JP2007537182A5 - - Google Patents
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- Publication number
- JP2007537182A5 JP2007537182A5 JP2007512054A JP2007512054A JP2007537182A5 JP 2007537182 A5 JP2007537182 A5 JP 2007537182A5 JP 2007512054 A JP2007512054 A JP 2007512054A JP 2007512054 A JP2007512054 A JP 2007512054A JP 2007537182 A5 JP2007537182 A5 JP 2007537182A5
- Authority
- JP
- Japan
- Prior art keywords
- propionyl
- acyl group
- acetyl
- compound according
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 125000002252 acyl group Chemical group 0.000 claims 3
- 150000001875 compounds Chemical class 0.000 claims 3
- -1 isobutyryl Chemical group 0.000 claims 3
- 125000001501 propionyl group Chemical group O=C([*])C([H])([H])C([H])([H])[H] 0.000 claims 3
- 125000002777 acetyl group Chemical group [H]C([H])([H])C(*)=O 0.000 claims 2
- 125000004063 butyryl group Chemical group O=C([*])C([H])([H])C([H])([H])C([H])([H])[H] 0.000 claims 1
- 125000003774 valeryl group Chemical group O=C([*])C([H])([H])C([H])([H])C([H])([H])C([H])([H])[H] 0.000 claims 1
Description
Claims (3)
- Ｃ2〜Ｃ8のアシル基が、アセチル、プロピオニル、ブチリル、イソブチリル、バレリル、イソバレリル、ピバロイル、カプロイルから選択される請求項１に記載の化合物。
- Ｃ2〜Ｃ8のアシル基が、アセチル又はプロピオニルである請求項２に記載の化合物。
- Ｃ2〜Ｃ8のアシル基が、プロピオニルである請求項３に記載の化合物。
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT000954A ITMI20040954A1 (it) | 2004-05-12 | 2004-05-12 | Derivati del 3,6-diazabiciclo 3.1.i.eptano ad attivita' analgesica |
| PCT/EP2005/004994 WO2005108402A1 (en) | 2004-05-12 | 2005-05-09 | 3,6-diazabicyclos[3.1.1]heptane derivatives with analgesic activity |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2007537182A JP2007537182A (ja) | 2007-12-20 |
| JP2007537182A5 true JP2007537182A5 (ja) | 2008-06-26 |
Family
ID=34969286
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007512054A Pending JP2007537182A (ja) | 2004-05-12 | 2005-05-09 | 鎮痛活性を有する３，６−ジアザビシクロ［３．１．１］ヘプタン誘導体 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US20070225492A1 (ja) |
| EP (1) | EP1751164A1 (ja) |
| JP (1) | JP2007537182A (ja) |
| IT (1) | ITMI20040954A1 (ja) |
| WO (1) | WO2005108402A1 (ja) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1395452B1 (it) * | 2009-02-25 | 2012-09-21 | Neuroscienze Pharmaness S C A Rl | Microemulsioni |
| IT1390850B1 (it) * | 2008-07-31 | 2011-10-19 | Neuroscienze Pharmaness S C A R L | Microemulsioni |
| IT1390848B1 (it) | 2008-07-31 | 2011-10-19 | Neuroscienze Pharmaness S C A R L | Composti farmaceutici |
| EP2149370A1 (en) | 2008-07-31 | 2010-02-03 | Neuroscienze Pharmaness S.C. A R.L. | Diazabicyclic compounds and microemulsions thereof |
| JP2013512922A (ja) * | 2009-12-07 | 2013-04-18 | ターガセプト，インコーポレイテッド | 神経型ニコチン性アセチルコリン受容体リガンドとしての３，６−ジアザビシクロ［３．１．１］ヘプタン |
| IT1396951B1 (it) | 2009-12-18 | 2012-12-20 | Neuroscienze Pharmaness S C A R L | Composti farmaceutici |
| WO2012125518A1 (en) | 2011-03-14 | 2012-09-20 | Targacept, Inc. | Salt forms of 3 - cyclopropylcarbonyl - 3, 6 - diazabicyclo [3.1.1] heptane |
| WO2014011863A1 (en) * | 2012-07-12 | 2014-01-16 | Targacept, Inc. | Method of treatment with 3-cyclopropylcarbonyl-3,6-diazabicyclo[3.1.1]heptane |
| DK3030561T3 (en) | 2013-08-07 | 2017-03-27 | Cadila Healthcare Ltd | N-CYANOMETHYLAMIDES AS INHIBITORS OF JANUS KINASE |
| WO2016054123A1 (en) | 2014-09-30 | 2016-04-07 | Lightner Derek | Methods of producing heteropolycycles via bis-epoxidation |
| CN111892599B (zh) * | 2020-08-14 | 2023-01-13 | 黄芳 | 一种2,5-二氮杂双环[2.2.2]辛烷-2-羧酸叔丁酯的合成方法 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1274018B (it) * | 1994-02-23 | 1997-07-14 | Riace Ets | Derivati del 3,8-diazabiciclo(3.2.1.)ottano ad attivita' analgesica |
| CN1636996A (zh) * | 1999-01-29 | 2005-07-13 | 艾博特公司 | 用作烟碱性乙酰胆碱受体配体的二氮杂二环衍生物 |
| ES2242749T3 (es) * | 2000-05-25 | 2005-11-16 | Targacept, Inc. | Hetoroarildiazabicycloalkanos como ligandos de receptores colinergicos nicotinicos. |
| US7358243B2 (en) * | 2002-07-26 | 2008-04-15 | Neurosearch A/S | Diazabicyclonane and-decane derivatives and their use as opioid receptor ligands |
-
2004
- 2004-05-12 IT IT000954A patent/ITMI20040954A1/it unknown
-
2005
- 2005-05-09 WO PCT/EP2005/004994 patent/WO2005108402A1/en active Application Filing
- 2005-05-09 JP JP2007512054A patent/JP2007537182A/ja active Pending
- 2005-05-09 EP EP05747942A patent/EP1751164A1/en not_active Withdrawn
- 2005-05-09 US US11/596,083 patent/US20070225492A1/en not_active Abandoned
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