JP2001524931A5 - - Google Patents
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- Publication number
- JP2001524931A5 JP2001524931A5 JP1998508118A JP50811898A JP2001524931A5 JP 2001524931 A5 JP2001524931 A5 JP 2001524931A5 JP 1998508118 A JP1998508118 A JP 1998508118A JP 50811898 A JP50811898 A JP 50811898A JP 2001524931 A5 JP2001524931 A5 JP 2001524931A5
- Authority
- JP
- Japan
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (9)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US69242096A | 1996-08-05 | 1996-08-05 | |
| US08/692,420 | 1996-08-05 | ||
| US72507396A | 1996-10-02 | 1996-10-02 | |
| US08/725,073 | 1996-10-02 | ||
| US79791597A | 1997-02-10 | 1997-02-10 | |
| US08/797,915 | 1997-02-10 | ||
| US4706797P | 1997-05-19 | 1997-05-19 | |
| US60/047,067 | 1997-05-19 | ||
| PCT/US1997/013622 WO1998005333A1 (en) | 1996-08-05 | 1997-08-05 | Use of beta-sheet mimetics as protease and kinase inhibitors and as inhibitors of transcription factors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2001524931A JP2001524931A (ja) | 2001-12-04 |
| JP2001524931A5 true JP2001524931A5 (https=) | 2005-04-07 |
Family
ID=27489127
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP50811898A Pending JP2001524931A (ja) | 1996-08-05 | 1997-08-05 | プロテアーゼおよびキナーゼのインヒビターとしてならびに転写因子のインヒビターとしてのβシート模倣物の使用 |
Country Status (11)
| Country | Link |
|---|---|
| EP (1) | EP0915700B1 (https=) |
| JP (1) | JP2001524931A (https=) |
| KR (1) | KR20000029838A (https=) |
| AT (1) | ATE320811T1 (https=) |
| AU (1) | AU732174B2 (https=) |
| CA (1) | CA2262900A1 (https=) |
| DE (1) | DE69735545T2 (https=) |
| ES (1) | ES2262184T3 (https=) |
| NO (1) | NO990522L (https=) |
| NZ (1) | NZ334227A (https=) |
| WO (1) | WO1998005333A1 (https=) |
Families Citing this family (26)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6184223B1 (en) | 1995-10-27 | 2001-02-06 | Molecumetics Ltd. | Reverse-turn mimetics and methods relating thereto |
| DE69810513T2 (de) * | 1998-02-12 | 2004-03-18 | Molecumetics, Ltd., Bellevue | Mimetika von beta-faltblatt und verfahren zur verwendung davon |
| US6323219B1 (en) | 1998-04-02 | 2001-11-27 | Ortho-Mcneil Pharmaceutical, Inc. | Methods for treating immunomediated inflammatory disorders |
| US8106094B2 (en) | 1998-07-06 | 2012-01-31 | Johnson & Johnson Consumer Companies, Inc. | Compositions and methods for treating skin conditions |
| US8093293B2 (en) | 1998-07-06 | 2012-01-10 | Johnson & Johnson Consumer Companies, Inc. | Methods for treating skin conditions |
| WO2000038683A1 (en) | 1998-12-23 | 2000-07-06 | Du Pont Pharmaceuticals Company | THROMBIN OR FACTOR Xa INHIBITORS |
| CZ20012722A3 (cs) | 1999-01-27 | 2002-08-14 | Ortho-Mcneil Pharmaceutical, Inc. | Peptidylové heterocyklické ketony pouľitelné jako inhibitory typtasy |
| US7309688B2 (en) | 2000-10-27 | 2007-12-18 | Johnson & Johnson Consumer Companies | Topical anti-cancer compositions and methods of use thereof |
| US7253169B2 (en) | 1999-11-12 | 2007-08-07 | Gliamed, Inc. | Aza compounds, pharmaceutical compositions and methods of use |
| US6417189B1 (en) * | 1999-11-12 | 2002-07-09 | Gpi Nil Holdings, Inc. | AZA compounds, pharmaceutical compositions and methods of use |
| EP1261611A2 (en) * | 2000-02-29 | 2002-12-04 | Bristol-Myers Squibb Pharma Company | Inhibitors of hepatitis c virus ns3 protease |
| US8431550B2 (en) | 2000-10-27 | 2013-04-30 | Johnson & Johnson Consumer Companies, Inc. | Topical anti-cancer compositions and methods of use thereof |
| DE10100053A1 (de) * | 2001-01-02 | 2002-08-22 | Keyneurotek Ag I G | Verwendung von Enzyminhibitoren der Dipeptidylpeptidase IV sowie der Aminopeptidase N und pharmazeutischen Zubereitungen daraus zur Prävention und/oder Therapie Ischämie-bedingter akuter und chronischer neurodegenerativer Prozesse und Erkrankungen |
| US7192615B2 (en) | 2001-02-28 | 2007-03-20 | J&J Consumer Companies, Inc. | Compositions containing legume products |
| US8080657B2 (en) | 2001-10-12 | 2011-12-20 | Choongwae Pharma Corporation | Compounds of reverse turn mimetics and the use thereof |
| US7671054B1 (en) | 2001-10-12 | 2010-03-02 | Choongwae Pharma Corporation | Reverse-turn mimetics and method relating thereto |
| US7576084B2 (en) | 2001-10-12 | 2009-08-18 | Choongwae Pharma Corporation | Reverse-turn mimetics and method relating thereto |
| US7232822B2 (en) | 2001-10-12 | 2007-06-19 | Choongwae Pharma Corporation | Reverse-turn mimetics and method relating thereto |
| US7566711B2 (en) | 2001-10-12 | 2009-07-28 | Choongwae Pharma Corporation | Reverse-turn mimetics and method relating thereto |
| WO2003055856A2 (en) | 2001-10-17 | 2003-07-10 | Bristol-Myers Squibb Company | BICYCLIC LACTAM DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES AND/OR TNF-α CONVERTING ENZYME (TACE) |
| TWI286476B (en) * | 2001-12-12 | 2007-09-11 | Tibotec Pharm Ltd | Combination of cytochrome P450 dependent protease inhibitors |
| CA2502644A1 (en) | 2002-10-17 | 2004-04-29 | Myriad Genetics, Inc. | Reverse-turn mimetics and composition and methods relating thereto |
| CN102906566A (zh) * | 2010-02-03 | 2013-01-30 | 株式会社棱镜生物实验室 | 与天然变性蛋白质结合的化合物及其筛选方法 |
| MX378266B (es) | 2014-10-06 | 2025-03-10 | Lighthouse Pharmaceuticals Inc | Inhibidores de gingipaina de lisina. |
| CN108602787A (zh) | 2015-11-09 | 2018-09-28 | 库特克希米公司 | 精氨酸牙龈卟啉菌蛋白酶的抑制剂 |
| CN109983012B (zh) | 2016-09-16 | 2023-12-01 | 莱特豪斯制药公司 | 赖氨酸牙龈蛋白酶的酮抑制剂 |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1600880A (en) * | 1978-05-23 | 1981-10-21 | Lilly Industries Ltd | Pharmaceutical compositions comprising hydantoin derivatives |
| IL60617A0 (en) * | 1979-07-23 | 1980-09-16 | Sparamedica Ag | Triazolopyridazine derivative,their preparation and pharmaceutical compositions containing them |
| US4594431A (en) * | 1983-08-01 | 1986-06-10 | Eli Lilly Company | Octahydroindolizinepropanoic acids and related compounds as enzyme inhibitors |
| JPH0676373B2 (ja) * | 1985-12-27 | 1994-09-28 | エーザイ株式会社 | グアニジノ安息香酸エステル誘導体 |
| AU653024B2 (en) * | 1991-05-30 | 1994-09-15 | Novartis Ag | Substituted diaminophthalimides and analogues |
| US5463063A (en) * | 1993-07-02 | 1995-10-31 | Celgene Corporation | Ring closure of N-phthaloylglutamines |
| US5716929A (en) * | 1994-06-17 | 1998-02-10 | Vertex Pharmaceuticals, Inc. | Inhibitors of interleukin-1β converting enzyme |
| AP9701004A0 (en) * | 1994-12-22 | 1997-07-31 | Iaf Biochem Int | Low molecular weight bicyclic thrombin inhibitors. |
| HU226558B1 (en) * | 1994-12-30 | 2009-03-30 | Celgene Corp | Immunotherapeutic imides/amides and their use for reducing levels of tnfalpha |
| JPH10508034A (ja) * | 1995-03-24 | 1998-08-04 | モレキュメティックス リミテッド | βシート模倣物および生物学的に活性なペプチドまたはタンパク質のインヒビターとしてのその使用 |
| WO1996030396A1 (en) * | 1995-03-24 | 1996-10-03 | Molecumetics Ltd. | β-SHEET MIMETICS AND USE THEREOF AS PROTEASE INHIBITORS |
| IT1277405B1 (it) * | 1995-08-01 | 1997-11-10 | Menarini Farma Ind | Derivati di lattami biciclici come inibitori della trombina |
-
1997
- 1997-08-05 NZ NZ334227A patent/NZ334227A/xx not_active IP Right Cessation
- 1997-08-05 AT AT97936371T patent/ATE320811T1/de not_active IP Right Cessation
- 1997-08-05 EP EP97936371A patent/EP0915700B1/en not_active Expired - Lifetime
- 1997-08-05 ES ES97936371T patent/ES2262184T3/es not_active Expired - Lifetime
- 1997-08-05 AU AU39058/97A patent/AU732174B2/en not_active Ceased
- 1997-08-05 WO PCT/US1997/013622 patent/WO1998005333A1/en not_active Ceased
- 1997-08-05 CA CA002262900A patent/CA2262900A1/en not_active Abandoned
- 1997-08-05 KR KR1019997000994A patent/KR20000029838A/ko not_active Ceased
- 1997-08-05 DE DE69735545T patent/DE69735545T2/de not_active Expired - Lifetime
- 1997-08-05 JP JP50811898A patent/JP2001524931A/ja active Pending
-
1999
- 1999-02-04 NO NO990522A patent/NO990522L/no unknown