JP2008524186A - ケモカイン受容体活性の調節のためのチアゾロピラミジン化合物 - Google Patents
ケモカイン受容体活性の調節のためのチアゾロピラミジン化合物 Download PDFInfo
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- JP2008524186A JP2008524186A JP2007546178A JP2007546178A JP2008524186A JP 2008524186 A JP2008524186 A JP 2008524186A JP 2007546178 A JP2007546178 A JP 2007546178A JP 2007546178 A JP2007546178 A JP 2007546178A JP 2008524186 A JP2008524186 A JP 2008524186A
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- alkyl
- pharmaceutically acceptable
- solvate
- formula
- acceptable salt
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
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Landscapes
- Health & Medical Sciences (AREA)
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- Chemical & Material Sciences (AREA)
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- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Rheumatology (AREA)
- Physical Education & Sports Medicine (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Immunology (AREA)
- Pain & Pain Management (AREA)
- Otolaryngology (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0427698A GB0427698D0 (en) | 2004-12-17 | 2004-12-17 | Compounds |
| GB0502542A GB0502542D0 (en) | 2005-02-08 | 2005-02-08 | Method |
| PCT/GB2005/004825 WO2006064228A2 (en) | 2004-12-17 | 2005-12-14 | Thiazolopyramidine compounds for the modulation of chemokine receptor activity |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2008524186A true JP2008524186A (ja) | 2008-07-10 |
| JP2008524186A5 JP2008524186A5 (enExample) | 2009-01-29 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007546178A Pending JP2008524186A (ja) | 2004-12-17 | 2005-12-14 | ケモカイン受容体活性の調節のためのチアゾロピラミジン化合物 |
Country Status (4)
| Country | Link |
|---|---|
| US (1) | US20090239882A1 (enExample) |
| EP (1) | EP1844054A2 (enExample) |
| JP (1) | JP2008524186A (enExample) |
| WO (1) | WO2006064228A2 (enExample) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2008535835A (ja) * | 2005-04-06 | 2008-09-04 | アストラゼネカ・アクチエボラーグ | 新規な５−置換された７−アミノ［１，３］チアゾロ［４，５−ｄ］ピリミジン誘導体 |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE9903544D0 (sv) | 1999-10-01 | 1999-10-01 | Astra Pharma Prod | Novel compounds |
| GB2359551A (en) | 2000-02-23 | 2001-08-29 | Astrazeneca Uk Ltd | Pharmaceutically active pyrimidine derivatives |
| GB0221828D0 (en) | 2002-09-20 | 2002-10-30 | Astrazeneca Ab | Novel compound |
| GB0328243D0 (en) | 2003-12-05 | 2004-01-07 | Astrazeneca Ab | Methods |
| TW200820973A (en) * | 2006-09-29 | 2008-05-16 | Astrazeneca Ab | Novel compounds 480 |
| NZ576519A (en) | 2006-09-29 | 2011-11-25 | Astrazeneca Ab | Novel 5,7-disubstituted [1, 3] thiazolo [4, 5-d] pyrimidin-2 (3h)-amine derivatives and their use in therapy |
| AU2010324249B2 (en) * | 2009-11-30 | 2014-08-28 | Jiangsu Hansoh Pharmaceutical Group Co., Ltd. | Azilsartan organic amine salts, preparation method and use thereof |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE9802729D0 (sv) * | 1998-08-13 | 1998-08-13 | Astra Pharma Prod | Novel Compounds |
| SE9903544D0 (sv) * | 1999-10-01 | 1999-10-01 | Astra Pharma Prod | Novel compounds |
| WO2001058906A1 (en) * | 2000-02-11 | 2001-08-16 | Astrazeneca Ab | Pyrimidine compounds and their use as modulators of chemokine receptor activity |
| AU2004278276B2 (en) * | 2003-10-07 | 2007-10-18 | Astrazeneca Ab | New 2-substituted, 4-amino-thiazolo(4,5-d) pyrimidines, useful as chemokine receptor antagonists, esp. CX3CR1 |
| WO2005082865A1 (ja) * | 2004-02-27 | 2005-09-09 | Astellas Pharma Inc. | 縮合二環性ピリミジン誘導体 |
-
2005
- 2005-12-14 JP JP2007546178A patent/JP2008524186A/ja active Pending
- 2005-12-14 WO PCT/GB2005/004825 patent/WO2006064228A2/en not_active Ceased
- 2005-12-14 US US11/721,583 patent/US20090239882A1/en not_active Abandoned
- 2005-12-14 EP EP05818307A patent/EP1844054A2/en not_active Withdrawn
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2008535835A (ja) * | 2005-04-06 | 2008-09-04 | アストラゼネカ・アクチエボラーグ | 新規な５−置換された７−アミノ［１，３］チアゾロ［４，５−ｄ］ピリミジン誘導体 |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2006064228A3 (en) | 2007-02-08 |
| US20090239882A1 (en) | 2009-09-24 |
| WO2006064228A2 (en) | 2006-06-22 |
| EP1844054A2 (en) | 2007-10-17 |
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