IT1176770B - DERIVATIVES OF BENZOSSAZOLONE AND BENZOTIAZOLONE PRO CEDIMENTS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOUND THAT CONTAINS THEM - Google Patents
DERIVATIVES OF BENZOSSAZOLONE AND BENZOTIAZOLONE PRO CEDIMENTS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOUND THAT CONTAINS THEMInfo
- Publication number
- IT1176770B IT1176770B IT2278584A IT2278584A IT1176770B IT 1176770 B IT1176770 B IT 1176770B IT 2278584 A IT2278584 A IT 2278584A IT 2278584 A IT2278584 A IT 2278584A IT 1176770 B IT1176770 B IT 1176770B
- Authority
- IT
- Italy
- Prior art keywords
- cediments
- benzotiazolone
- benzossazolone
- pro
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
- C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
- C07D263/58—Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB838325370A GB8325370D0 (en) | 1983-09-22 | 1983-09-22 | Benzoxazoline and benzothiazoline derivatives |
Publications (3)
Publication Number | Publication Date |
---|---|
IT8422785A0 IT8422785A0 (en) | 1984-09-21 |
IT8422785A1 IT8422785A1 (en) | 1986-03-21 |
IT1176770B true IT1176770B (en) | 1987-08-18 |
Family
ID=10549143
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IT2278584A IT1176770B (en) | 1983-09-22 | 1984-09-21 | DERIVATIVES OF BENZOSSAZOLONE AND BENZOTIAZOLONE PRO CEDIMENTS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOUND THAT CONTAINS THEM |
Country Status (4)
Country | Link |
---|---|
AU (1) | AU3431784A (en) |
GB (1) | GB8325370D0 (en) |
IT (1) | IT1176770B (en) |
WO (1) | WO1985001289A1 (en) |
Cited By (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2010129596A1 (en) * | 2009-05-04 | 2010-11-11 | Agios Pharmaceuticals, Inc. | Pmk2 modulators for use in the treatment of cancer |
US8742119B2 (en) | 2009-04-06 | 2014-06-03 | Agios Pharmaceuticals, Inc. | Pyruvate kinase M2 modulators, therapeutic compositions and related methods of use |
US8889667B2 (en) | 2010-12-29 | 2014-11-18 | Agios Pharmaceuticals, Inc | Therapeutic compounds and compositions |
US9115086B2 (en) | 2009-06-29 | 2015-08-25 | Agios Pharmaceuticals, Inc. | Therapeutic compositions and related methods of use |
US9181231B2 (en) | 2011-05-03 | 2015-11-10 | Agios Pharmaceuticals, Inc | Pyruvate kinase activators for use for increasing lifetime of the red blood cells and treating anemia |
US9221792B2 (en) | 2010-12-17 | 2015-12-29 | Agios Pharmaceuticals, Inc | N-(4-(azetidine-1-carbonyl) phenyl)-(hetero-) arylsulfonamide derivatives as pyruvate kinase M2 (PMK2) modulators |
US9328077B2 (en) | 2010-12-21 | 2016-05-03 | Agios Pharmaceuticals, Inc | Bicyclic PKM2 activators |
US9365545B2 (en) | 2013-03-15 | 2016-06-14 | Agios Pharmaceuticals, Inc | Therapeutic compounds and compositions |
US9980961B2 (en) | 2011-05-03 | 2018-05-29 | Agios Pharmaceuticals, Inc. | Pyruvate kinase activators for use in therapy |
US10029987B2 (en) | 2009-06-29 | 2018-07-24 | Agios Pharmaceuticals, Inc. | Therapeutic compounds and compositions |
US11234976B2 (en) | 2015-06-11 | 2022-02-01 | Agios Pharmaceuticals, Inc. | Methods of using pyruvate kinase activators |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK288287A (en) * | 1986-06-09 | 1987-12-10 | Pfizer | HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL PREPARATIONS FOR TREATMENT OF ALLERGIC OR INFLAMMATORY CONDITIONS |
JPH0283376A (en) * | 1988-09-19 | 1990-03-23 | Pfizer Pharmaceut Co Ltd | Benzoxazolone derivative and antiallergic or anti-inflammatory composition |
IL93473A0 (en) * | 1989-02-28 | 1990-11-29 | Pfizer | Antiinflammatory benzoxazolones |
FR2646350B1 (en) * | 1989-04-28 | 1991-06-28 | Adir | NOVEL BENZOTHIAZOLINON DERIVATIVES, THEIR PREPARATION PROCESS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME |
US5166353A (en) * | 1989-04-28 | 1992-11-24 | Adir Et Compagnie | Benzothiazolinone compounds |
JPH0678327B2 (en) * | 1989-07-20 | 1994-10-05 | ファイザー製薬株式会社 | 4,5,6,7, -tetrasubstituted benzoxazolones |
JPH06759B2 (en) * | 1989-09-22 | 1994-01-05 | ファイザー製薬株式会社 | Novel benzimidazole compound |
JPH0717589B2 (en) * | 1990-01-22 | 1995-03-01 | ファイザー製薬株式会社 | Novel 1,3-dicarbonyl compound and composition thereof |
US7022480B1 (en) | 2001-10-11 | 2006-04-04 | The Regents Of The University Of California | Exons of the hSKCa3/KCNN3 gene |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2244507A1 (en) * | 1973-06-26 | 1975-04-18 | Inst Nat Sante Rech Med | Chalcones and analogues - analgesics having low toxicity |
FR2244506B1 (en) * | 1973-06-26 | 1977-02-25 | Inst Nat Sante Rech Med | |
DE2634787C2 (en) * | 1976-08-03 | 1983-01-27 | Hoechst Ag, 6000 Frankfurt | Process for the preparation of sulfuric acid half-ester compounds and their use |
JPS5697268A (en) * | 1979-12-28 | 1981-08-05 | Fujisawa Pharmaceut Co Ltd | Lower alkanoic acid derivative, salt and preparation thereof and preventing agent and remedy for diabetic complication containing the same as active constituent |
FR2491066A1 (en) * | 1980-09-29 | 1982-04-02 | Cerm Cent Europ Rech Mauvernay | BENZOXAZOLINONES SUBSTITUTED IN 6 BY AN AMINOALCOHOL OR AMINOCETONE CHAIN, THEIR PREPARATION AND THEIR THERAPEUTIC USE |
-
1983
- 1983-09-22 GB GB838325370A patent/GB8325370D0/en active Pending
-
1984
- 1984-09-20 WO PCT/JP1984/000452 patent/WO1985001289A1/en unknown
- 1984-09-20 AU AU34317/84A patent/AU3431784A/en not_active Abandoned
- 1984-09-21 IT IT2278584A patent/IT1176770B/en active
Cited By (20)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US9657004B2 (en) | 2009-04-06 | 2017-05-23 | Agios Pharmaceuticals, Inc | Pyruvate kinase M2 modulators, therapeutic compositions and related methods of use |
US8742119B2 (en) | 2009-04-06 | 2014-06-03 | Agios Pharmaceuticals, Inc. | Pyruvate kinase M2 modulators, therapeutic compositions and related methods of use |
US9938259B2 (en) | 2009-04-06 | 2018-04-10 | Agios Pharmaceuticals, Inc. | Therapeutic compositions and related methods of use |
WO2010129596A1 (en) * | 2009-05-04 | 2010-11-11 | Agios Pharmaceuticals, Inc. | Pmk2 modulators for use in the treatment of cancer |
US10988448B2 (en) | 2009-06-29 | 2021-04-27 | Agios Pharmaceuticals, Inc. | Therapeutic compounds and compositions |
US11866411B2 (en) | 2009-06-29 | 2024-01-09 | Agios Pharmaceutical, Inc. | Therapeutic compounds and compositions |
USRE49582E1 (en) | 2009-06-29 | 2023-07-18 | Agios Pharmaceuticals, Inc. | Therapeutic compounds and compositions |
US9115086B2 (en) | 2009-06-29 | 2015-08-25 | Agios Pharmaceuticals, Inc. | Therapeutic compositions and related methods of use |
US10029987B2 (en) | 2009-06-29 | 2018-07-24 | Agios Pharmaceuticals, Inc. | Therapeutic compounds and compositions |
US9221792B2 (en) | 2010-12-17 | 2015-12-29 | Agios Pharmaceuticals, Inc | N-(4-(azetidine-1-carbonyl) phenyl)-(hetero-) arylsulfonamide derivatives as pyruvate kinase M2 (PMK2) modulators |
US9328077B2 (en) | 2010-12-21 | 2016-05-03 | Agios Pharmaceuticals, Inc | Bicyclic PKM2 activators |
US10087169B2 (en) | 2010-12-21 | 2018-10-02 | Agios Pharmaceuticals, Inc. | Bicyclic PKM2 activators |
US9199968B2 (en) | 2010-12-29 | 2015-12-01 | Agios Pharmaceuticals, Inc. | Therapeutic compounds and compositions |
US8889667B2 (en) | 2010-12-29 | 2014-11-18 | Agios Pharmaceuticals, Inc | Therapeutic compounds and compositions |
US10632114B2 (en) | 2011-05-03 | 2020-04-28 | Agios Pharmaceuticals, Inc. | Pyruvate kinase activators for use in therapy |
US9980961B2 (en) | 2011-05-03 | 2018-05-29 | Agios Pharmaceuticals, Inc. | Pyruvate kinase activators for use in therapy |
US9181231B2 (en) | 2011-05-03 | 2015-11-10 | Agios Pharmaceuticals, Inc | Pyruvate kinase activators for use for increasing lifetime of the red blood cells and treating anemia |
US11793806B2 (en) | 2011-05-03 | 2023-10-24 | Agios Pharmaceuticals, Inc. | Pyruvate kinase activators for use in therapy |
US9365545B2 (en) | 2013-03-15 | 2016-06-14 | Agios Pharmaceuticals, Inc | Therapeutic compounds and compositions |
US11234976B2 (en) | 2015-06-11 | 2022-02-01 | Agios Pharmaceuticals, Inc. | Methods of using pyruvate kinase activators |
Also Published As
Publication number | Publication date |
---|---|
GB8325370D0 (en) | 1983-10-26 |
WO1985001289A1 (en) | 1985-03-28 |
IT8422785A1 (en) | 1986-03-21 |
IT8422785A0 (en) | 1984-09-21 |
AU3431784A (en) | 1985-04-23 |
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