JP2006500337A - 塩酸ベナゼプリルの結晶多形形態および非晶質形態 - Google Patents
塩酸ベナゼプリルの結晶多形形態および非晶質形態 Download PDFInfo
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- JP2006500337A JP2006500337A JP2004525233A JP2004525233A JP2006500337A JP 2006500337 A JP2006500337 A JP 2006500337A JP 2004525233 A JP2004525233 A JP 2004525233A JP 2004525233 A JP2004525233 A JP 2004525233A JP 2006500337 A JP2006500337 A JP 2006500337A
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- phenylpropyl
- ethoxycarbonyl
- tetrahydro
- amino
- oxo
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
- C07D223/14—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D223/16—Benzazepines; Hydrogenated benzazepines
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
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- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP02405653 | 2002-07-26 | ||
| PCT/EP2003/007771 WO2004013105A1 (en) | 2002-07-26 | 2003-07-17 | Crystalline polymorphic and amorphous forms of benazepril hydrochloride |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2006500337A true JP2006500337A (ja) | 2006-01-05 |
| JP2006500337A5 JP2006500337A5 (enExample) | 2006-08-31 |
Family
ID=31198001
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004525233A Withdrawn JP2006500337A (ja) | 2002-07-26 | 2003-07-17 | 塩酸ベナゼプリルの結晶多形形態および非晶質形態 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20050107359A1 (enExample) |
| EP (1) | EP1525189A1 (enExample) |
| JP (1) | JP2006500337A (enExample) |
| AU (1) | AU2003250086A1 (enExample) |
| CA (1) | CA2492949A1 (enExample) |
| WO (1) | WO2004013105A1 (enExample) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2014506919A (ja) * | 2011-07-12 | 2014-03-20 | サムジン ファーマシューティカル カンパニー，リミテッド | クロピドグレル硫酸水素塩の球状粒子、これを含む薬学的組成物及びその製造方法 |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2005075467A2 (en) * | 2004-02-06 | 2005-08-18 | Ciba Specialty Chemicals Holding Inc. | Crystalline forms of zolmitriptan |
| WO2006084761A1 (en) * | 2005-02-11 | 2006-08-17 | Albemarle Corporation | Crystalline polymorphs of benazepril hydrochloride |
| US20090082559A1 (en) * | 2005-05-12 | 2009-03-26 | Lupin Limited | Process for Crystallization of Benazepril Hydrochloride |
| US9409913B2 (en) * | 2012-11-21 | 2016-08-09 | Enaltec Labs Private Limited | Polymorphic forms of alcaftadine |
| CN104788376A (zh) * | 2014-01-17 | 2015-07-22 | 海门慧聚药业有限公司 | 一种盐酸贝那普利的新晶型及其制备方法 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE18397T1 (de) * | 1981-08-11 | 1986-03-15 | Ciba Geigy Ag | Benzazepin-2-one, verfahren zu ihrer herstellung, pharmazeutische praeparate die diese verbindungen enthalten, sowie die verbindungen zur therapeutischen verwendung. |
| US4410520A (en) * | 1981-11-09 | 1983-10-18 | Ciba-Geigy Corporation | 3-Amino-[1]-benzazepin-2-one-1-alkanoic acids |
| US4575503A (en) * | 1983-02-10 | 1986-03-11 | Ciba-Geigy Corporation | 3-Amino-[1]-benzazepin-2-one-1-alkanoic acids |
| ES2247193T3 (es) * | 2000-10-31 | 2006-03-01 | Ciba Specialty Chemicals Holding Inc. | Formas cristalinas del fluvastatin sodico. |
| CN100338028C (zh) * | 2000-10-31 | 2007-09-19 | 山道士有限公司 | 盐酸文拉法辛的晶形 |
| WO2002050036A1 (en) * | 2000-12-21 | 2002-06-27 | Ciba Speciality Chemicals Holding Inc. | Crystalline forms of cerivastatin sodium |
| CA2454072A1 (en) * | 2001-08-03 | 2003-02-20 | Paul Adriaan Van Der Schaaf | Crystalline forms of fluvastatin sodium |
-
2003
- 2003-07-17 AU AU2003250086A patent/AU2003250086A1/en not_active Abandoned
- 2003-07-17 EP EP03766204A patent/EP1525189A1/en not_active Withdrawn
- 2003-07-17 WO PCT/EP2003/007771 patent/WO2004013105A1/en not_active Ceased
- 2003-07-17 JP JP2004525233A patent/JP2006500337A/ja not_active Withdrawn
- 2003-07-17 CA CA002492949A patent/CA2492949A1/en not_active Abandoned
- 2003-07-17 US US10/500,910 patent/US20050107359A1/en not_active Abandoned
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2014506919A (ja) * | 2011-07-12 | 2014-03-20 | サムジン ファーマシューティカル カンパニー，リミテッド | クロピドグレル硫酸水素塩の球状粒子、これを含む薬学的組成物及びその製造方法 |
Also Published As
| Publication number | Publication date |
|---|---|
| AU2003250086A1 (en) | 2004-02-23 |
| WO2004013105A1 (en) | 2004-02-12 |
| EP1525189A1 (en) | 2005-04-27 |
| CA2492949A1 (en) | 2004-02-12 |
| US20050107359A1 (en) | 2005-05-19 |
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