IT1397233B1 - Procedimento migliorativo per la sintesi del mono-acetil ganciclovir, intermedio chiave per la sintesi del valganciclovir. - Google Patents

Procedimento migliorativo per la sintesi del mono-acetil ganciclovir, intermedio chiave per la sintesi del valganciclovir.

Info

Publication number
IT1397233B1
IT1397233B1 ITMI2010A000006A ITMI20100006A IT1397233B1 IT 1397233 B1 IT1397233 B1 IT 1397233B1 IT MI2010A000006 A ITMI2010A000006 A IT MI2010A000006A IT MI20100006 A ITMI20100006 A IT MI20100006A IT 1397233 B1 IT1397233 B1 IT 1397233B1
Authority
IT
Italy
Prior art keywords
synthesis
acetil
valganciclovir
ganciclovir
mono
Prior art date
Application number
ITMI2010A000006A
Other languages
English (en)
Inventor
Emilio Vecchio
Claudio Fuganti
Original Assignee
Fidia Farmaceutici
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fidia Farmaceutici filed Critical Fidia Farmaceutici
Priority to ITMI2010A000006A priority Critical patent/IT1397233B1/it
Publication of ITMI20100006A1 publication Critical patent/ITMI20100006A1/it
Application granted granted Critical
Publication of IT1397233B1 publication Critical patent/IT1397233B1/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/18Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 one oxygen and one nitrogen atom, e.g. guanine

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ITMI2010A000006A 2010-01-08 2010-01-08 Procedimento migliorativo per la sintesi del mono-acetil ganciclovir, intermedio chiave per la sintesi del valganciclovir. IT1397233B1 (it)

Priority Applications (1)

Application Number Priority Date Filing Date Title
ITMI2010A000006A IT1397233B1 (it) 2010-01-08 2010-01-08 Procedimento migliorativo per la sintesi del mono-acetil ganciclovir, intermedio chiave per la sintesi del valganciclovir.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ITMI2010A000006A IT1397233B1 (it) 2010-01-08 2010-01-08 Procedimento migliorativo per la sintesi del mono-acetil ganciclovir, intermedio chiave per la sintesi del valganciclovir.

Publications (2)

Publication Number Publication Date
ITMI20100006A1 ITMI20100006A1 (it) 2011-07-09
IT1397233B1 true IT1397233B1 (it) 2013-01-04

Family

ID=42135919

Family Applications (1)

Application Number Title Priority Date Filing Date
ITMI2010A000006A IT1397233B1 (it) 2010-01-08 2010-01-08 Procedimento migliorativo per la sintesi del mono-acetil ganciclovir, intermedio chiave per la sintesi del valganciclovir.

Country Status (1)

Country Link
IT (1) IT1397233B1 (it)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN108373471A (zh) * 2018-04-29 2018-08-07 安徽海康药业有限责任公司 一种高纯度单乙酰更昔洛韦的合成方法
CN108383840A (zh) * 2018-04-29 2018-08-10 安徽海康药业有限责任公司 一种制备高纯度单乙酰更昔洛韦的方法
CN108503641A (zh) * 2018-04-29 2018-09-07 安徽海康药业有限责任公司 一种合成高纯度单乙酰更昔洛韦的方法
CN108503642A (zh) * 2018-04-29 2018-09-07 安徽海康药业有限责任公司 一种高纯度单乙酰更昔洛韦的制备方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5840890A (en) * 1996-01-26 1998-11-24 Syntex (U.S.A.) Inc. Process for preparing a 2-(2-amino-1,6-dihydro-6-oxo-purin-9-yl)methoxy-1,3-propanediol derivative

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN108373471A (zh) * 2018-04-29 2018-08-07 安徽海康药业有限责任公司 一种高纯度单乙酰更昔洛韦的合成方法
CN108383840A (zh) * 2018-04-29 2018-08-10 安徽海康药业有限责任公司 一种制备高纯度单乙酰更昔洛韦的方法
CN108503641A (zh) * 2018-04-29 2018-09-07 安徽海康药业有限责任公司 一种合成高纯度单乙酰更昔洛韦的方法
CN108503642A (zh) * 2018-04-29 2018-09-07 安徽海康药业有限责任公司 一种高纯度单乙酰更昔洛韦的制备方法

Also Published As

Publication number Publication date
ITMI20100006A1 (it) 2011-07-09

Similar Documents

Publication Publication Date Title
SMT201600216B (it) Ottaidropirrolo[3,4.c]pirroli disostituiti come modulatori del recettore di orexina
IT1403054B1 (it) Bottiglia.
IT1398484B1 (it) Dilatatore anatomico nasale.
IT1400982B1 (it) Collirio osmotico trans-epiteliale per la cura del cheratocono.
IT1402748B1 (it) Procedimento per la raffinazione del greggio
DK2241698T3 (da) Slagfast, forsænket loft
IT1393136B1 (it) Procedimento per la preparazione del bosentan
IT1398317B1 (it) Nuovo procedimento per la preparazione del dronedarone.
DK2618842T3 (da) Hidtil ukendt immunstimulerende fremgangsmåde
IT1398636B1 (it) Regolatore del getto
IT1397233B1 (it) Procedimento migliorativo per la sintesi del mono-acetil ganciclovir, intermedio chiave per la sintesi del valganciclovir.
DE112011104051A5 (de) Kombi-Radsatzpresse
ITTO20110857A1 (it) Procedimento per la produzione di cicloesanonossina.
IT1403438B1 (it) Rivestimento del manubrio.
IT1400666B1 (it) Procedimento per la sintesi di 5-amino, 1-fenil, 3-ciano, 4-trifluorometil sulfinil pirazoli.
IT1401345B1 (it) Bomboletta.
IT1397547B1 (it) Complessi azoturo dissimmetrici monocationici del tecnezio
FI20115978A (fi) Lukkojärjestely
ITRM20090257A1 (it) Trocar.
IT1404226B1 (it) Procedimento per la produzione di fibrocemento ecologico, fibrocemento ottenuto e suoi impieghi.
ES1079005Y (es) Carreton.
IT1398862B1 (it) Cerniera per occhiali, del tipo flex
IT1401800B1 (it) Astuccio telescopico, particolarmente per occhiali.
IT1403232B1 (it) Pannello del tipo sandwich e procedimento per la produzione di un siffatto pannello.
IT1398929B1 (it) Procedimento per la produzione di vetri stratificati.