IT1135270B - 3-amidino-ansamicine - Google Patents

3-amidino-ansamicine

Info

Publication number
IT1135270B
IT1135270B IT19473/81A IT1947381A IT1135270B IT 1135270 B IT1135270 B IT 1135270B IT 19473/81 A IT19473/81 A IT 19473/81A IT 1947381 A IT1947381 A IT 1947381A IT 1135270 B IT1135270 B IT 1135270B
Authority
IT
Italy
Prior art keywords
ansamicine
amidino
Prior art date
Application number
IT19473/81A
Other languages
English (en)
Italian (it)
Other versions
IT8119473A0 (it
Inventor
Leonardo Marsili
Giovanni Fraceschi
Aurora Sanfilippo
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of IT8119473A0 publication Critical patent/IT8119473A0/it
Application granted granted Critical
Publication of IT1135270B publication Critical patent/IT1135270B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • A61P31/06Antibacterial agents for tuberculosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pulmonology (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IT19473/81A 1980-04-12 1981-02-03 3-amidino-ansamicine IT1135270B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8012168 1980-04-12

Publications (2)

Publication Number Publication Date
IT8119473A0 IT8119473A0 (it) 1981-02-03
IT1135270B true IT1135270B (it) 1986-08-20

Family

ID=10512762

Family Applications (1)

Application Number Title Priority Date Filing Date
IT19473/81A IT1135270B (it) 1980-04-12 1981-02-03 3-amidino-ansamicine

Country Status (5)

Country Link
US (1) US4327096A (cg-RX-API-DMAC10.html)
JP (1) JPS56161392A (cg-RX-API-DMAC10.html)
BE (1) BE888310A (cg-RX-API-DMAC10.html)
DE (1) DE3106229A1 (cg-RX-API-DMAC10.html)
IT (1) IT1135270B (cg-RX-API-DMAC10.html)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4447432A (en) * 1981-11-17 1984-05-08 Farmitalia Carlo Erba S.P.A. Azino rifamycins
IT1201963B (it) * 1983-03-24 1989-02-02 Prodotti Antibiotici Spa Derivati delle rifamicine e procedimento per la loro preparazione
GB8308166D0 (en) * 1983-03-24 1983-05-05 Erba Farmitalia Preparation of azinomethyl-rifamycins
US4652644A (en) * 1985-04-29 1987-03-24 Bristol-Myers Company Process for preparation of N7 -amidino substituted mitomycin C derivatives
US4631290A (en) * 1985-08-29 1986-12-23 American Home Products Corporation Method of treating hepatitis
US4743619A (en) * 1985-08-29 1988-05-10 American Home Products Corporation Method of treating hepatitis
JPH02501926A (ja) * 1987-10-27 1990-06-28 チバ‐ガイギー アクチェンゲゼルシャフト 置換されたアザシクロヘキシル誘導体
US5003070A (en) * 1988-06-30 1991-03-26 Ciba-Geigy Corporation Substituted azacyclohexyl derivatives of rifamycins
DE69400631T2 (de) * 1993-05-05 1997-02-27 Palo Alto Medical Foundation, Palo Alto, Calif. Verwendung von rifamycinderivaten zur herstellung eines arzneimittels zur behandlung der toxoplasmose
US5529994A (en) * 1993-05-05 1996-06-25 Palo Alto Medical Foundation Treatment for toxoplasmosis
DE10216719B4 (de) * 2002-04-10 2007-09-20 Helmholtz-Zentrum Für Umweltforschung Gmbh - Ufz N-(3-Rifamycinyl)carbamate, Verfahren zu ihrer Herstellung und ihre Verwendung bei der Behandlung und Verhütung von Tuberkulose
US7247634B2 (en) * 2004-01-13 2007-07-24 Cumbre Pharmaceuticals Inc. Rifamycin derivatives effective against drug-resistant microbes

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH512510A (de) * 1965-08-24 1971-09-15 Ciba Geigy Ag Verfahren zur Herstellung von in 3-Stellung durch eine unsubstituierte oder substituierte Aminogruppe substituierten Derivaten von Rifamycin-S und Rifamycin-SV
IT1068367B (it) * 1975-11-12 1985-03-21 Archifar Ind Chim Trentino 3 aldimino rifamicine ad alta attivita antibiotica loro derivati e procedimento per ottenerle

Also Published As

Publication number Publication date
DE3106229A1 (de) 1981-12-10
IT8119473A0 (it) 1981-02-03
JPS6242916B2 (cg-RX-API-DMAC10.html) 1987-09-10
BE888310A (fr) 1981-07-31
JPS56161392A (en) 1981-12-11
US4327096A (en) 1982-04-27

Similar Documents

Publication Publication Date Title
BE891422A (fr) Degrilleur
FI811406L (fi) Faergtelevisionspresentationssystem
BR8107326A (pt) Container-tanque
IT1135270B (it) 3-amidino-ansamicine
JPS5754087A (ja) Shindoyokuseigatanohandorusochi
BR8101718A (pt) Microcentrais
BR8108640A (pt) Filatorio
BR8108621A (pt) Arpeu
BG33404A1 (bg) Registrovo aritmetichno ustrojjstvo
BE890439A (fr) Afdekbaanrol
BE891654A (fr) Schuifdeur
FI812149L (fi) Dispensionsanordning foer toalettapparater
FI811622L (fi) Elektroniskt taendroer foer projektiler
BG32324A1 (bg) Telopodavahho ustrojjstvo
JPS5754145A (ja) Jikarubonirukioryoshitabarupuroeetofukugotai
ES253183Y (es) Cantonera
BR8002799A (pt) Corredica
BR6001201U (pt) Veneziana
BR8007025A (pt) Vagonete monotrilho
BR8006091A (pt) Momicroencapsulacao
BR8006012A (pt) Vibra-som fasar
BR8005701A (pt) Conicaleira
BR8005450A (pt) Odontograma
BR8004979A (pt) Muchila bati-movel
DD150330A3 (de) Rechnerkoppelgeraet