JP2008530007A5 - - Google Patents
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- Publication number
- JP2008530007A5 JP2008530007A5 JP2007554134A JP2007554134A JP2008530007A5 JP 2008530007 A5 JP2008530007 A5 JP 2008530007A5 JP 2007554134 A JP2007554134 A JP 2007554134A JP 2007554134 A JP2007554134 A JP 2007554134A JP 2008530007 A5 JP2008530007 A5 JP 2008530007A5
- Authority
- JP
- Japan
- Prior art keywords
- compound according
- alkyl
- bond
- pharmaceutical composition
- cycloalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 150000001875 compounds Chemical class 0.000 claims 8
- 125000000217 alkyl group Chemical group 0.000 claims 5
- 125000000753 cycloalkyl group Chemical group 0.000 claims 3
- 239000008194 pharmaceutical composition Substances 0.000 claims 3
- 125000000923 (C1-C30) alkyl group Chemical group 0.000 claims 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 claims 1
- 239000003937 drug carrier Substances 0.000 claims 1
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims 1
- 125000001475 halogen functional group Chemical group 0.000 claims 1
- 229910052739 hydrogen Inorganic materials 0.000 claims 1
- 239000001257 hydrogen Substances 0.000 claims 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US65037605P | 2005-02-04 | 2005-02-04 | |
| US60/650,376 | 2005-02-04 | ||
| PCT/US2006/002436 WO2006083618A1 (en) | 2005-02-04 | 2006-01-24 | NANDROLONE 17ß-CARBONATES |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2008530007A JP2008530007A (ja) | 2008-08-07 |
| JP2008530007A5 true JP2008530007A5 (enExample) | 2008-11-27 |
| JP5227593B2 JP5227593B2 (ja) | 2013-07-03 |
Family
ID=36283873
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007554134A Expired - Fee Related JP5227593B2 (ja) | 2005-02-04 | 2006-01-24 | ナンドロロン１７β−カーボネート |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US7820642B2 (enExample) |
| EP (1) | EP1846434B1 (enExample) |
| JP (1) | JP5227593B2 (enExample) |
| AT (1) | ATE426610T1 (enExample) |
| AU (1) | AU2006211907B2 (enExample) |
| CA (1) | CA2596884C (enExample) |
| DE (1) | DE602006005901D1 (enExample) |
| WO (1) | WO2006083618A1 (enExample) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN109575098B (zh) * | 2019-01-18 | 2021-01-01 | 湖南成大生物科技有限公司 | 诺孕美特的合成方法 |
| CN110128529B (zh) * | 2019-04-11 | 2023-07-07 | 中国农业科学院兰州畜牧与兽药研究所 | 一种去甲睾酮人工抗原的合成方法 |
| WO2021252761A2 (en) * | 2020-06-11 | 2021-12-16 | The United States Of America, As Represented By The Secretary, Department Of Health And Human Services | Monomeric and oligomeric compound embodiments as contraceptives and therapies and methods of making and using the same |
Family Cites Families (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3056727A (en) * | 1960-10-27 | 1962-10-02 | Roussel Uclaf | Cyclohexylcarbonates of steroids |
| FR1215M (fr) * | 1961-03-28 | 1962-04-02 | Roussel Uclaf S A Soc | Nouveau médicament, notamment pour le traitement des troubles dus a une hyperestrogénie ou a une hypoandrogénie. |
| FR6576M (enExample) * | 1965-10-11 | 1968-12-30 | ||
| FR5913M (enExample) * | 1965-12-02 | 1968-04-01 | ||
| US3629244A (en) * | 1966-01-21 | 1971-12-21 | Roussel Uclaf | 17beta-ethers of delta 4 9 11-gonatrienes and compositions containing them |
| US3523126A (en) * | 1967-12-13 | 1970-08-04 | Du Pont | Testosterone and 19-nortestosterone(4'-methylbicyclo(2,2,2)octane - 1' - methyl)carbonate and selected derivatives |
| GB1291293A (en) | 1970-05-29 | 1972-10-04 | Du Pont | Steroid carbonates and their preparation |
| GB1355663A (en) * | 1970-06-17 | 1974-06-05 | Theramex | 19-nortestosterone 17- -p-substituted phenoxy-acetates |
| DE4025342A1 (de) * | 1990-08-10 | 1992-02-13 | Hoechst Ag | In 17-stellung substituierte corticoid-17-alkylcarbonate, verfahren zu deren herstellung und diese enthaltende arzneimittel |
| WO1993025197A1 (en) * | 1992-06-12 | 1993-12-23 | Affymax Technologies N.V. | Compositions and methods for enhanced drug delivery |
| US5622944A (en) * | 1992-06-12 | 1997-04-22 | Affymax Technologies N.V. | Testosterone prodrugs for improved drug delivery |
| US5952319A (en) * | 1997-11-26 | 1999-09-14 | Research Triangle Institute | Androgenic steroid compounds and a method of making and using the same |
| EP1272196B1 (en) * | 2000-03-31 | 2006-08-02 | THE GOVERNMENT OF THE UNITED STATES OF AMERICA, as represented by THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES | Methods of making the 4-n-butylcyclohexanoic and the undecanoic acid esters of (7 alpha,11 beta)-dimethyl-17 beta-hydroxy-4-estren-3-one and their medical use |
| US20030069215A1 (en) * | 2001-03-30 | 2003-04-10 | The Government Of The United States Of America, | Methods of making and using 7a,11b-dimethyl-17b-hydroxy-4-estren-3-one 17b-trans-4-n-butylcyclohexane carboxylate and 7a,11b-dimethyl-17b-hydroxyestr-4-en-3-one 17-undecanoate |
| US6740646B2 (en) * | 2002-01-16 | 2004-05-25 | Biotest Laboratories, Llc | Bioavailable prodrugs of androgenic steroids and related method |
| US20030134828A1 (en) * | 2002-01-16 | 2003-07-17 | Roberts William J. | Composition and method for increasing in vivo androgen concentration |
| US20030134831A1 (en) * | 2002-01-16 | 2003-07-17 | Roberts William J | Bioavailable prodrugs of androgenic steroids and related method |
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2006
- 2006-01-24 AT AT06719336T patent/ATE426610T1/de not_active IP Right Cessation
- 2006-01-24 DE DE602006005901T patent/DE602006005901D1/de active Active
- 2006-01-24 CA CA2596884A patent/CA2596884C/en not_active Expired - Fee Related
- 2006-01-24 AU AU2006211907A patent/AU2006211907B2/en not_active Ceased
- 2006-01-24 US US11/815,532 patent/US7820642B2/en active Active
- 2006-01-24 WO PCT/US2006/002436 patent/WO2006083618A1/en not_active Ceased
- 2006-01-24 JP JP2007554134A patent/JP5227593B2/ja not_active Expired - Fee Related
- 2006-01-24 EP EP06719336A patent/EP1846434B1/en not_active Not-in-force