JP2008512496A5 - - Google Patents

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Publication number
JP2008512496A5
JP2008512496A5 JP2007531440A JP2007531440A JP2008512496A5 JP 2008512496 A5 JP2008512496 A5 JP 2008512496A5 JP 2007531440 A JP2007531440 A JP 2007531440A JP 2007531440 A JP2007531440 A JP 2007531440A JP 2008512496 A5 JP2008512496 A5 JP 2008512496A5
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JP
Japan
Prior art keywords
carbon atoms
alkyl
cycloalkyl
aryl
carbon
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2007531440A
Other languages
English (en)
Japanese (ja)
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JP2008512496A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2005/032484 external-priority patent/WO2006031770A1/en
Publication of JP2008512496A publication Critical patent/JP2008512496A/ja
Publication of JP2008512496A5 publication Critical patent/JP2008512496A5/ja
Withdrawn legal-status Critical Current

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JP2007531440A 2004-09-10 2005-09-09 １，３，４，９−テトラヒドロピラノ［３，４−ｂ］インドール誘導体の大規模実施可能な合成方法 Withdrawn JP2008512496A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US60899504P 2004-09-10 2004-09-10
PCT/US2005/032484 WO2006031770A1 (en) 2004-09-10 2005-09-09 Process for the scalable synthesis of 1, 3, 4, 9-tetrahydropyrano[3, 4-b]-indole derivatives

Publications (2)

Publication Number Publication Date
JP2008512496A JP2008512496A (ja) 2008-04-24
JP2008512496A5 true JP2008512496A5 (https=) 2008-10-23

Family

ID=35478248

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007531440A Withdrawn JP2008512496A (ja) 2004-09-10 2005-09-09 １，３，４，９−テトラヒドロピラノ［３，４−ｂ］インドール誘導体の大規模実施可能な合成方法

Country Status (8)

Country Link
US (1) US20060058532A1 (https=)
EP (1) EP1786772A1 (https=)
JP (1) JP2008512496A (https=)
AU (1) AU2005285005A1 (https=)
BR (1) BRPI0514313A (https=)
CA (1) CA2573508A1 (https=)
MX (1) MX2007002837A (https=)
WO (1) WO2006031770A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PH12012501293A1 (en) * 2009-12-23 2013-01-07 Arqule Inc Purified pyrroloquinolinyl-pyrrolidine-2,5-dione compositions and methods for preparing and using same
CN102516151B (zh) * 2011-11-11 2013-09-11 华东师范大学 一种3-取代-3-羟基吲哚酮衍生物及其制备方法和应用
PL233259B1 (pl) * 2017-07-10 2019-09-30 Politechnika Poznanska Indolilooctany 1-alkilochininy, sposób ich otrzymywania oraz zastosowanie jako środki bakteriostatyczne i bakteriobójcze

Family Cites Families (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3974179A (en) * 1971-06-01 1976-08-10 American Home Products Corporation 1,3,4,9-Tetrahydropyrano[3,4-b]indole-1-acetamides and derivatives
US3939178A (en) * 1971-06-01 1976-02-17 American Home Products Corporation Certain pyrano [3,4-b]indoles and thiopyrano[3,4-b]indoles
US3843681A (en) * 1971-06-01 1974-10-22 American Home Prod 1-carboxamido pyrano(thiopyrano)(3,4-6)indole derivatives
US3880853A (en) * 1972-01-13 1975-04-29 Ayerst Mckenna & Harrison Pyrano-and thiopyranoindole
US4036842A (en) * 1972-05-16 1977-07-19 American Home Products Corporation Process for preparing polycyclic heterocycles having a pyran ring
US4012417A (en) * 1972-05-16 1977-03-15 American Home Products Corporation Process for preparing pyrano[3,4-b]indole or thio pyrano[3,4-b]indole derivatives
US4076831A (en) * 1972-05-16 1978-02-28 American Home Products Corporation Pyrano[3,4-b]-indole derivatives, pharmaceutical compositions and methods of use
US4070371A (en) * 1972-05-16 1978-01-24 American Home Products Corporation Derivatives of 1,3,4,9-tetrahydropyrano[3,4-b]indole-1-acetic acid
US4118394A (en) * 1976-10-18 1978-10-03 Ayerst, Mckenna & Harrison Limited Pyrano- and thiopyranoindole derivatives
US4179503A (en) * 1978-05-08 1979-12-18 American Home Products Corp. 1-Hydroxyalkanamine pyrano[3,4-b]indole derivatives
US4520203A (en) * 1983-08-16 1985-05-28 American Home Products Corporation Resolution of (±)-1,8-diethyl-1,3,4,9-tetrahydropyrano[3,4-b]indole-1-acetic acid using cinchonine
US4515961A (en) * 1983-08-16 1985-05-07 American Home Products Corporation Resolution of (±)-1,8-diethyl-1,3,4,9-tetrahydropyrano[3,4,-b] indole-1-acetic acid using enrichment crystallization
US4501899A (en) * 1983-08-16 1985-02-26 American Home Products Corporation Resolution of (+)-1,8-diethyl-1,3,4,9-tetrahydropyrano[3,4-b]indole-1-acetic acid using cholesteryl aniline
US4544757A (en) * 1984-02-16 1985-10-01 American Home Products Corporation Process for the resolution of pyrano[3,4-b]indole-1-acetic acids
US4585877A (en) * 1985-05-06 1986-04-29 American Home Products Corporation Process for preparing 1,8-diethyl-1,3,4,9-tetrahydropyrano(3,4-b)-indole-1-acetic acid, etodolac
US4775690A (en) * 1987-01-13 1988-10-04 American Home Products Corporation Substituted 1,3,4,9-tetrahydropyrano(3,4-b)indole-1-acetic acids
US4670462A (en) * 1986-03-11 1987-06-02 American Home Products Corporation Substituted 1,3,4,9-tetrahydropyrano(3,4-B)indole-1-acetic acids
US4686213A (en) * 1986-08-15 1987-08-11 American Home Products Corporation Substituted 1,3,4,9-tetrahydropyrano(3,4-b)indole-1-acetic acids
CA1319695C (en) * 1987-02-20 1993-06-29 Brian A. Mckittrick Substituted 1,3,4,9-tetrahydropyrano¬3,4-b|- indole-1-acetic acids
US4810699A (en) * 1987-02-20 1989-03-07 American Home Products Corporation Substituted 1,3,4,9-tetrahydropyrano[3,4,-b]indole-1-acetic acids, pharmaceutical compositions containing them, and methods for treating inflammatory conditions and for analgesic purposes using them
US4776967A (en) * 1987-02-27 1988-10-11 Idemitsu Kosan Company Limited Lubricating oil composition
US4824961A (en) * 1987-08-27 1989-04-25 American Home Products Corporation Production of substituted 1,3,4,9-tetrahydropyrano(3,4-b)indole-1-acetic acids
US4822781A (en) * 1987-10-08 1989-04-18 American Home Products Substituted-8-alkenyl-1,3,4,9-tetrahydropyrano-[3,4-b]indole-1-acetic acids
US4822893A (en) * 1988-02-08 1989-04-18 American Home Products Production of substituted 1,3,4,9-tetrahydropyrano[3,4-b]indole-1-acetic acids
US4960902A (en) * 1988-08-19 1990-10-02 American Home Products Corporation Trifluoromethoxy substituted 1,3,4,9-tetrahydropyrano-[3,4-b]indole-1-acetic acids
US4925955A (en) * 1989-02-28 1990-05-15 American Home Products Corporation Resolution of (1S,4R)-1-ethyl-1,3,4,9-tetrahydro-4-(phenylmethyl) pyrano[3,4-B]indole-1-acetic acid using brucine
US5830911A (en) * 1996-08-14 1998-11-03 American Home Products Corporation Pyranoindole and tetrahydrocarbazole inhibitors of COX-2

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