IT1149118B - Derivati di esteri arilici della 2-idrossipropilammina ad attivita' beta-bloccante - Google Patents
Derivati di esteri arilici della 2-idrossipropilammina ad attivita' beta-bloccanteInfo
- Publication number
- IT1149118B IT1149118B IT49477/82A IT4947782A IT1149118B IT 1149118 B IT1149118 B IT 1149118B IT 49477/82 A IT49477/82 A IT 49477/82A IT 4947782 A IT4947782 A IT 4947782A IT 1149118 B IT1149118 B IT 1149118B
- Authority
- IT
- Italy
- Prior art keywords
- hydroxypropilamine
- beta
- ester derivatives
- aryl ester
- blocking activity
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
- C07D295/215—Radicals derived from nitrogen analogues of carbonic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C275/00—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
- C07C275/04—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to acyclic carbon atoms
- C07C275/06—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to acyclic carbon atoms of an acyclic and saturated carbon skeleton
- C07C275/14—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to acyclic carbon atoms of an acyclic and saturated carbon skeleton being further substituted by nitrogen atoms not being part of nitro or nitroso groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C275/00—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
- C07C275/28—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/320,773 US4582855A (en) | 1981-11-12 | 1981-11-12 | Aromatic and esters of hydroxypropylamines |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IT8249477A0 IT8249477A0 (it) | 1982-11-12 |
| IT1149118B true IT1149118B (it) | 1986-12-03 |
Family
ID=23247815
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IT49477/82A IT1149118B (it) | 1981-11-12 | 1982-11-12 | Derivati di esteri arilici della 2-idrossipropilammina ad attivita' beta-bloccante |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US4582855A (it) |
| EP (1) | EP0093765B1 (it) |
| JP (2) | JPS6320424B1 (it) |
| AU (1) | AU562862B2 (it) |
| CA (1) | CA1201438A (it) |
| DE (1) | DE3274640D1 (it) |
| EG (1) | EG16198A (it) |
| ES (4) | ES8401014A1 (it) |
| GR (1) | GR78306B (it) |
| IL (1) | IL67243A0 (it) |
| IT (1) | IT1149118B (it) |
| NZ (1) | NZ202228A (it) |
| WO (1) | WO1983001770A1 (it) |
| ZA (1) | ZA827749B (it) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1988007044A1 (en) * | 1987-03-17 | 1988-09-22 | Insite Vision, Inc. | Timolol derivatives |
| JPH0662521B2 (ja) * | 1988-02-24 | 1994-08-17 | 日東紡績株式会社 | 新規コリン誘導体及びそれを用いた血清コリンエステラーゼ活性測定法 |
| US5064827A (en) * | 1988-12-15 | 1991-11-12 | Du Pont Merck Pharmaceutical Company | Polyhydroxybenzyloxpropanolamines |
| US4935422A (en) * | 1988-12-15 | 1990-06-19 | E. I. Du Pont De Nemours And Company | Acyloxypropanolamines |
| US4897417A (en) * | 1988-12-15 | 1990-01-30 | E. I. Du Pont De Nemours & Co. | Prodrugs of 3,4-hydroxy benzoyloxypropanolamines |
| US4966914A (en) * | 1988-12-15 | 1990-10-30 | E. I. Du Pont De Nemours And Company | Oculoselective beta-blockers as antiglaucoma agents |
| US5248808A (en) * | 1989-11-01 | 1993-09-28 | Avery Dennison Corporation | Vinyl functional reactive tackifiers for pressure-sensitive adhesives |
| JPH04343212A (ja) * | 1991-05-20 | 1992-11-30 | Hitachi Aic Inc | ヒューズ付コンデンサ |
| US5629345A (en) * | 1993-07-23 | 1997-05-13 | Vide Pharmaceuticals | Methods and compositions for ATP-sensitive K+ channel inhibition for lowering intraocular pressure |
| US5965620A (en) * | 1993-07-23 | 1999-10-12 | Vide Pharmaceuticals | Methods and compositions for ATP-sensitive K+ channel inhibition for lowering intraocular pressure |
| US5543083A (en) * | 1994-07-26 | 1996-08-06 | The Procter & Gamble Company | Fatty amine derivatives of butylated hydroxy toluene for the protection of surfaces from physical and chemical degradation |
| US5536749A (en) * | 1994-10-13 | 1996-07-16 | Sl Pharmaceuticals, Inc. | Method for attenuation of sympathetic nervous system activity or onset of migraine by selectively metabolized beta-blocking agents |
| JP2002511445A (ja) * | 1998-04-14 | 2002-04-16 | サムスン ファイン ケミカルズ カンパニー リミテッド | キラル（ｓ）−２，３−二置換−１−プロピルアミン誘導体の製造方法 |
| US8115031B2 (en) * | 2007-11-09 | 2012-02-14 | Yates Charles R | Anti-inflammatory quinic acid derivatives for oral administration |
| EP2096105A1 (en) * | 2008-02-28 | 2009-09-02 | Laboratorios Almirall, S.A. | Derivatives of 4-(2-amino-1-hydroxyethyl)phenol as agonists of the b2 adrenergic receptor |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US1476934A (en) * | 1922-02-13 | 1923-12-11 | Abbott Lab | Anaesthetic compound |
| US3129201A (en) * | 1959-10-30 | 1964-04-14 | Monsanto Chemicals | Alkyl 3-acyloxy-2-alkenoates and homopolymers thereof |
| NL301580A (it) * | 1962-12-11 | |||
| US4405642A (en) * | 1980-11-28 | 1983-09-20 | American Hospital Supply Corporation | Method for treatment or prophylaxis of cardiac disorders |
| US4387103A (en) * | 1980-11-28 | 1983-06-07 | American Hospital Supply Corporation | Method for treatment or prophylaxis of cardiac disorders |
-
1981
- 1981-11-12 US US06/320,773 patent/US4582855A/en not_active Expired - Lifetime
-
1982
- 1982-10-20 NZ NZ202228A patent/NZ202228A/en unknown
- 1982-10-22 ZA ZA827749A patent/ZA827749B/xx unknown
- 1982-10-28 WO PCT/US1982/001536 patent/WO1983001770A1/en active IP Right Grant
- 1982-10-28 DE DE8282903569T patent/DE3274640D1/de not_active Expired
- 1982-10-28 JP JP82503552A patent/JPS6320424B1/ja active Pending
- 1982-10-28 JP JP57503552A patent/JPS58501724A/ja active Pending
- 1982-10-28 AU AU10120/83A patent/AU562862B2/en not_active Ceased
- 1982-10-28 EP EP82903569A patent/EP0093765B1/en not_active Expired
- 1982-11-10 CA CA000415282A patent/CA1201438A/en not_active Expired
- 1982-11-10 GR GR69775A patent/GR78306B/el unknown
- 1982-11-11 ES ES517296A patent/ES8401014A1/es not_active Expired
- 1982-11-12 IL IL67243A patent/IL67243A0/xx not_active IP Right Cessation
- 1982-11-12 IT IT49477/82A patent/IT1149118B/it active
- 1982-11-13 EG EG671/82A patent/EG16198A/xx active
-
1983
- 1983-07-01 ES ES523804A patent/ES523804A0/es active Granted
- 1983-07-01 ES ES523805A patent/ES8500888A1/es not_active Expired
-
1984
- 1984-03-20 ES ES530788A patent/ES8505942A1/es not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| ES517296A0 (es) | 1983-12-01 |
| IT8249477A0 (it) | 1982-11-12 |
| NZ202228A (en) | 1985-10-11 |
| WO1983001770A1 (en) | 1983-05-26 |
| ES8500887A1 (es) | 1984-11-01 |
| EP0093765A4 (en) | 1984-04-27 |
| JPS6320424B1 (it) | 1988-04-27 |
| ES523805A0 (es) | 1984-11-01 |
| ES530788A0 (es) | 1985-06-01 |
| CA1201438A (en) | 1986-03-04 |
| GR78306B (it) | 1984-09-26 |
| EP0093765A1 (en) | 1983-11-16 |
| ES523804A0 (es) | 1984-11-01 |
| US4582855A (en) | 1986-04-15 |
| ES8505942A1 (es) | 1985-06-01 |
| AU562862B2 (en) | 1987-06-18 |
| ES8500888A1 (es) | 1984-11-01 |
| DE3274640D1 (de) | 1987-01-22 |
| EP0093765B1 (en) | 1986-12-10 |
| JPS58501724A (ja) | 1983-10-13 |
| ES8401014A1 (es) | 1983-12-01 |
| ZA827749B (en) | 1983-08-31 |
| IL67243A0 (en) | 1983-03-31 |
| EG16198A (en) | 1987-09-30 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| IT8448492A0 (it) | Derivati di gangliosidi | |
| IT1153080B (it) | Esteri ed amidi di 13,14-dideidro prostaglandine | |
| IT8519512A0 (it) | Derivati naturali ad attivita'farmacologica | |
| IT1149118B (it) | Derivati di esteri arilici della 2-idrossipropilammina ad attivita' beta-bloccante | |
| IT1097314B (it) | Derivati dell'imidazolo ad attivita' anticonvulsivante | |
| FI823795L (fi) | Foerfarande foer framstaellning av torkade nudlar och liknande | |
| IT1149117B (it) | Esteri di derivati della arilossi-propanolammina aventi attivita' beta-bloccante | |
| FR2646441B1 (fr) | Procede d'electrosynthese d'un ester beta gamma insature | |
| IT1159698B (it) | Derivati 5-nitro-imidazolici della piperazina ad attivita' antiprotozoica | |
| FR2579597B1 (fr) | Esters d'alceneamidocephalosporines | |
| IT8620037A1 (it) | Anello di sostegno | |
| IT7948449A0 (it) | Derivati di 3,3-dicloro-2-azetidino ne ad attivita' anti-infiammatoria | |
| IT8025285A0 (it) | Derivati di prostagliandina e prostaciclina ad attivita'farmacologica. | |
| IT1185514B (it) | Promedicinali di ossicam antiinfiammatorie | |
| IT7948802A0 (it) | Derivati di n-alchenilmoranolina aventi attivita' farmacologica | |
| IT1094287B (it) | Derivati della 2-idrossimetil-pirazina aventi attivita' ipolipemizzante | |
| IT8521236A0 (it) | Amminoacil derivati di 4(5)-imidazolidinoni ad attivita | |
| IT7950523A0 (it) | Derivati carbamoil-piperazinici dotati di attivita' farmacologica | |
| IT1221196B (it) | Rivelatore ottico di punti di fumo | |
| IT1162702B (it) | Derivati di 11-alcanoil-4"-isonitril-oleandomicina | |
| IT8519442A0 (it) | Derivati di fenilpropargilammine | |
| FI810094L (fi) | Anordning foer klyvning av trae | |
| IT1173454B (it) | Derivati della pantetina ad attivita' antidislipemica | |
| IT8448728A1 (it) | Derivati amidici dell'acido 2 - (p-aminobenzil) butirrico e relativi esteri provvisti di attivita' ipolipidemizzante | |
| IT8220271A1 (it) | Derivati di eterociclici azotati dotati di attivita' fitoregolatrice |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| TA | Fee payment date (situation as of event date), data collected since 19931001 |
Effective date: 19941027 |