IT8522645A0 - ENANTIOMERS OF PHENOXY DERIVATIVES OF BENZYLMORPHOLINE AND THEIR SALTS. - Google Patents
ENANTIOMERS OF PHENOXY DERIVATIVES OF BENZYLMORPHOLINE AND THEIR SALTS.Info
- Publication number
- IT8522645A0 IT8522645A0 IT8522645A IT2264585A IT8522645A0 IT 8522645 A0 IT8522645 A0 IT 8522645A0 IT 8522645 A IT8522645 A IT 8522645A IT 2264585 A IT2264585 A IT 2264585A IT 8522645 A0 IT8522645 A0 IT 8522645A0
- Authority
- IT
- Italy
- Prior art keywords
- benzylmorpholine
- enantiomers
- salts
- phenoxy derivatives
- phenoxy
- Prior art date
Links
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical compound C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 title 1
- -1 PHENOXY DERIVATIVES OF BENZYLMORPHOLINE Chemical class 0.000 title 1
- 150000003839 salts Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
- C07D265/30—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB08429546A GB2167407B (en) | 1984-11-22 | 1984-11-22 | Enantiomers of phenoxy derivatives of benzyl morpholine and salts thereof |
Publications (2)
Publication Number | Publication Date |
---|---|
IT8522645A0 true IT8522645A0 (en) | 1985-10-29 |
IT1190420B IT1190420B (en) | 1988-02-16 |
Family
ID=10570118
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IT22645/85A IT1190420B (en) | 1984-11-22 | 1985-10-29 | BENZYLMORPHOLINE-DERIVED PHENOXY-BASED ENANTIOMERS AND THEIR SALTS |
Country Status (5)
Country | Link |
---|---|
JP (1) | JPH0667916B2 (en) |
DE (1) | DE3540093A1 (en) |
FR (1) | FR2573425B1 (en) |
GB (1) | GB2167407B (en) |
IT (1) | IT1190420B (en) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IT1305322B1 (en) | 1998-04-23 | 2001-05-04 | Pharmacia & Upjohn Spa | Use of reboxetine for treating obsessive compulsive disorder and panic disorder |
EP1459749B1 (en) * | 1999-07-01 | 2005-10-05 | Pharmacia & Upjohn Company LLC | (S,S)-reboxetine for treating incontinence |
DK1632234T3 (en) | 1999-07-01 | 2007-09-17 | Pharmacia & Upjohn Co Llc | (S, S) reboxetine for the treatment of chronic fatigue syndrome |
CO5210862A1 (en) | 1999-09-15 | 2002-10-30 | Alza Corp | DOSAGE FORMS AND METHODS TO PROVIDE REBOXETINE EFFECTIVE THERAPY WITH DOSAGE ONCE A DAY |
CN101298440A (en) * | 2002-06-17 | 2008-11-05 | 辉瑞意大利公司 | Pharmaceutical salts of reboxetine |
ES2315525T3 (en) | 2002-08-23 | 2009-04-01 | Eli Lilly And Company | DERIVATIVES OF 2- (PHENYLTIOMETIL) -MORFOLINE FOR USE AS SELECTIVE INHIBITORS OF NOREPINEFRINE RECAPTATION. |
ATE327982T1 (en) | 2002-08-23 | 2006-06-15 | Lilly Co Eli | BENZYLMORPHOLINE DERIVATIVES |
GB0219687D0 (en) | 2002-08-23 | 2002-10-02 | Lilly Co Eli | Benzyl morpholine derivatives |
GB0319793D0 (en) | 2003-08-22 | 2003-09-24 | Lilly Co Eli | Pyridinylmorpholine derivatives |
WO2005053663A2 (en) * | 2003-11-24 | 2005-06-16 | Eli Lilly And Company | Norepinephrine reuptake inhibitors useful for treatment of cognitive failure |
AU2004305563C1 (en) | 2003-12-11 | 2011-07-07 | Sunovion Pharmaceuticals Inc. | Combination of a sedative and a neurotransmitter modulator, and methods for improving sleep quality and treating depression |
CA2556063A1 (en) * | 2004-02-20 | 2005-09-09 | Pharmacia & Upjohn Company Llc | Method for the preparation of aryl ethers |
WO2005082869A1 (en) * | 2004-02-20 | 2005-09-09 | Pharmacia & Upjohn Company Llc | Method for the preparation of aryl ethers |
GB0409744D0 (en) * | 2004-04-30 | 2004-06-09 | Pfizer Ltd | Novel compounds |
BRPI0510453A (en) * | 2004-04-30 | 2007-10-30 | Warner Lambert Co | Substituted Morpholine Compounds for the Treatment of Central Nervous System Disorders |
EP2076508B1 (en) | 2006-10-18 | 2011-01-05 | Pfizer Products Inc. | Biaryl ether urea compounds |
US20100069389A1 (en) * | 2008-09-06 | 2010-03-18 | Bionevia Pharmaceuticals, Inc. | Novel forms of reboxetine |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL56369A (en) * | 1978-01-20 | 1984-05-31 | Erba Farmitalia | Alpha-phenoxybenzyl propanolamine derivatives,their preparation and pharmaceutical compositions comprising them |
-
1984
- 1984-11-22 GB GB08429546A patent/GB2167407B/en not_active Expired
-
1985
- 1985-10-29 IT IT22645/85A patent/IT1190420B/en active
- 1985-11-12 DE DE19853540093 patent/DE3540093A1/en not_active Withdrawn
- 1985-11-20 JP JP60258816A patent/JPH0667916B2/en not_active Expired - Lifetime
- 1985-11-22 FR FR8517324A patent/FR2573425B1/en not_active Expired
Also Published As
Publication number | Publication date |
---|---|
IT1190420B (en) | 1988-02-16 |
JPH0667916B2 (en) | 1994-08-31 |
FR2573425A1 (en) | 1986-05-23 |
GB8429546D0 (en) | 1985-01-03 |
GB2167407A (en) | 1986-05-29 |
FR2573425B1 (en) | 1988-12-23 |
JPS61129174A (en) | 1986-06-17 |
GB2167407B (en) | 1988-05-11 |
DE3540093A1 (en) | 1986-05-28 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
TA | Fee payment date (situation as of event date), data collected since 19931001 |
Effective date: 19971024 |