JP2005507878A5 - - Google Patents

Download PDF

Info

Publication number
JP2005507878A5
JP2005507878A5 JP2003526920A JP2003526920A JP2005507878A5 JP 2005507878 A5 JP2005507878 A5 JP 2005507878A5 JP 2003526920 A JP2003526920 A JP 2003526920A JP 2003526920 A JP2003526920 A JP 2003526920A JP 2005507878 A5 JP2005507878 A5 JP 2005507878A5
Authority
JP
Japan
Prior art keywords
cyclopentylamino
pyrimidinyl
pyridin
cyclopentyl
amine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2003526920A
Other languages
English (en)
Japanese (ja)
Other versions
JP2005507878A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2002/027251 external-priority patent/WO2003022845A1/en
Publication of JP2005507878A publication Critical patent/JP2005507878A/ja
Publication of JP2005507878A5 publication Critical patent/JP2005507878A5/ja
Pending legal-status Critical Current

Links

JP2003526920A 2001-09-07 2002-08-27 ヘルペス感染症を治療するためのピラゾロ−ピリジン類 Pending JP2005507878A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US31820301P 2001-09-07 2001-09-07
PCT/US2002/027251 WO2003022845A1 (en) 2001-09-07 2002-08-27 Pyrazolo-pyridines for the treatment of herpes infections

Publications (2)

Publication Number Publication Date
JP2005507878A JP2005507878A (ja) 2005-03-24
JP2005507878A5 true JP2005507878A5 (cg-RX-API-DMAC7.html) 2005-11-17

Family

ID=23237109

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2003526920A Pending JP2005507878A (ja) 2001-09-07 2002-08-27 ヘルペス感染症を治療するためのピラゾロ−ピリジン類

Country Status (7)

Country Link
US (1) US20040214834A1 (cg-RX-API-DMAC7.html)
EP (1) EP1423389B1 (cg-RX-API-DMAC7.html)
JP (1) JP2005507878A (cg-RX-API-DMAC7.html)
AT (1) ATE364043T1 (cg-RX-API-DMAC7.html)
DE (1) DE60220525T2 (cg-RX-API-DMAC7.html)
ES (1) ES2286272T3 (cg-RX-API-DMAC7.html)
WO (1) WO2003022845A1 (cg-RX-API-DMAC7.html)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2005525382A (ja) 2002-03-07 2005-08-25 スミスクライン ビーチャム コーポレーション ピラゾロピリミジンおよびピラゾロトリアジン誘導体ならびにそれを含む医薬組成物
US20070155738A1 (en) 2005-05-20 2007-07-05 Alantos Pharmaceuticals, Inc. Heterobicyclic metalloprotease inhibitors
UA103319C2 (en) 2008-05-06 2013-10-10 Глаксосмитклайн Ллк Thiazole- and oxazole-benzene sulfonamide compounds
EP2402335A1 (en) 2010-06-29 2012-01-04 Basf Se Pyrazolopyridine compounds
EP2402336A1 (en) 2010-06-29 2012-01-04 Basf Se Pyrazolopyridine compounds
WO2017070089A1 (en) 2015-10-19 2017-04-27 Incyte Corporation Heterocyclic compounds as immunomodulators
US20170145025A1 (en) 2015-11-19 2017-05-25 Incyte Corporation Heterocyclic compounds as immunomodulators
LT3394033T (lt) 2015-12-22 2021-03-10 Incyte Corporation Heterocikliniai junginiai, kaip imunomoduliatoriai
US20170320875A1 (en) 2016-05-06 2017-11-09 Incyte Corporation Heterocyclic compounds as immunomodulators
US20170342060A1 (en) 2016-05-26 2017-11-30 Incyte Corporation Heterocyclic compounds as immunomodulators
HRP20221030T1 (hr) 2016-06-20 2022-11-11 Incyte Corporation Heterociklički spojevi kao imunomodulatori
WO2018013789A1 (en) 2016-07-14 2018-01-18 Incyte Corporation Heterocyclic compounds as immunomodulators
MA46045A (fr) 2016-08-29 2021-04-28 Incyte Corp Composés hétérocycliques utilisés comme immunomodulateurs
WO2018119236A1 (en) 2016-12-22 2018-06-28 Incyte Corporation Triazolo[1,5-a]pyridine derivatives as immunomodulators
JP7149276B2 (ja) 2016-12-22 2022-10-06 インサイト・コーポレイション Pd-l1内在化誘導物質としてのテトラヒドロイミダゾ[4,5-c]ピリジン誘導体
BR112019012993A2 (pt) 2016-12-22 2019-12-03 Incyte Corporation derivados de benzo-oxazol como imunomoduladores
EP3558963B1 (en) 2016-12-22 2022-03-23 Incyte Corporation Bicyclic heteroaromatic compounds as immunomodulators
WO2018119221A1 (en) 2016-12-22 2018-06-28 Incyte Corporation Pyridine derivatives as immunomodulators
MY210070A (en) 2018-03-30 2025-08-25 Incyte Corp Heterocyclic compounds as immunomodulators
PT3790877T (pt) 2018-05-11 2023-05-10 Incyte Corp Derivados de tetrahidro-imidazo[4,5-c]piridina como imunomoduladores pd-l1
TW202115059A (zh) 2019-08-09 2021-04-16 美商英塞特公司 Pd—1/pd—l1抑制劑之鹽
BR112022005826A2 (pt) 2019-09-30 2022-06-21 Incyte Corp Compostos de pirido[3,2-d]pirimidina como imunomoduladores
BR112022009031A2 (pt) 2019-11-11 2022-10-11 Incyte Corp Sais e formas cristalinas de um inibidor de pd-1/pd-l1
TW202233615A (zh) 2020-11-06 2022-09-01 美商英塞特公司 Pd—1/pd—l1抑制劑之結晶形式
WO2022099018A1 (en) 2020-11-06 2022-05-12 Incyte Corporation Process of preparing a pd-1/pd-l1 inhibitor
MX2023005362A (es) 2020-11-06 2023-06-22 Incyte Corp Proceso para hacer un inhibidor de proteina de muerte programada 1 (pd-1)/ligando de muerte programada 1 (pd-l1) y sales y formas cristalinas del mismo.

Family Cites Families (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0151962A3 (en) * 1984-01-25 1985-10-02 Beecham Group Plc Pyrazolopyridine derivatives
GB8404584D0 (en) * 1984-02-22 1984-03-28 Beecham Group Plc Compounds
GB8404586D0 (en) * 1984-02-22 1984-03-28 Beecham Group Plc Compounds
US4925849A (en) * 1987-06-15 1990-05-15 Fujisawa Pharmaceutical Company, Ltd. Pharmaceutically useful pyrazolopyridines
US5155114A (en) * 1989-01-23 1992-10-13 Fujisawa Pharmaceutical Company, Ltd. Method of treatment using pyrazolopyridine compound
GB8901423D0 (en) * 1989-01-23 1989-03-15 Fujisawa Pharmaceutical Co Pyrazolopyridine compound and processes for preparation thereof
AU622330B2 (en) * 1989-06-23 1992-04-02 Takeda Chemical Industries Ltd. Condensed heterocyclic compounds having a nitrogen atom in the bridgehead for use as fungicides
GB9015764D0 (en) * 1990-07-18 1990-09-05 Fujisawa Pharmaceutical Co Pyrazolopyridine compound and processes for preparation thereof
GB9107513D0 (en) * 1991-04-10 1991-05-29 Fujisawa Pharmaceutical Co Pyrazolopyridine compound and processes for preparation thereof
US5300478A (en) * 1993-01-28 1994-04-05 Zeneca Limited Substituted fused pyrazolo compounds
US5552422A (en) * 1995-01-11 1996-09-03 Merck Frosst Canada, Inc. Aryl substituted 5,5 fused aromatic nitrogen compounds as anti-inflammatory agents
US5700816A (en) * 1995-06-12 1997-12-23 Isakson; Peter C. Treatment of inflammation and inflammation-related disorders with a combination of a cyclooxygenase-2 inhibitor and a leukotriene A4 hydrolase inhibitor
CA2224517A1 (en) * 1995-06-12 1996-12-27 G.D. Searle & Co. Compositions comprising a cyclooxygenase-2 inhibitor and a 5-lipoxygenase inhibitor
FR2757166B1 (fr) * 1996-12-12 1999-01-29 Rhone Poulenc Rorer Sa Derives du pyrrole, leur preparation et les compositions pharmaceutiques qui les contiennent
US20020156104A1 (en) * 1997-06-13 2002-10-24 Jerry L. Adams Novel pyrazole and pyrazoline substituted compounds
NZ511349A (en) * 1998-11-03 2003-10-31 Glaxo Group Ltd Pyrazolopyridine derivatives useful as selective COX-2 inhibitors
ES2216631T3 (es) * 1999-02-27 2004-10-16 Glaxo Group Limited Pirazolpiridinas.
ES2245380T3 (es) * 2000-12-15 2006-01-01 Glaxo Group Limited Pirazolopiridinas.
DE60112330T2 (de) * 2000-12-15 2006-04-13 Glaxo Group Ltd., Greenford Pyrazolopyridinderivate
US7153855B2 (en) * 2001-03-08 2006-12-26 Smithkline Beecham Corporation Pyrazolopyridinyl pyrimidine therapeutic compounds
EP1372642A1 (en) * 2001-03-30 2004-01-02 SmithKline Beecham Corporation Use of pyrazolopyridines as therapeutic compounds
ATE332301T1 (de) * 2001-04-10 2006-07-15 Smithkline Beecham Corp Antivirale pyrazolopyridin verbindungen
US6962914B2 (en) * 2001-04-27 2005-11-08 Smithkline Beecham Corporation Pyrazolopyridinyl pyridine and pyrimidine therapeutic compounds

Similar Documents

Publication Publication Date Title
JP2005507878A5 (cg-RX-API-DMAC7.html)
JP2005508955A5 (cg-RX-API-DMAC7.html)
CA2446435A1 (en) 4-amino-5-phenyl-7-cyclobutyl-pyrrolo[2,3-d]pyrimidine derivatives
RU94013439A (ru) Гетероциклические соединения, способ их получения, фармацевтическая композиция и способ лечения
GB0211649D0 (en) Organic compounds
GB9104890D0 (en) Compositions
HUP0203437A3 (en) Use of resorcinol derivatives for producing pharmaceutical compositions for treatment of immune diseases
WO2005023759A3 (en) Heterocyclic inhibitors of mek and methods of use thereof
WO2005005414A3 (en) Pyrazolyl-indole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
MY142019A (en) Pyrazolo-quinazoline derivatives, process for their preparation and their use as kinase inhibitors
HUP0104867A3 (en) Heterocyclic compounds useful in the treatment of inflammatory diseases, process for their preparation, pharmaceutical compositions comprising thereof and their use
PT1235826E (pt) Acrilamidas de quinuclidina
HUP0200493A3 (en) Pharmaceutical compositions comprising sulphonyl-amino-carbonyl derivatives for the treatment of nuclear factor-kappa b mediated diseases
EE200200211A (et) Bitsüklilised aminohapped kui farmatseutilised toimeained
EE04854B1 (et) Oksabispidiinühendid, nende valmistamise meetod ning ravimvorm kasutamiseks südame arütmia raviks ja profülaktikaks
JP2002510633A5 (cg-RX-API-DMAC7.html)
BRPI0413438A (pt) derivados de pirimidilpirrol ativos como inibidores de cinase
JP2004517098A5 (cg-RX-API-DMAC7.html)
GB2285219A (en) Use of norastemizole for the treatment of allergic disorders
MY148125A (en) Compounds
HUP0002963A3 (en) Use of pyrazolo-[4,3-d] pyrimidinon derivatives for the production of pharmaceutical compositions for treating diseases of the eye field
PL356932A1 (en) Pyrrole-type compounds, compositions, and methods for treating cancer or viral diseases
AU7731700A (en) Low dose ifn-gamma for treatment of disease
IL146133A0 (en) Preparations for the application of anti-inflammatory agents
SE9902935D0 (sv) Pharmaceutical compositions