ITMI20030312A1 - Derivati di acidi 2-fenil-2-alchil-acetici per il trattamento della malattia di alzheimer. - Google Patents

Derivati di acidi 2-fenil-2-alchil-acetici per il trattamento della malattia di alzheimer.

Info

Publication number
ITMI20030312A1
ITMI20030312A1 IT000312A ITMI20030312A ITMI20030312A1 IT MI20030312 A1 ITMI20030312 A1 IT MI20030312A1 IT 000312 A IT000312 A IT 000312A IT MI20030312 A ITMI20030312 A IT MI20030312A IT MI20030312 A1 ITMI20030312 A1 IT MI20030312A1
Authority
IT
Italy
Prior art keywords
alchyl
fenyl
derivatives
treatment
alzheimer disease
Prior art date
Application number
IT000312A
Other languages
English (en)
Inventor
Bruno Pietro Imbimbo
Ilaria Peretto
Stefano Radaelli
Luca Raveglia
Andrea Rizzi
Gino Villetti
Original Assignee
Chiesi Farma Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chiesi Farma Spa filed Critical Chiesi Farma Spa
Priority to IT000312A priority Critical patent/ITMI20030312A1/it
Priority to PCT/EP2004/001595 priority patent/WO2004073705A1/en
Publication of ITMI20030312A1 publication Critical patent/ITMI20030312A1/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D257/00Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
    • C07D257/02Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D257/04Five-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C57/00Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms
    • C07C57/52Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms containing halogen
    • C07C57/58Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms containing halogen containing six-membered aromatic rings
IT000312A 2003-02-21 2003-02-21 Derivati di acidi 2-fenil-2-alchil-acetici per il trattamento della malattia di alzheimer. ITMI20030312A1 (it)

Priority Applications (2)

Application Number Priority Date Filing Date Title
IT000312A ITMI20030312A1 (it) 2003-02-21 2003-02-21 Derivati di acidi 2-fenil-2-alchil-acetici per il trattamento della malattia di alzheimer.
PCT/EP2004/001595 WO2004073705A1 (en) 2003-02-21 2004-02-19 1-phenyl-2- monoalkyl carboxylic acid derivatives for the treatment of neurodegenerative diseases

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT000312A ITMI20030312A1 (it) 2003-02-21 2003-02-21 Derivati di acidi 2-fenil-2-alchil-acetici per il trattamento della malattia di alzheimer.

Publications (1)

Publication Number Publication Date
ITMI20030312A1 true ITMI20030312A1 (it) 2004-08-22

Family

ID=32894162

Family Applications (1)

Application Number Title Priority Date Filing Date
IT000312A ITMI20030312A1 (it) 2003-02-21 2003-02-21 Derivati di acidi 2-fenil-2-alchil-acetici per il trattamento della malattia di alzheimer.

Country Status (2)

Country Link
IT (1) ITMI20030312A1 (it)
WO (1) WO2004073705A1 (it)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005110963A1 (en) * 2004-05-19 2005-11-24 Cellzome Ag (biphenyl-3-yl)-carboxylic acids and derivatives thereof and their use in therapy
EP1604970A1 (en) * 2004-05-19 2005-12-14 Cellzome Ag 2-(Biphenyl-3-yl)-carboxylic acids of gamma-secretase-modulating activity
EP1650183A1 (en) * 2004-10-21 2006-04-26 Cellzome Ag (Benzyloxy-biphenyl) acetic acids and derivatives thereof and their use in therapy
US20110040094A1 (en) * 2007-09-14 2011-02-17 Envivo Pharmaceuticals, Inc. 1,3,4-trisubstituted benzenes
CA2742897A1 (en) 2008-11-06 2010-05-14 Astrazeneca Ab Modulators of amyloid beta.
BR112012026803A2 (pt) 2010-04-21 2016-07-12 Chiesi Farma Spa composto
DK3004080T3 (da) 2013-06-04 2019-01-02 Acturum Real Estate Ab Triazolforbindelser og deres anvendelse som gamma-sekretase-modulatorer
JP6368776B2 (ja) 2013-06-04 2018-08-01 アクチュラム・ライフ・サイエンス・アクチエボラーグ トリアゾール化合物およびガンマセクレターゼモジュレーターとしてのその使用
NO3004079T3 (it) 2013-06-04 2018-06-16

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5994379A (en) * 1998-02-13 1999-11-30 Merck Frosst Canada, Inc. Bisaryl COX-2 inhibiting compounds, compositions and methods of use
DE19907895A1 (de) * 1999-02-24 2000-11-16 Paz Arzneimittelentwicklung Verwendung von R-Arylpropionsäuren zur Herstellung von Arzneimitteln zur Behandlung von Erkrankungen bei Mensch und Tier, welche durch die Hemmung der Aktivierung von NF-kB therapeutisch beeinflußt werden können
CA2406383A1 (en) * 2000-04-13 2001-10-25 Mayo Foundation For Medical Education And Research A.beta.42 lowering agents

Also Published As

Publication number Publication date
WO2004073705A1 (en) 2004-09-02

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