IT1170307B - CEPHALOSPORINIC DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION - Google Patents

CEPHALOSPORINIC DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION

Info

Publication number
IT1170307B
IT1170307B IT47826/83A IT4782683A IT1170307B IT 1170307 B IT1170307 B IT 1170307B IT 47826/83 A IT47826/83 A IT 47826/83A IT 4782683 A IT4782683 A IT 4782683A IT 1170307 B IT1170307 B IT 1170307B
Authority
IT
Italy
Prior art keywords
cephalosporinic
derivatives
procedure
preparation
cephalosporinic derivatives
Prior art date
Application number
IT47826/83A
Other languages
Italian (it)
Other versions
IT8347826A0 (en
Inventor
Shimpei Aburaki
Hajime Kamachi
Yukio Marita
Jun Okumura
Takayuki Naito
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/354,851 external-priority patent/US4406899A/en
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of IT8347826A0 publication Critical patent/IT8347826A0/en
Application granted granted Critical
Publication of IT1170307B publication Critical patent/IT1170307B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/247-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/38Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof
    • C07D501/46Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof with the 7-amino radical acylated by carboxylic acids containing hetero rings
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
IT47826/83A 1982-03-04 1983-03-01 CEPHALOSPORINIC DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION IT1170307B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/354,851 US4406899A (en) 1982-03-04 1982-03-04 Cephalosporins
US35753482A 1982-03-12 1982-03-12

Publications (2)

Publication Number Publication Date
IT8347826A0 IT8347826A0 (en) 1983-03-01
IT1170307B true IT1170307B (en) 1987-06-03

Family

ID=26998584

Family Applications (1)

Application Number Title Priority Date Filing Date
IT47826/83A IT1170307B (en) 1982-03-04 1983-03-01 CEPHALOSPORINIC DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION

Country Status (29)

Country Link
KR (1) KR870001986B1 (en)
AT (2) AT382155B (en)
AU (1) AU562776B2 (en)
BE (1) BE896086A (en)
CA (1) CA1213882A (en)
CH (1) CH654313A5 (en)
CS (1) CS249512B2 (en)
DD (1) DD210280A5 (en)
DE (1) DE3307550A1 (en)
DK (1) DK156900C (en)
EG (1) EG15934A (en)
ES (2) ES8403919A1 (en)
FI (1) FI74973C (en)
FR (1) FR2522659B1 (en)
GB (1) GB2116180B (en)
GR (1) GR77916B (en)
HU (1) HU193158B (en)
IE (1) IE56647B1 (en)
IL (1) IL68011A0 (en)
IT (1) IT1170307B (en)
LU (1) LU84674A1 (en)
MY (1) MY8700943A (en)
NL (2) NL193284C (en)
NZ (1) NZ203312A (en)
PH (1) PH18002A (en)
PT (1) PT76330B (en)
SE (1) SE453091B (en)
SU (1) SU1250173A3 (en)
YU (2) YU43822B (en)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3409431A1 (en) * 1983-10-08 1985-04-18 Hoechst Ag, 6230 Frankfurt CEPHALOSPORINE DERIVATIVES AND METHOD FOR THEIR PRODUCTION
DE3404906A1 (en) * 1984-02-11 1985-08-14 Bayer Ag, 5090 Leverkusen 1-OXADETHIACEPHALOSPORINE DERIVATIVES AND METHOD FOR THE PRODUCTION THEREOF
DE3419013A1 (en) * 1984-05-22 1985-11-28 Bayer Ag, 5090 Leverkusen NEW CEPHALOSPORINE AND METHOD FOR THEIR PRODUCTION
GB8424692D0 (en) * 1984-10-01 1984-11-07 Glaxo Group Ltd Chemical compounds
US4698336A (en) * 1985-01-30 1987-10-06 Eisai Co., Ltd. 3-(pyrrolidinio)methyl-3-cephem derivatives
FR2585705B1 (en) * 1985-08-05 1989-01-13 Bristol Myers Co CEPHALOSPORIN SALTS AND INJECTABLE COMPOSITIONS
US4910301A (en) * 1985-08-05 1990-03-20 Bristol-Myers Company Cefepime cephalosporin salts
US4808617A (en) * 1985-12-18 1989-02-28 Bristol-Myers Company Lyophilized or precipitated cephalosporin zwitterion and salt combination
DE3789466T2 (en) * 1986-03-17 1994-07-28 Fujisawa Pharmaceutical Co 3,7-disubstituted-3-cephem compounds and process for their preparation.
CA2011116C (en) * 1989-03-06 1999-11-16 Murray A. Kaplan Lyophilized bmy-28142 dihydrochloride for parenteral use
DE69231815T2 (en) 1991-03-08 2001-09-27 Biochemie Gmbh Process for the preparation of cephalosporins and intermediates in this process
MY108872A (en) * 1991-09-10 1996-11-30 Bristol Myers Squibb Co Preparation of a cephalosporin antibiotic using the syn-isomer of a thiazolyl intermediate.
YU81692A (en) * 1991-09-10 1995-03-27 Bristol-Myers Co. PROCEDURE FOR THE PRODUCTION OF CEPHALOSPORIN ANTIBIOTICS
US5523400A (en) * 1993-04-16 1996-06-04 Hoffmann-La Roche Inc. Cephalosporin antibiotics
EP1699804B1 (en) * 2003-12-23 2008-02-06 Sandoz Gmbh Process for production of intermediates for use in cefalosporin synthesis

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2715385A1 (en) * 1976-04-14 1977-11-10 Takeda Chemical Industries Ltd CEPHALOSPORIN DERIVATIVES, THE PROCESS FOR THEIR MANUFACTURING AND MEDICINAL PRODUCTS CONTAINING THEM
GB1591439A (en) * 1976-10-01 1981-06-24 Glaxo Operations Ltd 7-syn (oxyimino -acylamido) cephalosporins
AR228726A1 (en) * 1978-05-26 1983-04-15 Glaxo Group Ltd PROCEDURE FOR THE PREPARATION OF ANTIBIOTIC (6R, 7R) -7 - ((Z) -2- (2-AMINOTIAZOL-4-IL) -2- (2-CARBOXIPROP-2-OXIIMINO) ACETAMIDO) -3- (1- PIRIDINIOMETIL) CEF-3-EM-4-CARBOXILATO
CA1131618A (en) * 1978-10-27 1982-09-14 Cynthia H. O'callaghan Cephalosporin compounds
US4443444A (en) * 1980-08-11 1984-04-17 Fujisawa Pharmaceutical Co., Ltd. Cephem compounds

Also Published As

Publication number Publication date
GR77916B (en) 1984-09-25
KR870001986B1 (en) 1987-10-24
FI74973C (en) 1988-04-11
ATA228285A (en) 1987-05-15
DE3307550A1 (en) 1983-09-15
DK156900C (en) 1990-03-12
DK156900B (en) 1989-10-16
GB2116180A (en) 1983-09-21
LU84674A1 (en) 1983-11-17
EG15934A (en) 1987-10-30
PH18002A (en) 1985-02-28
IL68011A0 (en) 1983-06-15
BE896086A (en) 1983-09-05
HU193158B (en) 1987-08-28
DD210280A5 (en) 1984-06-06
GB8305940D0 (en) 1983-04-07
YU52383A (en) 1986-02-28
CS249512B2 (en) 1987-03-12
AU562776B2 (en) 1987-06-18
MY8700943A (en) 1987-12-31
CH654313A5 (en) 1986-02-14
FI830689L (en) 1983-09-05
ES526397A0 (en) 1985-09-16
ES8507557A1 (en) 1985-09-16
AT384612B (en) 1987-12-10
NL990039I1 (en) 2000-01-03
FI74973B (en) 1987-12-31
KR840004118A (en) 1984-10-06
IE830455L (en) 1983-09-04
YU149685A (en) 1986-02-28
NL8300755A (en) 1983-10-03
ES520224A0 (en) 1984-04-01
AT382155B (en) 1987-01-26
PT76330A (en) 1983-04-01
NZ203312A (en) 1985-12-13
NL193284C (en) 1999-05-06
ATA76183A (en) 1986-06-15
DK86283D0 (en) 1983-02-24
AU1130483A (en) 1983-09-08
NL990039I2 (en) 2000-04-03
FI830689A0 (en) 1983-03-01
GB2116180B (en) 1985-09-18
SE453091B (en) 1988-01-11
SE8301178L (en) 1983-09-05
FR2522659B1 (en) 1986-10-24
SE8301178D0 (en) 1983-03-03
FR2522659A1 (en) 1983-09-09
PT76330B (en) 1986-02-04
DK86283A (en) 1983-09-05
IT8347826A0 (en) 1983-03-01
IE56647B1 (en) 1991-10-23
DE3307550C2 (en) 1988-11-24
CA1213882A (en) 1986-11-12
NL193284B (en) 1999-01-04
YU43822B (en) 1989-12-31
YU44777B (en) 1991-02-28
SU1250173A3 (en) 1986-08-07
ES8403919A1 (en) 1984-04-01

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Legal Events

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TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19970329