JP2000514456A5 - - Google Patents

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Publication number
JP2000514456A5
JP2000514456A5 JP1998506095A JP50609598A JP2000514456A5 JP 2000514456 A5 JP2000514456 A5 JP 2000514456A5 JP 1998506095 A JP1998506095 A JP 1998506095A JP 50609598 A JP50609598 A JP 50609598A JP 2000514456 A5 JP2000514456 A5 JP 2000514456A5
Authority
JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
JP1998506095A
Other languages
English (en)
Japanese (ja)
Other versions
JP2000514456A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US1997/011845 external-priority patent/WO1998002436A1/en
Publication of JP2000514456A publication Critical patent/JP2000514456A/ja
Publication of JP2000514456A5 publication Critical patent/JP2000514456A5/ja
Ceased legal-status Critical Current

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JP10506095A 1996-07-15 1997-07-08 ファルネシルプロテイントランスフェラーゼのチアジオキソベンゾジアゼピン阻害剤 Ceased JP2000514456A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US2178696P 1996-07-15 1996-07-15
US60/021,786 1996-07-15
PCT/US1997/011845 WO1998002436A1 (en) 1996-07-15 1997-07-08 Thiadioxobenzodiazepine inhibitors of farnesyl protein transferase

Publications (2)

Publication Number Publication Date
JP2000514456A JP2000514456A (ja) 2000-10-31
JP2000514456A5 true JP2000514456A5 (cg-RX-API-DMAC10.html) 2005-02-10

Family

ID=21806140

Family Applications (1)

Application Number Title Priority Date Filing Date
JP10506095A Ceased JP2000514456A (ja) 1996-07-15 1997-07-08 ファルネシルプロテイントランスフェラーゼのチアジオキソベンゾジアゼピン阻害剤

Country Status (6)

Country Link
US (1) US6624157B2 (cg-RX-API-DMAC10.html)
EP (1) EP0918771A4 (cg-RX-API-DMAC10.html)
JP (1) JP2000514456A (cg-RX-API-DMAC10.html)
AU (1) AU709409B2 (cg-RX-API-DMAC10.html)
CA (1) CA2260216A1 (cg-RX-API-DMAC10.html)
WO (1) WO1998002436A1 (cg-RX-API-DMAC10.html)

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US8293769B2 (en) 2007-05-21 2012-10-23 Novartis Ag CSF-1R inhibitors, compositions, and methods of use
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WO2010057006A1 (en) 2008-11-13 2010-05-20 Link Medicine Corporation Azaquinolinone derivatives and uses thereof
US8691825B2 (en) 2009-04-01 2014-04-08 Merck Sharp & Dohme Corp. Inhibitors of AKT activity
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US8765747B2 (en) 2009-06-12 2014-07-01 Dana-Farber Cancer Institute, Inc. Fused 2-aminothiazole compounds
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US9180127B2 (en) 2009-12-29 2015-11-10 Dana-Farber Cancer Institute, Inc. Type II Raf kinase inhibitors
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US8999957B2 (en) 2010-06-24 2015-04-07 Merck Sharp & Dohme Corp. Heterocyclic compounds as ERK inhibitors
EP2601293B1 (en) 2010-08-02 2017-12-06 Sirna Therapeutics, Inc. RNA INTERFERENCE MEDIATED INHIBITION OF CATENIN (CADHERIN-ASSOCIATED PROTEIN), BETA 1 (CTNNB1) GENE EXPRESSION USING SHORT INTERFERING NUCLEIC ACID (siNA)
CN103282497B (zh) 2010-08-17 2018-07-10 瑟纳治疗公司 使用短干扰核酸(siNA)的乙型肝炎病毒(HBV)基因表达的RNA干扰介导的抑制
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US11993602B2 (en) 2018-08-07 2024-05-28 Merck Sharp & Dohme Llc PRMT5 inhibitors
US11981701B2 (en) 2018-08-07 2024-05-14 Merck Sharp & Dohme Llc PRMT5 inhibitors
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JP7660063B2 (ja) 2018-12-28 2025-04-10 ダナ-ファーバー キャンサー インスティテュート, インコーポレイテッド サイクリン依存性キナーゼ7のインヒビターおよびそれらの使用
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US20240325409A1 (en) * 2023-02-27 2024-10-03 Enanta Pharmaceuticals, Inc. Fused Heterotetracyclic Antiviral Agents
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Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2920385B2 (ja) * 1988-08-18 1999-07-19 武田薬品工業株式会社 1,2,5‐ベンゾチアジアゼピン誘導体,その製造法および用途
JPH02111766A (ja) * 1988-10-20 1990-04-24 Taiho Yakuhin Kogyo Kk ベンゾチアジアゼピン誘導体及びその塩
AU6909194A (en) * 1993-05-14 1994-12-12 Board Of Regents, The University Of Texas System Preparation of n-cyanodithioimino-carbonates and 3-mercapto-5-amino-1h-1,2,4-triazole
US6011029A (en) * 1996-02-26 2000-01-04 Bristol-Myers Squibb Company Inhibitors of farnesyl protein transferase
US6156746A (en) * 1998-08-25 2000-12-05 Bristol-Myers Squibb Company 1,2,5-benzothiadiazepine-1,1-dioxides with n-2 imidazolylalkyl substituents

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