IT1262990B - Derivati peptidici, loro preparazione e loro impiego come medicamenti,in particolare antagonisti dell'lh-rh - Google Patents
Derivati peptidici, loro preparazione e loro impiego come medicamenti,in particolare antagonisti dell'lh-rhInfo
- Publication number
- IT1262990B IT1262990B ITRM920677A ITRM920677A IT1262990B IT 1262990 B IT1262990 B IT 1262990B IT RM920677 A ITRM920677 A IT RM920677A IT RM920677 A ITRM920677 A IT RM920677A IT 1262990 B IT1262990 B IT 1262990B
- Authority
- IT
- Italy
- Prior art keywords
- drugs
- peptide derivatives
- antagonists
- preparation
- compounds
- Prior art date
Links
- 239000003814 drug Substances 0.000 title abstract 2
- 229940079593 drug Drugs 0.000 title abstract 2
- 108090000765 processed proteins & peptides Proteins 0.000 title abstract 2
- 101000904177 Clupea pallasii Gonadoliberin-1 Proteins 0.000 title 1
- 239000000579 Gonadotropin-Releasing Hormone Substances 0.000 title 1
- 101000857870 Squalus acanthias Gonadoliberin Proteins 0.000 title 1
- 239000005557 antagonist Substances 0.000 title 1
- XLXSAKCOAKORKW-AQJXLSMYSA-N gonadorelin Chemical compound C([C@@H](C(=O)NCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N1[C@@H](CCC1)C(=O)NCC(N)=O)NC(=O)[C@H](CO)NC(=O)[C@H](CC=1C2=CC=CC=C2NC=1)NC(=O)[C@H](CC=1N=CNC=1)NC(=O)[C@H]1NC(=O)CC1)C1=CC=C(O)C=C1 XLXSAKCOAKORKW-AQJXLSMYSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- 125000003277 amino group Chemical group 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 150000002170 ethers Chemical class 0.000 abstract 1
- 239000002474 gonadorelin antagonist Substances 0.000 abstract 1
- 150000002431 hydrogen Chemical class 0.000 abstract 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
Landscapes
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
L'invenzione riguarda derivati peptidici di un antagonista dell'LH-RH e comprendenti, legato ad un gruppo ammino di questi composti, almeno a) un resto glucidico o b) un resto di formula (b1) o (b2) (FORMULA b1 o b2) in cui uno dei simboli Yi e Y2 significa l'idrogeno e l'altro un gruppo idrossi, oppure ambedue significano l'idrogeno, f ed g significano ciascuno indipendentemente 0 o 1, e gli eteri fisiologicamente accettabili e gli esteri fisiologicamente idrolizzabili e fisiologicamente accettabili di questi composti c) una qualsiasi combinazione di a) e b), Questi composti possono venire impiegati come medicamenti.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ITRM920677A IT1262990B (it) | 1992-09-16 | 1992-09-16 | Derivati peptidici, loro preparazione e loro impiego come medicamenti,in particolare antagonisti dell'lh-rh |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ITRM920677A IT1262990B (it) | 1992-09-16 | 1992-09-16 | Derivati peptidici, loro preparazione e loro impiego come medicamenti,in particolare antagonisti dell'lh-rh |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| ITRM920677A0 ITRM920677A0 (it) | 1992-09-16 |
| ITRM920677A1 ITRM920677A1 (it) | 1994-03-16 |
| IT1262990B true IT1262990B (it) | 1996-07-23 |
Family
ID=11401191
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ITRM920677A IT1262990B (it) | 1992-09-16 | 1992-09-16 | Derivati peptidici, loro preparazione e loro impiego come medicamenti,in particolare antagonisti dell'lh-rh |
Country Status (1)
| Country | Link |
|---|---|
| IT (1) | IT1262990B (it) |
-
1992
- 1992-09-16 IT ITRM920677A patent/IT1262990B/it active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| ITRM920677A1 (it) | 1994-03-16 |
| ITRM920677A0 (it) | 1992-09-16 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| NZ244021A (en) | Benzylthiazolidinedione derivatives, preparation and pharmaceutical compositions thereof | |
| NZ232853A (en) | Heterocyclyl-substituted-fluorobenzoyl derivatives and pharmaceutical compositions | |
| ZA948670B (en) | New benzoyl guanidine derivatives,the preparation thereof and their use in pharmaceutical compositions | |
| AU2337197A (en) | Cinnamic acid derivatives and their use as integrin antagonists | |
| NZ247201A (en) | Substituted sulphonylamido- or sulphonamidocarbonyl-pyridine-2-carboxamide derivatives and pharmaceutical compositions | |
| IL108520A0 (en) | Imidazopyridine derivatives, processes for the preparation thereof, and pharmaceutical compositions containing them | |
| AU7535798A (en) | Novel cyclosporin derivatives, preparation and pharmaceutical compositions containing same | |
| IE901862L (en) | Inclusion compound of imipramine | |
| GR3023516T3 (en) | Stable hydrated cephalosporin dry powder for oral suspension formulation. | |
| DE69317877D1 (en) | 4''-deoxyerythromycinderivate | |
| IL102814A0 (en) | Pyrazine derivatives,their preparation and pharmaceutical compositions comprising them | |
| GB9424766D0 (en) | Pharmaceutical composition | |
| IL96636A0 (en) | Piperidine derivatives and pharmaceutical compositions containing them | |
| DE3369983D1 (en) | Isoquinoline derivatives, process for their preparation, pharmaceutical compositions containing them and their use | |
| TW252979B (it) | ||
| IL114968A (en) | 1,4-dihydropyridine compounds and pharmaceutical compositions containing them | |
| IT1262990B (it) | Derivati peptidici, loro preparazione e loro impiego come medicamenti,in particolare antagonisti dell'lh-rh | |
| IL66960A0 (en) | 4-phenyl-quinazoline derivatives,their preparation and pharmaceutical compositions containing them | |
| TW261605B (it) | ||
| ES2091570T3 (es) | Nuevos derivados peptidicos antagonistas de la bradiquidina, su procedimiento de preparacion y composiciones farmaceuticas que los contienen. | |
| GR3023941T3 (en) | Cyclic derivatives of angiopeptin, their preparation and their pharmaceutical compositions. | |
| GR1002385B (el) | Καθαρη μορφη στρεπτογραμινων, παρασκευη αυτης και φαρμακευτικες συνθεσεις που την περιεχουν. | |
| ES8605819A1 (es) | Procedimiento de preparacion de nuevos derivados nucleosidos. | |
| ES2007745A6 (es) | Proceddimiento de preparacion de nuevos derivados triazoles ciclicos condensados. | |
| HU901631D0 (en) | Process for the preparation of thienyl-piperazine derivatives and pharmaceutical compositions containing them |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 0001 | Granted |