JP2005516004A5 - - Google Patents

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Publication number
JP2005516004A5
JP2005516004A5 JP2003550776A JP2003550776A JP2005516004A5 JP 2005516004 A5 JP2005516004 A5 JP 2005516004A5 JP 2003550776 A JP2003550776 A JP 2003550776A JP 2003550776 A JP2003550776 A JP 2003550776A JP 2005516004 A5 JP2005516004 A5 JP 2005516004A5
Authority
JP
Japan
Prior art keywords
pharmaceutical composition
receptor
affinity
composition according
agonist
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2003550776A
Other languages
English (en)
Japanese (ja)
Other versions
JP2005516004A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2002/039310 external-priority patent/WO2003049727A1/en
Publication of JP2005516004A publication Critical patent/JP2005516004A/ja
Publication of JP2005516004A5 publication Critical patent/JP2005516004A5/ja
Pending legal-status Critical Current

Links

JP2003550776A 2001-12-07 2002-12-09 新形成の治療 Pending JP2005516004A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US33673201P 2001-12-07 2001-12-07
PCT/US2002/039310 WO2003049727A1 (en) 2001-12-07 2002-12-09 Treatment of neoplasia

Publications (2)

Publication Number Publication Date
JP2005516004A JP2005516004A (ja) 2005-06-02
JP2005516004A5 true JP2005516004A5 (enExample) 2006-02-02

Family

ID=23317407

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2003550776A Pending JP2005516004A (ja) 2001-12-07 2002-12-09 新形成の治療

Country Status (6)

Country Link
US (1) US20040259936A1 (enExample)
EP (1) EP1461027A4 (enExample)
JP (1) JP2005516004A (enExample)
AU (1) AU2002357114B2 (enExample)
CA (1) CA2468794A1 (enExample)
WO (1) WO2003049727A1 (enExample)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7632955B2 (en) * 2001-12-13 2009-12-15 National Health Research Institutes Indole compounds
US7528165B2 (en) * 2001-12-13 2009-05-05 National Health Research Institutes Indole compounds
WO2005023232A2 (en) * 2003-09-04 2005-03-17 Affibody Ab Therapeutic, screening and diagnostic methods based on the effect of cb1 receptor modulation on lymphoproliferative disorders.
EP1736775A4 (en) * 2004-04-12 2008-03-12 Takeda Pharmaceutical NEW LIGAND OF A G-PROTEIN-COUPLED RECEPTOR PROTEIN AND USE THEREOF
TWI360539B (en) 2004-10-28 2012-03-21 Shionogi & Co 3-carbamoyl-2-pyridone derivatives
US7456289B2 (en) * 2004-12-31 2008-11-25 National Health Research Institutes Anti-tumor compounds
MX2009005071A (es) * 2006-11-13 2009-05-25 Novartis Ag Compuestos de pirazol y triazol sustituidos como inhibidores de ksp.
EP2470508A1 (en) 2009-08-28 2012-07-04 Arena Pharmaceuticals, Inc. Cannabinoid receptor modulators
CA2789151A1 (en) 2010-02-08 2011-08-11 Allergan, Inc. Pyridazine derivatives useful as cannabinoid-2 agonists
US9597340B2 (en) 2011-02-25 2017-03-21 Arena Pharmaceuticals, Inc. Cannabinoid receptor modulators
MX392150B (es) 2011-02-25 2025-03-21 Arena Pharm Inc Moduladores de receptores canabinoides.
JP5945554B2 (ja) 2011-02-25 2016-07-05 アリーナ ファーマシューティカルズ, インコーポレイテッド 縮合型アザ環の結晶形およびその調製プロセス(カンナビノイド受容体モジュレーター)
WO2016085941A1 (en) 2014-11-25 2016-06-02 Arena Pharmaceuticals, Inc. Processes for the preparation of cannabinoid receptor modulators
CN114096241A (zh) * 2019-05-16 2022-02-25 技术研究及发展基金有限公司 大麻素及其用途
CN115282279B (zh) * 2022-08-08 2024-03-12 暨南大学附属第一医院(广州华侨医院) CNR2通过介导DCs成熟及功能作为脓毒症急性肺损伤治疗靶点的应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1271266B (it) * 1994-12-14 1997-05-27 Valle Francesco Della Impiego terapeutico di ammidi di acidi mono e bicarbossilici con amminoalcoli,selettivamente attive sul recettore periferico dei cannabinoidi
FR2735774B1 (fr) * 1995-06-21 1997-09-12 Sanofi Sa Utilisation de composes agonistes du recepteur cb2 humain pour la preparation de medicaments immunomodulateurs, nouveaux composes agonistes du recepteur cb2 et les compositions pharmaceutiques les contenant
CA2340444A1 (en) * 1998-05-04 1999-11-11 The University Of Connecticut Cannabinoids selective for the cb2 receptor
CA2387892A1 (en) * 1999-10-18 2001-04-26 University Of Connecticut Pyrazole derivatives as cannabinoid receptor antagonists
FR2800372B1 (fr) * 1999-11-03 2001-12-07 Sanofi Synthelabo Derives tricycliques d'acide 1-benzylpyrazole-3- carboxylique, leur preparation, les medicaments en contenant
JP2004502642A (ja) * 2000-02-11 2004-01-29 ブリストル−マイヤーズ スクイブ カンパニー カンナビノイドレセプターモジュレーター、それらの製造方法、および呼吸系および非呼吸系疾患の処置のためのカンナビノイドレセプターモジュレーターの使用

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