inc. Viscosity determination apparatus, systems, and methods

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7517895B2 (en) * 2001-08-24 2009-04-14 Board Of Regents, The University Of Texas System Synthetic diazonamides
US7022720B2 (en) * 2001-08-24 2006-04-04 Board Of Regents, The University Of Texas System Synthetic diazonamides as novel anti-mitotic agents

Also Published As

Publication number Publication date
US20070149583A1 (en) 2007-06-28
BRPI0618136A2 (pt) 2011-08-16
US7538129B2 (en) 2009-05-26
EP1948169A4 (en) 2009-11-04
CR10038A (es) 2008-09-12
JP2009513710A (ja) 2009-04-02
AU2006308849A1 (en) 2007-05-10
EP1948169A2 (en) 2008-07-30
EA013692B1 (ru) 2010-06-30
WO2007053650A2 (en) 2007-05-10
WO2007053650A3 (en) 2007-11-22

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Legal Events

Date Code Title Description
MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ BY KZ KG MD TJ TM RU