IT1171091B - BIOLOGICALLY ACTIVE 2,5-PIPERAZINDION DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM - Google Patents
BIOLOGICALLY ACTIVE 2,5-PIPERAZINDION DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEMInfo
- Publication number
 - IT1171091B IT1171091B IT23058/83A IT2305883A IT1171091B IT 1171091 B IT1171091 B IT 1171091B IT 23058/83 A IT23058/83 A IT 23058/83A IT 2305883 A IT2305883 A IT 2305883A IT 1171091 B IT1171091 B IT 1171091B
 - Authority
 - IT
 - Italy
 - Prior art keywords
 - piperazindion
 - derivatives
 - contain
 - processes
 - preparation
 - Prior art date
 
Links
Classifications
- 
        
- C—CHEMISTRY; METALLURGY
 - C07—ORGANIC CHEMISTRY
 - C07D—HETEROCYCLIC COMPOUNDS
 - C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
 - C07D241/36—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems
 - C07D241/38—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems with only hydrogen or carbon atoms directly attached to the ring nitrogen atoms
 
 - 
        
- A—HUMAN NECESSITIES
 - A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
 - A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
 - A61P25/00—Drugs for disorders of the nervous system
 
 
Landscapes
- Chemical & Material Sciences (AREA)
 - Organic Chemistry (AREA)
 - Health & Medical Sciences (AREA)
 - Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
 - Pharmacology & Pharmacy (AREA)
 - Neurosurgery (AREA)
 - Biomedical Technology (AREA)
 - Chemical Kinetics & Catalysis (AREA)
 - General Chemical & Material Sciences (AREA)
 - Medicinal Chemistry (AREA)
 - Bioinformatics & Cheminformatics (AREA)
 - Engineering & Computer Science (AREA)
 - Neurology (AREA)
 - Life Sciences & Earth Sciences (AREA)
 - Animal Behavior & Ethology (AREA)
 - General Health & Medical Sciences (AREA)
 - Public Health (AREA)
 - Veterinary Medicine (AREA)
 - Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
 - Peptides Or Proteins (AREA)
 - Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
 - Nitrogen Condensed Heterocyclic Rings (AREA)
 - Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
 
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title | 
|---|---|---|---|
| CS827012A CS231227B1 (en) | 1982-10-01 | 1982-10-01 | 2,5-pierazindion derivatives | 
Publications (3)
| Publication Number | Publication Date | 
|---|---|
| IT8323058A0 IT8323058A0 (en) | 1983-09-29 | 
| IT8323058A1 IT8323058A1 (en) | 1985-03-29 | 
| IT1171091B true IT1171091B (en) | 1987-06-10 | 
Family
ID=5418454
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date | 
|---|---|---|---|
| IT23058/83A IT1171091B (en) | 1982-10-01 | 1983-09-29 | BIOLOGICALLY ACTIVE 2,5-PIPERAZINDION DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM | 
Country Status (12)
| Country | Link | 
|---|---|
| JP (1) | JPS5989671A (en) | 
| AT (1) | AT388161B (en) | 
| BE (1) | BE897843A (en) | 
| CH (1) | CH655929A5 (en) | 
| CS (1) | CS231227B1 (en) | 
| DE (1) | DE3335891C2 (en) | 
| FR (1) | FR2533919B1 (en) | 
| GB (1) | GB2127807B (en) | 
| HU (1) | HU193047B (en) | 
| IT (1) | IT1171091B (en) | 
| SE (1) | SE466654B (en) | 
| YU (1) | YU44751B (en) | 
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title | 
|---|---|---|---|---|
| CS277405B6 (en) * | 1986-06-12 | 1993-03-17 | Vyzk Ustav Farm Biochem Sp | Peptides with 1-amino-1-cycloalkane carboxylic acid | 
| US5182285A (en) * | 1986-11-07 | 1993-01-26 | Spojene Podniky Pro Zdravotnickou Vyrobu | Cell-protective composition for preventing or treating of peptic ulcer | 
| GB8822674D0 (en) * | 1988-09-27 | 1988-11-02 | Tate & Lyle Plc | Preparation of acylated sucrose derivatives | 
| US7202279B1 (en) * | 1998-02-11 | 2007-04-10 | Georgetown University | Cyclic dipeptides and azetidinone compounds and their use in treating CNS injury and neurodegenerative disorders | 
| NZ519183A (en) | 1999-12-03 | 2005-02-25 | Ono Pharmaceutical Co | Triazaspiro[5.5]undecane derivatives and pharmaceutical compositions comprising thereof, as an active ingredient | 
| CA2441162A1 (en) * | 2001-03-19 | 2002-09-26 | Ono Pharmaceutical Co., Ltd. | Pharmaceutical composition comprising, as an active ingredient, triazaspiro[5.5]undecane derivative | 
| JP3975226B2 (en) | 2006-01-11 | 2007-09-12 | 生化学工業株式会社 | Cycloalkylcarbonylamino acid derivative and process for producing the same | 
| JP4047365B2 (en) | 2006-01-11 | 2008-02-13 | 生化学工業株式会社 | Cycloalkanecarboxamide derivative and method for producing the same | 
| AU2007205578B2 (en) | 2006-01-11 | 2012-06-28 | Seikagaku Corporation | Cycloalkylcarbonylamino acid ester derivative and process for producing the same | 
| WO2013020527A1 (en) | 2011-08-11 | 2013-02-14 | University Of Veterinary And Pharmaceutical Sciences Brno Faculty Of Pharmacy | Utilization of alaptide as transdermal penetration modifier in pharmaceutical compositions for human and veterinary applications containing anti-inflammatory drugs and/or antimicrobial chemotherapeutics | 
| WO2014019556A1 (en) | 2012-08-02 | 2014-02-06 | University Of Veterinary And Pharmaceutical Sciences Brno Faculty Of Pharmacy | Alaptide : methods of effecting its solubility, membrane permeation and pharmaceutical compositions for human and/or veterinary applications | 
| CN107903303B (en) * | 2017-11-20 | 2021-06-04 | 陕西慧康生物科技有限责任公司 | A kind of liquid phase synthesis method of cyclic peptide Alaptide | 
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title | 
|---|---|---|---|---|
| GB1459488A (en) * | 1974-03-19 | 1976-12-22 | Wyeth John & Brother Ltd | Piperazinedione derivatives | 
- 
        1982
        
- 1982-10-01 CS CS827012A patent/CS231227B1/en unknown
 
 - 
        1983
        
- 1983-09-14 GB GB08324683A patent/GB2127807B/en not_active Expired
 - 1983-09-21 AT AT0336683A patent/AT388161B/en not_active IP Right Cessation
 - 1983-09-23 SE SE8305157A patent/SE466654B/en not_active IP Right Cessation
 - 1983-09-26 CH CH5208/83A patent/CH655929A5/en not_active IP Right Cessation
 - 1983-09-27 BE BE0/211589A patent/BE897843A/en not_active IP Right Cessation
 - 1983-09-29 IT IT23058/83A patent/IT1171091B/en active
 - 1983-09-29 YU YU1952/83A patent/YU44751B/en unknown
 - 1983-09-30 FR FR8315599A patent/FR2533919B1/en not_active Expired
 - 1983-09-30 HU HU833419A patent/HU193047B/en not_active IP Right Cessation
 - 1983-10-01 JP JP58181834A patent/JPS5989671A/en active Granted
 - 1983-10-03 DE DE3335891A patent/DE3335891C2/en not_active Expired - Fee Related
 
 
Also Published As
| Publication number | Publication date | 
|---|---|
| DE3335891A1 (en) | 1984-04-05 | 
| FR2533919A1 (en) | 1984-04-06 | 
| GB2127807B (en) | 1987-02-25 | 
| CH655929A5 (en) | 1986-05-30 | 
| SE8305157D0 (en) | 1983-09-23 | 
| GB8324683D0 (en) | 1983-10-19 | 
| YU44751B (en) | 1991-02-28 | 
| CS231227B1 (en) | 1984-10-15 | 
| IT8323058A1 (en) | 1985-03-29 | 
| YU195283A (en) | 1986-10-31 | 
| BE897843A (en) | 1984-01-16 | 
| ATA336683A (en) | 1988-10-15 | 
| CS701282A1 (en) | 1984-01-16 | 
| HU193047B (en) | 1987-08-28 | 
| JPH0526782B2 (en) | 1993-04-19 | 
| DE3335891C2 (en) | 1993-11-11 | 
| GB2127807A (en) | 1984-04-18 | 
| FR2533919B1 (en) | 1986-10-03 | 
| SE466654B (en) | 1992-03-16 | 
| AT388161B (en) | 1989-05-10 | 
| IT8323058A0 (en) | 1983-09-29 | 
| SE8305157L (en) | 1984-04-02 | 
| JPS5989671A (en) | 1984-05-23 | 
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Legal Events
| Date | Code | Title | Description | 
|---|---|---|---|
| TA | Fee payment date (situation as of event date), data collected since 19931001 | 
             Effective date: 19960928  |