JP2005523268A - グルココルチコイドおよびβ２−アドレナリン受容体アゴニストを含む吸入用製剤 - Google Patents
グルココルチコイドおよびβ２−アドレナリン受容体アゴニストを含む吸入用製剤 Download PDFInfo
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- JP2005523268A JP2005523268A JP2003565457A JP2003565457A JP2005523268A JP 2005523268 A JP2005523268 A JP 2005523268A JP 2003565457 A JP2003565457 A JP 2003565457A JP 2003565457 A JP2003565457 A JP 2003565457A JP 2005523268 A JP2005523268 A JP 2005523268A
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/007—Pulmonary tract; Aromatherapy
- A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
- A61K9/0075—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/18—Sulfonamides
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
- A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/007—Pulmonary tract; Aromatherapy
- A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
- A61K9/008—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy comprising drug dissolved or suspended in liquid propellant for inhalation via a pressurized metered dose inhaler [MDI]
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
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- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
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- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Pulmonology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Otolaryngology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Immunology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US10/066,961 US6537983B1 (en) | 2001-04-07 | 2002-02-04 | Anti-inflammatory androstane derivatives |
| PCT/GB2003/000485 WO2003066033A1 (en) | 2002-02-04 | 2003-02-04 | Formulation for inhalation comprising a glucocorticoid and a beta 2-adrenoreceptor agonist |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2005523268A true JP2005523268A (ja) | 2005-08-04 |
| JP2005523268A5 JP2005523268A5 (enExample) | 2006-01-05 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003565457A Withdrawn JP2005523268A (ja) | 2002-02-04 | 2003-02-04 | グルココルチコイドおよびβ２−アドレナリン受容体アゴニストを含む吸入用製剤 |
Country Status (7)
| Country | Link |
|---|---|
| EP (1) | EP1471895B2 (enExample) |
| JP (1) | JP2005523268A (enExample) |
| AT (1) | ATE396716T1 (enExample) |
| AU (1) | AU2003205855A1 (enExample) |
| DE (1) | DE60321311D1 (enExample) |
| ES (1) | ES2305438T5 (enExample) |
| WO (1) | WO2003066033A1 (enExample) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2005527496A (ja) * | 2002-02-04 | 2005-09-15 | グラクソ グループ リミテッド | 炎症状態およびアレルギー状態の治療のためのアンドロスタン誘導体およびβ２−アドレナリン受容体を含む吸入投与用の医薬製剤 |
| JP2013542940A (ja) * | 2010-10-12 | 2013-11-28 | シプラ・リミテッド | 医薬組成物 |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2389530B (en) | 2002-06-14 | 2007-01-10 | Cipla Ltd | Pharmaceutical compositions |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL95590A (en) † | 1989-09-08 | 1996-06-18 | Glaxo Group Ltd | Medicinal preparations containing Salmetrol and Pluticasone Propionate |
| GB9903759D0 (en) † | 1999-02-18 | 1999-04-14 | Novartis Ag | Organic compounds |
| CA2417826A1 (en) * | 2000-08-05 | 2002-02-14 | Glaxo Group Limited | 17.beta.-carbothioate 17.alpha.-arylcarbonyloxyloxy androstane derivative as anti-inflammatory agents |
| GB0103630D0 (en) * | 2001-02-14 | 2001-03-28 | Glaxo Group Ltd | Chemical compounds |
| WO2002070490A1 (en) * | 2001-03-08 | 2002-09-12 | Glaxo Group Limited | Agonists of beta-adrenoceptors |
| EP1370521B1 (en) * | 2001-03-22 | 2007-12-19 | Glaxo Group Limited | Formanilide derivatives as beta2-adrenoreceptor agonists |
| UA77656C2 (en) † | 2001-04-07 | 2007-01-15 | Glaxo Group Ltd | S-fluoromethyl ester of 6-alpha, 9-alpha-difluoro-17-alpha-[(2-furanylcarbonyl)oxy]-11-beta-hydroxy-16- alpha-methyl-3-oxoandrosta-1,4-dien-17-beta-carbothioacid as anti-inflammatory agent |
-
2003
- 2003-02-04 EP EP03702732A patent/EP1471895B2/en not_active Expired - Lifetime
- 2003-02-04 AU AU2003205855A patent/AU2003205855A1/en not_active Abandoned
- 2003-02-04 AT AT03702732T patent/ATE396716T1/de not_active IP Right Cessation
- 2003-02-04 DE DE60321311T patent/DE60321311D1/de not_active Expired - Lifetime
- 2003-02-04 ES ES03702732T patent/ES2305438T5/es not_active Expired - Lifetime
- 2003-02-04 JP JP2003565457A patent/JP2005523268A/ja not_active Withdrawn
- 2003-02-04 WO PCT/GB2003/000485 patent/WO2003066033A1/en not_active Ceased
Cited By (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2005527496A (ja) * | 2002-02-04 | 2005-09-15 | グラクソ グループ リミテッド | 炎症状態およびアレルギー状態の治療のためのアンドロスタン誘導体およびβ２−アドレナリン受容体を含む吸入投与用の医薬製剤 |
| JP2013542940A (ja) * | 2010-10-12 | 2013-11-28 | シプラ・リミテッド | 医薬組成物 |
| JP2017039746A (ja) * | 2010-10-12 | 2017-02-23 | シプラ・リミテッド | 医薬組成物 |
| US10179139B2 (en) | 2010-10-12 | 2019-01-15 | Cipla Limited | Pharmaceutical composition |
Also Published As
| Publication number | Publication date |
|---|---|
| EP1471895A1 (en) | 2004-11-03 |
| ES2305438T3 (es) | 2008-11-01 |
| WO2003066033A1 (en) | 2003-08-14 |
| ATE396716T1 (de) | 2008-06-15 |
| AU2003205855A1 (en) | 2003-09-02 |
| DE60321311D1 (de) | 2008-07-10 |
| ES2305438T5 (es) | 2012-06-05 |
| EP1471895B1 (en) | 2008-05-28 |
| EP1471895B2 (en) | 2012-03-14 |
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