IT1195267B - Derivati teofillinmetildiossolanici,procedimento per la loro preparazione e relative composizioni farmaceutiche - Google Patents

Derivati teofillinmetildiossolanici,procedimento per la loro preparazione e relative composizioni farmaceutiche

Info

Publication number
IT1195267B
IT1195267B IT21370/80A IT2137080A IT1195267B IT 1195267 B IT1195267 B IT 1195267B IT 21370/80 A IT21370/80 A IT 21370/80A IT 2137080 A IT2137080 A IT 2137080A IT 1195267 B IT1195267 B IT 1195267B
Authority
IT
Italy
Prior art keywords
theofillinmethylsoxananic
derivatives
procedure
preparation
pharmaceutical compositions
Prior art date
Application number
IT21370/80A
Other languages
English (en)
Italian (it)
Other versions
IT8021370A0 (it
Inventor
Ugo Chiodoni
Jose Sebastian Franzone
Silvano Spinelli
Original Assignee
Abc Ist Biolog Chem Spa
Unibios Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abc Ist Biolog Chem Spa, Unibios Spa filed Critical Abc Ist Biolog Chem Spa
Priority to IT21370/80A priority Critical patent/IT1195267B/it
Publication of IT8021370A0 publication Critical patent/IT8021370A0/it
Priority to US06/251,485 priority patent/US4378359A/en
Priority to FR8107075A priority patent/FR2480286A1/fr
Priority to DE19813114130 priority patent/DE3114130A1/de
Priority to GB8111536A priority patent/GB2078717B/en
Priority to JP56056896A priority patent/JPS5827796B2/ja
Priority to BE0/204481A priority patent/BE888417A/fr
Application granted granted Critical
Publication of IT1195267B publication Critical patent/IT1195267B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
    • C07D473/06Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
    • C07D473/08Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3 with methyl radicals in positions 1 and 3, e.g. theophylline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/14Antitussive agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IT21370/80A 1980-04-15 1980-04-15 Derivati teofillinmetildiossolanici,procedimento per la loro preparazione e relative composizioni farmaceutiche IT1195267B (it)

Priority Applications (7)

Application Number Priority Date Filing Date Title
IT21370/80A IT1195267B (it) 1980-04-15 1980-04-15 Derivati teofillinmetildiossolanici,procedimento per la loro preparazione e relative composizioni farmaceutiche
US06/251,485 US4378359A (en) 1980-04-15 1981-04-06 Theophyllinylmethyldioxolane derivatives, methods for their preparation and pharmaceutical compositions containing them
FR8107075A FR2480286A1 (fr) 1980-04-15 1981-04-08 Nouveaux derives de theophyllinylmethyldioxolane, leurs procedes de preparation et leur application en therapeutique
DE19813114130 DE3114130A1 (de) 1980-04-15 1981-04-08 Neue theophyllinylmethyldioxolan-derivate, verfahren zu ihrer herstellung und sie enthaltende pharmazeutische ansaetze
GB8111536A GB2078717B (en) 1980-04-15 1981-04-13 Theophyllinyl methyl dioxolanes
JP56056896A JPS5827796B2 (ja) 1980-04-15 1981-04-14 テオフイリニルメチルジオキソラン誘導体およびその製法
BE0/204481A BE888417A (fr) 1980-04-15 1981-04-14 Nouveaux derives de theophyllinylmethyldioxolane, leur procedes de preparation et leur application en therapeutique,

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT21370/80A IT1195267B (it) 1980-04-15 1980-04-15 Derivati teofillinmetildiossolanici,procedimento per la loro preparazione e relative composizioni farmaceutiche

Publications (2)

Publication Number Publication Date
IT8021370A0 IT8021370A0 (it) 1980-04-15
IT1195267B true IT1195267B (it) 1988-10-12

Family

ID=11180793

Family Applications (1)

Application Number Title Priority Date Filing Date
IT21370/80A IT1195267B (it) 1980-04-15 1980-04-15 Derivati teofillinmetildiossolanici,procedimento per la loro preparazione e relative composizioni farmaceutiche

Country Status (7)

Country Link
US (1) US4378359A (enExample)
JP (1) JPS5827796B2 (enExample)
BE (1) BE888417A (enExample)
DE (1) DE3114130A1 (enExample)
FR (1) FR2480286A1 (enExample)
GB (1) GB2078717B (enExample)
IT (1) IT1195267B (enExample)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3138397A1 (de) * 1981-09-26 1983-04-07 Hoechst Ag, 6230 Frankfurt "arzneimittel, darin enthaltene vicinale dihydroxyalkylxanthine und herstellungsverfahren fuer diese xanthinverbindungen"
HU190377B (en) * 1982-03-12 1986-08-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing theophyllinyl-alkyl-oxadiazoles
EP0171005B1 (en) * 1984-07-27 1989-11-23 BOEHRINGER BIOCHEMIA ROBIN S.p.A. Xanthinylmethylthiazolidines, process for their preparation and pharmaceutical compositions containing them
IT1197516B (it) * 1986-12-24 1988-11-30 Abc Ist Biolog Chem Spa Derivati teofillinmetilanici e teofillinmetilditianici procedimento per la loro preparazione e composizioni farmaceutiche che li comprendono
HU198933B (en) * 1987-11-02 1989-12-28 Chinoin Gyogyszer Es Vegyeszet Process for producing new xanthine derivatives and pharmaceutical compositions comprising same as active ingredient
JP2500277B2 (ja) * 1990-11-27 1996-05-29 三井東圧化学株式会社 フェノ―ル系樹脂パイプの押出成型方法および装置
US5786360A (en) 1996-11-19 1998-07-28 Link Technology Incorporated A1 adenosine receptor antagonists
WO2004074247A2 (en) 2003-02-19 2004-09-02 Endacea, Inc. A1 adenosine receptor antagonists
EP1636229A4 (en) * 2003-06-06 2008-07-30 Endacea Inc ADENOSINE A1 RECEPTOR ANTAGONISTS
EP1636230A4 (en) * 2003-06-09 2010-06-16 Endacea Inc ADENOSINE A1 RECEPTOR ANTAGONISTS

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2761861A (en) * 1953-09-11 1956-09-04 Hoffmann La Roche Process for the manufacture of novel xanthine bases and salts thereof
US2840559A (en) * 1954-06-22 1958-06-24 Krantz Jr Nuclearly substituted 8-theophyllines and method of making the same
FR1523273A (fr) * 1967-03-13 1968-05-03 Soc Ind Fab Antibiotiques Sifa Nouveaux dérivés de théophylline et procédé de préparation
GB1289287A (enExample) * 1969-03-28 1972-09-13
IT1113122B (it) * 1978-04-06 1986-01-20 Abc Ist Biolog Chem Spa Composizione farmaceutica ad attivita' antibrocospastica e antitosse

Also Published As

Publication number Publication date
GB2078717A (en) 1982-01-13
IT8021370A0 (it) 1980-04-15
BE888417A (fr) 1981-07-31
FR2480286B1 (enExample) 1984-03-30
GB2078717B (en) 1984-02-15
JPS56164191A (en) 1981-12-17
DE3114130A1 (de) 1982-01-28
JPS5827796B2 (ja) 1983-06-11
US4378359A (en) 1983-03-29
FR2480286A1 (fr) 1981-10-16

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