IT1394407B1 - Procedimento per la preparazione di fosinopril e suoi intermedi - Google Patents
Procedimento per la preparazione di fosinopril e suoi intermediInfo
- Publication number
- IT1394407B1 IT1394407B1 ITMI2009A000918A ITMI20090918A IT1394407B1 IT 1394407 B1 IT1394407 B1 IT 1394407B1 IT MI2009A000918 A ITMI2009A000918 A IT MI2009A000918A IT MI20090918 A ITMI20090918 A IT MI20090918A IT 1394407 B1 IT1394407 B1 IT 1394407B1
- Authority
- IT
- Italy
- Prior art keywords
- fosinopril
- intermediates
- procedure
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic System
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/30—Phosphinic acids R2P(=O)(OH); Thiophosphinic acids, i.e. R2P(=X)(XH) (X = S, Se)
- C07F9/32—Esters thereof
- C07F9/3258—Esters thereof the ester moiety containing a substituent or a structure which is considered as characteristic
- C07F9/3264—Esters with hydroxyalkyl compounds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic System
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/30—Phosphinic acids R2P(=O)(OH); Thiophosphinic acids, i.e. R2P(=X)(XH) (X = S, Se)
- C07F9/306—Arylalkanephosphinic acids, e.g. Ar-(CH2)n-P(=X)(R)(XH), (X = O,S, Se; n>=1)
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic System
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
- C07F9/572—Five-membered rings
Priority Applications (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ITMI2009A000918A IT1394407B1 (it) | 2009-05-25 | 2009-05-25 | Procedimento per la preparazione di fosinopril e suoi intermedi |
| EP10158731A EP2264039A1 (en) | 2009-05-25 | 2010-03-31 | Process for the preparation of fosinopril and intermediates thereof |
| US12/785,746 US20100297711A1 (en) | 2009-05-25 | 2010-05-24 | Process for the synthesis of fosinopril and intermediates thereof |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ITMI2009A000918A IT1394407B1 (it) | 2009-05-25 | 2009-05-25 | Procedimento per la preparazione di fosinopril e suoi intermedi |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ITMI20090918A1 ITMI20090918A1 (it) | 2010-11-26 |
| IT1394407B1 true IT1394407B1 (it) | 2012-06-15 |
Family
ID=41467076
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ITMI2009A000918A IT1394407B1 (it) | 2009-05-25 | 2009-05-25 | Procedimento per la preparazione di fosinopril e suoi intermedi |
Country Status (3)
| Country | Link |
|---|---|
| US (1) | US20100297711A1 (it) |
| EP (1) | EP2264039A1 (it) |
| IT (1) | IT1394407B1 (it) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1406151B1 (it) * | 2010-12-06 | 2014-02-14 | Dipharma Francis Srl | Procedimento per la preparazione di fosinopril e suoi intermedi |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4337201A (en) | 1980-12-04 | 1982-06-29 | E. R. Squibb & Sons, Inc. | Phosphinylalkanoyl substituted prolines |
| US4912231A (en) | 1987-06-15 | 1990-03-27 | E. R. Squibb & Sons, Inc. | Process for preparing (trans)-4-phenyl-L-proline derivatives |
| US4873356A (en) * | 1987-09-30 | 1989-10-10 | E. R. Squibb & Sons, Inc. | Method for preparing phosphinic acids used in preparing ace inhibitors and intermediates produced thereby |
| US4937355A (en) | 1989-01-17 | 1990-06-26 | E. R. Squibb & Sons, Inc. | Process for preparing (trans)-4-substituted-dl-proline derivatives |
| US5008399A (en) | 1990-01-19 | 1991-04-16 | E. R. Squibb & Sons, Inc. | Diastereoselective preparation of phosphinate esters |
| US6426354B1 (en) * | 1998-04-23 | 2002-07-30 | Novartis Ag | Certain heteroaryl substituted thiol inhibitors of endothelin-converting enzyme |
| EP1290208B1 (en) * | 2000-06-01 | 2010-10-13 | SK Holdings Co., Ltd. | Method for optically resolving a racemic alpha-substituted heterocyclic carboxylic acid using enzyme |
| WO2004094452A2 (en) * | 2003-04-16 | 2004-11-04 | Bristol-Myers Squibb Company | Macrocyclic isoquinoline peptide inhibitors of hepatitis c virus |
| CN100497335C (zh) * | 2005-10-27 | 2009-06-10 | 上海医药工业研究院 | 取代氧膦基乙酸的光学拆分方法 |
| CN100488969C (zh) * | 2005-10-27 | 2009-05-20 | 上海医药工业研究院 | 光学活性的取代氧膦基乙酸盐及其用途 |
-
2009
- 2009-05-25 IT ITMI2009A000918A patent/IT1394407B1/it active
-
2010
- 2010-03-31 EP EP10158731A patent/EP2264039A1/en not_active Withdrawn
- 2010-05-24 US US12/785,746 patent/US20100297711A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| ITMI20090918A1 (it) | 2010-11-26 |
| EP2264039A1 (en) | 2010-12-22 |
| US20100297711A1 (en) | 2010-11-25 |
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